Herbicidal sulfonamides

ABSTRACT

Benzenesulfonamide compounds such as N-[(4,6-dimethoxy-1,3,5-triazin-2-yl)aminocarbonyl]-1,4-dihydro-3-methyl-4-oxo-1-phenyl-indeno[1,2-C]-pyrazole-5-sulfonamide and N-[(4-methoxy-6-methyl-pyrimidin-2-yl)aminocarbonyl]-1,4-dihydro-3-methyl-4-oxo-1-phenyl-indeno[1,2-C]pyrazole-5-sulfonamide, agricultural compositions containing them, and their herbicidal utility are disclosed.

RELATED APPLICATION

This application is a continuation-in-part of my copending applicationU.S. Ser. No. 710,458, filed Mar. 11, 1985, now abandoned.

BACKGROUND OF THE INVENTION

The invention relates to novel benzenesulfonamide compounds,agriculturally suitable compositions containing them, and theirmethod-of-use as general and selective preemergent and postemergentherbicides.

European Patent Application (EP-A) No. 83,975 (published July 20, 1983)discloses herbicidal benzenesulfonamides of formula ##STR1## wherein Qis selected from various five or six-membered aromatic or partiallyunsaturated heterocyclic rings containing 2 or 3 heteroatoms selectedfrom O, S or NR.

EP-A-No. 85,476 (published Aug. 10, 1983) discloses herbicidalbenzenesulfonamides of formulae ##STR2## wherein Q is selected fromvarious 5-membered aromatic heterocycles, and their dihydro andtetrahydro analogs, which contain one heteroatom selected from O, S orNR, or Q is a saturated or partially unsaturated 6-membered ringcontaining one heteroatom selected from O or S; and

Q¹ is a 6-membered aromatic heterocycle containing one to three N atoms.

South African Patent Application No. 83/8416 (published May 12, 1984)discloses herbicidal benzenesulfonamides of formula ##STR3## wherein Ais an unsaturated or only partially saturated 5- or 6-memberedheterocyclic ring system which is bonded through a carbon atom andcontains 1, 2 or 3 heteroatoms.

EP-A-No. 79,683 (published May 25, 1983) discloses herbicidalbenzenesulfonamides including those of general Formulae I and II:##STR4## wherein Q is O, S or SO₂ ;

R₂ is H or C₁ -C₃ alkyl;

R₃ is H or CH₃ ;

R₄ is H or CH₃ ; and

A is a pyrimidinyl or triazinyl heterocyclic ring.

EP-A-No. 107,979 (published May 9, 1984) teaches herbicidal sulfonamidesof formula ##STR5## where J is, among other values, ##STR6## wherein nis 0, 1 or 2.

EP-A-No. 82,681 (published June 29, 1983) discloses herbicidal indane,1,3-benzodioxole and 1,4-benzodioxanesulfonylureas.

South African Patent Application No. 83/5165 (published Jan. 16, 1984)discloses herbicidal sulfonylureas of the general structure shown below:##STR7## wherein A is an unsubstituted or substituted bridge of 3 or 4atoms which contains 1 or 2 oxygen, sulfur or nitrogen atoms and,together with the linking carbon atom, forms a non-aromatic 5- or6-membered heterocyclic ring system, with the proviso that two oxygenatoms are separated by at least one carbon atom and that oxygen andsulfur atoms are only linked to each other if the sulfur atom takes theform of the --SO-- or SO₂ -- group.

SUMMARY OF THE INVENTION

This invention pertains to novel compounds of Formula I, agriculturallysuitable compositions containing them and their method of use as generaland/or selective preemergent and/or postemergent herbicides or plantgrowth regulants. ##STR8## wherein W is O or S:

Q is ##STR9## G is CH₂, CH₂ CH₂, O, S, NH, NCH₃ or CH═CH; G₁ is CH₂, CH₂CH₂ or CH═CH;

J is CH₂, C═O, S(O)_(m), O, NH, NCH₃, CHOH, CHOCH₃, CH(CH₃) or C(CH₃)OH;

J₁ is CH₂, C═O or SO₂ ;

n and n₁ are independently 0 or 1;

m is 0, 1 or 2;

E is a bridge of 3 or 4 atoms containing 0 to 2 heteroatoms selectedfrom the group consisting of oxygen, sulfur or nitrogen, wherein 1 atomof sulfur may take the form of SO or SO₂, said bridge also containing 1to 4 atoms of carbon wherein 1 atom of carbon may take the form of C═O,said bridge together with two attachment sites forming a non-aromaticheterocyclic or carbocyclic ring optionally substituted by 1 to 3substituent groups selected from the group L, or E is a bridge of 3 or 4atoms containing 0-1 heteroatoms of oxygen or sulfur and 0-3 heteroatomsof nigrogen, said bridge also containing 0-4 atoms of carbon, saidbridge together with two attachment sites forming an aromaticheterocyclic or carbocyclic ring optionally substituted by 1 to 3substituents selected from the group L, with the proviso that when Econtains two oxygen atoms or two sulfur atoms said atoms must beseparated by at least one atom of carbon and that oxygen and sulfur areonly linked to each other if the sulfur is in the form of SO or SO₂ ;

L is C₁ -C₄ alkyl, C₁ -C₄ haloalkyl, C₁ -C₄ alkoxy, C₁ -C₄ haloalkoxy,C₂ -C₈ alkoxyalkoxy, halogen, N(CH₃)₂, cyano, nitro, phenyl or phenylsubstituted with C₁ -C₃ alkyl, C₁ -C₃ haloalkyl, halogen, NO₂, C₁ -C₃alkoxy, C₁ -C₃ alkylthio, C₁ -C₃ alkylsulfinyl or C₁ -C₃ alkylsulfonyl;

R is H or CH₃ ;

R₁ is H, C₁ -C₃ alkyl, C₁ -C₃ haloalkyl, halogen, nitro, C₁ -C₃ alkoxy,SO₂ NR^(I) R^(II), C₁ -C₃ alkylthio, C₁ -C₃ alkylsulfinyl, C₁ -C₃alkylsulfonyl, CO₂ R^(III) or NR_(a) R_(b) ;

R^(I) is H, C₁ -C₄ alkyl, C₂ -C₃ cyanoalkyl, methoxy or ethoxy;

R^(II) is H, C₁ -C₄ alkyl or C₃ -C₄ alkenyl; or

R^(I) and R^(II) may be taken together as --(CH₂)₃ --, --(CH₂)₄ --,--(CH₂)₅ -- or --CH₂ CH₂ OCH₂ CH₂ --;

R^(III) is C₁ -C₄ alkyl, C₃ -C₄ alkenyl, C₃ -C₄ alkynyl, C₂ -C₄haloalkyl, C₁ -C₃ cyanoalkyl, C₅ -C₆ cycloalkyl, C₄ -C₇ cycloalkylalkylor C₂ -C₄ alkoxyalkyl;

R_(a) and R_(b) are independently H or C₁ -C₂ alkyl; A is ##STR10## X isH, C₁ -C₄ alkyl, C₁ -C₄ alkoxy, C₁ -C₄ haloalkoxy, C₁ -C₄ haloalkyl, C₁-C₄ haloalkylthio, C₁ -C₄ alkylthio, halogen, C₂ -C₅ alkoxyalkyl, C₂ -C₅alkoxyalkoxy, amino, C₁ -C₃ alkylamino or di(C₁ -C₃ alkyl)amino;

Y is H, C₁ -C₄ alkyl, C₁ -C₄ alkoxy, C₁ -C₄ haloalkoxy, haloalkylthio,C₁ -C₄ alkylthio, C₂ -C₅ alkoxyalkyl, C₂ -C₅ alkoxyalkoxy, amino, C₁ -C₃alkylamino, di(C₁ -C₃ alkyl)amino, C₃ -C₄ alkenyloxy, C₃ -C₄ alkynyloxy,C₂ -C₅ alkylthioalkyl, C₁ -C₄ haloalkyl, C₃ -C₅ cycloalkyl, C₂ -C₄alkynyl, N(OCH₃)CH₃, ##STR11## p is 2 or 3; L₁ and L₂ are independentlyO or S;

R₂ and R₃ are independently C₁ -C₂ alkyl;

R₄ is H or CH₃ ;

Z is CH or N;

Y₁ is O or CH₂ ;

X₁ is CH₃, OCH₃, OC₂ H₅ or OCF₂ H;

Y₂ is H or CH₃ ;

X₂ is CH₃, OCH₃ or SCH₃ ;

Y₃ is CH₃, CH₂ CH₃ or CH₂ CF₃ ;

X₃ is CH₃ or OCH₃ ;

X₄ is CH₃, OCH₃, OC₂ H₅, CH₂ OCH₃ or Cl; and

Y₄ is CH₃, OCH₃, OC₂ H₅ or Cl;

and their agriculturally suitable salts; provided that

(a) when X is Cl, F, Br or I, then Z is CH and Y is OCH₃, OC₂ H₅,N(OCH₃)CH₃, NHCH₃, N(CH₃)₂ or OCF₂ H;

(b) when X or Y is C₁ haloalkoxy, then Z is CH;

(c) n and n₁ cannot simultaneously be O;

(d) when G or G₁ is CH₂ CH₂ or CH═CH, then n is O;

(e) when Q is Q₁ and n is 1, then E must contain at least one heteroatomselected from oxygen, sulfur or nitrogen;

(f) when W is S, then A is A-1, R is H, and Y is CH₃, OCH₃, OC₂ H₅, CH₂OCH₃, C₂ H₅, CF₃, SCH₃, OCH₂ CH═CH₂, OCH₂ C.tbd.CH, OCH₂ CH₂ OCH₃,CH(OCH₃)₂ or ##STR12## and (g) X₄ and Y₄ cannot simultaneously be Cl.

In the above definitions, the term "alkyl" used either alone or incompound words such as "alkylthio" or "haloalkyl", denotes straightchain or branched alkyl, e.g., methyl, ethyl, n-propyl, isopropyl or thedifferent butyl isomers.

Alkoxy denotes methoxy, ethoxy, n-propoxy, isopropoxy and the differentbutyl isomers.

Alkenyl denotes straight chain or branched alkenes, e.g., vinyl,1-propenyl, 2-propenyl, 3-propenyl or the different butenyl isomers.

Alkynyl denotes straight chain or branched alkynes, e.g., ethynyl,1-propynyl, 2-propynyl and the different butynyl isomers.

Alkylsulfonyl denotes methylsulfonyl, ethylsulfonyl or the differentpropylsulfonyl isomers.

Alkylthio, alkylsulfinyl, alkylamino, etc. are defined in an analogousmanner.

Cycloalkyl means cyclopropyl, cyclobutyl, cyclopentyl and cyclohexyl.

The term "halogen", either alone or in compound words such as"haloalkyl", denotes fluorine, chlorine, bromine or iodine.

The total number of carbon atoms in a substituent group is indicated bythe C_(i) -C_(j) prefix where i and j are numbers from 1 to 7. Forexample, C₁ -C₃ alkylsulfonyl would designate methylsulfonyl throughpropylsulfonyl, C₂ alkoxyalkoxy would designate OCH₂ OCH₃, C₂ cyanoalkylwould designate CH₂ CN and C₃ cyanoalkyl would designate CH₂ CH₂ CN andCH(CN)CH₃. The term C₄ -C₇ cycloalkylalkyl is meant to definecyclopropylmethyl through cyclohexylmethyl or cyclopropylbutyl and thevarious structural isomers embraced therein.

Preferred for reasons of increased ease of synthesis and/or greaterherbicidal efficacy are:

(1) Compounds of Formula I where W is O; G and G₁ are CH₂, CH₂ CH₂ orCH═CH; J is CO, SO₂ or CH₂ ; R is H; X is CH₃, OCH₃, OCH₂ CH₃, Cl, F,Br, I, OCF₂ H, CH₂ F, OCH₂ CH₂ F, OCH₂ CHF₂, OCH₂ CF₃, CF₃, CH₂ Cl orCH₂ Br; Y is H, CH₃, OCH₃, OC₂ H₅, CH₂ OCH₃, NHCH₃, N(OCH₃)CH₃, N(CH₃)₂,CH₂ CH₃, CF₃, SCH₃, OCH₂ CH═CH₂, OCH₂ C.tbd.CH, CH₂ OCH₂ CH₃, OCH₂ CH₂OCH₃, CH₂ SCH₃, ##STR13## OCF₂ H, SCF₂ H, cyclopropyl, C.tbd.CH or orC.tbd.CCH₃ ; (2) Compounds of Preferred 1 where R₁ is H, CH₃, halogen,OCH₃, SCH₃ or SO₂ CH₃ ; A is A-1; and L is halogen, CH₃, OCH₃, SCH₃,NO₂, N(CH₃)₂ or phenyl.

(3) Compounds of Preferred 2 where Q is ##STR14## R₅ is H or CH₃ ; R₆ isH, CH₃ or phenyl;

R₇ is H or CH₃ ;

R₈ is H or CH₃ ;

R₉ is H, CH₃ or phenyl;

R₁₀ is H or CH₃ ;

R₁₁ is SCH₃, OCH₃, N(CH₃)₂ or CH₃ ;

R₁₂ is H or CH₃ ;

R₁₃ is H, CH₃, OCH₃ or SCH₃ ; and

R₁₄ is H, Cl, Br, F, CH₃, OCH₃ or NO₂.

(4) Compounds of Preferred 3 where X is CH₃, OCH₃, OCH₂ CH₃, Cl, OCF₂ Hor OCH₂ CF₃ ; and Y is CH₃, OCH₃, CH₂ CH₃, CH₂ OCH₃, NHCH₃ or CH(OCH₃)₂.

(5) Compounds of Preferred 4 where n is O.

(6) Compounds of Preferred 4 where n₁ is O.

(7) Compounds of Preferred 5 where Q is Q₁ -4, Q₁ -6, Q₁ -17, Q₁ -18, Q₁-19, Q₁ -21, Q₁ -22, Q₁ -23, Q₂ -1 or Q₃ -1.

(8) Compounds of Preferred 6 where Q is Q₁ -2, Q₁ -3 or Q₁ -14.

(9) Compounds of Preferred 5 where Q is Q₁ -1.

(10) Compounds of Preferred 5 where Q is Q₁ -2.

(11) Compounds of Preferred 5 where Q is Q₁ -3.

(12) Compounds of Preferred 5 where Q is Q₁ -4.

(13) Compounds of Preferred 5 where Q is Q₁ -5.

(14) Compounds of Preferred 5 where Q is Q₁ -6.

(15) Compounds of Preferred 5 where Q is Q₁ -7.

(16) Compounds of Preferred 5 where Q is Q₁ -8.

(17) Compounds of Preferred 5 where Q is Q₁ -9.

(18) Compounds of Preferred 5 where Q is Q₁ -10.

(19) Compounds of Preferred 5 where Q is Q₁ -11.

(20) Compounds of Preferred 5 where Q is Q₁ -12.

(21) Compounds of Preferred 5 where Q is Q₁ -13.

(22) Compounds of Preferred 5 where Q is Q₁ -14.

(23) Compounds of Preferred 5 where Q is Q₁ -16.

(24) Compounds of Preferred 5 where Q is Q₁ -17.

(25) Compounds of Preferred 5 where Q is Q₁ -18.

(26) Compounds of Preferred 5 where Q is Q₁ -19.

(27) Compounds of Preferred 5 where Q is Q₁ -20.

(28) Compounds of Preferred 5 where Q is Q₁ -21.

(29) Compounds of Preferred 5 where Q is Q₁ -22.

(30) Compounds of Preferred 5 where Q is Q₁ -23.

(31) Compounds of Preferred 5 where Q is Q₁ -24.

(32) Compounds of Preferred 5 where Q is Q₂ -1.

(33) Compounds of Preferred 5 where Q is Q₂ -2.

(34) Compounds of Preferred 5 where Q is Q₂ -3.

(35) Compounds of Preferred 5 where Q is Q₃ -1.

(36) Compounds of Preferred 5 where Q is Q₃ -2.

(37) Compounds of Preferred 5 where Q is Q₃ -3.

(38) Compounds of Preferred 6 where Q is Q₁ -1.

(39) Compounds of Preferred 6 where Q is Q₁ -2.

(40) Compounds of Preferred 6 where Q is Q₁ -3.

(41) Compounds of Preferred 6 where Q is Q₁ -4.

(42) Compounds of Preferred 6 where Q is Q₁ -5.

(43) Compounds of Preferred 6 where Q is Q₁ -6.

(44) Compounds of Preferred 6 where Q is Q₁ -7.

(45) Compounds of Preferred 6 where Q is Q₁ -8.

(46) Compounds of Preferred 6 where Q is Q₁ -9.

(47) Compounds of Preferred 6 where Q is Q₁ -10.

(48) Compounds of Preferred 6 where Q is Q₁ -11.

(49) Compounds of Preferred 6 where Q is Q₁ -12.

(50) Compounds of Preferred 6 where Q is Q₁ -13.

(51) Compounds of Preferred 6 where Q is Q₁ -14.

(52) Compounds of Preferred 6 where Q is Q₁ -16.

(53) Compounds of Preferred 6 where Q is Q₁ -17.

(54) Compounds of Preferred 6 where Q is Q₁ -18.

(55) Compounds of Preferred 6 where Q is Q₁ -19.

(56) Compounds of Preferred 6 where Q is Q₁ -20.

(57) Compounds of Preferred 6 where Q is Q₁ -21.

(58) Compounds of Preferred 6 where Q is Q₁ -22.

(59) Compounds of Preferred 6 where Q is Q₁ -23.

(60) Compounds of Preferred 6 where Q is Q₁ -24.

(61) Compounds of Preferred 6 where Q is Q₂ -1.

(62) Compounds of Preferred 6 where Q is Q₂ -2.

(63) Compounds of Preferred 6 where Q is Q₂ -3.

(64) Compounds of Preferred 6 where Q is Q₃ -1.

(65) Compounds of Preferred 6 where Q is Q₃ -2.

(66) Compounds of Preferred 6 where Q is Q₃ -3.

(67) Compounds of Preferred 4 where Q is Q₁ -15.

Specifically preferred for reasons of greatest ease of synthesis and/orgreatest herbicidal efficacy are:

N-[(4,6-dimethoxypyrimidin-2-yl)aminocarbonyl]-1-phenyl-1H-[1]benzothieno[3,2-C]pyrazole-5-sulfonamide,4,4-dioxide, m.p. 243°-248° C.

4,5-dihydro-N-[(4,6-dimethoxypyrimidin-2-yl)aminocarbonyl]naphth[2,1-D]isoxazole-9-sulfonamide,m.p. 189°-192° C.(d).

4,5-dihydro-N-[(4-methoxy-6-methylpyrimidin-2-yl)aminocarbonyl]naphth[2,1-D]isoxazole-9-sulfonamide,m.p. 186°-189° C.

4,5-dihydro-N-[(4,6-dimethoxy-1,3,5-triazin-2-yl)aminocarbonyl]naphth[2,1-D]isoxazole-9-sulfonamide,m.p. 147°-150° C.

DETAILED DESCRIPTION OF THE INVENTION Synthesis

The compounds of Formula 1 can be prepared by one or more of the methodsdescribed below in Equations 1, 2, 3 and 4.

As shown in Equation 1, compounds of Formula 1 can be prepared byreacting a sulfonyl isocyanate or sulfonyl isothiocyanate of Formula 2with an appropriate heterocyclic amine of Formula 3. ##STR15##

The reaction is carried out at 25° to 100° C. in an inert aproticsolvent such as methylene chloride or xylene for 0.5 to 24 hours astaught in U.S. Pat. No. 4,127,405.

Compounds of Formula 1 can also be prepared by reacting the sulfonamidesof Formula 4 with a phenylcarbamate or phenylthiocarbamate of Formula 5in the presence of DBU and in solvents such as methylene chloride oracetonitrile as taught in European Patent Application No. 70,804.##STR16##

Alternatively, compounds of Formula 1 where W is O can be prepared byreacting sulfonamides of Formula 4 with a methyl carbamate of Formula 6in the presence of an equimolar quantity of trimethylaluminum as shownin Equation 3. ##STR17##

The reaction is carried out at 25°-40° C. in a solvent such as methylenechloride, for 10-96 hours, under an inert atmosphere as taught inEP-A-83,975. The required carbamates (5) are prepared by reacting thecorresponding amines (3) with dimethyl carbonate or methyl chloroformatein the presence of a strong base.

Compounds of Formula 1 can also be prepared by reacting a sulfonylcarbamate or thiocarbamate of Formula 7 with an appropriate amine ofFormula 3 as shown in Equation 4. ##STR18##

The reaction is carried out at 50°-100° C. in a solvent such as dioxanefor 0.5 to 24 hours as taught in EP-A-44,807. The required carbamatesand thiocarbamates (7) can be prepared by methods, or modificationsthereof known to those skilled in the art, described in South AfricanPatent Application No. 82/5671 and South African Patent Application No.82/5045.

As shown in Equation 5, many of the sulfonyl isocyanates of Formula 2can be prepared by the reaction of sulfonamides of Formula 4 withphosgene, in the presence of n-butylisocyanate and a tertiary aminecatalyst, such as 1,4-diazabicyclo[2.2.2]-octane (DABCO), at reflux, ina solvent such as xylene by the method of U.S. Pat. No. 4,238,621.##STR19##

Many of the sulfonyl isocyanates can be prepared from the sulfonamidesby a two-step procedure involving (a) reacting the sulfonamides withn-butylisocyanate in the presence of a base such as K₂ CO₃ at reflux inan inert solvent such as 2-butanone forming an n-butylsulfonylurea; and(b) reacting this compound with phosgene and a tertiary amine catalystat reflux in xylene solvent. The method is similar to a procedure taughtby Ulrich and Sayigh, Newer Methods of Preparative Organic Chemistry,Vol. VI, p. 223-241, Academic Press, New York and London, W. Foerst, Ed.

Alternatively, many of the sulfonyl isocyanates of Formula 2 can beprepared by reacting the corresponding sulfonyl chlorides (8) withcyanic acid salt. ##STR20##

The reaction is carried out at 25°-100° in an inert aprotic solvent suchas acetonitrile for 0.5-24 hours in the presence of phosphorouspentoxide and an alkali metal salt such as lithium iodide according tothe teachings of Japanese Patent No. 76/26,816 (Chem. Abst. 85:77892e(1976)).

Sulfonyl isothiocyanates (2, W is S) are known in the art and areprepared from the corresponding sulfonamides (4) by reaction with carbondisulfide and potassium hydroxide followed by treatment of the resultingdipotassium salt with phosgene. Such a procedure is described in Arch.Pharm. 299, 174 (1966).

The sulfonamides of Formula 4 of Equations 2, 3, 4, 5 and 7 areimportant intermediates for the preparation of compounds of thisinvention. As shown in Equation 7, many of the sulfonamides of Formula 4can be prepared from the corresponding sulfonyl chlorides of Formula 8by contacting with either anhydrous or aqueous ammonia. ##STR21##

Preparation of sulfonamides from sulfonyl chlorides is widely reportedin the literature, for reviews see F. Hawking and J. S. Lawrence "TheSulfonamides", H. K. Lewis and Co., London, 1950, and E. H. Northey "TheSulfonamides and Allied Compounds", Reinhold Publishing Corp., New York,1948.

Many of the sulfonyl chlorides of Formula 8 of Equations 6 and 7 can beprepared from the corresponding amines of Formula 9 by the method shownin Equation 8. ##STR22##

The reaction involves diazotization of the amine 9 with sodiumnitrite/HCl followed by reaction of the diazonium salt with sulfurdioxide and cupric chloride in acetic acid analogous to the teachings ofYale and Sowinski, J. Org. Chem., 25, 1824 (1960).

Alternatively, many of the sulfonyl chlorides of Formula 8 can beprepared by a modification of the above procedure whereby thediazotization reaction is carried out in dilute sulfuric acid and theresulting diazonium salt is reacted with sulfur dioxide, HCl and cupricchloride is a co-solvent mixture consisting of acetic acid-water (1:1)and an immiscible inert solvent such as 1-chlorobutane or methylenechloride at 0°-40° C. for 1-24 hours.

Some of the amines of the Formula 9 in Equation 8 can be prepared fromthe corresponding nitro compounds (10). The reduction reaction ofEquation 9 can be run by methods known in the literature. ##STR23##

For example, the reduction can be carried out with stannous chloride ortin and hydrochloric acid either neat or in an inert solvent such asmethanol at about 25° to 80° C. for 0.5 to 10 hours. For details, referto similar procedures described in G. Corsi et al., Bull. Chim. Farm.,103, 115 (1964), A. Quilico et al, Gass. Chim. Ital., 76, 87 (1946) andM. Kahn and J. Polya, J. Chem. Soc., 85 (1970).

Many of the sulfonyl chorides of Formula 8 can be prepared from thebromo compounds of Formula 11 as shown in Equation 10. ##STR24##

According to Equation 10 a lithium salt, prepared by reaction of thebromide of Formula 11 with butyl lithium in ether at about -70° C., isadded to sulfuryl chloride in hexane at -30° to -20° C. and stirred for0.5 to 10 hours to yield the sulfonyl chloride 8 according to theteachings of S. N. Battacharya et al., J. Chem. Soc. C. 1265 (1968).

Many of the sulfonyl chlorides of Formula 8 can be prepared from thechloro compounds of Formula 12 by the two-step sequence shown inEquation 11. ##STR25## wherein RS.sup.⊖ M.sup.⊕ represents an alkyl orbenzyl mercaptide salt.

The first step involves nucleophilic displacement of the chlorine atomwith an alkyl or benzyl mercaptide to give an intermediate sulfide. Thereaction can be carried out at 25° to 80° C. in a polar solvent such asDMF for 0.5 to 24 hours. The sulfide is then oxidatively chlorinated tothe desired sulfonyl chloride 8 by the addition of molecular chlorine ora chlorine equivalent to the sulfide in the presence of water at 15° to80° C. in an aliphatic carboxylic acid solvent such as acetic acid or aninert organic solvent such as dichloroethane for 1 to 24 hours.

The tricyclic intermediates of Formulae 9, 10, 11 and 12 are known orcan be prepared by one skilled in the art.

The synthesis of heterocyclic amines such as those represented byFormula 3 has been reviewed in "The Chemistry of HeterocyclicCompounds," a series published by Interscience Publ., New York andLondon. Aminopyrimidines are described by D. J. Brown in "ThePyrimidines", Vol. XVI of the series, mentioned above which is hereinincorporated by reference. The 2-amino-1,3,5-triazines of Formula 3,where A is A-1 and Z is N, can be prepared according to methodsdescribed by E. M. Smolin and L. Rapaport in "s-Triazines andDerivatives," Vol. XIII.

Pyrimidines of Formula 3, where A is A-1 and Y is an acetal orthioacetal substituent, can be prepared by methods taught in EuropeanPatent Application No. 84,224 (published July 27, 1983).

Pyrimidines of Formula 3, where A is A-1 and Y is cyclopropyl or OCF₂ H,can be synthesized according to the methods taught in South AfricanPatent Application No. 83/7434 and South African Publication No.82/5045, respectively.

Compounds of Formula 3, where A is A-2 or A-3, can be prepared byprocedures disclosed in U.S. Pat. No. 4,339,267.

Compounds of Formula 3, where A is A-5, can be prepared by methodstaught in U.S. Pat. No. 4,421,550.

Compounds of Formula 3, where A is A-6, can be prepared by methodstaught in European Patent Application No. 94,260 (published Nov. 16,1983).

Agriculturally suitable salts of compounds of Formula 1 are also usefulherbicides and can be prepared in a number of ways known to the art. Forexample, metal salts can be made by treating compounds of Formula 1 witha solution of an alkali or alkaline earth metal salt having asufficiently basic anion (e.g., hydroxide, alkoxide, carbonate orhydride). Quaternary amine salts can be made by similar techniques.Detailed examples of such techniques are given in U.S. Pat. No.4,127,405.

The preparation of the compounds of this invention is furtherillustrated by the following examples.

EXAMPLES EXAMPLE 1 2-Acetyl-4-nitro 1,3-indanedione

To a solution of 100 g of 3-nitrophthalic acid in 100 mL of pyridine wasadded 0.8 mL of piperdine followed by 500 g of 2,4-pentanedione at roomtemperature. The mixture was stirred at 35°-40° C. for 6 hours and thendiluted with 100 mL ether. The pyridine salt was filtered oft, washedwith 100 ml of ether, dried, suspended in waer, and acidified with 400mL of 6N HCl. The title compound was filtered off, dried,andrecrystallized from ethanol to yield 84 g of yellow crystals, m.p.148°-150°.

200 MHz NMR (CDCL₃)δ7.8-8.08 (m.3H aromatic) δ2.6 (S, CH₃).

IR(nujol) 3460, 3360, 1690 cm⁻¹.

EXAMPLE 2 2-Acetyl-4-amino 1,3 indanedione

To a suspension of 20.0 g of 4-nitro-1,3-indanedione in 100 mLtetrahydrofuran and 20 mL of ethanol, 1.0 g of 10% Pd/C catalyst wasadded and the mixture hydrogenated at 50 psi until three molarequivalents of hydrogen were taken up. The catalyst was filtered off andsolvent was removed from the filtrate under reduced pressure.Recrystallization from ethanol afforded 14.8 g of the title compound,m.p. 126°-128°.

IR(nujol) 3460, 3340, 1690 cm⁻¹,

EXAMPLE 3 1-phenyl-5-aminoindenopyrazol-4-one

To a solution of 4.7 g of 4-amino-1,3-indanedione in 500 mL ethanol wasadded 2 mL of phenylhydrazine at room temperature and the mixture washeated at reflux for 2 hours. The mixture was then cooled to roomtemperature and 4 mL concentrated hydrochloric acid was added. Themixture was then refluxed for an additional 2 hours. The mixture wasthen concentrated in vacuo and the crystals that separated were filteredoff and dried, to yield 3.4 g of the title compound, m.p. 200°-202° C.

200 MHz NMR (CDCl₃)δ: 6.5-6.58 (m, Aromatic 2H), 7.06-7.1 (m, Aromatic1H), 7.51-7.65 (m, Aromatic 5H), 2.26 (s, CH₃), 4.2 (br, NH₂).

IR(nujol) 3420 and 3310. 1665 cm⁻¹.

EXAMPLE 4 1-phenylindenopyrazol-4-one-5-sulfonylchloride

A suspension of 36 g of aminopyrazolone of Example 3 in 130 mLconcentrated hydrochloric acid and 250 mL of glacial acetic acid wascooled to 0°-5° C. and 10 g of sodium nitrite was added in portionswhile maintaining the temperature at 0°-5°. After stirring for 30minutes, the suspension was added in portions to a preformed mixturecontaining 200 mL acetic acid, 15 g of cuprous chloride, and 150 mLconcentrated hydrochloric acid at 10° C. The mixture was stirred at 10°for 30 minutes and then at 40°-50° for 3 hours. The suspension was addedto 1000 mL ice water, stirred and extracted with 250 mL of methylenechloride. The methylene chloride layer was washed with water, dilutebircarbonate solution and water and then dried. The solvent was removedunder reduced pressure to yield 25 g of the crude sulfonyl chloride.

IR(nujol) 1700, 1380, 1165 cm⁻¹.

EXAMPLE 5 1-phenylindenopyrazolone-4-one-5-sulfonamide

A solution of 10 g of the sulfonyl chloride prepared in Example 4 in 75mL of tetrahydrofuran was cooled in an ice bath and treated cautiouslywith 40 mL of concentrated ammonium hydroxide, while maintaining thetemperature at 0°-5° C. The resulting suspension was stirred at roomtemperature for 8 hours. The solvent was then removed under reducedpressure. The residue was stirred in 500 mL water and filtered. Thesolids obtained were recrystallized from a mixture of acetonitrile andwater to give 6.9 g of the title compound as yellow crystals, m.p.247°-249°.

200 MHz NMR (CDCl₃) δ: 6.5-6.58 (m, Aromatic, 2H), 7.06-7.1 (m,Aromatic, 1H), 7.51-7.65 (m, Aromatic, 5H), 2.26 (s, CH₃), 4.2 (s, NH₂).

IR(nujol) 3310, 3420, 1665 cm⁻¹.

EXAMPLE 6N[(4,6,Dimethyl-1,3,5-triazin-2-yl)aminocarbonyl]-1-phenylidenopyrazol-4-one-5-sulfonamide

To a suspension 0.27 g ofN-phenoxycarbonyl-4,6-dimethoxy-2-aminotriazine in 20 mL ofacetronitrile was added 0.327 g of the sulfonamide described in Example5 followed by 0.2 mL of 1,8-diazabicyclo-[5.4.0]-undec-7-ene. Themixture was then stirred at room temperature for 2 hours. The mixturewas added to 50 mL water containing 2 mL conc. hydrochloric acid andextracted with methylene chloride. The methylene chloride extract wasdried and stripped of solvent under reduced pressure to furnish a yellowsolid which was triturated with chlorobutane and filtered to give 0.12 gof yellow crystals, m.p. 152°-155°.

NMR 200 MHz (CDCl₃)δ: 13.2 (broad s, 1H, NH), 8.06 (s, 1H, NH), 7.2-7.6(m, 8H, Aromatic), 4.23 (s, 3H, OCH₃), 2.38 (s, 3H, CH₃).

IR(nujol) 1725, 1710, 1360, 1170 cm⁻¹.

EXAMPLE 7 5-amino-1-methylindenopyrazol-4-one

To a solution 25 g of 4-amino-1,3-indanedione, described in Example 2,in 200 mL ethanol was added 5.5 mL of methyl hydrazine at roomtemperature and then heated to reflux for 2 hours. The mixture wastreated with 4 mL concentrated hydrochloric acid and again heated atreflux for 2 hours. The mixture was then cooled and the solvent wasremoved. The residue was triturated with water, filtered and dried.Recrystalliztion from ethanol and water yielded 18.9 g of yellowcrystals. m.p. 225°-227°.

NMR 200 MHz (CDCl₃) δ: (m. 7.02-7.10, 1H, Aromatic), (m, 6.5-6.6, 2H,Aromatic), (br s, 5.32, 2H, NH₂), (s, 3.89, 3H, NCH₃), (s, 2.31, 3H,CH₃).

IR(nujol) 3420, 3310, 1665 cm⁻¹.

EXAMPLE 8 1-Methyl-indenopyrazol-4-one 5-sulfonylchloride

A suspension of 12.5 g of the aminopyrazolone of Example 7 in 65 mL ofconcentrated hydrochloric acid and 125 mL of glacial acetic acid wascooled to 0° to 5° and then 5 g of sodium nitrite was added in portionswhile maintaining the temperature at 0°-5°. After 30 minutes, thesuspension was added to a preformed mixture of 100 mL glacial aceticacid, 7.5 g of cuprous chloride, and 75 mL of concentrated hydrochloricacid at 0°-5°. The mixture was stirred at that temperature for 30minutes and then was heated at 40° to 50° for 3 hours. The suspensionwas poured into 5000 mL ice water and extracted with 250 mL methylenechloride. The methylene chloride extract was washed with water and thendried. The solvent was striped under reduced pressure to afford thecrude sulfonyl chloride as a yellow solid.

IR(nujol) 1700, 1380, 1165 cm⁻¹.

EXAMPLE 9 1-Methyl-indenopyrazol-4-one-5-sulfonamide

A solution of 5 g of the sulfonyl chloride of Example 8 in 40 mLtetrahydrofuran was cooled in a ice water bath and treated cautiouslywith 20 mL of concentrated ammonium hydroxide, added slowly maintainingthe temperature at 0° to 5° C. The resulting suspension was stirred atroom temperature for 8 hours and then stripped of the solvent underreduced pressure. The residue was stirred in 200 mL water, filtered,washed with hot ethanol and dried to afford 1.8 g of yellow crystals,m.p. 260°-265°

NMR 200 MHz δ: 7.7-7.82 (m, 3H, aromatic), 3.95 (s, 3H, NCH₃), 2.2 (s,3H, CH₃).

IR(nujol) 3350, 3260, 1700, 1370, 1160 cm⁻¹.

EXAMPLE 10N-[(4,6-Dimethoxypyrimidin-2-yl)aminocarbonyl]-methylindenopyrazol-4-one-5-sulfonamide

To a suspension of 0.2 g ofN-phenoxycarbonyl-4,6-dimethoxyaminopyrimidine in 15 mL of acetonitrilewas added 0.2 g of methylindenopyrazolone-5-sulfonamide, followed by theaddition of 0.2 mL of 1,8-diazabicyclo[5.4.0]undec-7-ene and the mixturewas stirred at room temperature for 2 hours. The mixture was added to 50mL water containing 2 mL concentrated hydrochloric acid and extractedwith 50 mL methylene chloride. The methylene chloride extract was driedand the solvent was removed. The residue was triturated withchlorobutane, filtered and dried to give 0.21 g of the title compound,m.p. 224°-230°.

NMR 200 MHz (CDCl₃)δ: (s, 12.75, 1H, NH), (s, 8.12, 1H, NH), (m 7.4-7.63H, Aromatic), (s, 5.83, 1H, CH), (s, 4.17, 3H, CH₃), (s, 3.98, 3H,NCH₃), (s, 2.27, 3H, CH₃).

IR(nujol) 1700, 1370, 1160 cm⁻¹.

EXAMPLE 11N-(1,1-Dimethylethyl)-5,6,7,8-tetrahydro-8-hydroxy-1-naphthalenesulfonamide

To a solution of 25.2 g (93.5 mmol) of a 1:1 mixture ofN-(1,1-dimethylethyl)-5,6,7,8-tetrahydro-1-naphthalenesulfonamide andN-(1,1-dimethylethyl)-5,6,7,8-tetrahydro-2-naphthalenesulfonamide in 450mL of tetrahydrofuran at -10° C., was added dropwise 75 mL (187 mmol) ofa 2.5M solution of n-butyllithium in hexanes. After 90 minutes at thistemperature the reaction mixture had turned red. The reaction mixturewas cooled to -78° C. and oxygen was bubbled through for 15 minutesuntil the red color disappeared. After an additional 15 minutes, 200 mLof 5% NaHSO₃ was added. The reaction mixture was extracted with ethylacetate, dried (Na₂ SO₄) and the solvent was removed with a rotaryevaporator. The residue was purified by flash chromatography to give 6.0g of the title compound as a sticky solid; m.p. 100°-111° C.

¹ H NMR (CDCl₃)δ1.24 (s, 9H), 1.8 (m, 2H), 2.0 (m, 2H), 2.8 (m, 2H), 3.5(d, 1H), 5.2 (br, 1H), 5.55 (m, 1H), 7.3 (m, 2H), 7.99 (d, 1H).

EXAMPLE 12N-(1,1-Dimethylethyl)-5,6,7,8-tetrahydro-8-oxo-1-naphthalenesulfonamide

To a solution of 5.49 g (19.4 mmol) of material prepared in Example 11in 250 mL of methylene chloride was added 8.35 g (39 mmol) ofpyridiniumchlorochromate. After 3 hours the reaction mixture was dilutedwith ether and passed through a plug of fluorosil to give 5.3 g of thetitle compound as a colorless oil.

¹ NMR (CDCl₃)δ1.27 (s, 9H), 2.1 (m, 2H), 2.26 (dd, 2H), 3.00 (dd, 2H),6.77 (br, 1H), 7.54 (m, 2H), 8.13 (dd, 1H).

EXAMPLE 13N-(1,1-Dimethylethyl)-5,6,7,8-tetrahydro-7-(hydroxymethylene)-8-oxo-1-naphthanesulfonamide

1.0 g (43.5 g-atom) of sodium was added to 25 mL of ethanol. When all ofthe sodium had reacted the ethanol was removed with a rotary evaporator.25 mL of benzene was added. The reaction mixture was cooled in an icebath and 2.5 mL of ethyl formate was added. 4.82 g (17.1 mmol) ofmaterial prepared in Example 12 was added in 25 mL of benzene. Thereaction mixture was allowed to stand at room temperature for 16 hours.The reaction mixture was extracted with 100 mL of water. This aqueouslayer was acidified with 5% HCl and was extracted with ethyl acetate.The organic layer was dried (Na₂ SO₄) and the solvent was removed with arotary evaporator to give 4.30 g of the title compound as a yellowsolid.

¹ H NMR (CDCl₃)δ1.30 (s, 9H), 2.49 (t, 2H), 2.95 (t, 2H), 6.79 (br, 1H),7.54 (m, 3H), 8.16 (d, 1H).

EXAMPLE 14N-(1,1-Dimethylethyl)-3,4-dihydronaphth((2,1-D))-isoxazole-9-sulfonamide

A mixture of 0.7 g (2.85 mmol) of material prepared in Example 13 and0.4 g (5.8 mmol) of hydroxylamine hydrochloride was dissolved in 20 mLof acetic acid. The reaction mixture was placed in an oil bath at 125°C. for 15 minutes. After cooling, water and 1-chlorobutane were added.After extraction with 1-chlorobutane, the organic layer was washed withsaturated NaHCO₃, dried (Na₂ SO₄) and the solvent was removed with arotary evaporator. The residue was purified by flash chromatography togive 0.26 g of an orange solid.

¹ NMR (CDCl₃)δ1.21 (s, 9H), 2.78 (m, 2H), 3.10 (m, 2H), 5.73 (br, 1H),7.48 (m, 2H), 8.15 (d, 1H), 8.27 (s, 1H).

EXAMPLE 15 3,4-Dihydronaphth((2,1-D))isoxazole-9-sulfonamide

0.20 g of material prepared in Example 14 was dissolved in 5 mL oftrifluoroacetic acid. After 1 hour the volatiles were removed with arotary evaporator. The residue was purified by flash chromatography togive 0.09 g of a brown solid.

¹ H NMR (d₆ -DMSO)δ2.71 (m, 2H), 3.03 (m, 2H), 7.36 (s, 2H), 7.52 (dd,1H), 7.62 (d, 1H), 7.90 (d, 1H), 8.62 (s, 1H).

EXAMPLE 16N-((4,6-Dimethoxypyrimidinyl-2-yl)aminocarbonyl)-3,4-dihydronaphth((2,1-D))isoxazole-9-sulfonamide

To a solution of 45 mg of material prepared in Example 15 and 50 mgphenyl 4,6-dimethoxypyrimidin-2-yl carbamate in 1 mL of acetonitrile wasadded 0.027 mL of 1,8-diazabicyclo[5.4.0]undec-7-ene. After 1 hour, 1 mLof water and 0.5 mL of 5% HCl were added. The brown solid whichprecipitated out was collected to give 45 mg of the title compound; m.p.189-192(d).

¹ H NMR (d₆ -DMSO)δ2.77 (m, 2H), 3.07 (m, 2H), 3.99 (s, 6H), 5.99 (s,1H), 7.61 (dd, 1H), 7.79 (d, 1H), 8.05 (d, 1H), 8.60 (s, 1H), 10.6 (br,1H), 13.1 (br, 1H).

Using the techniques described in Equations 1-12 and Examples 1-16 thefollowing compounds of Tables 1 through 28 can be prepared.

Unless otherwise indicated, all temperatures are in °C.

    ______________________________________                                        General Formulas for Tables                                                   ______________________________________                                        General Formula 1a                                                                     ##STR26##                                                            General Formula 1b                                                                     ##STR27##                                                            General Formula 1c                                                                     ##STR28##                                                            General Formula 1d                                                                     ##STR29##                                                            General Formula 1e                                                                     ##STR30##                                                            General Formula 1f                                                                     ##STR31##                                                            General Formula 1g                                                                     ##STR32##                                                            General Formula 1h                                                                     ##STR33##                                                            General Formula 2a                                                                     ##STR34##                                                            General Formula 2b                                                                     ##STR35##                                                            General Formula 3a                                                                     ##STR36##                                                            General Formula 3b                                                                     ##STR37##                                                            General Formula 4a                                                                     ##STR38##                                                            General Formula 4b                                                                     ##STR39##                                                            General Formula 5a                                                                     ##STR40##                                                            General Formula 5b                                                                     ##STR41##                                                            General Formula 6                                                                      ##STR42##                                                            General Formula 7                                                                      ##STR43##                                                            General Formula 8                                                                      ##STR44##                                                            General Formula 9                                                                      ##STR45##                                                            General Formula 10                                                                     ##STR46##                                                            General Formula 11                                                                     ##STR47##                                                            General Formula 12                                                                     ##STR48##                                                            General  Formula 13                                                                    ##STR49##                                                            General Formula 14                                                                     ##STR50##                                                            General Formula 15                                                                     ##STR51##                                                            General Formula 16                                                                     ##STR52##                                                            General Formula 17                                                                     ##STR53##                                                            General Formula 18                                                                     ##STR54##                                                            General Formula 19                                                                     ##STR55##                                                            General Formula 20                                                                     ##STR56##                                                            General Formula 21                                                                     ##STR57##                                                            General Formula 22                                                                     ##STR58##                                                            General Formula 23                                                                     ##STR59##                                                            General Formula 24                                                                     ##STR60##                                                            General Formula 25                                                                     ##STR61##                                                            General Formula 26                                                                     ##STR62##                                                            General Formula 27                                                                     ##STR63##                                                            General Formula 28                                                                     ##STR64##                                                            ______________________________________                                    

In general Formulas 1-28, the position of the substituent R₁ isdesignated as follows: ##STR65##

                                      TABLE Ia                                    __________________________________________________________________________    General Formula Ia                                                            R.sub.1                                                                            J   R.sub.6  R.sub.7                                                                          X    Y        Z  m.p. (°C.)                       __________________________________________________________________________    H    C═H                                                                           H        CH.sub.3                                                                         CH.sub.3                                                                           CH.sub.3 CH 226-230                                 H    C═O                                                                           H        CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.3                                                                              CH 248-250                                 H    C═O                                                                           H        CH.sub.3                                                                         OCH.sub.3                                                                          OCH.sub.3                                                                              CH 242-246                                 H    C═O                                                                           H        CH.sub.3                                                                         Cl   OCH.sub.3                                                                              CH 245-251                                 H    C═O                                                                           H        CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.3                                                                              N  218-221                                 H    C═O                                                                           H        CH.sub.3                                                                         OCH.sub.3                                                                          OCH.sub.3                                                                              N  222-227                                 H    C═O                                                                           CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           CH.sub.3 CH 238-240                                 H    C═O                                                                           CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.3                                                                              CH 238-240                                 H    C═O                                                                           CH.sub.3 CH.sub.3                                                                         OCH.sub.3                                                                          OCH.sub.3                                                                              CH 224-230                                 H    C═O                                                                           CH.sub.3 CH.sub.3                                                                         Cl   OCH.sub.3                                                                              CH 250-255                                 H    C═O                                                                           CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.3                                                                              N  232-234                                 H    C═O                                                                           CH.sub.3 CH.sub.3                                                                         OCH.sub.3                                                                          OCH.sub.3                                                                              N  232-235                                 H    C═O                                                                           CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           CH.sub.3 N                                          H    C═O                                                                           C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         CH.sub.3                                                                           CH.sub.3 CH 212-214                                 H    C═O                                                                           C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         OCH.sub.3                                                                          CH.sub.3 CH 185-189                                 H    C═O                                                                           C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         OCH.sub.3                                                                          OCH.sub.3                                                                              CH 215-217                                 H    C═O                                                                           C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         Cl   OCH.sub.3                                                                              CH 202-204                                 H    C═O                                                                           C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.3                                                                              N  168-171                                 H    C═O                                                                           C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         OCH.sub.3                                                                          OCH.sub.3                                                                              N  152-155                                 H    C═O                                                                           C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         CH.sub.3                                                                           CH.sub.3 N  205-208                                 H    C═O                                                                           C.sub.6 H.sub.5                                                                        H  CH.sub.3                                                                           CH.sub.3 CH                                         H    C═O                                                                           C.sub.6 H.sub.5                                                                        H  CH.sub.3                                                                           OCH.sub.3                                                                              CH                                         H    C═O                                                                           C.sub.6 H.sub.5                                                                        H  OCH.sub.3                                                                          OCH.sub.3                                                                              CH                                         H    C═O                                                                           C.sub.6 H.sub.5                                                                        H  Cl   OCH.sub.3                                                                              CH                                         H    C═O                                                                           C.sub.6 H.sub.5                                                                        H  CH.sub.3                                                                           OCH.sub.3                                                                              N                                          H    C═O                                                                           C.sub.6 H.sub.5                                                                        H  OCH.sub.3                                                                          OCH.sub.3                                                                              N                                          H    C═O                                                                           C.sub.6 H.sub.5                                                                        H  CH.sub.3                                                                           CH.sub.3 N                                          H    C═O                                                                           4-Cl--C.sub.6 H.sub.5                                                                  CH.sub.3                                                                         CH.sub.3                                                                           CH.sub.3 CH 227-231                                 H    C═O                                                                           4-Cl--C.sub.6 H.sub.5                                                                  CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.3                                                                              CH 236-238                                 H    C═O                                                                           4-Cl--C.sub.6 H.sub.5                                                                  CH.sub.3                                                                         OCH.sub.3                                                                          OCH.sub.3                                                                              CH 248-250                                 H    C═O                                                                           4-Cl--C.sub.6 H.sub.5                                                                  CH.sub.3                                                                         Cl   OCH.sub.3                                                                              CH 229-232                                 H    C═O                                                                           4-Cl--C.sub.6 H.sub.5                                                                  CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.3                                                                              N                                          H    C═O                                                                           4-Cl--C.sub.6 H.sub.5                                                                  CH.sub.3                                                                         OCH.sub.3                                                                          OCH.sub.3                                                                              N  206-210                                 H    C═O                                                                           4-Cl--C.sub.6 H.sub.5                                                                  CH.sub.3                                                                         CH.sub.3                                                                           CH.sub.3 N                                          H    C═O                                                                           4-OCH.sub.3 --C.sub.6 H.sub.5                                                          CH.sub.3                                                                         CH.sub.3                                                                           CH.sub.3 CH                                         H    C═O                                                                           4-OCH.sub.3 --C.sub.6 H.sub.5                                                          CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.3                                                                              CH                                         H    C═O                                                                           4-OCH.sub.3 --C.sub.6 H.sub.5                                                          CH.sub.3                                                                         OCH.sub.3                                                                          OCH.sub.3                                                                              CH 228-230                                 H    C═O                                                                           4-OCH.sub.3 --C.sub.6 H.sub.5                                                          CH.sub.3                                                                         Cl   OCH.sub.3                                                                              CH                                         H    C═O                                                                           4-OCH.sub.3 --C.sub.6 H.sub.5                                                          CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.3                                                                              N                                          H    C═O                                                                           4-OCH.sub.3 --C.sub.6 H.sub.5                                                          CH.sub.3                                                                         OCH.sub.3                                                                          OCH.sub.3                                                                              N                                          H    C═O                                                                           4-OCH.sub.3 --C.sub.6 H.sub.5                                                          CH.sub.3                                                                         CH.sub.3                                                                           CH.sub.3 N                                          H    C═O                                                                           4-SO.sub.2 CH.sub.3 --C.sub.6 H.sub.5                                                  CH.sub.3                                                                         CH.sub.3                                                                           CH.sub.3 CH 172-176                                 H    C═O                                                                           4-SO.sub.2 CH.sub.3 --C.sub.6 H.sub.5                                                  CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.3                                                                              CH 166-169                                 H    C═O                                                                           4-SO.sub.2 CH.sub.3 --C.sub.6 H.sub.5                                                  CH.sub.3                                                                         OCH.sub.3                                                                          OCH.sub.3                                                                              CH 204-208                                 H    C═O                                                                           4-SO.sub.2 CH.sub.3 --C.sub.6 H.sub.5                                                  CH.sub.3                                                                         Cl   OCH.sub.3                                                                              CH                                         H    C═O                                                                           4-SO.sub.2 CH.sub.3 --C.sub.6 H.sub.5                                                  CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.3                                                                              N                                          H    C═O                                                                           4-SO.sub.2 CH.sub.3 --C.sub.6 H.sub.5                                                  CH.sub.3                                                                         OCH.sub.3                                                                          OCH.sub.3                                                                              N  104-109                                 H    C═O                                                                           4-SO.sub.2 CH.sub.3 --C.sub.6 H.sub.5                                                  CH.sub.3                                                                         CH.sub.3                                                                           CH.sub.3 N                                          H    C═O                                                                           4-NO.sub.2 --C.sub.6 H.sub.5                                                           CH.sub.3                                                                         CH.sub.3                                                                           CH.sub.3 CH                                         H    C═O                                                                           4-NO.sub.2 --C.sub.6 H.sub.5                                                           CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.3                                                                              CH                                         H    C═O                                                                           4-NO.sub.2 --C.sub.6 H.sub.5                                                           CH.sub.3                                                                         OCH.sub.3                                                                          OCH.sub.3                                                                              CH                                         H    C═O                                                                           4-NO.sub.2 --C.sub.6 H.sub.5                                                           CH.sub.3                                                                         Cl   OCH.sub.3                                                                              CH                                         H    C═O                                                                           4-NO.sub.2 --C.sub.6 H.sub.5                                                           CH.sub.3                                                                         OCH.sub.3                                                                          CH.sub.3 N                                          H    C═O                                                                           4-NO.sub.2 --C.sub.6 H.sub.5                                                           CH.sub.3                                                                         OCH.sub.3                                                                          OCH.sub.3                                                                              N                                          H    C═O                                                                           4-NO.sub.2 --C.sub.6 H.sub.5                                                           CH.sub.3                                                                         CH.sub.3                                                                           CH.sub.3 N                                          H    C═O                                                                           4-CH.sub.3 --C.sub.6 H.sub.5                                                           CH.sub.3                                                                         CH.sub.3                                                                           CH.sub.3 CH                                         H    C═O                                                                           4-CH.sub.3 --C.sub.6 H.sub.5                                                           CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.3                                                                              CH                                         H    C═O                                                                           4-CH.sub.3 --C.sub.6 H.sub.5                                                           CH.sub.3                                                                         OCH.sub.3                                                                          OCH.sub.3                                                                              CH                                         H    C═O                                                                           4-CH.sub.3 --C.sub.6 H.sub.5                                                           CH.sub.3                                                                         Cl   OCH.sub.3                                                                              CH                                         H    C═O                                                                           4-CH.sub.3 --C.sub.6 H.sub.5                                                           CH.sub.3                                                                         OCH.sub.3                                                                          CH.sub.3 N                                          H    C═O                                                                           4-CH.sub.3 --C.sub.6 H.sub.5                                                           CH.sub.3                                                                         OCH.sub.3                                                                          OCH.sub.3                                                                              N                                          H    C═O                                                                           4-CH.sub.3 --C.sub.6 H.sub.5                                                           CH.sub.3                                                                         OH.sub.3                                                                           CH.sub.3 N                                          H    C═O                                                                           2-pyridyl                                                                              H  CH.sub.3                                                                           CH.sub.3 CH 158-160                                 H    C═O                                                                           2-pyridyl                                                                              H  CH.sub.3                                                                           OCH.sub.3                                                                              CH 160-164                                 H    C═O                                                                           2-pyridyl                                                                              H  OCH.sub.3                                                                          OCH.sub.3                                                                              CH 203-207                                 H    C═O                                                                           2-pyridyl                                                                              H  Cl   OCH.sub.3                                                                              CH 145-151                                 H    C═O                                                                           2-pyridyl                                                                              H  CH.sub.3                                                                           OCH.sub.3                                                                              N  135-141                                 H    C═O                                                                           2-pyridyl                                                                              H  OCH.sub.3                                                                          OCH.sub.3                                                                              N  148-153                                 H    C═O                                                                           2-pyridyl                                                                              H  CH.sub.3                                                                           CH.sub.3 N                                          H    C═O                                                                           2-pyridyl                                                                              CH.sub.3                                                                         CH.sub.3                                                                           CH.sub.3 CH                                         H    C═O                                                                           2-pyridyl                                                                              CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.3                                                                              CH                                         H    C═O                                                                           2-pyridyl                                                                              CH.sub.3                                                                         OCH.sub.3                                                                          OCH.sub.3                                                                              CH                                         H    C═O                                                                           2-pyridyl                                                                              CH.sub.3                                                                         Cl   OCH.sub.3                                                                              CH                                         H    C═O                                                                           2-pyridyl                                                                              CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.3                                                                              N                                          H    C═O                                                                           2-pyridyl                                                                              CH.sub.3                                                                         OCH.sub.3                                                                          OCH.sub.3                                                                              N                                          H    C═O                                                                           2-pyridyl                                                                              CH.sub.3                                                                         CH.sub.3                                                                           CH.sub.3 N                                          H    SO.sub.2                                                                          2-pyridyl                                                                              CH.sub.3                                                                         CH   CH.sub.3 CH                                         H    SO.sub.2                                                                          2-pyridyl                                                                              CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.3                                                                              CH                                         H    SO.sub.2                                                                          2-pyridyl                                                                              CH.sub.3                                                                         OCH.sub.3                                                                          OCH.sub.3                                                                              CH                                         H    SO.sub.2                                                                          2-pyridyl                                                                              CH.sub.3                                                                         Cl   OCH.sub.3                                                                              CH                                         H    SO.sub.2                                                                          2-pyridyl                                                                              CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.3                                                                              N                                          H    SO.sub.2                                                                          2-pyridyl                                                                              CH.sub.3                                                                         OCH.sub.3                                                                          OCH.sub.3                                                                              N                                          H    SO.sub.2                                                                          2-pyridyl                                                                              CH.sub.3                                                                         CH.sub.3                                                                           CH.sub.3 N                                          H    C═O                                                                           CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.2 CH.sub.3                                                                     CH                                         H    C═O                                                                           CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           NH.sub.2 CH                                         H    C═O                                                                           CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           NHCH.sub.3                                                                             CH                                         H    C═O                                                                           CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           N(CH.sub.3).sub.2                                                                      CH                                         H    C═O                                                                           CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           CH.sub.2 CH.sub.3                                                                      CH                                         H    C═O                                                                           CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           CH.sub.2 CH.sub.3                                                                      CH                                         H    C═O                                                                           CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           CF.sub.3 CH                                         H    C═O                                                                           CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           SCH.sub.3                                                                              CH                                         H    C═O                                                                           CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.2 CH═CH.sub.2                                                              CH                                         H    C═O                                                                           CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.2 CH═CH.sub.2                                                              CH                                         H    C═O                                                                           CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.2 C.tbd. CH                                                                    CH                                         H    C═O                                                                           CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.2 CF.sub.3                                                                     CH                                         H    C═O                                                                           CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.2 CH.sub.2 OCH.sub.3                                                           CH                                         H    C═O                                                                           CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           CH(OCH.sub.3).sub.2                                                                    CH                                         H    C═O                                                                           CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           1,3-dioxolan-2-yl                                                                      CH                                         H    C═O                                                                           CH.sub.3 CH.sub.2                                                                         CH.sub.3                                                                           CH.sub.2 OCH.sub.3                                                                     CH                                         H    C═O                                                                           CH.sub.3 CH.sub.3                                                                         F    OCH.sub.3                                                                              CH                                         H    C═O                                                                           CH.sub.3 CH.sub.3                                                                         Br   OCH.sub.3                                                                              CH                                         H    C═O                                                                           CH.sub.3 CH.sub.3                                                                         OCH.sub.2 F                                                                        OCH.sub.3                                                                              CH                                         H    C═O                                                                           CH.sub.3 CH.sub.3                                                                         OCF.sub.3                                                                          OCH.sub.3                                                                              CH                                         H    C═O                                                                           CH.sub.3 CH.sub.3                                                                         CF.sub.3                                                                           OCH.sub.3                                                                              CH                                         H    C═O                                                                           CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           4-methyl-1,3-                                                                          CH                                                                   dioxolan-2-yl                                       H    C═O                                                                           CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.2 F                                                                            CH                                         H    C═O                                                                           CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           CN       CH                                         H    C═O                                                                           CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           CH(OCH.sub.2 CH.sub.3).sub.2                                                           CH                                         H    C═O                                                                           CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           OCF.sub.2 CHClF                                                                        CH                                         H    C═O                                                                           CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           SCH.sub.2 F                                                                            CH                                         H    C═O                                                                           CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           OCF.sub.2 CHBrF                                                                        CH                                         H    C═O                                                                           CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           OCF.sub.2 CHFCF.sub.3                                                                  CH                                         H    C═O                                                                           C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.2 CH.sub.3                                                                     CH                                         H    C═O                                                                           C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         CH.sub.3                                                                           NHCH.sub.3                                                                             CH                                         H    C═O                                                                           C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         CH.sub.3                                                                           N(CH.sub.3).sub.2                                                                      CH                                         H    C═O                                                                           C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         CH.sub.3                                                                           CH.sub.2 CH.sub.3                                                                      CH                                         H    C═O                                                                           C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         CH.sub.3                                                                           SCH.sub.3                                                                              CH                                         H    C═O                                                                           C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.2 C.tbd.CH                                                                     CH                                         H    C═O                                                                           C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.2 CH.sub.2 OCH.sub.3                                                           CH                                         H    C═O                                                                           C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         CH.sub.3                                                                           CH(OCH.sub.3).sub.2                                                                    CH                                         H    C═O                                                                           C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         CH.sub.3                                                                           SCH.sub.2 F                                                                            CH                                         H    C═O                                                                           C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         CH.sub.3                                                                           1,3-dioxolan-2-yl                                                                      CH                                         H    C═O                                                                           C.sub.6 H.sub. 5                                                                       CH.sub.3                                                                         CH.sub.3                                                                           OCF.sub.2 CHClF                                                                        CH                                         H    C═O                                                                           C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         CH.sub.3                                                                           CN       CH                                         H    SO.sub.2                                                                          H        H  CH.sub.3                                                                           CH.sub.3 CH                                         H    SO.sub.2                                                                          H        H  CH.sub.3                                                                           OCH.sub.3                                                                              CH                                         H    SO.sub.2                                                                          H        H  OCH.sub.3                                                                          OCH.sub.3                                                                              CH                                         H    SO.sub.2                                                                          H        H  Cl   OCH.sub.3                                                                              CH                                         H    SO.sub.2                                                                          H        H  CH.sub.3                                                                           OCH.sub.3                                                                              N                                          H    SO.sub.2                                                                          H        H  OCH.sub.3                                                                          OCH.sub.3                                                                              N                                          H    SO.sub.2                                                                          H        H  CH.sub.3                                                                           CH.sub.3 N                                          H    SO.sub.2                                                                          CH.sub.3 H  CH.sub.3                                                                           CH.sub.3 CH 262-266                                 H    SO.sub.2                                                                          CH.sub.3 H  CH.sub.3                                                                           OCH.sub.3                                                                              CH 238-242                                 H    SO.sub.2                                                                          CH.sub.3 H  OCH.sub.3                                                                          OCH.sub.3                                                                              CH 232-235                                 H    SO.sub.2                                                                          CH.sub.3 H  Cl   OCH.sub.3                                                                              CH 245-247                                 H    SO.sub.2                                                                          CH.sub.3 H  CH.sub.3                                                                           OCH.sub.3                                                                              N  227-230                                 H    SO.sub.2                                                                          CH.sub.3 H  OCH.sub.3                                                                          OCH.sub.3                                                                              N  228-231                                 H    SO.sub.2                                                                          CH.sub.3 H  CH.sub.3                                                                           CH.sub.3 N                                          H    SO.sub.2                                                                          C.sub.6 H.sub.5                                                                        H  CH.sub.3                                                                           CH.sub.3 CH 244-247                                 H    SO.sub.2                                                                          C.sub.6 H.sub. 5                                                                       H  CH.sub.3                                                                           OCH.sub.3                                                                              CH 250-253                                 H    SO.sub.2                                                                          C.sub.6 H.sub.5                                                                        H  OCH.sub.3                                                                          OCH.sub.3                                                                              CH 243-248                                 H    SO.sub.2                                                                          C.sub.6 H.sub.5                                                                        H  Cl   OCH.sub.3                                                                              CH 236-240                                 H    SO.sub.2                                                                          C.sub.6 H.sub.5                                                                        H  CH.sub.3                                                                           OCH.sub.3                                                                              N  215-226                                 H    SO.sub.2                                                                          C.sub.6 H.sub.5                                                                        H  OCH.sub.3                                                                          OCH.sub.3                                                                              N  212-213                                 H    SO.sub.2                                                                          C.sub.6 H.sub.5                                                                        H  CH.sub.3                                                                           CH.sub.3 N                                          H    SO.sub.2                                                                          H        CH.sub.3                                                                         CH.sub.3                                                                           CH.sub.3 CH                                         H    SO.sub.2                                                                          H        CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.3                                                                              CH                                         H    SO.sub.2                                                                          H        CH.sub.3                                                                         OCH.sub.3                                                                          OCH.sub.3                                                                              CH                                         H    SO.sub.2                                                                          H        CH.sub.3                                                                         Cl   OCH.sub.3                                                                              CH                                         H    SO.sub.2                                                                          H        CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.3                                                                              N                                          H    SO.sub.2                                                                          H        CH.sub.3                                                                         OCH.sub.3                                                                          OCH.sub.3                                                                              N                                          H    SO.sub.2                                                                          H        CH.sub.3                                                                         CH.sub.3                                                                           CH.sub.3 N                                          H    SO.sub.2                                                                          CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           CH.sub.3 CH                                         H    SO.sub.2                                                                          CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.3                                                                              CH 245-247                                 H    SO.sub.2                                                                          CH.sub.3 CH.sub.3                                                                         OCH.sub.3                                                                          OCH.sub.3                                                                              CH 259-262                                 H    SO.sub.2                                                                          CH.sub.3 CH.sub.3                                                                         Cl   OCH.sub.3                                                                              CH                                         H    SO.sub.2                                                                          CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.3                                                                              N  220-224                                 H    SO.sub.2                                                                          CH.sub.3 CH.sub.3                                                                         OCH.sub.3                                                                          OCH.sub.3                                                                              N  240-243                                 H    SO.sub.2                                                                          C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         CH.sub.3                                                                           CH.sub.3 CH 255-258                                 H    SO.sub.2                                                                          C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.3                                                                              CH 264-266                                 H    SO.sub.2                                                                          C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         OCH.sub.3                                                                          OCH.sub.3                                                                              CH 260-264                                 H    SO.sub.2                                                                          C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         Cl   OCH.sub.3                                                                              CH 262-266                                 H    SO.sub.2                                                                          C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         OCH.sub.3                                                                          OCH.sub.3                                                                              N  217-219                                 H    SO.sub.2                                                                          C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.3                                                                              N  214-218                                 H    SO.sub.2                                                                          C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         CH.sub.3                                                                           CH.sub.3 N                                          H    NH  H        CH.sub.3                                                                         CH.sub.3                                                                           CH.sub.3 CH                                         H    NH  H        CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.3                                                                              CH                                         H    NH  H        CH.sub.3                                                                         OCH.sub.3                                                                          OCH.sub.3                                                                              CH                                         H    NH  H        CH.sub.3                                                                         Cl   OCH.sub.3                                                                              CH                                         H    NH  H        CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.3                                                                              N                                          H    NH  H        CH.sub.3                                                                         OCH.sub. 3                                                                         OCH.sub.3                                                                              N                                          H    NH  H        CH.sub.3                                                                         CH.sub.3                                                                           CH.sub.3 N                                          H    NH  CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           CH.sub.3 CH                                         H    NH  CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.3                                                                              CH                                         H    NH  CH.sub.3 CH.sub.3                                                                         OCH.sub.3                                                                          OCH.sub.3                                                                              CH                                         H    NH  CH.sub.3 CH.sub.3                                                                         Cl   OCH.sub.3                                                                              CH                                         H    NH  CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.3                                                                              N                                          H    NH  CH.sub.3 CH.sub.3                                                                         OCH.sub.3                                                                          OCH.sub.3                                                                              N                                          H    NH  CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           CH.sub.3 N                                          H    NH  C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         CH.sub.3                                                                           CH.sub.3 CH                                         H    NH  C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.3                                                                              CH                                         H    NH  C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         OCH.sub.3                                                                          OCH.sub.3                                                                              CH                                         H    NH  C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         Cl   OCH.sub.3                                                                              CH                                         H    NH  C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.3                                                                              N                                          H    NH  C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         OCH.sub.3                                                                          OCH.sub.3                                                                              N                                          H    NH  C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         CH.sub.3                                                                           CH.sub.3 N                                          H    SO.sub.2                                                                          C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.2 CH.sub.3                                                                     CH                                         H    SO.sub.2                                                                          C.sub. 6 H.sub.5                                                                       CH.sub.3                                                                         CH.sub.3                                                                           NH.sub.2 CH                                         H    SO.sub.2                                                                          C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         CH.sub.3                                                                           NHCH.sub.3                                                                             CH                                         H    SO.sub.2                                                                          C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         CH.sub.3                                                                           N(CH.sub.3).sub.2                                                                      CH                                         H    SO.sub.2                                                                          C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         CH.sub.3                                                                           CH.sub.2 CH.sub.3                                                                      CH                                         H    SO.sub.2                                                                          C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         CH.sub.3                                                                           CF.sub.3 CH                                         H    SO.sub.2                                                                          C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         CH.sub.3                                                                           SCH.sub.3                                                                              CH                                         H    SO.sub.2                                                                          C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.2 CH═CH.sub.2                                                              CH                                         H    SO.sub.2                                                                          C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.2 CH.tbd.CH                                                                    CH                                         H    SO.sub.2                                                                          C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.2 CF.sub.3                                                                     CH                                         H    SO.sub.2                                                                          C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.2 CH.sub.2 OCH.sub.3                                                           CH                                         H    SO.sub.2                                                                          C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         CH.sub.3                                                                           CH(OCH.sub.3).sub.2                                                                    CH                                         H    SO.sub.2                                                                          C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         CH.sub.3                                                                           1,3-dioxolan-2-yl                                                                      CH                                         H    SO.sub.2                                                                          C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         CH.sub.3                                                                           CH.sub.2 OCH.sub.3                                                                     CH                                         H    SO.sub.2                                                                          C.sub. 6 H.sub.5                                                                       CH.sub.3                                                                         OCH.sub.3                                                                          N(CH.sub.3).sub.2                                                                      CH                                         H    SO.sub.2                                                                          C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         Br   OCH.sub.3                                                                              CH                                         H    SO.sub.2                                                                          C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         OCH.sub.2 F                                                                        OCH.sub.3                                                                              CH                                         H    SO.sub.2                                                                          C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         CF.sub.3                                                                           OCH.sub.3                                                                              CH                                         H    SO.sub.2                                                                          C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.2 F                                                                            CH                                         H    SO.sub.2                                                                          C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         CH.sub.3                                                                           CN       CH                                         H    SO.sub.2                                                                          C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         CH.sub.3                                                                           CH(OCH.sub.2 CH.sub.3).sub.2                                                           CH                                         H    SO.sub.2                                                                          C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         CH.sub.3                                                                           SCH.sub.2 F                                                                            CH                                         H    SO.sub.2                                                                          C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.2 CFBrF                                                                        CH                                         H    SO.sub.2                                                                          C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.2 CHFCF.sub.3                                                                  CH                                         H    S   CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.2 CH.sub.3                                                                     CH                                         H    S   CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           NH.sub.2 CH                                         H    S   CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           NHCH.sub.3                                                                             CH                                         H    S   CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           N(CH.sub.3).sub.2                                                                      CH                                         H    S   CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           CH.sub.2 CH.sub.3                                                                      CH                                         H    S   CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           CF.sub.3 CH                                         H    S   CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           SCH.sub.3                                                                              CH                                         H    S   CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.2 CH═CH.sub.2                                                              CH                                         H    S   CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.2 C.tbd.CH                                                                     CH                                         H    S   CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.2 CF.sub.3                                                                     CH                                         H    S   CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.2 CH.sub.2 OCH.sub.3                                                           CH                                         H    S   CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           CH(OCH.sub.3).sub.2                                                                    CH                                         H    S   CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           1,3-dioxolan-2-yl                                                                      CH                                         H    S   CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           CH.sub.2 OCH.sub.3                                                                     CH                                         H    S   CH.sub.3 CH.sub.3                                                                         Br   OCH.sub.3                                                                              CH                                         H    S   CH.sub.3 CH.sub.3                                                                         OCH.sub.2 F                                                                        OCH.sub.3                                                                              CH                                         H    S   CH.sub.3 CH.sub.3                                                                         CF.sub.3                                                                           OCH.sub.3                                                                              CH                                         H    S   CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.2 F                                                                            CH                                         H    S   CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           CN       CH                                         H    S   CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           CH(OCH.sub.2 CH.sub.3).sub.2                                                           CH                                         H    S   CH.sub. 3                                                                              CH.sub.3                                                                         CH.sub.3                                                                           OCF.sub.2 CHClF                                                                        CH                                         H    S   CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           SCH.sub.2 F                                                                            CH                                         H    S   CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.2 CFBrF                                                                        CH                                         H    S   CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           OCF.sub.2 CHFCF.sub.3                                                                  CH                                         H    S   CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.2 CH.sub.3                                                                     CH                                         H    SO.sub.2                                                                          CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           NH.sub.2 CH                                         H    SO.sub.2                                                                          CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           NHCH.sub.3                                                                             CH                                         H    SO.sub.2                                                                          CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           N(CH.sub.3).sub.2                                                                      CH                                         H    SO.sub.2                                                                          CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           CH.sub.2 CH.sub.3                                                                      CH                                         H    SO.sub.2                                                                          CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           CF.sub.3 CH                                         H    SO.sub.2                                                                          CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           SCH.sub.3                                                                              CH                                         H    SO.sub.2                                                                          CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.2 CH═CH.sub.2                                                              CH                                         H    SO.sub.2                                                                          CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.2 C.tbd.CH                                                                     CH                                         H    SO.sub.2                                                                          CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.2 CF.sub.3                                                                     CH                                         H    SO.sub.2                                                                          CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.2 CH.sub.2 OCH.sub.3                                                           CH                                         H    SO.sub.2                                                                          CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           CH(OCH.sub.3).sub.2                                                                    CH                                         H    SO.sub.2                                                                          CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           1,3-dioxolan-2-yl                                                                      CH                                         H    SO.sub.2                                                                          CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           CH.sub.2 OCH.sub.3                                                                     CH                                         H    SO.sub.2                                                                          CH.sub.3 CH.sub.3                                                                         Br   OCH.sub.3                                                                              CH                                         H    SO.sub.2                                                                          CH.sub.3 CH.sub.3                                                                         OCH.sub.2 F                                                                        OCH.sub.3                                                                              CH                                         H    SO.sub.2                                                                          CH.sub.3 CH.sub.3                                                                         CF.sub.3                                                                           OCH.sub.3                                                                              CH                                         H    SO.sub.2                                                                          CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.2 F                                                                            CH                                         H    SO.sub.2                                                                          CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           CN       CH                                         H    SO.sub.2                                                                          CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           CH(OCH.sub.2 CH.sub.3)                                                                 CH                                         H    SO.sub.2                                                                          CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           OCF.sub.2 CH ClF)                                                                      CH                                         H    SO.sub.2                                                                          CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           SCH.sub.2 F                                                                            CH                                         H    SO.sub.2                                                                          CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.2 CFBrF                                                                        CH                                         H    SO.sub.2                                                                          CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           OCF.sub.2 CHFCF.sub.3                                                                  CH                                         H    CH.sub.2                                                                          C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.2 CH.sub.3                                                                     CH                                         H    CH.sub.2                                                                          C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         CH.sub.3                                                                           NH.sub.2 CH                                         H    CH.sub.2                                                                          C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         CH.sub.3                                                                           NHCH.sub.3                                                                             CH                                         H    CH.sub.2                                                                          C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         CH.sub.3                                                                           N(CH.sub.3).sub.2                                                                      CH                                         H    CH.sub.2                                                                          C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         CH.sub.3                                                                           CH.sub.2 CH.sub.3                                                                      CH                                         H    CH.sub.2                                                                          C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         CH.sub.3                                                                           CF.sub.3 CH                                         H    CH.sub.2                                                                          C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         CH.sub.3                                                                           SCH.sub.3                                                                              CH                                         H    CH.sub.2                                                                          C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.2 CH═CH.sub.2                                                              CH                                         H    CH.sub.2                                                                          C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.2 C.tbd.CH                                                                     CH                                         H    CH.sub.2                                                                          C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.2 CF.sub.3                                                                     CH                                         H    CH.sub.2                                                                          C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.2 CH.sub.2 OCH.sub.3                                                           CH                                         H    CH.sub.2                                                                          C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         CH.sub.3                                                                           CH(OCH.sub.3).sub.2                                                                    CH                                         H    CH.sub.2                                                                          C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         CH.sub.3                                                                           1,3-dioxolan-2-yl                                                                      CH                                         H    CH.sub.2                                                                          C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         CH.sub.3                                                                           CH.sub.2 OCH.sub.3                                                                     CH                                         H    CH.sub.2                                                                          C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         Br   OCH.sub.3                                                                              CH                                         H    CH.sub.2                                                                          C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         OCH.sub.2 F                                                                        OCH.sub.3                                                                              CH                                         H    CH.sub.2                                                                          C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         CF.sub.3                                                                           OCH.sub.3                                                                              CH                                         H    CH.sub.2                                                                          C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.2 F                                                                            CH                                         H    CH.sub.2                                                                          C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         CH.sub.3                                                                           CN       CH                                         H    CH.sub.2                                                                          C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         CH.sub.3                                                                           CH(OCH.sub.2 CH.sub.3).sub.2                                                           CH                                         H    CH.sub.2                                                                          C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         CH.sub.3                                                                           SCH.sub.2 F                                                                            CH                                         H    CH.sub.2                                                                          C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.2 CFBrF                                                                        CH                                         H    CH.sub.2                                                                          C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         CH.sub.3                                                                           OCF.sub.2 CHFCF.sub.3                                                                  CH                                         H    CH.sub.2                                                                          CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.2 CH.sub.3                                                                     CH                                         H    CH.sub.2                                                                          CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           NH.sub.2 CH                                         H    CH.sub.2                                                                          CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           NHCH.sub.3                                                                             CH                                         H    CH.sub.2                                                                          CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           N(CH.sub.3).sub.2                                                                      CH                                         H    CH.sub.2                                                                          CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           CH.sub.2 CH.sub.3                                                                      CH                                         H    CH.sub. 2                                                                         CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           CF.sub.3 CH                                         H    CH.sub.2                                                                          CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           SCH.sub.3                                                                              CH                                         H    CH.sub.2                                                                          CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.2 CH═CH.sub.2                                                              CH                                         H    CH.sub.2                                                                          CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.2 C.tbd.CH                                                                     CH                                         H    CH.sub.2                                                                          CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.2 CF.sub.3                                                                     CH                                         H    CH.sub.2                                                                          CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.2 CH.sub.2 OCH.sub.3                                                           CH                                         H    CH.sub.2                                                                          CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           CH(OCH.sub.3).sub.2                                                                    CH                                         H    CH.sub.2                                                                          CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           1,3-dioxolan-2-yl                                                                      CH                                         H    CH.sub.2                                                                          CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           CH.sub.2 OCH.sub.3                                                                     CH                                         H    CH.sub.2                                                                          CH.sub.3 CH.sub.3                                                                         Br   OCH.sub.3                                                                              CH                                         H    CH.sub.2                                                                          CH.sub.3 CH.sub.3                                                                         OCH.sub.2 F                                                                        OCH.sub.3                                                                              CH                                         H    CH.sub.2                                                                          CH.sub.3 CH.sub.3                                                                         CF.sub.3                                                                           OCH.sub.3                                                                              CH                                         H    CH.sub.2                                                                          CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.2 F                                                                            CH                                         H    CH.sub.2                                                                          CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           CN       CH                                         H    CH.sub.2                                                                          CH.sub.3 CH.sub. 3                                                                        CH.sub.3                                                                           CH(OCH.sub.2 CH.sub.3).sub.2                                                           CH                                         H    CH.sub.2                                                                          CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           OCF.sub.2 CHClF                                                                        CH                                         H    CH.sub.2                                                                          CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           SCH.sub.2 F                                                                            CH                                         H    CH.sub.2                                                                          CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.2 CFBrF                                                                        CH                                         H    CH.sub.2                                                                          CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           OCF.sub.2 CHFCF.sub.3                                                                  CH                                         6-CH.sub.3                                                                         C═O                                                                           H        CH.sub.3                                                                         CH.sub.3                                                                           CH.sub.3 CH                                         6-CH.sub.3                                                                         C═O                                                                           H        CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.3                                                                              CH                                         6-CH.sub.3                                                                         C═O                                                                           H        CH.sub.3                                                                         OCH.sub.3                                                                          OCH.sub.3                                                                              CH                                         6-CH.sub.3                                                                         C═O                                                                           H        CH.sub.3                                                                         Cl   OCH.sub.3                                                                              CH                                         6-CH.sub.3                                                                         C═O                                                                           H        CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.3                                                                              N                                          6-CH.sub.3                                                                         C═O                                                                           H        CH.sub.3                                                                         OCH.sub.3                                                                          OCH.sub.3                                                                              N                                          6-CH.sub.3                                                                         C═O                                                                           H        CH.sub.3                                                                         CH.sub.3                                                                           CH.sub.3 N                                          6-CH.sub.3                                                                         C═O                                                                           C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         CH.sub.3                                                                           CH.sub.3 CH                                         6-CH.sub.3                                                                         C═O                                                                           C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.3                                                                              CH                                         6-CH.sub.3                                                                         C═O                                                                           C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         OCH.sub.3                                                                          OCH.sub. 3                                                                             CH                                         6-CH.sub.3                                                                         C═O                                                                           C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         Cl   OCH.sub.3                                                                              CH                                         6-CH.sub.3                                                                         C═O                                                                           C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.3                                                                              N                                          6-CH.sub.3                                                                         C═O                                                                           C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         OCH.sub.3                                                                          OCH.sub.3                                                                              N                                          6-CH.sub.3                                                                         C═O                                                                           C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         CH.sub.3                                                                           CH.sub.3 N                                          6-CH.sub.3                                                                         C═O                                                                           C.sub.6 H.sub.5                                                                        H  CH.sub.3                                                                           CH.sub.3 N                                          6-CH.sub.3                                                                         C═O                                                                           C.sub.6 H.sub.5                                                                        H  CH.sub.3                                                                           OCH.sub.3                                                                              CH                                         6-CH.sub.3                                                                         C═O                                                                           C.sub.6 H.sub.5                                                                        H  OCH.sub.3                                                                          OCH.sub.3                                                                              CH                                         6-CH.sub.3                                                                         C═O                                                                           C.sub.6 H.sub.5                                                                        H  Cl   OCH.sub.3                                                                              CH                                         6-CH.sub.3                                                                         C═O                                                                           C.sub.6 H.sub.5                                                                        H  CH.sub.3                                                                           OCH.sub.3                                                                              N                                          6-CH.sub.3                                                                         C═O                                                                           C.sub.6 H.sub.5                                                                        H  OCH.sub.3                                                                          OCH.sub.3                                                                              N                                          6-CH.sub.3                                                                         C═O                                                                           C.sub.6 H.sub.5                                                                        H  CH.sub.3                                                                           CH.sub.3 N                                          6-CH.sub.3                                                                         C═O                                                                           H        CH.sub.3                                                                         CH.sub.3                                                                           CH.sub.3 CH                                         6-CH.sub.3                                                                         C═O                                                                           H        CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.3                                                                              CH                                         6-CH.sub.3                                                                         C═O                                                                           H        CH.sub.3                                                                         OCH.sub.3                                                                          OCH.sub.3                                                                              CH                                         6-CH.sub.3                                                                         C═O                                                                           H        CH.sub. 3                                                                        Cl   OCH.sub.3                                                                              CH                                         6-CH.sub.3                                                                         C═O                                                                           H        CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.3                                                                              N                                          6-CH.sub.3                                                                         C═O                                                                           H        CH.sub.3                                                                         OCH.sub.3                                                                          OCH.sub.3                                                                              N                                          6-CH.sub.3                                                                         C═O                                                                           H        CH.sub.3                                                                         CH.sub.3                                                                           CH.sub.3 N                                          6-CH.sub.3                                                                         C═O                                                                           CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           CH.sub.3 CH                                         6-CH.sub.3                                                                         C═O                                                                           CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.3                                                                              CH                                         6-CH.sub.3                                                                         C═O                                                                           CH.sub.3 CH.sub.3                                                                         OCH.sub.3                                                                          OCH.sub.3                                                                              CH                                         6-CH.sub.3                                                                         C═O                                                                           CH.sub.3 CH.sub.3                                                                         Cl   OCH.sub.3                                                                              CH                                         6-CH.sub.3                                                                         C═O                                                                           CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.3                                                                              N                                          6-CH.sub.3                                                                         C═O                                                                           CH.sub.3 CH.sub.3                                                                         OCH.sub.3                                                                          OCH.sub.3                                                                              N                                          6-CH.sub.3                                                                         C═O                                                                           CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           CH.sub.3 N                                          6-CH.sub.3                                                                         C═O                                                                           CH.sub.3 H  CH.sub.3                                                                           CH.sub.3 CH                                         6-CH.sub.3                                                                         C═O                                                                           CH.sub.3 H  CH.sub.3                                                                           OCH.sub.3                                                                              CH                                         6-CH.sub.3                                                                         C═O                                                                           CH.sub.3 H  OCH.sub.3                                                                          OCH.sub.3                                                                              CH                                         6-CH.sub.3                                                                         C═O                                                                           CH.sub.3 H  Cl   OCH.sub.3                                                                              CH                                         6-CH.sub.3                                                                         C═O                                                                           CH.sub.3 H  CH.sub.3                                                                           OCH.sub.3                                                                              N                                          6-CH.sub.3                                                                         C═O                                                                           CH.sub.3 H  OCH.sub.3                                                                          OCH.sub. 3                                                                             N                                          6-CH.sub.3                                                                         C═O                                                                           CH.sub.3 H  CH.sub.3                                                                           CH.sub.3 N                                          6-CH.sub.3                                                                         C═O                                                                           H        H  CH.sub.3                                                                           OCH.sub.3                                                                              CH                                         6-CH.sub.3                                                                         C═O                                                                           H        H  OCH.sub.3                                                                          OCH.sub.3                                                                              CH                                         6-CH.sub.3                                                                         C═O                                                                           H        H  Cl   OCH.sub.3                                                                              CH                                         6-CH.sub.3                                                                         C═O                                                                           H        H  CH.sub.3                                                                           OCH.sub.3                                                                              N                                          6-CH.sub.3                                                                         C═O                                                                           H        H  OCH.sub.3                                                                          OCH.sub.3                                                                              N                                          6-CH.sub.3                                                                         C═O                                                                           H        H  CH.sub.3                                                                           CH.sub.3 N                                          6-CH.sub.3                                                                         C═O                                                                           2-pyridyl                                                                              CH.sub.3                                                                         CH.sub.3                                                                           CH.sub.3 CH                                         6-CH.sub.3                                                                         C═O                                                                           2-pyridyl                                                                              CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.3                                                                              CH                                         6-CH.sub.3                                                                         C═O                                                                           2-pyridyl                                                                              CH.sub.3                                                                         OCH.sub.3                                                                          OCH.sub.3                                                                              CH                                         6-CH.sub.3                                                                         C═O                                                                           2-pyridyl                                                                              CH.sub.3                                                                         Cl   OCH.sub.3                                                                              CH                                         6-CH.sub.3                                                                         C═O                                                                           2-pyridyl                                                                              CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.3                                                                              N                                          6-CH.sub.3                                                                         C═O                                                                           2-pyridyl                                                                              CH.sub.3                                                                         OCH.sub.3                                                                          OCH.sub.3                                                                              N                                          6-CH.sub.3                                                                         C═O                                                                           2-pyridyl                                                                              CH.sub.3                                                                         CH.sub.3                                                                           CH.sub.3 N                                          6-CH.sub.3                                                                         C═O                                                                           4-Cl--C.sub.6 H.sub.5                                                                  CH.sub.3                                                                         CH.sub.3                                                                           CH.sub.3 CH                                         6-CH.sub.3                                                                         C═O                                                                           4-Cl--C.sub.6 H.sub.5                                                                  CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.3                                                                              CH                                         6-CH.sub.3                                                                         C═O                                                                           4-Cl--C.sub. 6 H.sub.5                                                                 CH.sub.3                                                                         OCH.sub.3                                                                          OCH.sub.3                                                                              CH                                         6-CH.sub.3                                                                         C═O                                                                           4-Cl--C.sub.6 H.sub.5                                                                  CH.sub.3                                                                         Cl   OCH.sub.3                                                                              CH                                         6-CH.sub.3                                                                         C═O                                                                           4-Cl--C.sub.6 H.sub.5                                                                  CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.3                                                                              N                                          6-CH.sub.3                                                                         C═O                                                                           4-Cl--C.sub.6 H.sub.5                                                                  CH.sub.3                                                                         OCH.sub.3                                                                          OCH.sub.3                                                                              N                                          6-CH.sub.3                                                                         C═O                                                                           4-Cl--C.sub.6 H.sub.5                                                                  CH.sub.3                                                                         CH.sub.3                                                                           CH.sub.3 N                                          6-CH.sub.3                                                                         C═O                                                                           4-Cl--C.sub.6 H.sub.5                                                                  H  CH.sub.3                                                                           CH.sub.3 CH                                         6-CH.sub.3                                                                         C═O                                                                           2-pyridyl                                                                              H  CH.sub.3                                                                           OCH.sub.3                                                                              CH                                         6-CH.sub.3                                                                         C═O                                                                           2-pyridyl                                                                              H  OCH.sub.3                                                                          OCH.sub.3                                                                              CH                                         6-CH.sub.3                                                                         C═O                                                                           2-pyridyl                                                                              H  Cl   OCH.sub.3                                                                              CH                                         6-CH.sub.3                                                                         C═O                                                                           2-pyridyl                                                                              H  CH.sub.3                                                                           OCH.sub.3                                                                              N                                          6-CH.sub.3                                                                         C═O                                                                           2-pyridyl                                                                              H  OCH.sub.3                                                                          OCH.sub.3                                                                              N                                          6-CH.sub.3                                                                         C═O                                                                           2-pyridyl                                                                              H  CH.sub.3                                                                           CH.sub.3 N                                          6-Cl C═O                                                                           H        CH.sub.3                                                                         CH.sub.3                                                                           CH.sub.3 CH                                         6-Cl C═O                                                                           H        CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.3                                                                              CH                                         6-Cl C═O                                                                           H        CH.sub.3                                                                         OCH.sub.3                                                                          OCH.sub.3                                                                              CH                                         6-Cl C═O                                                                           H        CH.sub.3                                                                         Cl   OCH.sub.3                                                                              CH                                         6-Cl C═O                                                                           H        CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.3                                                                              N                                          6-Cl C═O                                                                           H        CH.sub.3                                                                         OCH.sub.3                                                                          OCH.sub.3                                                                              N                                          6-Cl C═O                                                                           H        CH.sub.3                                                                         CH.sub.3                                                                           CH.sub.3 N                                          6-Cl C═O                                                                           C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         CH.sub.3                                                                           CH.sub.3 CH                                         6-Cl C═O                                                                           C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.3                                                                              CH                                         6-Cl C═O                                                                           C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         OCH.sub.3                                                                          OCH.sub.3                                                                              CH                                         6-Cl C═O                                                                           C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         Cl   OCH.sub.3                                                                              CH                                         6-Cl C═O                                                                           C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.3                                                                              N                                          6-Cl C═O                                                                           C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         OCH.sub.3                                                                          OCH.sub.3                                                                              N                                          6-Cl C═O                                                                           C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         CH.sub.3                                                                           CH.sub.3 N                                          6-Cl C═O                                                                           C.sub.6 H.sub.5                                                                        H  CH.sub.3                                                                           CH.sub.3 CH                                         6-Cl C═O                                                                           C.sub.6 H.sub.5                                                                        H  CH.sub.3                                                                           OCH.sub.3                                                                              CH                                         6-Cl C═O                                                                           C.sub.6 H.sub.5                                                                        H  OCH.sub.3                                                                          OCH.sub.3                                                                              CH                                         6-Cl C═O                                                                           C.sub.6 H.sub.5                                                                        H  Cl   OCH.sub.3                                                                              CH                                         6-Cl C═O                                                                           C.sub.6 H.sub.5                                                                        H  CH.sub.3                                                                           OCH.sub.3                                                                              N                                          6-Cl C═O                                                                           C.sub.6 H.sub.5                                                                        H  OCH.sub.3                                                                          OCH.sub.3                                                                              N                                          6-Cl C═O                                                                           C.sub.6 H.sub.5                                                                        H  CH.sub.3                                                                           CH.sub.3 N                                          6-Cl C═O                                                                           CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           CH.sub.3 CH                                         6-Cl C═O                                                                           CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.3                                                                              CH                                         6-Cl C═O                                                                           H        CH.sub.3                                                                         OCH.sub.3                                                                          OCH.sub.3                                                                              CH                                         6-Cl C═O                                                                           H        CH.sub.3                                                                         Cl   OCH.sub.3                                                                              CH                                         6-Cl C═O                                                                           H        CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.3                                                                              N                                          6-Cl C═O                                                                           H        CH.sub.3                                                                         OCH.sub.3                                                                          OCH.sub.3                                                                              N                                          6-Cl C═O                                                                           H        CH.sub.3                                                                         CH.sub.3                                                                           CH.sub.3 N                                          6-Cl C═O                                                                           CH.sub.3 H  CH.sub.3                                                                           CH.sub.3 CH                                         6-Cl C═O                                                                           CH.sub.3 H  CH.sub.3                                                                           OCH.sub.3                                                                              CH                                         6-Cl C═O                                                                           CH.sub.3 H  OCH.sub.3                                                                          OCH.sub.3                                                                              CH                                         6-Cl C═O                                                                           CH.sub.3 CH.sub.3                                                                         Cl   OCH.sub.3                                                                              CH                                         6-Cl C═O                                                                           CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.3                                                                              N                                          6-Cl C═O                                                                           CH.sub.3 CH.sub.3                                                                         OCH.sub.3                                                                          OCH.sub.3                                                                              N                                          6-Cl C═O                                                                           CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           CH.sub.3 N                                          6-Cl C═O                                                                           CH.sub.3 H  CH.sub.3                                                                           CH.sub.3 CH                                         6-Cl C═O                                                                           H        H  CH.sub.3                                                                           OCH.sub.3                                                                              CH                                         6-Cl C═O                                                                           H        H  OCH.sub.3                                                                          OCH.sub.3                                                                              CH                                         6-Cl C═O                                                                           H        H  Cl   OCH.sub.3                                                                              CH                                         6-Cl C═O                                                                           H        H  CH.sub.3                                                                           OCH.sub.3                                                                              N                                          6-Cl C═O                                                                           H        H  OCH.sub.3                                                                          OCH.sub.3                                                                              N                                          6-Cl C═O                                                                           H        H  CH.sub.3                                                                           CH.sub.3 N                                          6-Cl C═O                                                                           2-pyridyl                                                                              CH.sub.3                                                                         CH.sub.3                                                                           CH.sub.3 CH                                         6-Cl C═O                                                                           2-pyridyl                                                                              CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.3                                                                              CH                                         6-Cl C═O                                                                           2-pyridyl                                                                              CH.sub.3                                                                         OCH.sub.3                                                                          OCH.sub.3                                                                              CH                                         6-Cl C═O                                                                           2-pyridyl                                                                              CH.sub.3                                                                         Cl   OCH.sub.3                                                                              CH                                         6-Cl C═O                                                                           2-pyridyl                                                                              CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.3                                                                              N                                          6-Cl C═O                                                                           2-pyridyl                                                                              CH.sub.3                                                                         OCH.sub.3                                                                          OCH.sub.3                                                                              N                                          6-Cl C═O                                                                           2-pyridyl                                                                              CH.sub.3                                                                         CH.sub.3                                                                           CH.sub.3 N                                          6-Cl C═O                                                                           4-Cl--phenyl                                                                           CH.sub.3                                                                         CH.sub.3                                                                           CH.sub.3 CH                                         6-Cl C═O                                                                           4-Cl--phenyl                                                                           CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.3                                                                              CH                                         6-Cl C═O                                                                           4-Cl--phenyl                                                                           CH.sub.3                                                                         OCH.sub.3                                                                          OCH.sub.3                                                                              CH                                         6-Cl C═O                                                                           4-Cl--phenyl                                                                           CH.sub.3                                                                         Cl   OCH.sub.3                                                                              CH                                         6-Cl C═O                                                                           4-Cl--phenyl                                                                           CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.3                                                                              N                                          6-Cl C═O                                                                           4-Cl--phenyl                                                                           CH.sub.3                                                                         OCH.sub.3                                                                          OCH.sub.3                                                                              N                                          6-Cl C═O                                                                           4-Cl--phenyl                                                                           CH.sub.3                                                                         CH.sub.3                                                                           CH.sub.3 N                                          6-Cl C═O                                                                           2-pyridyl                                                                              H  CH.sub.3                                                                           CH.sub.3 CH                                         6-Cl C═O                                                                           2-pyridyl                                                                              H  CH.sub.3                                                                           OCH.sub.3                                                                              CH                                         6-Cl C═O                                                                           2-pyridyl                                                                              H  OCH.sub.3                                                                          OCH.sub.3                                                                              CH                                         6-Cl C═O                                                                           2-pyridyl                                                                              H  Cl   OCH.sub.3                                                                              CH                                         6-Cl C═O                                                                           2-pyridyl                                                                              H  CH.sub.3                                                                           OCH.sub.3                                                                              N                                          6-Cl C═O                                                                           2-pyridyl                                                                              H  OCH.sub.3                                                                          OCH.sub.3                                                                              N                                          6-Cl C═O                                                                           2-pyridyl                                                                              H  CH.sub.3                                                                           CH.sub.3 N                                          5-NO.sub.2                                                                         C═O                                                                           H        CH.sub.3                                                                         CH.sub.3                                                                           CH.sub.3 CH                                         5-NO.sub.2                                                                         C═O                                                                           H        CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.3                                                                              CH                                         5-NO.sub.2                                                                         C═O                                                                           H        CH.sub.3                                                                         OCH.sub.3                                                                          OCH.sub.3                                                                              CH                                         5-NO.sub.2                                                                         C═O                                                                           H        CH.sub.3                                                                         Cl   OCH.sub.3                                                                              CH                                         5-NO.sub.2                                                                         C═O                                                                           H        CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.3                                                                              N                                          5-NO.sub.2                                                                         C═O                                                                           H        CH.sub.3                                                                         OCH.sub.3                                                                          OCH.sub.3                                                                              N                                          5-NO.sub.2                                                                         C═O                                                                           H        CH.sub.3                                                                         CH.sub.3                                                                           CH.sub.3 N                                          5-NO.sub.2                                                                         C═O                                                                           C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         CH.sub.3                                                                           CH.sub.3 CH                                         5-NO.sub.2                                                                         C═O                                                                           C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.3                                                                              CH                                         5-NO.sub.2                                                                         C═O                                                                           C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         OCH.sub.3                                                                          OCH.sub.3                                                                              CH                                         5-NO.sub.2                                                                         C═O                                                                           C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         Cl   OCH.sub.3                                                                              CH                                         5-NO.sub.2                                                                         C═O                                                                           C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.3                                                                              N                                          5-NO.sub.2                                                                         C═O                                                                           C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         OCH.sub.3                                                                          OCH.sub.3                                                                              N                                          5-NO.sub.2                                                                         C═O                                                                           C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         CH.sub.3                                                                           CH.sub.3 N                                          5-NO.sub.2                                                                         C═O                                                                           C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         CH.sub.3                                                                           CH.sub.3 CH                                         5-NO.sub.2                                                                         C═O                                                                           CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.3                                                                              CH                                         5-NO.sub.2                                                                         C═O                                                                           CH.sub.3 CH.sub.3                                                                         OCH.sub.3                                                                          OCH.sub.3                                                                              CH                                         5-NO.sub.2                                                                         C═O                                                                           CH.sub.3 CH.sub.3                                                                         Cl   OCH.sub.3                                                                              CH                                         5-NO.sub.2                                                                         C═O                                                                           CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.3                                                                              N                                          5-NO.sub.2                                                                         C═O                                                                           CH.sub.3 CH.sub.3                                                                         OCH.sub.3                                                                          OCH.sub.3                                                                              N                                          5-NO.sub.2                                                                         C═O                                                                           CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           CH.sub.3 N                                          5-SCH.sub.3                                                                        C═O                                                                           H        CH.sub.3                                                                         CH.sub.3                                                                           CH.sub.3 CH                                         5-SCH.sub.3                                                                        C═O                                                                           H        CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.3                                                                              CH                                         5-SCH.sub.3                                                                        C═O                                                                           H        CH.sub.3                                                                         OCH.sub.3                                                                          OCH.sub.3                                                                              CH                                         5-SCH.sub.3                                                                        C═O                                                                           H        CH.sub.3                                                                         Cl   OCH.sub.3                                                                              CH                                         5-SCH.sub.3                                                                        C═O                                                                           H        CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.3                                                                              N                                          5-SCH.sub.3                                                                        C═O                                                                           H        CH.sub.3                                                                         OCH.sub.3                                                                          OCH.sub.3                                                                              N                                          5-SCH.sub.3                                                                        C═O                                                                           H        CH.sub.3                                                                         CH.sub.3                                                                           CH.sub.3 N                                          5-SCH.sub.3                                                                        C═O                                                                           C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         CH.sub.3                                                                           CH.sub.3 CH                                         5-SCH.sub.3                                                                        C═O                                                                           C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.3                                                                              CH                                         5-SCH.sub.3                                                                        C═O                                                                           C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         OCH.sub.3                                                                          OCH.sub.3                                                                              CH                                         5-SCH.sub.3                                                                        C═O                                                                           C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         Cl   OCH.sub.3                                                                              CH                                         5-SCH.sub.3                                                                        C═O                                                                           C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.3                                                                              N                                          5-SCH.sub.3                                                                        C═O                                                                           C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         OCH.sub.3                                                                          OCH.sub.3                                                                              N                                          5-SCH.sub.3                                                                        C═O                                                                           C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         CH.sub.3                                                                           CH.sub.3 N                                          5-SCH.sub.3                                                                        C═O                                                                           CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           CH.sub.3 CH                                         5-SCH.sub.3                                                                        C═O                                                                           CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.3                                                                              CH                                         5-SCH.sub.3                                                                        C═O                                                                           CH.sub.3 CH.sub.3                                                                         OCH.sub.3                                                                          OCH.sub.3                                                                              CH                                         5-SCH.sub.3                                                                        C═O                                                                           CH.sub.3 CH.sub. 3                                                                        Cl   OCH.sub.3                                                                              CH                                         5-SCH.sub.3                                                                        C═O                                                                           CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.3                                                                              N                                          5-SCH.sub.3                                                                        C═O                                                                           CH.sub.3 CH.sub.3                                                                         OCH.sub.3                                                                          OCH.sub.3                                                                              N                                          5-SCH.sub.3                                                                        C═O                                                                           CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           CH.sub.3 N                                          6-F  C═O                                                                           H        CH.sub.3                                                                         CH.sub.3                                                                           CH.sub.3 CH                                         6-F  C═O                                                                           H        CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.3                                                                              CH                                         6-F  C═O                                                                           H        CH.sub.3                                                                         OCH.sub.3                                                                          OCH.sub.3                                                                              CH                                         6-F  C═O                                                                           H        CH.sub.3                                                                         Cl   OCH.sub.3                                                                              CH                                         6-F  C═O                                                                           H        CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.3                                                                              N                                          6-F  C═O                                                                           H        CH.sub.3                                                                         OCH.sub.3                                                                          OCH.sub.3                                                                              N                                          6-F  C═O                                                                           H        CH.sub.3                                                                         CH.sub.3                                                                           CH.sub.3 N                                          5-F  C═O                                                                           C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         CH.sub.3                                                                           CH.sub.3 CH                                         5-F  C═O                                                                           C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.3                                                                              CH                                         5-F  C═O                                                                           C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         OCH.sub.3                                                                          OCH.sub.3                                                                              CH                                         5-F  C═O                                                                           C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         Cl   OCH.sub.3                                                                              CH                                         5-F  C═O                                                                           C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.3                                                                              N                                          5-F  C═O                                                                           C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         OCH.sub.3                                                                          OCH.sub.3                                                                              N                                          5-F  C═O                                                                           C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         CH.sub.3                                                                           CH.sub.3 N                                          6-F  C═O                                                                           C.sub.6 H.sub.5                                                                        CH.sub.3                                                                         CH.sub.3                                                                           CH.sub.3 CH                                         6-F  C═O                                                                           CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.3                                                                              CH                                         6-F  C═O                                                                           CH.sub.3 CH.sub.3                                                                         OCH.sub.3                                                                          OCH.sub.3                                                                              CH                                         6-F  C═O                                                                           CH.sub.3 CH.sub.3                                                                         Cl   OCH.sub.3                                                                              CH                                         6-F  C═O                                                                           CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           OCH.sub.3                                                                              N                                          6-F  C═O                                                                           CH.sub.3 CH.sub.3                                                                         OCH.sub.3                                                                          OCH.sub.3                                                                              N                                          6-F  C═O                                                                           CH.sub.3 CH.sub.3                                                                         CH.sub.3                                                                           CH.sub.3 N                                          H    SO.sub.2                                                                          CH.sub.2 CH.sub.2 CH.sub.3                                                             H  OCH.sub.3                                                                          OCH.sub.3                                                                              CH 244-247                                 H    SO.sub.2                                                                          CH.sub.2 CH.sub.2 CH.sub.3                                                             H  CH.sub.3                                                                           OCH.sub.3                                                                              CH                                         H    SO.sub.2                                                                          CH.sub.2 CH.sub.2 CH.sub.3                                                             H  Cl   OCH.sub.3                                                                              CH 245-250                                 H    SO.sub.2                                                                          CH.sub.2 CH.sub.2 CH.sub.3                                                             H  OCH.sub.3                                                                          OCH.sub.3                                                                              N  213-216                                 H    SO.sub.2                                                                          CH.sub.2 CH.sub.2 CH.sub.3                                                             H  CH.sub.3                                                                           OCH.sub.3                                                                              N  210-212                                 H    SO.sub.2                                                                          CH.sub.2 C.sub.6 H.sub.5                                                               H  OCH.sub.3                                                                          OCH.sub.3                                                                              CH 214- 216                                H    SO.sub.2                                                                          CH.sub.2 C.sub.6 H.sub.5                                                               H  CH.sub.3                                                                           OCH.sub.3                                                                              CH 227-231                                 H    SO.sub.2                                                                          CH.sub.2 C.sub.6 H.sub.5                                                               H  CH.sub.3                                                                           CH.sub.3 CH 237-243                                 H    SO.sub.2                                                                          CH.sub.2 C.sub.6 H.sub.5                                                               H  OCH.sub.3                                                                          OCH.sub.3                                                                              N  221-225                                 H    SO.sub.2                                                                          CH.sub.2 C.sub.6 H.sub.5                                                               H  CH.sub.3                                                                           OCH.sub.3                                                                              N  237-243                                 H    SO.sub.2                                                                          3-F--C.sub.6 H.sub.5                                                                   H  OCH.sub.3                                                                          OCH.sub.3                                                                              CH 208-210                                 H    SO.sub.2                                                                          3-F--C.sub.6 H.sub.5                                                                   H  CH.sub.3                                                                           OCH.sub.3                                                                              CH 215-220                                 H    SO.sub.2                                                                          CH.sub.2 C.sub.6 H.sub.5                                                               H  Cl   OCH.sub.3                                                                              CH 202-205                                 __________________________________________________________________________

                  TABLE Ib                                                        ______________________________________                                        General Formula Ib                                                            R.sub.1                                                                              J        R.sub.6 X.sub.1 Y.sub.1                                                                            m.p. (°C.)                        ______________________________________                                        H      C═O  H       CH.sub.3                                                                              O                                             H      C═O  H       OCH.sub.3                                                                             O                                             H      C═O  H       OC.sub.2 H.sub.5                                                                      O                                             H      C═O  H       OCF.sub.2 H                                                                           O                                             H      C═O  CH.sub.3                                                                              CH.sub.3                                                                              O                                             H      C═O  CH.sub.3                                                                              OCH.sub.3                                                                             O                                             H      C═O  CH.sub.3                                                                              OC.sub.2 H.sub.5                                                                      O                                             H      C═O  CH.sub.3                                                                              OCF.sub.2 H                                                                           O                                             H      C═O  C.sub.6 H.sub.5                                                                       CH.sub.3                                                                              O                                             H      C═O  C.sub.6 H.sub.5                                                                       OCH.sub.3                                                                             O                                             H      C═O  C.sub.6 H.sub.5                                                                       OC.sub.2 H.sub.5                                                                      O                                             H      C═O  C.sub.6 H.sub.5                                                                       OCF.sub.2 H                                                                           O                                             H      C═O  CH.sub.3                                                                              CH.sub.3                                                                              CH.sub.2                                      H      C═O  CH.sub.3                                                                              OCH.sub.3                                                                             CH.sub.2                                      H      C═O  CH.sub.3                                                                              OC.sub.2 H.sub.5                                                                      CH.sub.2                                      H      C═O  CH.sub.3                                                                              OCF.sub.2 H                                                                           CH.sub.2                                      H      C═O  C.sub.6 H.sub.5                                                                       CH.sub.3                                                                              CH.sub.2                                      H      C═O  C.sub.6 H.sub.5                                                                       OCH.sub.3                                                                             CH.sub.2                                      H      C═O  C.sub.6 H.sub.5                                                                       OC.sub.2 H.sub.5                                                                      CH.sub.2                                      H      C═O  C.sub.6 H.sub.5                                                                       OCF.sub.2 H                                                                           CH.sub.2                                      H      SO.sub.2 H       CH.sub.3                                                                              O                                             H      SO.sub.2 H       OCH.sub.3                                                                             O                                             H      SO.sub.2 H       OC.sub.2 H.sub.5                                                                      O                                             H      SO.sub.2 H       OCF.sub.2 H                                                                           O                                             H      SO.sub.2 CH.sub.3                                                                              CH.sub.3                                                                              O                                             H      SO.sub.2 CH.sub.3                                                                              OCH.sub.3                                                                             O                                             H      SO.sub.2 CH.sub.3                                                                              OC.sub.2 H.sub.5                                                                      O                                             H      SO.sub.2 CH.sub.3                                                                              OCF.sub.2 H                                                                           O                                             H      SO.sub.2 C.sub.6 H.sub.5                                                                       CH.sub.3                                                                              O                                             H      SO.sub.2 C.sub.6 H.sub.5                                                                       OCH.sub.3                                                                             O                                             H      SO.sub.2 C.sub.6 H.sub.5                                                                       OC.sub.2 H.sub.5                                                                      O                                             H      SO.sub.2 C.sub.6 H.sub.5                                                                       OCF.sub.2 H                                                                           O                                             H      SO.sub.2 CH.sub.3                                                                              CH.sub.3                                                                              CH.sub.2                                      H      SO.sub.2 CH.sub.3                                                                              OCH.sub.3                                                                             CH.sub.2                                      H      SO.sub.2 CH.sub.3                                                                              OC.sub.2 H.sub.5                                                                      CH.sub.2                                      H      SO.sub.2 CH.sub.3                                                                              OCF.sub.2 H                                                                           CH.sub.2                                      H      SO.sub.2 C.sub.6 H.sub.5                                                                       CH.sub.3                                                                              CH.sub.2                                      H      SO.sub.2 C.sub.6 H.sub.5                                                                       OCH.sub.3                                                                             CH.sub.2                                      H      SO.sub.2 C.sub.6 H.sub.5                                                                       OC.sub.2 H.sub.5                                                                      CH.sub.2                                      H      SO.sub.2 C.sub.6 H.sub.5                                                                       OCF.sub.2 H                                                                           CH.sub.2                                      ______________________________________                                    

                  TABLE Ic                                                        ______________________________________                                        General Formula Ic                                                            R.sub.1                                                                              J         R.sub.6  X.sub.1                                                                              m.p. (°C.)                            ______________________________________                                        H      C═O   H        CH.sub.3                                            H      C═O   H        OCH.sub.3                                           H      C═O   H        OC.sub.2 H.sub.5                                    H      C═O   H        OCF.sub.2 H                                         H      C═O   CH.sub.3 CH.sub.3                                            H      C═O   CH.sub.3 OCH.sub.3                                           H      C═O   CH.sub.3 OC.sub.2 H.sub.5                                    H      C═O   CH.sub.3 OCF.sub.2 H                                         H      C═O   C.sub.6 H.sub.5                                                                        CH.sub.3                                            H      C═O   C.sub.6 H.sub.5                                                                        OCH.sub.3                                           H      C═O   C.sub.6 H.sub.5                                                                        OC.sub.2 H.sub.5                                    H      C═O   C.sub.6 H.sub.5                                                                        OCF.sub.2 H                                         H      SO.sub.2  CH.sub.3 CH.sub.3                                            H      SO.sub.2  CH.sub.3 OCH.sub.3                                           H      SO.sub.2  CH.sub.3 OC.sub.2 H.sub.5                                    H      SO.sub.2  CH.sub.3 OCF.sub.2 H                                         H      SO.sub.2  C.sub.6 H.sub.5                                                                        CH.sub.3                                            H      SO.sub.2  C.sub.6 H.sub.5                                                                        OCH.sub.3                                           H      SO.sub.2  C.sub.6 H.sub.5                                                                        OC.sub.2 H.sub.5                                    H      SO.sub.2  C.sub.6 H.sub.5                                                                        OCF.sub.2 H                                         ______________________________________                                    

                  TABLE Id                                                        ______________________________________                                        General Formula Id                                                            R.sub.1                                                                              J        R.sub.6 X.sub.1 Y.sub.2                                                                            m.p. (°C.)                        ______________________________________                                        H      C═O  H       CH.sub.3                                                                              CH.sub.3                                      H      C═O  H       OCH.sub.3                                                                             CH.sub.3                                      H      C═O  H       OC.sub.2 H.sub.5                                                                      CH.sub.3                                      H      C═O  H       OCF.sub.2 H                                                                           CH.sub.3                                      H      C═O  CH.sub.3                                                                              CH.sub.3                                                                              H                                             H      C═O  CH.sub.3                                                                              OCH.sub.3                                                                             H                                             H      C═O  CH.sub.3                                                                              OC.sub.2 H.sub.5                                                                      H                                             H      C═O  CH.sub.3                                                                              OCF.sub.2 H                                                                           H                                             H      C═O  C.sub.6 H.sub.5                                                                       CH.sub.3                                                                              H                                             H      C═O  C.sub.6 H.sub.5                                                                       OCH.sub.3                                                                             H                                             H      C═O  C.sub.6 H.sub.5                                                                       OC.sub.2 H.sub.5                                                                      H                                             H      C═O  C.sub.6 H.sub.5                                                                       OCF.sub.2 H                                                                           H                                             H      SO.sub.2 CH.sub.3                                                                              CH.sub.3                                                                              CH.sub.3                                      H      SO.sub.2 CH.sub.3                                                                              OCH.sub.3                                                                             CH.sub.3                                      H      SO.sub.2 CH.sub.3                                                                              OC.sub.2 H.sub.5                                                                      CH.sub.3                                      H      SO.sub.2 CH.sub.3                                                                              OCF.sub.2 H                                                                           CH.sub.3                                      H      SO.sub.2 C.sub.6 H.sub.5                                                                       CH.sub.3                                                                              H                                             H      SO.sub. 2                                                                              C.sub.6 H.sub.5                                                                       OCH.sub.3                                                                             H                                             H      SO.sub.2 C.sub.6 H.sub.5                                                                       OC.sub.2 H.sub.5                                                                      H                                             H      SO.sub.2 C.sub.6 H.sub.5                                                                       OCF.sub.2 H                                                                           H                                             ______________________________________                                    

                  TABLE Ie                                                        ______________________________________                                        General Formula Ie                                                            R.sub.1                                                                              J        R.sub.6 X.sub.2                                                                              Y.sub.3 m.p.(°C.)                       ______________________________________                                        H      C═O  C.sub.6 H.sub.5                                                                       CH.sub.3                                                                             CH.sub.3                                       H      C═O  C.sub.6 H.sub.5                                                                       OCH.sub.3                                                                            CH.sub.3                                       H      C═O  C.sub.6 H.sub.5                                                                       SCH.sub.3                                                                            CH.sub.3                                       H      C═O  H       CH.sub.3                                                                             C.sub.2 H.sub.5                                H      C═O  H       OCH.sub.3                                                                            C.sub.2 H.sub.5                                H      C═O  H       SCH.sub.3                                                                            C.sub.2 H.sub.5                                H      C═O  CH.sub.3                                                                              CH.sub.3                                                                             CH.sub.2 CF.sub.3                              H      C═O  CH.sub.3                                                                              OCH.sub.3                                                                            CH.sub.2 CF.sub.3                              H      C═O  CH.sub.3                                                                              SCH.sub.3                                                                            CH.sub.2 CF.sub.3                              H      C═O  H       CH.sub.3                                                                             CH.sub.3                                       H      C═O  H       OCH.sub.3                                                                            CH.sub.3                                       H      C═O  H       SCH.sub.3                                                                            CH.sub.3                                       H      C═O  CH.sub.3                                                                              CH.sub.3                                                                             C.sub.2 H.sub.5                                H      C═O  CH.sub.3                                                                              OCH.sub.3                                                                            C.sub.2 H.sub.5                                H      C═O  CH.sub.3                                                                              SCH.sub.3                                                                            C.sub.2 H.sub.5                                H      C═O  C.sub.6 H.sub.5                                                                       CH.sub.3                                                                             CH.sub.2 CF.sub.3                              H      C═O  C.sub.6 H.sub.5                                                                       OCH.sub.3                                                                            CH.sub.2 CF.sub.3                              H      C═O  C.sub.6 H.sub.5                                                                       SCH.sub.3                                                                            CH.sub.2 CF.sub.3                              H      C═O  CH.sub.3                                                                              CH.sub.3                                                                             CH.sub.3                                       H      C═O  CH.sub.3                                                                              OCH.sub.3                                                                            CH.sub.3                                       H      C═O  CH.sub.3                                                                              SCH.sub.3                                                                            CH.sub.3                                       H      C═O  C.sub.6 H.sub.5                                                                       CH.sub.3                                                                             C.sub.2 H.sub.5                                H      C═O  C.sub.6 H.sub.5                                                                       OCH.sub.3                                                                            C.sub.2 H.sub.5                                H      C═O  C.sub.6 H.sub.5                                                                       SCH.sub.3                                                                            C.sub.2 H.sub.5                                H      C═O  H       CH.sub.3                                                                             CH.sub.2 CF.sub.3                              H      C═O  H       OCH.sub.3                                                                            CH.sub.2 CF.sub.3                              H      C═O  H       SCH.sub.3                                                                            CH.sub.2 CF.sub.3                              H      SO.sub.2 C.sub.6 H.sub.5                                                                       CH.sub.3                                                                             CH.sub.3                                       H      SO.sub.2 C.sub.6 H.sub.5                                                                       OCH.sub.3                                                                            CH.sub.3                                       H      SO.sub.2 C.sub.6 H.sub.5                                                                       SCH.sub.3                                                                            CH.sub.3                                       H      SO.sub.2 H       CH.sub.3                                                                             C.sub.2 H.sub.5                                H      SO.sub.2 H       OCH.sub.3                                                                            C.sub.2 H.sub.5                                H      SO.sub.2 H       SCH.sub.3                                                                            C.sub.2 H.sub.5                                H      SO.sub.2 CH.sub.3                                                                              CH.sub.3                                                                             CH.sub.2 CF.sub.3                              H      SO.sub.2 CH.sub.3                                                                              OCH.sub.3                                                                            CH.sub.2 CF.sub.3                              H      SO.sub.2 CH.sub.3                                                                              SCH.sub.3                                                                            CH.sub.2 CF.sub.3                              H      SO.sub.2 H       CH.sub.3                                                                             CH.sub.3                                       H      SO.sub.2 H       OCH.sub.3                                                                            CH.sub.3                                       H      SO.sub.2 H       SCH.sub.3                                                                            CH.sub.3                                       H      SO.sub.2 CH.sub.3                                                                              CH.sub.3                                                                             C.sub.2 H.sub.5                                H      SO.sub.2 CH.sub.3                                                                              OCH.sub.3                                                                            C.sub.2 H.sub.5                                H      SO.sub.2 CH.sub.3                                                                              SCH.sub.3                                                                            C.sub.2 H.sub.5                                H      SO.sub.2 C.sub.6 H.sub.5                                                                       CH.sub.3                                                                             CH.sub.2 CF.sub.3                              H      SO.sub.2 C.sub.6 H.sub.5                                                                       OCH.sub.3                                                                            OH.sub.2 CF.sub.3                              H      SO.sub.2 C.sub.6 H.sub.5                                                                       SCH.sub.3                                                                            CH.sub.2 CF.sub.3                              H      SO.sub.2 CH.sub.3                                                                              CH.sub.3                                                                             CH.sub.3                                       H      SO.sub.2 CH.sub.3                                                                              OCH.sub.3                                                                            CH.sub.3                                       H      SO.sub.2 CH.sub.3                                                                              SCH.sub.3                                                                            CH.sub.3                                       H      SO.sub.2 C.sub.6 H.sub.5                                                                       CH.sub.3                                                                             C.sub.2 H.sub.5                                H      SO.sub.2 C.sub.6 H.sub.5                                                                       OCH.sub.3                                                                            C.sub.2 H.sub.5                                H      SO.sub.2 C.sub.6 H.sub.5                                                                       SCH.sub.3                                                                            C.sub.2 H.sub.5                                ______________________________________                                    

                  TABLE If                                                        ______________________________________                                        General Structure If                                                          R.sub.1 J         R.sub.6  X.sub.3                                                                             m.p.(°C.)                             ______________________________________                                        H       C═O   H        CH.sub.3                                           H       C═O   H        OCH.sub.3                                          H       C═O   CH.sub.3 CH.sub.3                                           H       C═O   CH.sub.3 OCH.sub.3                                          H       C═O   C.sub.6 H.sub.5                                                                        CH.sub.3                                           H       C═O   C.sub.6 H.sub.5                                                                        OCH.sub.3                                          H       SO.sub.2  H        CH.sub.3                                           H       SO.sub.2  H        OCH.sub.3                                          H       SO.sub.2  CH.sub.3 CH.sub.3                                           H       SO.sub.2  CH.sub.3 OCH.sub.3                                          H       SO.sub.2  C.sub.6 H.sub.5                                                                        CH.sub.3                                           H       SO.sub.2  C.sub.6 H.sub.5                                                                        OCH.sub.3                                          ______________________________________                                    

                  TABLE Ig                                                        ______________________________________                                        General Structure Ig                                                          R.sub.1                                                                             G      J       R.sub.6                                                                            X     Y     Z    m.p.(°C.)                   ______________________________________                                        H     CH.sub.2                                                                             C═O H    CH.sub.3                                                                            CH.sub.3                                                                            CH                                      H     CH.sub.2                                                                             C═O H    CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H     CH.sub.2                                                                             C═O H    OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      H     CH.sub.2                                                                             C═O H    Cl    OCH.sub.3                                                                           CH                                      H     CH.sub.2                                                                             C═O H    CH.sub.3                                                                            OCH.sub.3                                                                           N                                       H     CH.sub.2                                                                             C═O H    OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       H     CH.sub.2                                                                             C═O H    CH.sub.3                                                                            CH.sub.3                                                                            N                                       H     CH.sub.2                                                                             C═O H    CH.sub.3                                                                            CH.sub.3                                                                            CH                                      H     CH.sub.2                                                                             C═O H    CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H     CH.sub.2                                                                             C═O H    OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      H     CH.sub.2                                                                             C═O H    Cl    OCH.sub.3                                                                           CH                                      H     CH.sub.2                                                                             C═O H    CH.sub.3                                                                            OCH.sub.3                                                                           N                                       H     CH.sub.2                                                                             C═O H    OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       H     CH.sub.2                                                                             C═O H    CH.sub.3                                                                            CH.sub.3                                                                            N                                       H     CH.sub.2                                                                             C═O H    CH    CH.sub.3                                                                            CH                                      H     CH.sub.2                                                                             C═O H    CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H     CH.sub.2                                                                             C═O H    OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      H     CH.sub.2                                                                             C═O H    Cl    OCH.sub.3                                                                           CH                                      H     CH.sub.2                                                                             C═O CH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           N                                       H     CH.sub.2                                                                             C═O CH.sub.3                                                                           CH.sub.3                                                                            CH.sub.3                                                                            N                                       H     CH.sub.2                                                                             C═O CH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       ______________________________________                                    

                  TABLE Ih                                                        ______________________________________                                        General Structure Ih                                                          R.sub.1                                                                            G        R.sub.6                                                                              R.sub.7                                                                            X     Y     Z    m.p. (°C.)                  ______________________________________                                        H    CH.sub.2 H      CH.sub.3                                                                           CH.sub.3                                                                            CH.sub.3                                                                            CH                                      H    CH.sub.2 H      CH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H    CH.sub.2 H      CH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      H    CH.sub.2 H      CH.sub.3                                                                           Cl    OCH.sub.3                                                                           CH                                      H    CH.sub.2 H      CH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           N                                       H    CH.sub.2 H      CH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       H    CH.sub.2 H      CH.sub.3                                                                           CH.sub.3                                                                            CH.sub.3                                                                            N                                       H    CH.sub.2 CH.sub.3                                                                             CH.sub.3                                                                           CH.sub.3                                                                            CH.sub.3                                                                            CH                                      H    CH.sub.2 CH.sub.3                                                                             CH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H    CH.sub.2 CH.sub.3                                                                             CH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      H    CH.sub.2 CH.sub.3                                                                             CH.sub.3                                                                           Cl    OCH.sub.3                                                                           CH                                      H    CH.sub.2 CH.sub.3                                                                             CH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           N                                       H    CH.sub.2 CH.sub.3                                                                             CH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       H    CH.sub.2 CH.sub.3                                                                             CH.sub.3                                                                           CH.sub.3                                                                            CH.sub.3                                                                            N                                       H    CH.sub.2 C.sub.6 H.sub.5                                                                      CH.sub.3                                                                           CH.sub.3                                                                            CH.sub.3                                                                            CH                                      H    CH.sub.2 C.sub.6 H.sub.5                                                                      CH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H    CH.sub.2 C.sub.6 H.sub.5                                                                      CH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      H    CH.sub.2 C.sub.6 H.sub.5                                                                      CH.sub.3                                                                           Cl    OCH.sub.3                                                                           CH                                      H    CH.sub.2 C.sub.6 H.sub.5                                                                      CH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           N                                       H    CH.sub.2 C.sub.6 H.sub.5                                                                      CH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       H    CH.sub.2 C.sub.6 H.sub.5                                                                      CH.sub.3                                                                           CH.sub.3                                                                            CH.sub.3                                                                            N                                       H    CH.sub.2 H      H    CH.sub.3                                                                            CH.sub.3                                                                            CH                                      H    CH.sub.2 H      H    CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H    CH.sub.2 H      H    OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      H    CH.sub.2 H      H    Cl    OCH.sub.3                                                                           CH                                      H    CH.sub.2 H      H    CH.sub.3                                                                            OCH.sub.3                                                                           N                                       H    CH.sub.2 H      H    OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       H    CH.sub.2 H      H    CH.sub.3                                                                            CH.sub.3                                                                            N                                       H    CH.sub.2 C.sub.6 H.sub.5                                                                      H    CH.sub.3                                                                            CH.sub.3                                                                            CH                                      H    CH.sub.2 C.sub.6 H.sub.5                                                                      H    CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H    CH.sub.2 C.sub.6 H.sub.5                                                                      H    OCH.sub.3                                                                           OCH.sub. 3                                                                          CH                                      H    CH.sub.2 C.sub.6 H.sub.5                                                                      H    Cl    OCH.sub.3                                                                           CH                                      H    CH.sub.2 C.sub.6 H.sub.5                                                                      H    CH.sub.3                                                                            OCH.sub.3                                                                           N                                       H    CH.sub.2 C.sub.6 H.sub.5                                                                      H    OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       H    CH.sub.2 C.sub.6 H.sub.5                                                                      H    CH.sub.3                                                                            CH.sub.3                                                                            N                                       6-Cl CH.sub.2 CH.sub.3                                                                             H    CH.sub.3                                                                            CH.sub.3                                                                            CH                                      6-Cl CH.sub.2 CH.sub.3                                                                             H    CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-Cl CH.sub.2 CH.sub.3                                                                             H    OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      6-Cl CH.sub.2 CH.sub.3                                                                             H    Cl    OCH.sub.3                                                                           CH                                      6-Cl CH.sub.2 CH.sub.3                                                                             H    CH.sub.3                                                                            OCH.sub.3                                                                           N                                       6-Cl CH.sub.2 CH.sub.3                                                                             H    OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       6-Cl CH.sub.2 C.sub.6 H.sub.5                                                                      H    CH.sub.3                                                                            CH.sub.3                                                                            CH                                      6-Cl CH.sub.2 C.sub.6 H.sub.5                                                                      H    CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-Cl CH.sub.2 C.sub.6 H.sub.5                                                                      H    OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      6-Cl CH.sub.2 C.sub.6 H.sub.5                                                                      H    Cl    OCH.sub.3                                                                           CH                                      6-Cl CH.sub.2 C.sub.6 H.sub.5                                                                      H    CH.sub.3                                                                            OCH.sub.3                                                                           N                                       6-Cl CH.sub.2 C.sub.6 H.sub.5                                                                      H    OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       H    CH.sub.2 CH.sub.2                                                                      H      CH.sub.3                                                                           CH.sub.3                                                                            CH.sub.3                                                                            CH                                      H    CH.sub.2 CH.sub.2                                                                      H      CH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H    CH.sub.2 CH.sub.2                                                                      H      CH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      H    CH.sub.2 CH.sub.2                                                                      H      CH.sub.3                                                                           Cl    OCH.sub.3                                                                           CH                                      H    CH.sub.2 CH.sub.2                                                                      H      CH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           N                                       H    CH.sub.2 CH.sub.2                                                                      H      CH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       H    CH.sub.2 CH.sub.2                                                                      H      CH.sub.3                                                                           CH.sub.3                                                                            CH.sub.3                                                                            N                                       H    CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             CH.sub.3                                                                           CH.sub.3                                                                            CH.sub.3                                                                            CH                                      H    CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             CH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H    CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             CH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      H    CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             CH.sub.3                                                                           Cl    OCH.sub.3                                                                           CH                                      H    CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             CH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           N                                       H    CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             CH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       H    CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             CH.sub.3                                                                           CH.sub.3                                                                            CH.sub.3                                                                            N                                       H    CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      CH.sub.3                                                                           CH.sub.3                                                                            CH.sub.3                                                                            CH                                      H    CH.sub. 2 CH.sub.2                                                                     C.sub.6 H.sub.5                                                                      CH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H    CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      CH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      H    CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      CH.sub.3                                                                           Cl    OCH.sub.3                                                                           CH                                      H    CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      CH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           N                                       H    CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      CH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       H    CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      CH.sub.3                                                                           CH.sub.3                                                                            CH.sub.3                                                                            N                                       H    CH.sub.2 CH.sub.2                                                                      H      H    CH.sub.3                                                                            CH.sub.3                                                                            CH                                      H    CH.sub.2 CH.sub.2                                                                      H      H    CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H    CH.sub.2 CH.sub.2                                                                      H      H    OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      H    CH.sub.2 CH.sub.2                                                                      H      H    Cl    OCH.sub.3                                                                           CH                                      H    CH.sub.2 CH.sub.2                                                                      H      H    CH.sub.3                                                                            OCH.sub.3                                                                           N                                       H    CH.sub.2 CH.sub.2                                                                      H      H    OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       H    CH.sub.2 CH.sub.2                                                                      H      H    CH.sub.3                                                                            CH.sub.3                                                                            N                                       H    CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      H    CH.sub.3                                                                            CH.sub.3                                                                            CH                                      H    CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      H    CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H    CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      H    OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      H    CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      H    Cl    OCH.sub.3                                                                           CH                                      H    CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      H    CH.sub.3                                                                            OCH.sub.3                                                                           N                                       H    CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      H    OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       H    CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      H    CH.sub.3                                                                            CH.sub.3                                                                            N                                       6-Cl CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             H    CH.sub.3                                                                            CH.sub.3                                                                            CH                                      6-Cl CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             H    CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-Cl CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             H    OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      6-Cl CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             H    Cl    OCH.sub.3                                                                           CH                                      6-Cl CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             H    CH.sub.3                                                                            OCH.sub.3                                                                           N                                       6-Cl CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             H    OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       6-Cl CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      H    CH.sub.3                                                                            CH.sub.3                                                                            CH                                      6-Cl CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      H    CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-Cl CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      H    OCH.sub.3                                                                           OCH.sub. 3                                                                          CH                                      6-Cl CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      H    Cl    OCH.sub.3                                                                           CH                                      6-Cl CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      H    CH.sub.3                                                                            OCH.sub.3                                                                           N                                       6-Cl CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      H    OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       H    CH═CH                                                                              H      CH.sub.3                                                                           CH.sub.3                                                                            CH.sub.3                                                                            CH                                      H    CH═CH                                                                              H      CH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H    CH═CH                                                                              H      CH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      H    CH═CH                                                                              H      CH.sub.3                                                                           Cl    OCH.sub.3                                                                           CH                                      H    CH═CH                                                                              H      CH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           N                                       H    CH═CH                                                                              H      CH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       H    CH═CH                                                                              H      CH.sub.3                                                                           CH.sub.3                                                                            CH.sub.3                                                                            N                                       H    CH═CH                                                                              CH.sub.3                                                                             CH.sub.3                                                                           CH.sub.3                                                                            CH.sub.3                                                                            CH                                      H    CH═CH                                                                              CH.sub.3                                                                             CH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H    CH═CH                                                                              CH.sub.3                                                                             CH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      H    CH═CH                                                                              CH.sub.3                                                                             CH.sub.3                                                                           Cl    OCH.sub.3                                                                           CH                                      H    CH═CH                                                                              CH.sub.3                                                                             CH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           N                                       H    CH═CH                                                                              CH.sub.3                                                                             CH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       H    CH═CH                                                                              CH.sub.3                                                                             CH.sub.3                                                                           CH.sub.3                                                                            CH.sub.3                                                                            N                                       H    CH═CH                                                                              C.sub.6 H.sub.5                                                                      CH.sub.3                                                                           CH.sub.3                                                                            CH.sub.3                                                                            CH                                      H    CH═CH                                                                              C.sub.6 H.sub.5                                                                      CH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H    CH═CH                                                                              C.sub.6 H.sub.5                                                                      CH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      H    CH═CH                                                                              C.sub.6 H.sub.5                                                                      CH.sub.3                                                                           Cl    OCH.sub.3                                                                           CH                                      H    CH═CH                                                                              C.sub.6 H.sub.5                                                                      CH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           N                                       H    CH═CH                                                                              C.sub.6 H.sub.5                                                                      CH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       H    CH═CH                                                                              C.sub.6 H.sub.5                                                                      CH.sub.3                                                                           CH.sub.3                                                                            CH.sub.3                                                                            N                                       H    CH═CH                                                                              H      H    CH.sub.3                                                                            CH.sub.3                                                                            CH                                      H    CH═CH                                                                              H      H    CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H    CH═CH                                                                              H      H    OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      H    CH═CH                                                                              H      H    Cl    OCH.sub.3                                                                           CH                                      H    CH═CH                                                                              H      H    CH.sub.3                                                                            OCH.sub.3                                                                           N                                       H    CH═CH                                                                              H      H    OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       H    CH═CH                                                                              H      H    CH.sub.3                                                                            CH.sub.3                                                                            N                                       H    CH═CH                                                                              C.sub.6 H.sub.5                                                                      H    CH.sub.3                                                                            CH.sub.3                                                                            CH                                      H    CH═CH                                                                              C.sub.6 H.sub.5                                                                      H    CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H    CH═CH                                                                              C.sub.6 H.sub.5                                                                      H    OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      H    CH═CH                                                                              C.sub.6 H.sub.5                                                                      H    Cl    OCH.sub.3                                                                           CH                                      H    CH═CH                                                                              C.sub.6 H.sub.5                                                                      H    CH.sub.3                                                                            OCH.sub.3                                                                           N                                       H    CH═CH                                                                              C.sub.6 H.sub.5                                                                      H    OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       H    CH═CH                                                                              C.sub.6 H.sub.5                                                                      H    CH.sub.3                                                                            CH.sub.3                                                                            N                                       6-Cl CH═CH                                                                              CH.sub.3                                                                             H    CH.sub.3                                                                            CH.sub.3                                                                            CH                                      6-Cl CH═CH                                                                              CH.sub.3                                                                             H    CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-Cl CH═CH                                                                              CH.sub.3                                                                             H    OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      6-Cl CH═CH                                                                              CH.sub.3                                                                             H    Cl    OCH.sub.3                                                                           CH                                      6-Cl CH═CH                                                                              CH.sub.3                                                                             H    CH.sub.3                                                                            OCH.sub.3                                                                           N                                       6-Cl CH═CH                                                                              CH.sub.3                                                                             H    OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       6-Cl CH═CH                                                                              C.sub.6 H.sub.5                                                                      H    CH.sub.3                                                                            CH.sub.3                                                                            CH                                      6-Cl CH═CH                                                                              C.sub.6 H.sub.5                                                                      H    CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-Cl CH═CH                                                                              C.sub.6 H.sub.5                                                                      H    OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      6-Cl CH═CH                                                                              C.sub.6 H.sub.5                                                                      H    Cl    OCH.sub.3                                                                           CH                                      6-Cl CH═CH                                                                              C.sub.6 H.sub.5                                                                      H    CH.sub.3                                                                            OCH.sub.3                                                                           N                                       6-Cl CH═CH                                                                              C.sub.6 H.sub.5                                                                      H    OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       H    CH.sub.2 CH.sub.3                                                                             H    OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      H    CH.sub.2 CH.sub.3                                                                             H    OCH.sub.3                                                                           CH.sub.3                                                                            CH                                      H    CH.sub.2 CH.sub.3                                                                             H    CH.sub.3                                                                            CH.sub.3                                                                            CH                                      H    CH.sub.2 CH.sub.3                                                                             H    OCH.sub.3                                                                           Cl.sub.3                                                                            CH                                      H    CH.sub.2 CH.sub.3                                                                             H    OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       H    CH.sub.2 CH.sub.3                                                                             H    OCH.sub.3                                                                           CH.sub.3                                                                            N                                       H    CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             H    OCH.sub.3                                                                           OCH.sub.3                                                                           CH   221-223(d)                         H    CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             H    OCH.sub.3                                                                           CH.sub.3                                                                            CH                                      H    CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             H    CH.sub.3                                                                            CH.sub.3                                                                            CH                                      H    CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             H    OCH.sub.3                                                                           Cl.sub.3                                                                            CH                                      H    CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             H    OCH.sub.3                                                                           CH.sub.3                                                                            N                                       H    CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             H    OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       H    CH═CH                                                                              CH.sub.3                                                                             H    OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      H    CH═CH                                                                              CH.sub.3                                                                             H    OCH.sub.3                                                                           CH.sub.3                                                                            CH                                      H    CH═CH                                                                              CH.sub. 3                                                                            H    CH.sub.3                                                                            CH.sub.3                                                                            CH                                      H    CH═CH                                                                              CH.sub.3                                                                             H    OCH.sub.3                                                                           Cl.sub.3                                                                            CH                                      H    CH═CH                                                                              CH.sub.3                                                                             H    OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       H    CH═CH                                                                              CH.sub.3                                                                             H    OCH.sub.3                                                                           CH.sub.3                                                                            N                                       ______________________________________                                    

                  TABLE 2a                                                        ______________________________________                                        General Formula 2a                                                            R.sub.1                                                                              J       W'    R.sub.9                                                                            X     Y     Z    m.p.(°C.)                   ______________________________________                                        H      C═O O     H    CH.sub.3                                                                            CH.sub.3                                                                            CH                                      H      C═O O     H    CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H      C═O O     H    OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      H      C═O O     H    Cl    OCH.sub.3                                                                           CH                                      H      C═O O     H    CH.sub.3                                                                            OCH.sub.3                                                                           N                                       H      C═O O     H    OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       H      C═O O     H    CH.sub.3                                                                            CH.sub.3                                                                            N                                       H      C═O O     CH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H      C═O O     CH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      H      C═O O     CH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H      C═O O     CH.sub.3                                                                           Cl    OCH.sub.3                                                                           CH                                      H      C═O O     CH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           N                                       H      C═O O     CH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       H      C═O O     CH.sub.3                                                                           CH.sub.3                                                                            CH.sub.3                                                                            N                                       H      C═O O     C.sub.6 H.sub.5                                                                    CH.sub.3                                                                            CH.sub.3                                                                            CH                                      H      C═O O     C.sub.6 H.sub.5                                                                    CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H      C═O O     C.sub.6 H.sub.5                                                                    OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      H      C═O O     C.sub.6 H.sub.5                                                                    Cl    OCH.sub.3                                                                           CH                                      H      C═O O     C.sub.6 H.sub.5                                                                    CH.sub.3                                                                            OCH.sub.3                                                                           N                                       H      C═O O     C.sub.6 H.sub.5                                                                    OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       H      C═O O     C.sub.6 H.sub.5                                                                    CH.sub.3                                                                            CH.sub.3                                                                            N                                       H      C═O S     H    CH.sub.3                                                                            CH.sub.3                                                                            CH                                      H      C═O S     H    CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H      C═O S     H    OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      H      C═O S     H    Cl    OCH.sub.3                                                                           CH                                      H      C═O S     H    CH.sub.3                                                                            OCH.sub.3                                                                           N                                       H      C═O S     H    OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       H      C═O S     H    CH.sub.3                                                                            CH.sub.3                                                                            N                                       H      C═O S     CH.sub.3                                                                           CH.sub.3                                                                            CH.sub.3                                                                            CH                                      H      C═O S     CH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H      C═O S     CH.sub.3                                                                           OCH   OCH.sub.3                                                                           CH                                      H      C═O S     CH.sub.3                                                                           Cl    OCH.sub.3                                                                           CH                                      H      C═O S     CH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           N                                       H      C═O S     CH.sub.3                                                                           OCH.sub. 3                                                                          OCH.sub.3                                                                           N                                       H      C═O S     CH.sub.3                                                                           CH.sub.3                                                                            CH.sub.3                                                                            N                                       H      C═O S     C.sub.6 H.sub.5                                                                    CH.sub.3                                                                            CH.sub.3                                                                            CH                                      H      C═O S     C.sub.6 H.sub.5                                                                    CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H      C═O S     C.sub.6 H.sub.5                                                                    OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      H      C═O S     C.sub.6 H.sub.5                                                                    Cl    OCH.sub.3                                                                           CH                                      H      C═O S     C.sub.6 H.sub.5                                                                    CH.sub.3                                                                            OCH.sub.3                                                                           N                                       H      C═O S     C.sub.6 H.sub.5                                                                    OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       H      C═O S     C.sub.6 H.sub.5                                                                    CH.sub.3                                                                            CH.sub.3                                                                            N                                       H      CH.sub.2                                                                              O     CH.sub.3                                                                           CH.sub.3                                                                            CH.sub.3                                                                            CH                                      H      CH.sub.2                                                                              O     CH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H      CH.sub.2                                                                              O     CH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      H      CH.sub.2                                                                              O     CH.sub.3                                                                           Cl    OCH.sub.3                                                                           CH                                      H      CH.sub.2                                                                              O     CH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           N                                       H      CH.sub.2                                                                              O     CH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       H      CH.sub.2                                                                              O     CH.sub.3                                                                           CH.sub.3                                                                            CH.sub.3                                                                            N                                       H      CH.sub.2                                                                              S     CH.sub.3                                                                           CH.sub.3                                                                            CH.sub.3                                                                            CH                                      H      CH.sub.2                                                                              S     CH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H      CH.sub.2                                                                              S     CH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      H      CH.sub.2                                                                              S     CH.sub.3                                                                           Cl    OCH.sub.3                                                                           CH                                      H      CH.sub.2                                                                              S     CH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           N                                       H      CH.sub.2                                                                              S     CH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       H      CH.sub.2                                                                              S     CH.sub.3                                                                           CH.sub.3                                                                            CH.sub.3                                                                            N                                       H      CH.sub.2                                                                              S     C.sub.6 H.sub.5                                                                    CH.sub.3                                                                            CH.sub.3                                                                            CH                                      H      CH.sub.2                                                                              S     C.sub.6 H.sub.5                                                                    CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H      CH.sub.2                                                                              S     C.sub.6 H.sub.5                                                                    OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      H      CH.sub.2                                                                              S     C.sub.6 H.sub.5                                                                    Cl    OCH.sub.3                                                                           CH                                      H      CH.sub.2                                                                              S     C.sub.6 H.sub.5                                                                    CH.sub.3                                                                            OCH.sub.3                                                                           N                                       H      CH.sub.2                                                                              S     C.sub.6 H.sub.5                                                                    OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       H      CH.sub.2                                                                              S     C.sub.6 H.sub.5                                                                    CH.sub.3                                                                            CH.sub.3                                                                            N                                       H      SO.sub.2                                                                              O     H    CH.sub.3                                                                            CH.sub.3                                                                            CH                                      H      SO.sub.2                                                                              O     H    CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H      SO.sub.2                                                                              O     H    OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      H      SO.sub.2                                                                              O     H    Cl    OCH.sub.3                                                                           CH                                      H      SO.sub.2                                                                              O     H    CH.sub.3                                                                            OCH.sub.3                                                                           N                                       H      SO.sub.2                                                                              O     H    OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       H      SO.sub.2                                                                              O     H    CH.sub.3                                                                            CH.sub.3                                                                            N                                       H      SO.sub.2                                                                              S     H    CH.sub.3                                                                            CH.sub.3                                                                            CH                                      H      SO.sub.2                                                                              S     H    CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H      SO.sub.2                                                                              S     H    OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      H      SO.sub.2                                                                              S     H    Cl    OCH.sub.3                                                                           CH                                      H      SO.sub.2                                                                              S     H    CH.sub.3                                                                            OCH.sub.3                                                                           N                                       H      SO.sub.2                                                                              S     H    OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       H      SO.sub.2                                                                              S     H    CH.sub.3                                                                            CH.sub.3                                                                            N                                       H      SO.sub.2                                                                              S     CH.sub.3                                                                           CH.sub.3                                                                            CH.sub.3                                                                            CH                                      H      SO.sub.2                                                                              S     CH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H      SO.sub.2                                                                              S     CH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      H      SO.sub.2                                                                              S     CH.sub.3                                                                           Cl    OCH.sub.3                                                                           CH                                      H      SO.sub.2                                                                              S     CH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           N                                       H      SO.sub.2                                                                              S     CH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       H      SO.sub.2                                                                              S     CH.sub.3                                                                           CH.sub.3                                                                            CH.sub.3                                                                            N                                       H      O       O     CH.sub.3                                                                           CH.sub.3                                                                            CH.sub.3                                                                            CH                                      H      O       O     CH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H      O       O     CH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      H      O       O     CH.sub.3                                                                           Cl    OCH.sub.3                                                                           CH                                      H      O       O     CH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           N                                       H      O       O     CH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       H      O       O     CH.sub.3                                                                           CH.sub.3                                                                            CH.sub.3                                                                            N                                       H      O       S     CH.sub.3                                                                           CH.sub.3                                                                            CH.sub.3                                                                            CH                                      H      O       S     CH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H      O       S     CH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      H      O       S     CH.sub.3                                                                           Cl    OCH.sub.3                                                                           CH                                      H      O       S     CH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           N                                       H      O       S     CH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       H      O       S     CH.sub.3                                                                           CH.sub.3                                                                            CH.sub.3                                                                            N                                       H      O       S     C.sub.6 H.sub.5                                                                    CH    CH.sub.3                                                                            CH                                      H      O       S     C.sub.6 H.sub.5                                                                    CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H      O       S     C.sub.6 H.sub.5                                                                    OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      H      O       S     C.sub.6 H.sub.5                                                                    Cl    OCH.sub.3                                                                           CH                                      H      O       S     C.sub.6 H.sub.5                                                                    CH.sub.3                                                                            OCH.sub.3                                                                           N                                       H      O       S     C.sub.6 H.sub.5                                                                    OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       H      O       S     C.sub.6 H.sub.5                                                                    CH.sub.3                                                                            CH.sub.3                                                                            N                                       6-Cl   C═O O     H    CH.sub.3                                                                            CH.sub.3                                                                            CH                                      6-Cl   C═O O     H    CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-Cl   C═O O     H    OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      6-Cl   C═O O     H    Cl    OCH.sub.3                                                                           CH                                      6-Cl   C═O O     H    CH.sub.3                                                                            OCH.sub.3                                                                           N                                       6-Cl   C═O O     H    OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       6-Cl   C═O O     H    CH.sub.3                                                                            CH.sub.3                                                                            N                                       6-CH.sub.3                                                                           C═O O     CH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-CH.sub.3                                                                           C═O O     CH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      6-CH.sub.3                                                                           C═O O     CH.sub.3                                                                           Cl    OCH.sub.3                                                                           CH                                      6-CH.sub.3                                                                           C═O O     CH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           N                                       6-CH.sub.3                                                                           C═O O     CH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       6-CH.sub.3                                                                           C═O O     CH.sub.3                                                                           CH.sub.3                                                                            CH.sub.3                                                                            N                                       6-CH.sub.3                                                                           C═O O     C.sub.6 H.sub.5                                                                    CH.sub.3                                                                            CH.sub.3                                                                            CH                                      6-CH.sub.3                                                                           C═O O     C.sub.6 H.sub.5                                                                    CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-CH.sub.3                                                                           C═O O     C.sub.6 H.sub.5                                                                    OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      6-CH.sub.3                                                                           C═O O     C.sub.6 H.sub.5                                                                    Cl    OCH.sub.3                                                                           CH                                      6-CH.sub.3                                                                           C═O O     C.sub.6 H.sub.5                                                                    CH.sub.3                                                                            OCH.sub.3                                                                           N                                       6-CH.sub.3                                                                           C═O O     C.sub.6 H.sub.5                                                                    OCH.sub. 3                                                                          OCH.sub.3                                                                           N                                       6-CH.sub.3                                                                           C═O O     6.sub.6 H.sub.5                                                                    CH.sub.3                                                                            CH.sub.3                                                                            N                                       5-NO.sub.2                                                                           C═O S     H    CH.sub.3                                                                            CH.sub.3                                                                            CH                                      5-NO.sub.2                                                                           C═O S     H    CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      5-NO.sub.2                                                                           C═O S     H    OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      5-NO.sub.2                                                                           C═O S     H    Cl    OCH.sub.3                                                                           CH                                      5-NO.sub.2                                                                           C═O S     H    CH.sub.3                                                                            OCH.sub.3                                                                           N                                       5-NO.sub.2                                                                           C═O S     H    OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       5-NO.sub.2                                                                           C═O S     H    CH.sub.3                                                                            CH.sub.3                                                                            N                                       5-SCH.sub.3                                                                          C═O S     CH.sub.3                                                                           CH.sub.3                                                                            CH.sub.3                                                                            CH                                      5-SCH.sub.3                                                                          C═O S     CH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      5-SCH.sub.3                                                                          C═O S     CH.sub.3                                                                           OCH   OCH.sub.3                                                                           CH                                      5-SCH.sub.3                                                                          C═O S     CH.sub.3                                                                           Cl    OCH.sub.3                                                                           CH                                      5-SCH.sub.3                                                                          C═O S     CH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           N                                       5-SCH.sub.3                                                                          C═O S     CH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       5-SCH.sub.3                                                                          C═O S     CH.sub.3                                                                           CH.sub.3                                                                            CH.sub.3                                                                            N                                       5-NO.sub.2                                                                           C═O S     C.sub.6 H.sub.5                                                                    CH.sub.3                                                                            CH.sub.3                                                                            CH                                      5-NO.sub.2                                                                           C═O S     C.sub.6 H.sub.5                                                                    CH.sub. 3                                                                           OCH.sub.3                                                                           CH                                      5-NO.sub.2                                                                           C═O S     C.sub.6 H.sub.5                                                                    OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      5-NO.sub.2                                                                           C═O S     C.sub.6 H.sub.5                                                                    Cl    OCH.sub.3                                                                           CH                                      5-NO.sub.2                                                                           C═O S     C.sub.6 H.sub.5                                                                    CH.sub.3                                                                            OCH.sub.3                                                                           N                                       5-NO.sub.2                                                                           C═O S     C.sub.6 H.sub.5                                                                    OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       5-NO.sub.2                                                                           C═O S     C.sub.6 H.sub.5                                                                    CH.sub.3                                                                            CH.sub.3                                                                            N                                       6-Cl   CH.sub.2                                                                              O     CH.sub.3                                                                           CH.sub.3                                                                            CH.sub.3                                                                            CH                                      6-Cl   CH.sub.2                                                                              O     CH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-Cl   CH.sub.2                                                                              O     CH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      6-Cl   CH.sub.2                                                                              O     CH.sub.3                                                                           Cl    OCH.sub.3                                                                           CH                                      6-Cl   CH.sub.2                                                                              O     CH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           N                                       6-Cl   CH.sub.2                                                                              O     CH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       6-Cl   CH.sub.2                                                                              O     CH.sub.3                                                                           CH.sub.3                                                                            CH.sub.3                                                                            N                                       6-Cl   CH.sub.2                                                                              S     CH.sub.3                                                                           CH.sub.3                                                                            CH.sub.3                                                                            CH                                      6-Cl   CH.sub.2                                                                              S     CH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-Cl   CH.sub.2                                                                              S     CH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      6-Cl   CH.sub.2                                                                              S     CH.sub.3                                                                           Cl    OCH.sub.3                                                                           CH                                      6-Cl   CH.sub.2                                                                              S     CH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           N                                       6-Cl   CH.sub.2                                                                              S     CH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       6-Cl   CH.sub.2                                                                              S     CH.sub.3                                                                           CH.sub.3                                                                            CH.sub.3                                                                            N                                       6-Cl   CH.sub.2                                                                              S     C.sub.6 H.sub.5                                                                    CH    CH.sub.3                                                                            CH                                      6-Cl   CH.sub.2                                                                              S     C.sub.6 H.sub.5                                                                    CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-Cl   CH.sub.2                                                                              S     C.sub.6 H.sub.5                                                                    OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      6-Cl   CH.sub.2                                                                              S     C.sub.6 H.sub.5                                                                    Cl    OCH.sub.3                                                                           CH                                      6-Cl   CH.sub.2                                                                              S     C.sub.6 H.sub.5                                                                    CH.sub.3                                                                            OCH.sub.3                                                                           N                                       6-Cl   CH.sub.2                                                                              S     C.sub.6 H.sub.5                                                                    OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       6-Cl   CH.sub.2                                                                              S     C.sub.6 H.sub.5                                                                    CH.sub.3                                                                            CH.sub.3                                                                            N                                       6-CH.sub.3                                                                           SO.sub.2                                                                              O     H    CH.sub.3                                                                            CH.sub.3                                                                            CH                                      6-CH.sub.3                                                                           SO.sub.2                                                                              O     H    CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-CH.sub.3                                                                           SO.sub.2                                                                              O     H    OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      6-CH.sub.3                                                                           SO.sub.2                                                                              O     H    Cl    OCH.sub.3                                                                           CH                                      6-CH.sub.3                                                                           SO.sub.2                                                                              O     H    CH.sub.3                                                                            OCH.sub.3                                                                           N                                       6-CH.sub.3                                                                           SO.sub.2                                                                              O     H    OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       6-CH.sub.3                                                                           SO.sub.2                                                                              O     H    CH.sub.3                                                                            CH.sub.3                                                                            N                                       6-CH.sub.3                                                                           SO.sub.2                                                                              S     H    CH.sub.3                                                                            CH.sub.3                                                                            CH                                      6-CH.sub.3                                                                           SO.sub.2                                                                              S     H    CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-CH.sub.3                                                                           SO.sub.2                                                                              S     H    OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      6-CH.sub.3                                                                           SO.sub.2                                                                              S     H    Cl    OCH.sub.3                                                                           CH                                      6-CH.sub.3                                                                           SO.sub.2                                                                              S     H    CH.sub.3                                                                            OCH.sub.3                                                                           N                                       6-CH.sub.3                                                                           SO.sub.2                                                                              S     H    OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       6-CH.sub.3                                                                           SO.sub.2                                                                              S     H    CH.sub.3                                                                            CH.sub.3                                                                            N                                       5-NO.sub.2                                                                           SO.sub.2                                                                              S     CH.sub.3                                                                           CH.sub.3                                                                            CH.sub.3                                                                            CH                                      5-NO.sub.2                                                                           SO.sub.2                                                                              S     CH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      5-NO.sub.2                                                                           SO.sub.2                                                                              S     CH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      5-NO.sub.2                                                                           SO.sub.2                                                                              S     CH.sub.3                                                                           Cl    OCH.sub.3                                                                           CH                                      5-NO.sub.2                                                                           SO.sub.2                                                                              S     CH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           N                                       5-NO.sub.2                                                                           SO.sub.2                                                                              S     CH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       5-NO.sub.2                                                                           SO.sub.2                                                                              S     CH.sub.3                                                                           CH.sub.3                                                                            CH.sub.3                                                                            N                                       6-CH.sub.3                                                                           O       O     CH.sub.3                                                                           CH.sub.3                                                                            CH.sub.3                                                                            CH                                      6-CH.sub.3                                                                           O       O     CH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-CH.sub.3                                                                           O       O     CH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      6-CH.sub.3                                                                           O       O     CH.sub.3                                                                           Cl    OCH.sub.3                                                                           CH                                      6-CH.sub.3                                                                           O       O     CH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           N                                       6-CH.sub.3                                                                           O       O     CH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       6-CH.sub.3                                                                           O       O     CH.sub.3                                                                           CH.sub.3                                                                            CH.sub.3                                                                            N                                       6-Cl   O       S     CH.sub.3                                                                           CH.sub.3                                                                            CH.sub.3                                                                            CH                                      6-Cl   O       S     CH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-Cl   O       S     CH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      6-Cl   O       S     CH.sub.3                                                                           Cl    OCH.sub.3                                                                           CH                                      6-Cl   O       S     CH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           N                                       6-Cl   O       S     CH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       6-Cl   O       S     CH.sub.3                                                                           CH.sub.3                                                                            CH.sub.3                                                                            N                                       5-NO.sub.2                                                                           O       S     C.sub.6 H.sub.5                                                                    CH.sub.3                                                                            CH.sub.3                                                                            CH                                      5-NO.sub.2                                                                           O       S     C.sub.6 H.sub.5                                                                    CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      5-NO.sub.2                                                                           O       S     C.sub.6 H.sub.5                                                                    OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      5-NO.sub.2                                                                           O       S     C.sub.6 H.sub.5                                                                    Cl    OCH.sub.3                                                                           CH                                      5-NO.sub.2                                                                           O       S     C.sub.6 H.sub.5                                                                    CH.sub.3                                                                            OCH.sub.3                                                                           N                                       5-NO.sub.2                                                                           O       S     C.sub.6 H.sub.5                                                                    OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       5-NO.sub.2                                                                           O       S     C.sub.6 H.sub.5                                                                    CH.sub.3                                                                            CH.sub.3                                                                            N                                       ______________________________________                                    

                  TABLE 2b                                                        ______________________________________                                        General Formula 2b                                                                                                          m.p.                            R.sub.1                                                                            G         W'      R.sub.9                                                                            X      Y     Z    (°C.)                    ______________________________________                                        H    CH.sub.2  O       H    CH.sub.3                                                                             CH.sub.3                                                                            CH                                   H    CH.sub.2  O       H    CH.sub.3                                                                             OCH.sub.3                                                                           CH                                   H    CH.sub.2  O       H    OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                   H    CH.sub.2  O       H    Cl     OCH.sub.3                                                                           CH                                   H    CH.sub.2  O       H    CH.sub.3                                                                             OCH.sub.3                                                                           N                                    H    CH.sub.2  O       H    OCH.sub.3                                                                            OCH.sub.3                                                                           N                                    H    CH.sub.2  O       H    CH.sub.3                                                                             CH.sub.3                                                                            N                                    H    CH.sub.2  S       CH.sub.3                                                                           CH.sub.3                                                                             CH.sub.3                                                                            CH                                   H    CH.sub.2  S       CH.sub.3                                                                           CH.sub.3                                                                             OCH.sub.3                                                                           CH                                   H    CH.sub.2  S       CH.sub.3                                                                           OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                   H    CH.sub.2  S       CH.sub.3                                                                           Cl     OCH.sub.3                                                                           CH                                   H    CH.sub.2  S       CH.sub.3                                                                           CH.sub.3                                                                             OCH.sub.3                                                                           N                                    H    CH.sub.2  S       CH.sub.3                                                                           OCH.sub.3                                                                            OCH.sub.3                                                                           N                                    H    CH.sub.2  S       CH.sub.3                                                                           CH.sub.3                                                                             CH.sub.3                                                                            N                                    H    CH.sub.2  NH      H    CH.sub.3                                                                             CH.sub.3                                                                            CH                                   H    CH.sub.2  NH      H    CH.sub.3                                                                             OCH.sub.3                                                                           CH                                   H    CH.sub.2  NH      H    OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                   H    CH.sub.2  NH      H    Cl     OCH.sub.3                                                                           CH                                   H    CH.sub.2  NH      H    CH.sub.3                                                                             OCH.sub.3                                                                           N                                    H    CH.sub.2  NH      H    OCH.sub.3                                                                            OCH.sub.3                                                                           N                                    H    CH.sub.2  NH      H    CH.sub.3                                                                             CH.sub.3                                                                            N                                    6-Cl CH.sub.2  O       H    CH.sub.3                                                                             CH.sub.3                                                                            CH                                   6-Cl CH.sub.2  O       H    CH.sub.3                                                                             OCH.sub.3                                                                           CH                                   6-Cl CH.sub.2  O       H    OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                   6-Cl CH.sub.2  O       H    Cl     OCH.sub.3                                                                           CH                                   6-Cl CH.sub.2  O       H    CH.sub.3                                                                             OCH.sub.3                                                                           N                                    6-Cl CH.sub.2  O       H    OCH.sub.3                                                                            OCH.sub.3                                                                           N                                    6-Cl CH.sub.2  O       H    CH.sub.3                                                                             CH.sub.3                                                                            N                                    6-Cl CH.sub.2  S       CH.sub.3                                                                           CH.sub.3                                                                             CH.sub.3                                                                            CH                                   6-Cl CH.sub.2  S       CH.sub.3                                                                           CH.sub.3                                                                             OCH.sub.3                                                                           CH                                   6-Cl CH.sub.2  S       CH.sub.3                                                                           OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                   6-Cl CH.sub.2  S       CH.sub.3                                                                           Cl     OCH.sub.3                                                                           CH                                   6-Cl CH.sub.2  S       CH.sub.3                                                                           CH.sub.3                                                                             OCH.sub.3                                                                           N                                    6-Cl CH.sub.2  S       CH.sub.3                                                                           OCH.sub.3                                                                            OCH.sub. 3                                                                          N                                    6-Cl CH.sub.2  S       CH.sub.3                                                                           CH.sub.3                                                                             CH.sub.3                                                                            N                                    6-Cl CH.sub.2  NH      H    CH     CH.sub.3                                                                            CH                                   6-Cl CH.sub.2  NH      H    CH.sub.3                                                                             OCH.sub.3                                                                           CH                                   6-Cl CH.sub.2  NH      H    OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                   6-Cl CH.sub.2  NH      H    Cl     OCH.sub.3                                                                           CH                                   6-Cl CH.sub.2  NH      H    CH.sub.3                                                                             OCH.sub.3                                                                           N                                    6-Cl CH.sub.2  NH      H    OCH.sub.3                                                                            OCH.sub.3                                                                           N                                    6-Cl CH.sub.2  NH      H    CH.sub.3                                                                             CH.sub.3                                                                            N                                    H    CH.sub.2  S       H    OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                   H    CH.sub.2  S       H    CH.sub.3                                                                             OCH.sub.3                                                                           CH                                   H    CH.sub.2  S       H    CH.sub.3                                                                             CH.sub.3                                                                            CH                                   H    CH.sub.2  S       H    CH.sub.3                                                                             OCH.sub.3                                                                           N                                    H    CH.sub.2  S       H    OCH.sub.3                                                                            OCH.sub.3                                                                           N                                    H    CH.sub.2  S       H    Cl     OCH.sub.3                                                                           CH                                   H    CH.sub.2  NCH.sub.3                                                                             H    OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                   H    CH.sub.2  NCH.sub.3                                                                             H    CH.sub.3                                                                             OCH.sub.3                                                                           N                                    H    CH.sub.2 CH.sub.2                                                                       O       H    CH.sub.3                                                                             CH.sub.3                                                                            CH                                   H    CH.sub.2 CH.sub.2                                                                       O       H    CH.sub.3                                                                             OCH.sub.3                                                                           CH                                   H    CH.sub.2 CH.sub.2                                                                       O       H    OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                   H    CH.sub. 2 CH.sub.2                                                                      O       H    Cl     OCH.sub.3                                                                           CH                                   H    CH.sub.2 CH.sub.2                                                                       O       H    CH.sub.3                                                                             OCH.sub.3                                                                           N                                    H    CH.sub.2 CH.sub.2                                                                       O       H    OCH.sub.3                                                                            OCH.sub.3                                                                           N                                    H    CH.sub.2 CH.sub.2                                                                       O       H    CH.sub.3                                                                             CH.sub.3                                                                            N                                    H    CH.sub.2 CH.sub.2                                                                       S       CH.sub.3                                                                           CH.sub.3                                                                             CH.sub.3                                                                            CH                                   H    CH.sub.2 CH.sub.2                                                                       S       CH.sub.3                                                                           CH.sub.3                                                                             OCH.sub.3                                                                           CH                                   H    CH.sub.2 CH.sub.2                                                                       S       CH.sub.3                                                                           OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                   H    CH.sub.2 CH.sub.2                                                                       S       CH.sub.3                                                                           Cl     OCH.sub.3                                                                           CH                                   H    CH.sub.2 CH.sub.2                                                                       S       CH.sub.3                                                                           CH.sub.3                                                                             OCH.sub.3                                                                           N                                    H    CH.sub.2 CH.sub.2                                                                       S       CH.sub.3                                                                           OCH.sub.3                                                                            OCH.sub.3                                                                           N                                    H    CH.sub.2 CH.sub.2                                                                       S       CH.sub.3                                                                           CH.sub.3                                                                             CH.sub.3                                                                            N                                    H    CH.sub.2 CH.sub.2                                                                       NH      H    CH.sub.3                                                                             CH.sub.3                                                                            CH                                   H    CH.sub.2 CH.sub.2                                                                       NH      H    CH.sub.3                                                                             OCH.sub.3                                                                           CH                                   H    CH.sub.2 CH.sub.2                                                                       NH      H    OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                   H    CH.sub.2 CH.sub.2                                                                       NH      H    Cl     OCH.sub.3                                                                           CH                                   H    CH.sub.2 CH.sub.2                                                                       NH      H    CH.sub.3                                                                             OCH.sub.3                                                                           N                                    H    CH.sub.2 CH.sub.2                                                                       NH      H    OCH.sub.3                                                                            OCH.sub.3                                                                           N                                    H    CH.sub.2 CH.sub.2                                                                       NH      H    CH.sub.3                                                                             CH.sub.3                                                                            N                                    6-Cl CH.sub.2 CH.sub.2                                                                       O       H    CH.sub.3                                                                             CH.sub.3                                                                            CH                                   6-Cl CH.sub.2 CH.sub.2                                                                       O       H    CH.sub.3                                                                             OCH.sub.3                                                                           CH                                   6-Cl CH.sub.2 CH.sub.2                                                                       O       H    OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                   6-Cl CH.sub.2 CH.sub.2                                                                       O       H    Cl     OCH.sub.3                                                                           CH                                   6-Cl CH.sub.2 CH.sub.2                                                                       O       H    CH.sub.3                                                                             OCH.sub.3                                                                           N                                    6-Cl CH.sub.2 CH.sub.2                                                                       O       H    OCH.sub.3                                                                            OCH.sub.3                                                                           N                                    6-Cl CH.sub.2 CH.sub.2                                                                       O       H    CH.sub.3                                                                             CH.sub.3                                                                            N                                    6-Cl CH.sub.2 CH.sub.2                                                                       S       CH.sub.3                                                                           CH.sub.3                                                                             CH.sub.3                                                                            CH                                   6-Cl CH.sub.2 CH.sub.2                                                                       S       CH.sub.3                                                                           CH.sub.3                                                                             OCH.sub.3                                                                           CH                                   6-Cl CH.sub.2 CH.sub.2                                                                       S       CH.sub.3                                                                           OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                   6-Cl CH.sub.2 CH.sub.2                                                                       S       CH.sub.3                                                                           Cl     OCH.sub.3                                                                           CH                                   6-Cl CH.sub.2 CH.sub.2                                                                       S       CH.sub.3                                                                           CH.sub.3                                                                             OCH.sub.3                                                                           N                                    6-Cl CH.sub.2 CH.sub.2                                                                       S       CH.sub.3                                                                           OCH.sub.3                                                                            OCH.sub.3                                                                           N                                    6-Cl CH.sub.2 CH.sub.2                                                                       S       CH.sub.3                                                                           CH.sub.3                                                                             CH.sub.3                                                                            N                                    6-Cl CH.sub.2 CH.sub.2                                                                       NH      H    CH     CH.sub. 3                                                                           CH                                   6-Cl CH.sub.2 CH.sub.2                                                                       NH      H    CH.sub.3                                                                             OCH.sub.3                                                                           CH                                   6-Cl CH.sub.2 CH.sub.2                                                                       NH      H    OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                   6-Cl CH.sub.2 CH.sub.2                                                                       NH      H    Cl     OCH.sub.3                                                                           CH                                   6-Cl CH.sub.2 CH.sub.2                                                                       NH      H    CH.sub.3                                                                             OCH.sub.3                                                                           N                                    6-Cl CH.sub.2 CH.sub.2                                                                       NH      H    OCH.sub.3                                                                            OCH.sub.3                                                                           N                                    6-Cl CH.sub.2 CH.sub.2                                                                       NH      H    CH.sub.3                                                                             CH.sub.3                                                                            N                                    H    CH.sub.2 CH.sub.2                                                                       S       H    OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                   H    CH.sub.2 CH.sub.2                                                                       S       H    CH.sub.3                                                                             OCH.sub.3                                                                           CH                                   H    CH.sub.2 CH.sub.2                                                                       S       H    CH.sub.3                                                                             CH.sub.3                                                                            CH                                   H    CH.sub.2 CH.sub.2                                                                       S       H    CH.sub.3                                                                             OCH.sub.3                                                                           N                                    H    CH.sub.2 CH.sub.2                                                                       S       H    OCH.sub.3                                                                            OCH.sub.3                                                                           N                                    H    CH.sub.2 CH.sub.2                                                                       S       H    Cl     OCH.sub.3                                                                           CH                                   H    CH.sub.2 CH.sub.2                                                                       NCH.sub.3                                                                             H    OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                   H    CH.sub.2 CH.sub.2                                                                       NCH.sub.3                                                                             H    CH.sub.3                                                                             OCH.sub.3                                                                           N                                    H    CH═CH O       H    CH.sub.3                                                                             CH.sub.3                                                                            CH                                   H    CH═CH O       H    CH.sub.3                                                                             OCH.sub.3                                                                           CH                                   H    CH═CH O       H    OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                   H    CH═CH O       H    Cl     OCH.sub.3                                                                           CH                                   H    CH═CH O       H    CH.sub.3                                                                             OCH.sub.3                                                                           N                                    H    CH═CH O       H    OCH.sub.3                                                                            OCH.sub.3                                                                           N                                    H    CH═CH O       H    CH.sub.3                                                                             CH.sub.3                                                                            N                                    H    CH═CH S       CH.sub.3                                                                           CH.sub.3                                                                             CH.sub.3                                                                            CH                                   H    CH═CH S       CH.sub.3                                                                           CH.sub.3                                                                             OCH.sub.3                                                                           CH                                   H    CH═CH S       CH.sub.3                                                                           OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                   H    CH═CH S       CH.sub.3                                                                           Cl     OCH.sub.3                                                                           CH                                   H    CH═CH S       CH.sub.3                                                                           CH.sub.3                                                                             OCH.sub.3                                                                           N                                    H    CH═CH S       CH.sub.3                                                                           OCH.sub.3                                                                            OCH.sub.3                                                                           N                                    H    CH═CH S       CH.sub.3                                                                           CH.sub.3                                                                             CH.sub.3                                                                            N                                    H    CH═CH NH      H    CH.sub.3                                                                             CH.sub.3                                                                            CH                                   H    CH═CH NH      H    CH.sub.3                                                                             OCH.sub.3                                                                           CH                                   H    CH═CH NH      H    OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                   H    CH═CH NH      H    Cl     OCH.sub.3                                                                           CH                                   H    CH═CH NH      H    CH.sub.3                                                                             OCH.sub.3                                                                           N                                    H    CH═CH NH      H    OCH.sub.3                                                                            OCH.sub.3                                                                           N                                    H    CH═CH NH      H    CH.sub.3                                                                             CH.sub.3                                                                            N                                    6-Cl CH═CH O       H    CH.sub.3                                                                             CH.sub.3                                                                            CH                                   6-Cl CH═CH O       H    CH.sub. 3                                                                            OCH.sub.3                                                                           CH                                   6-Cl CH═CH O       H    OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                   6-Cl CH═CH O       H    Cl     OCH.sub.3                                                                           CH                                   6-Cl CH═CH O       H    CH.sub.3                                                                             OCH.sub.3                                                                           N                                    6-Cl CH═CH O       H    OCH.sub.3                                                                            OCH.sub.3                                                                           N                                    6-Cl CH═CH O       H    CH.sub.3                                                                             CH.sub.3                                                                            N                                    6-Cl CH═CH S       CH.sub.3                                                                           CH.sub.3                                                                             CH.sub.3                                                                            CH                                   6-Cl CH═CH S       CH.sub.3                                                                           CH.sub.3                                                                             OCH.sub.3                                                                           CH                                   6-Cl CH═CH S       CH.sub.3                                                                           OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                   6-Cl CH═CH S       CH.sub.3                                                                           Cl     OCH.sub.3                                                                           CH                                   6-Cl CH═CH S       CH.sub.3                                                                           CH.sub.3                                                                             OCH.sub.3                                                                           N                                    6-Cl CH═CH S       CH.sub.3                                                                           OCH.sub.3                                                                            OCH.sub.3                                                                           N                                    6-Cl CH═CH S       CH.sub.3                                                                           CH.sub.3                                                                             CH.sub.3                                                                            N                                    6-Cl CH═CH NH      H    CH     CH.sub.3                                                                            CH                                   6-Cl CH═CH NH      H    CH.sub.3                                                                             OCH.sub.3                                                                           CH                                   6-Cl CH═CH NH      H    OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                   6-Cl CH═CH NH      H    Cl     OCH.sub.3                                                                           CH                                   6-Cl CH═CH NH      H    CH.sub.3                                                                             OCH.sub.3                                                                           N                                    6-Cl CH═CH NH      H    OCH.sub.3                                                                            OCH.sub.3                                                                           N                                    6-Cl CH═CH NH      H    CH.sub.3                                                                             CH.sub.3                                                                            N                                    H    CH═CH S       H    OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                   H    CH═CH S       H    CH.sub.3                                                                             OCH.sub.3                                                                           CH                                   H    CH═CH S       H    CH.sub.3                                                                             CH.sub.3                                                                            CH                                   H    CH═CH S       H    CH.sub.3                                                                             OCH.sub.3                                                                           N                                    H    CH═CH S       H    OCH.sub.3                                                                            OCH.sub.3                                                                           N                                    H    CH═CH S       H    Cl     OCH.sub.3                                                                           CH                                   H    CH═CH NCH.sub.3                                                                             H    OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                   H    CH═CH NCH.sub.3                                                                             H    CH.sub.3                                                                             OCH.sub.3                                                                           N                                    ______________________________________                                    

                  TABLE 3a                                                        ______________________________________                                        General Formula 3a                                                            R.sub.1                                                                              J       R.sub.10                                                                             X      Y     Z     m.p.(°C.)                     ______________________________________                                        H      C═O H      CH.sub.3                                                                             CH.sub.3                                                                            CH                                         H      C═O H      CH.sub.3                                                                             OCH.sub.3                                                                           CH                                         H      C═O H      OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                         H      C═O H      Cl     OCH.sub.3                                                                           CH                                         H      C═O H      CH.sub.3                                                                             OCH.sub.3                                                                           N                                          H      C═O H      OCH.sub.3                                                                            OCH.sub.3                                                                           N                                          H      C═O H      CH.sub.3                                                                             CH.sub.3                                                                            N                                          H      C═O CH.sub.3                                                                             CH.sub.3                                                                             CH.sub.3                                                                            CH                                         H      C═O CH.sub.3                                                                             CH.sub.3                                                                             OCH.sub.3                                                                           CH                                         H      C═O CH.sub.3                                                                             OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                         H      C═O CH.sub.3                                                                             Cl     OCH.sub.3                                                                           CH                                         H      C═O CH.sub.3                                                                             CH.sub.3                                                                             OCH.sub.3                                                                           N                                          H      C═O CH.sub.3                                                                             OCH.sub.3                                                                            OCH.sub.3                                                                           N                                          H      C═O CH.sub.3                                                                             CH.sub.3                                                                             CH.sub.3                                                                            N                                          H      CH.sub.2                                                                              CH.sub.3                                                                             CH.sub.3                                                                             CH.sub.3                                                                            CH                                         H      CH.sub.2                                                                              CH.sub.3                                                                             CH.sub.3                                                                             OCH.sub.3                                                                           CH                                         H      CH.sub.2                                                                              CH.sub.3                                                                             OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                         H      CH.sub.2                                                                              CH.sub.3                                                                             Cl     OCH.sub. 3                                                                          CH                                         H      CH.sub.2                                                                              CH.sub.3                                                                             CH.sub.3                                                                             OCH.sub.3                                                                           N                                          H      CH.sub.2                                                                              CH.sub.3                                                                             OCH.sub.3                                                                            OCH.sub.3                                                                           N                                          H      CH.sub.2                                                                              CH.sub.3                                                                             CH.sub.3                                                                             CH.sub.3                                                                            N                                          H      S       H      CH.sub.3                                                                             CH.sub.3                                                                            CH                                         H      S       H      CH.sub.3                                                                             OCH.sub.3                                                                           CH                                         H      S       H      OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                         H      S       H      Cl     OCH.sub.3                                                                           CH                                         H      S       H      CH.sub.3                                                                             OCH.sub.3                                                                           N                                          H      S       H      OCH.sub.3                                                                            OCH.sub.3                                                                           N                                          H      S       H      CH.sub.3                                                                             CH.sub.3                                                                            N                                          H      SO.sub.2                                                                              H      CH.sub.3                                                                             CH.sub.3                                                                            CH                                         H      SO.sub.2                                                                              H      CH.sub.3                                                                             OCH.sub.3                                                                           CH                                         H      SO.sub.2                                                                              H      CH.sub.3                                                                             OCH.sub.3                                                                           CH                                         H      SO.sub.2                                                                              H      OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                         H      SO.sub.2                                                                              H      Cl     OCH.sub.3                                                                           CH                                         H      SO.sub.2                                                                              H      CH.sub.3                                                                             OCH.sub.3                                                                           N                                          H      SO.sub.2                                                                              H      OCH.sub.3                                                                            OCH.sub.3                                                                           N                                          H      SO.sub.2                                                                              H      CH.sub.3                                                                             CH.sub.3                                                                            N                                          H      O       CH.sub.3                                                                             CH.sub.3                                                                             CH.sub.3                                                                            CH                                         H      O       CH.sub.3                                                                             CH.sub.3                                                                             OCH.sub.3                                                                           CH                                         H      O       CH.sub.3                                                                             OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                         H      O       CH.sub.3                                                                             Cl     OCH.sub.3                                                                           CH                                         H      O       CH.sub.3                                                                             CH.sub.3                                                                             OCH.sub. 3                                                                          N                                          H      O       CH.sub.3                                                                             OCH.sub.3                                                                            OCH.sub.3                                                                           N                                          H      O       CH.sub.3                                                                             CH.sub.3                                                                             CH.sub.3                                                                            N                                          6-CH.sub.3                                                                           C═O H      CH.sub.3                                                                             CH.sub.3                                                                            CH                                         6-CH.sub.3                                                                           C═O H      CH.sub.3                                                                             OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                           C═O H      OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                           C═O H      Cl     OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                           C═O H      CH.sub.3                                                                             OCH.sub.3                                                                           N                                          6-CH.sub.3                                                                           C═O H      OCH.sub.3                                                                            OCH.sub.3                                                                           N                                          6-CH.sub.3                                                                           C═O H      CH.sub.3                                                                             CH.sub.3                                                                            N                                          6-CH.sub.3                                                                           C═O CH.sub.3                                                                             CH.sub.3                                                                             CH.sub.3                                                                            CH                                         6-CH.sub.3                                                                           C═O CH.sub.3                                                                             CH.sub.3                                                                             OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                           C═O CH.sub.3                                                                             OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                           C═O CH.sub.3                                                                             Cl     OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                           C═O CH.sub.3                                                                             CH.sub.3                                                                             OCH.sub.3                                                                           N                                          6-CH.sub.3                                                                           C═O CH.sub.3                                                                             OCH.sub.3                                                                            OCH.sub.3                                                                           N                                          6-CH.sub.3                                                                           C═O CH.sub.3                                                                             CH.sub.3                                                                             CH.sub.3                                                                            N                                          6-CH.sub.3                                                                           CH.sub.2                                                                              CH.sub.3                                                                             CH.sub.3                                                                             CH.sub.3                                                                            CH                                         6-CH.sub.3                                                                           CH.sub.2                                                                              CH.sub.3                                                                             CH.sub.3                                                                             OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                           CH.sub.2                                                                              CH.sub.3                                                                             OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                           CH.sub.2                                                                              CH.sub.3                                                                             Cl     OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                           CH.sub.2                                                                              CH.sub.3                                                                             CH.sub.3                                                                             OCH.sub.3                                                                           N                                          6-CH.sub.3                                                                           CH.sub.2                                                                              CH.sub.3                                                                             OCH.sub.3                                                                            OCH.sub.3                                                                           N                                          6-CH.sub.3                                                                           CH.sub.2                                                                              CH.sub.3                                                                             CH.sub.3                                                                             CH.sub.3                                                                            N                                          6-CH.sub.3                                                                           S       H      CH.sub.3                                                                             CH.sub.3                                                                            CH                                         6-CH.sub.3                                                                           S       H      CH.sub.3                                                                             OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                           S       H      OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                           S       H      Cl     OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                           S       H      CH.sub.3                                                                             OCH.sub.3                                                                           N                                          6-CH.sub.3                                                                           S       H      OCH.sub.3                                                                            OCH.sub.3                                                                           N                                          6-CH.sub.3                                                                           S       H      CH.sub.3                                                                             CH.sub.3                                                                            N                                          6-CH.sub.3                                                                           SO.sub.2                                                                              H      CH.sub.3                                                                             CH.sub.3                                                                            CH                                         6-CH.sub.3                                                                           SO.sub.2                                                                              H      CH.sub.3                                                                             OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                           SO.sub.2                                                                              H      OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                           SO.sub.2                                                                              H      Cl     OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                           SO.sub.2                                                                              H      CH.sub.3                                                                             OCH.sub.3                                                                           N                                          6-CH.sub.3                                                                           SO.sub.2                                                                              H      OCH.sub.3                                                                            OCH.sub.3                                                                           N                                          6-CH.sub.3                                                                           SO.sub.2                                                                              H      CH.sub.3                                                                             CH.sub.3                                                                            N                                          6-CH.sub.3                                                                           O       CH.sub.3                                                                             CH.sub.3                                                                             CH.sub.3                                                                            CH                                         6-CH.sub.3                                                                           O       CH.sub.3                                                                             CH.sub.3                                                                             OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                           O       CH.sub.3                                                                             OCH.sub.3                                                                            OCH.sub. 3                                                                          CH                                         6-CH.sub.3                                                                           O       CH.sub.3                                                                             Cl     OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                           O       CH.sub.3                                                                             CH.sub.3                                                                             OCH.sub.3                                                                           N                                          6-CH.sub.3                                                                           O       CH.sub.3                                                                             OCH.sub.3                                                                            OCH.sub.3                                                                           N                                          6-CH.sub.3                                                                           O       CH.sub.3                                                                             CH.sub.3                                                                             CH.sub.3                                                                            N                                          6-Cl   C═O H      CH.sub.3                                                                             CH.sub.3                                                                            CH                                         6-Cl   C═O H      CH.sub.3                                                                             OCH.sub.3                                                                           CH                                         6-Cl   C═O H      OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                         6-Cl   C═O H      Cl     OCH.sub.3                                                                           CH                                         6-Cl   C═O H      CH.sub.3                                                                             OCH.sub.3                                                                           N                                          6-Cl   C═O H      OCH.sub.3                                                                            OCH.sub.3                                                                           N                                          6-Cl   C═O H      CH.sub.3                                                                             CH.sub.3                                                                            N                                          6-Cl   C═O CH.sub.3                                                                             CH.sub.3                                                                             CH.sub.3                                                                            CH                                         6-Cl   C═O CH.sub.3                                                                             CH.sub.3                                                                             OCH.sub.3                                                                           CH                                         6-Cl   C═O CH.sub.3                                                                             OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                         6-Cl   C═O CH.sub.3                                                                             Cl     OCH.sub.3                                                                           CH                                         6-Cl   C═O CH.sub.3                                                                             CH.sub.3                                                                             OCH.sub.3                                                                           N                                          6-Cl   C═O CH.sub.3                                                                             OCH.sub.3                                                                            OCH.sub.3                                                                           N                                          6-Cl   C═O CH.sub.3                                                                             CH.sub.3                                                                             CH.sub.3                                                                            N                                          6-Cl   CH.sub.2                                                                              CH.sub.3                                                                             CH.sub.3                                                                             CH.sub.3                                                                            CH                                         6-Cl   CH.sub.2                                                                              CH.sub.3                                                                             CH.sub.3                                                                             OCH.sub.3                                                                           CH                                         6-Cl   CH.sub.2                                                                              CH.sub.3                                                                             OCH.sub.3                                                                            OCH.sub. 3                                                                          CH                                         6-Cl   CH.sub.2                                                                              CH.sub.3                                                                             Cl     OCH.sub.3                                                                           CH                                         6-Cl   CH.sub.2                                                                              CH.sub.3                                                                             CH.sub.3                                                                             OCH.sub.3                                                                           N                                          6-Cl   CH.sub.2                                                                              CH.sub.3                                                                             OCH.sub.3                                                                            OCH.sub.3                                                                           N                                          6-Cl   CH.sub.2                                                                              CH.sub.3                                                                             CH.sub.3                                                                             CH.sub.3                                                                            N                                          6-Cl   S       H      CH.sub.3                                                                             CH.sub.3                                                                            CH                                         6-Cl   S       H      CH.sub.3                                                                             OCH.sub.3                                                                           CH                                         6-Cl   S       H      OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                         6-Cl   S       H      Cl     OCH.sub.3                                                                           CH                                         6-Cl   S       H      CH.sub.3                                                                             OCH.sub.3                                                                           N                                          6-Cl   S       H      OCH.sub.3                                                                            OCH.sub.3                                                                           N                                          6-Cl   S       H      CH.sub.3                                                                             CH.sub.3                                                                            N                                          6-Cl   SO.sub.2                                                                              H      CH.sub.3                                                                             CH.sub.3                                                                            CH                                         6-Cl   SO.sub.2                                                                              H      CH.sub.3                                                                             OCH.sub.3                                                                           CH                                         6-Cl   SO.sub.2                                                                              H      OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                         6-Cl   SO.sub.2                                                                              H      Cl     OCH.sub.3                                                                           CH                                         6-Cl   SO.sub.2                                                                              H      CH.sub.3                                                                             OCH.sub.3                                                                           N                                          6-Cl   SO.sub.2                                                                              H      OCH.sub.3                                                                            OCH.sub.3                                                                           N                                          6-Cl   SO.sub.2                                                                              H      CH.sub.3                                                                             CH.sub.3                                                                            N                                          6-Cl   O       CH.sub.3                                                                             CH.sub.3                                                                             CH.sub.3                                                                            CH                                         6-Cl   O       CH.sub.3                                                                             CH.sub.3                                                                             OCH.sub.3                                                                           CH                                         6-Cl   O       CH.sub.3                                                                             OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                         6-Cl   O       CH.sub.3                                                                             Cl     OCH.sub.3                                                                           CH                                         6-Cl   O       CH.sub.3                                                                             CH.sub.3                                                                             OCH.sub. 3                                                                          N                                          6-Cl   O       CH.sub.3                                                                             OCH.sub.3                                                                            OCH.sub.3                                                                           N                                          6-Cl   O       CH.sub.3                                                                             CH.sub.3                                                                             CH.sub.3                                                                            N                                          ______________________________________                                    

                  TABLE 3b                                                        ______________________________________                                        General Formula 3b                                                            R.sub.1                                                                             G        R.sub.10                                                                              X     Y      Z    m.p.(°C.)                     ______________________________________                                        H     CH.sub.2 H       CH.sub.3                                                                            CH.sub.3                                                                             CH                                        H     CH.sub.2 H       CH.sub.3                                                                            OCH.sub.3                                                                            CH                                        H     CH.sub.2 H       OCH.sub.3                                                                           OCH.sub.3                                                                            CH                                        H     CH.sub.2 H       Cl    OCH.sub.3                                                                            CH                                        H     CH.sub.2 H       CH.sub.3                                                                            OCH.sub.3                                                                            N                                         H     CH.sub.2 H       OCH.sub.3                                                                           OCH.sub.3                                                                            N                                         H     CH.sub.2 H       CH.sub.3                                                                            CH.sub.3                                                                             N                                         H     CH.sub.2 CH.sub.3                                                                              CH.sub.3                                                                            CH.sub.3                                                                             CH                                        H     CH.sub.2 CH.sub.3                                                                              CH.sub.3                                                                            OCH.sub.3                                                                            CH                                        H     CH.sub.2 CH.sub.3                                                                              OCH.sub.3                                                                           OCH.sub.3                                                                            CH                                        H     CH.sub.2 CH.sub.3                                                                              Cl    OCH.sub.3                                                                            CH                                        H     CH.sub.2 CH.sub.3                                                                              CH.sub.3                                                                            OCH.sub.3                                                                            N                                         H     CH.sub.2 CH.sub.3                                                                              OCH.sub.3                                                                           OCH.sub.3                                                                            N                                         H     CH.sub.2 CH.sub.3                                                                              CH.sub.3                                                                            CH.sub.3                                                                             N                                         H     CH.sub.2 C.sub.6 H.sub.5                                                                       CH.sub.3                                                                            CH.sub.3                                                                             CH                                        H     CH.sub.2 C.sub.6 H.sub.5                                                                       CH.sub.3                                                                            OCH.sub.3                                                                            CH                                        H     CH.sub.2 C.sub.6 H.sub.5                                                                       OCH.sub.3                                                                           OCH.sub.3                                                                            CH                                        H     CH.sub.2 C.sub.6 H.sub.5                                                                       Cl    OCH.sub.3                                                                            CH                                        H     CH.sub.2 C.sub.6 H.sub.5                                                                       CH.sub.3                                                                            OCH.sub.3                                                                            N                                         H     CH.sub.2 C.sub.6 H.sub.5                                                                       OCH.sub.3                                                                           OCH.sub.3                                                                            N                                         H     CH.sub.2 C.sub.6 H.sub.5                                                                       CH.sub.3                                                                            CH.sub.3                                                                             N                                         6-CH.sub.3                                                                          CH.sub.2 H       CH.sub.3                                                                            CH.sub.3                                                                             CH                                        6-CH.sub.3                                                                          CH.sub.2 H       CH.sub.3                                                                            OCH.sub.3                                                                            CH                                        6-CH.sub.3                                                                          CH.sub.2 H       OCH.sub.3                                                                           OCH.sub.3                                                                            CH                                        6-CH.sub.3                                                                          CH.sub.2 H       Cl    OCH.sub.3                                                                            CH                                        6-CH.sub.3                                                                          CH.sub.2 H       CH.sub.3                                                                            OCH.sub.3                                                                            N                                         6-CH.sub.3                                                                          CH.sub.2 H       OCH.sub.3                                                                           OCH.sub.3                                                                            N                                         6-CH.sub.3                                                                          CH.sub.2 H       CH.sub.3                                                                            CH.sub.3                                                                             N                                         6-CH.sub.3                                                                          CH.sub.2 CH.sub.3                                                                              CH.sub.3                                                                            CH.sub.3                                                                             CH                                        6-CH.sub.3                                                                          CH.sub.2 CH.sub.3                                                                              OCH.sub.3                                                                           CH.sub.3                                                                             CH                                        6-CH.sub.3                                                                          CH.sub.2 CH.sub.3                                                                              OCH.sub.3                                                                           OCH.sub.3                                                                            CH                                        6-CH.sub.3                                                                          CH.sub.2 CH.sub.3                                                                              Cl    OCH.sub.3                                                                            CH                                        6-CH.sub.3                                                                          CH.sub.2 CH.sub.3                                                                              CH.sub.3                                                                            OCH.sub.3                                                                            N                                         6-CH.sub.3                                                                          CH.sub.2 CH.sub.3                                                                              OCH.sub.3                                                                           OCH.sub.3                                                                            N                                         6-CH.sub.3                                                                          CH.sub.2 CH.sub.3                                                                              CH.sub.3                                                                            CH.sub.3                                                                             N                                         6-CH.sub.3                                                                          CH.sub.2 C.sub.6 H.sub.5                                                                       CH.sub. 3                                                                           CH.sub.3                                                                             CH                                        6-CH.sub.3                                                                          CH.sub.2 C.sub.6 H.sub.5                                                                       CH.sub.3                                                                            OCH.sub.3                                                                            CH                                        6-CH.sub.3                                                                          CH.sub.2 C.sub.6 H.sub.5                                                                       OCH.sub.3                                                                           OCH.sub.3                                                                            CH                                        6-CH.sub.3                                                                          CH.sub.2 C.sub.6 H.sub.5                                                                       Cl    OCH.sub.3                                                                            CH                                        6-CH.sub.3                                                                          CH.sub.2 C.sub.6 H.sub.5                                                                       CH.sub.3                                                                            OCH.sub.3                                                                            N                                         6-CH.sub.3                                                                          CH.sub.2 C.sub.6 H.sub.5                                                                       OCH.sub.3                                                                           OCH.sub.3                                                                            N                                         6-CH.sub.3                                                                          CH.sub.2 C.sub.6 H.sub.5                                                                       CH.sub.3                                                                            CH.sub.3                                                                             N                                         6-Cl  CH.sub.2 H       CH.sub.3                                                                            CH.sub.3                                                                             CH                                        6-Cl  CH.sub.2 H       CH.sub.3                                                                            OCH.sub.3                                                                            CH                                        6-Cl  CH.sub.2 H       OCH.sub.3                                                                           OCH.sub.3                                                                            CH                                        6-Cl  CH.sub.2 H       Cl    OCH.sub.3                                                                            CH                                        6-Cl  CH.sub.2 H       CH.sub.3                                                                            OCH.sub.3                                                                            N                                         6-Cl  CH.sub.2 H       OCH.sub.3                                                                           OCH.sub.3                                                                            N                                         6-Cl  CH.sub.2 H       CH.sub.3                                                                            CH.sub.3                                                                             N                                         6-Cl  CH.sub.2 CH.sub.3                                                                              CH.sub.3                                                                            CH.sub.3                                                                             CH                                        6-Cl  CH.sub.2 CH.sub.3                                                                              OCH.sub.3                                                                           CH.sub.3                                                                             CH                                        6-Cl  CH.sub.2 CH.sub.3                                                                              OCH.sub.3                                                                           OCH.sub.3                                                                            CH                                        6-Cl  CH.sub.2 CH.sub.3                                                                              Cl    OCH.sub.3                                                                            CH                                        6-Cl  CH.sub.2 CH.sub.3                                                                              CH.sub.3                                                                            OCH.sub.3                                                                            N                                         6-Cl  CH.sub.2 CH.sub.3                                                                              OCH.sub.3                                                                           OCH.sub. 3                                                                           N                                         6-Cl  CH.sub.2 CH.sub.3                                                                              CH.sub.3                                                                            CH.sub.3                                                                             N                                         6-Cl  CH.sub.2 C.sub.6 H.sub.5                                                                       CH.sub.3                                                                            CH.sub.3                                                                             CH                                        6-Cl  CH.sub.2 C.sub.6 H.sub.5                                                                       CH.sub.3                                                                            OCH.sub.3                                                                            CH                                        6-Cl  CH.sub.2 C.sub.6 H.sub.5                                                                       OCH.sub.3                                                                           OCH.sub.3                                                                            CH                                        6-Cl  CH.sub.2 C.sub.6 H.sub.5                                                                       Cl    OCH.sub.3                                                                            CH                                        6-Cl  CH.sub.2 C.sub.6 H.sub.5                                                                       CH.sub.3                                                                            OCH.sub.3                                                                            N                                         6-Cl  CH.sub.2 C.sub.6 H.sub.5                                                                       OCH.sub.3                                                                           OCH.sub.3                                                                            N                                         6-Cl  CH.sub.2 C.sub.6 H.sub.5                                                                       CH.sub.3                                                                            CH.sub.3                                                                             N                                         H     CH.sub.2 CH.sub.2                                                                      H       CH.sub.3                                                                            CH.sub.3                                                                             CH                                        H     CH.sub.2 CH.sub.2                                                                      H       CH.sub.3                                                                            OCH.sub.3                                                                            CH                                        H     CH.sub.2 CH.sub.2                                                                      H       OCH.sub.3                                                                           OCH.sub.3                                                                            CH                                        H     CH.sub.2 CH.sub.2                                                                      H       Cl    OCH.sub.3                                                                            CH                                        H     CH.sub.2 CH.sub.2                                                                      H       CH.sub.3                                                                            OCH.sub.3                                                                            N                                         H     CH.sub.2 CH.sub.2                                                                      H       OCH.sub.3                                                                           OCH.sub.3                                                                            N                                         H     CH.sub.2 CH.sub.2                                                                      H       CH.sub.3                                                                            CH.sub.3                                                                             N                                         H     CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              CH.sub.3                                                                            CH.sub.3                                                                             CH                                        H     CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              CH.sub.3                                                                            OCH.sub.3                                                                            CH                                        H     CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              OCH.sub.3                                                                           OCH.sub.3                                                                            CH                                        H     CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              Cl    OCH.sub.3                                                                            CH                                        H     CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              CH.sub.3                                                                            OCH.sub.3                                                                            N                                         H     CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              OCH.sub.3                                                                           OCH.sub.3                                                                            N                                         H     CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              CH.sub.3                                                                            CH.sub.3                                                                             N                                         H     CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                       CH.sub.3                                                                            CH.sub.3                                                                             CH                                        H     CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                       CH.sub.3                                                                            OCH.sub.3                                                                            CH                                        H     CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                       OCH.sub.3                                                                           OCH.sub.3                                                                            CH                                        H     CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                       Cl    OCH.sub.3                                                                            CH                                        H     CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                       CH.sub.3                                                                            OCH.sub.3                                                                            N                                         H     CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                       OCH.sub.3                                                                           OCH.sub.3                                                                            N                                         H     CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                       CH.sub.3                                                                            CH.sub.3                                                                             N                                         6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                      H       CH.sub.3                                                                            CH.sub.3                                                                             CH                                        6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                      H       CH.sub.3                                                                            OCH.sub.3                                                                            CH                                        6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                      H       OCH.sub.3                                                                           OCH.sub.3                                                                            CH                                        6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                      H       Cl    OCH.sub.3                                                                            CH                                        6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                      H       CH.sub.3                                                                            OCH.sub.3                                                                            N                                         6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                      H       OCH.sub.3                                                                           OCH.sub.3                                                                            N                                         6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                      H       CH.sub.3                                                                            CH.sub.3                                                                             N                                         6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              CH.sub.3                                                                            CH.sub.3                                                                             CH                                        6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              OCH.sub.3                                                                           CH.sub.3                                                                             CH                                        6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              OCH.sub.3                                                                           OCH.sub.3                                                                            CH                                        6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              Cl    OCH.sub.3                                                                            CH                                        6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              CH.sub.3                                                                            OCH.sub.3                                                                            N                                         6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              OCH.sub.3                                                                           OCH.sub.3                                                                            N                                         6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              CH.sub.3                                                                            CH.sub.3                                                                             N                                         6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                       CH.sub.3                                                                            CH.sub.3                                                                             CH                                        6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                       CH.sub.3                                                                            OCH.sub.3                                                                            CH                                        6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                       OCH.sub.3                                                                           OCH.sub.3                                                                            CH                                        6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                       Cl    OCH.sub.3                                                                            CH                                        6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                       CH.sub.3                                                                            OCH.sub.3                                                                            N                                         6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                       OCH.sub.3                                                                           OCH.sub.3                                                                            N                                         6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                       CH.sub.3                                                                            CH.sub.3                                                                             N                                         6-Cl  CH.sub.2 CH.sub.2                                                                      H       CH.sub.3                                                                            CH.sub.3                                                                             CH                                        6-Cl  CH.sub.2 CH.sub.2                                                                      H       CH.sub.3                                                                            OCH.sub.3                                                                            CH                                        6-Cl  CH.sub.2 CH.sub.2                                                                      H       OCH.sub.3                                                                           OCH.sub.3                                                                            CH                                        6-Cl  CH.sub.2 CH.sub.2                                                                      H       Cl    OCH.sub.3                                                                            CH                                        6-Cl  CH.sub.2 CH.sub.2                                                                      H       CH.sub.3                                                                            OCH.sub.3                                                                            N                                         6-Cl  CH.sub.2 CH.sub.2                                                                      H       OCH.sub.3                                                                           OCH.sub.3                                                                            N                                         6-Cl  CH.sub.2 CH.sub.2                                                                      H       CH.sub.3                                                                            CH.sub.3                                                                             N                                         6-Cl  CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              CH.sub.3                                                                            CH.sub.3                                                                             CH                                        6-Cl  CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              OCH.sub.3                                                                           CH.sub.3                                                                             CH                                        6-Cl  CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              OCH.sub.3                                                                           OCH.sub.3                                                                            CH                                        6-Cl  CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              Cl    OCH.sub.3                                                                            CH                                        6-Cl  CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              CH.sub.3                                                                            OCH.sub.3                                                                            N                                         6-Cl  CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              OCH.sub.3                                                                           OCH.sub.3                                                                            N                                         6-Cl  CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              CH.sub.3                                                                            CH.sub.3                                                                             N                                         6-Cl  CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                       CH.sub.3                                                                            CH.sub.3                                                                             CH                                        6-Cl  CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                       CH.sub.3                                                                            OCH.sub.3                                                                            CH                                        6-Cl  CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                       OCH.sub.3                                                                           OCH.sub.3                                                                            CH                                        6-Cl  CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                       Cl    OCH.sub.3                                                                            CH                                        6-Cl  CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                       CH.sub.3                                                                            OCH.sub.3                                                                            N                                         6-Cl  CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                       OCH.sub.3                                                                           OCH.sub.3                                                                            N                                         6-Cl  CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                       CH.sub.3                                                                            CH.sub.3                                                                             N                                         H     CH═CH                                                                              H       CH.sub.3                                                                            CH.sub.3                                                                             CH                                        H     CH═CH                                                                              H       CH.sub.3                                                                            OCH.sub.3                                                                            CH                                        H     CH═CH                                                                              H       OCH.sub.3                                                                           OCH.sub.3                                                                            CH                                        H     CH═CH                                                                              H       Cl    OCH.sub.3                                                                            CH                                        H     CH═CH                                                                              H       CH.sub.3                                                                            OCH.sub.3                                                                            N                                         H     CH═CH                                                                              H       OCH.sub.3                                                                           OCH.sub.3                                                                            N                                         H     CH═CH                                                                              H       CH.sub.3                                                                            CH.sub.3                                                                             N                                         H     CH═CH                                                                              CH.sub.3                                                                              CH.sub.3                                                                            CH.sub.3                                                                             CH                                        H     CH═CH                                                                              CH.sub.3                                                                              CH.sub.3                                                                            OCH.sub.3                                                                            CH                                        H     CH═CH                                                                              CH.sub.3                                                                              OCH.sub.3                                                                           OCH.sub.3                                                                            CH                                        H     CH═CH                                                                              CH.sub.3                                                                              Cl    OCH.sub.3                                                                            CH                                        H     CH═CH                                                                              CH.sub.3                                                                              CH.sub.3                                                                            OCH.sub.3                                                                            N                                         H     CH═CH                                                                              CH.sub.3                                                                              OCH.sub.3                                                                           OCH.sub.3                                                                            N                                         H     CH═CH                                                                              CH.sub.3                                                                              CH.sub.3                                                                            CH.sub.3                                                                             N                                         H     CH═CH                                                                              C.sub.6 H.sub.5                                                                       CH.sub.3                                                                            CH.sub.3                                                                             CH                                        H     CH═CH                                                                              C.sub.6 H.sub.5                                                                       CH.sub.3                                                                            OCH.sub.3                                                                            CH                                        H     CH═CH                                                                              C.sub.6 H.sub.5                                                                       OCH.sub.3                                                                           OCH.sub.3                                                                            CH                                        H     CH═CH                                                                              C.sub.6 H.sub.5                                                                       Cl    OCH.sub.3                                                                            CH                                        H     CH═CH                                                                              C.sub.6 H.sub.5                                                                       CH.sub.3                                                                            OCH.sub.3                                                                            N                                         H     CH═CH                                                                              C.sub.6 H.sub.5                                                                       OCH.sub.3                                                                           OCH.sub.3                                                                            N                                         H     CH═CH                                                                              C.sub.6 H.sub.5                                                                       CH.sub.3                                                                            CH.sub.3                                                                             N                                         6-CH.sub.3                                                                          CH═CH                                                                              H       CH.sub.3                                                                            CH.sub.3                                                                             CH                                        6-CH.sub.3                                                                          CH═CH                                                                              H       CH.sub.3                                                                            OCH.sub.3                                                                            CH                                        6-CH.sub.3                                                                          CH═CH                                                                              H       OCH.sub.3                                                                           OCH.sub.3                                                                            CH                                        6-CH.sub.3                                                                          CH═CH                                                                              H       Cl    OCH.sub.3                                                                            CH                                        6-CH.sub.3                                                                          CH═CH                                                                              H       CH.sub.3                                                                            OCH.sub.3                                                                            N                                         6-CH.sub.3                                                                          CH═CH                                                                              H       OCH.sub.3                                                                           OCH.sub.3                                                                            N                                         6-CH.sub.3                                                                          CH═CH                                                                              H       CH.sub.3                                                                            CH.sub.3                                                                             N                                         6-CH.sub.3                                                                          CH═CH                                                                              CH.sub.3                                                                              CH.sub.3                                                                            CH.sub.3                                                                             CH                                        6-CH.sub.3                                                                          CH═CH                                                                              CH.sub.3                                                                              OCH.sub.3                                                                           CH.sub.3                                                                             CH                                        6-CH.sub.3                                                                          CH═CH                                                                              CH.sub.3                                                                              OCH.sub.3                                                                           OCH.sub.3                                                                            CH                                        6-CH.sub.3                                                                          CH═CH                                                                              CH.sub.3                                                                              Cl    OCH.sub.3                                                                            CH                                        6-CH.sub.3                                                                          CH═CH                                                                              CH.sub.3                                                                              CH.sub.3                                                                            OCH.sub.3                                                                            N                                         6-CH.sub.3                                                                          CH═CH                                                                              CH.sub.3                                                                              OCH.sub.3                                                                           OCH.sub.3                                                                            N                                         6-CH.sub.3                                                                          CH═CH                                                                              CH.sub.3                                                                              CH.sub.3                                                                            CH.sub.3                                                                             N                                         6-CH.sub.3                                                                          CH═CH                                                                              C.sub.6 H.sub.5                                                                       CH.sub.3                                                                            CH.sub.3                                                                             CH                                        6-CH.sub.3                                                                          CH═CH                                                                              C.sub.6 H.sub.5                                                                       CH.sub.3                                                                            OCH.sub.3                                                                            CH                                        6-CH.sub.3                                                                          CH═CH                                                                              C.sub.6 H.sub.5                                                                       OCH.sub.3                                                                           OCH.sub.3                                                                            CH                                        6-CH.sub.3                                                                          CH═CH                                                                              C.sub.6 H.sub.5                                                                       Cl    OCH.sub.3                                                                            CH                                        6-CH.sub.3                                                                          CH═CH                                                                              C.sub.6 H.sub.5                                                                       CH.sub.3                                                                            OCH.sub.3                                                                            N                                         6-CH.sub.3                                                                          CH═CH                                                                              C.sub.6 H.sub.5                                                                       OCH.sub.3                                                                           OCH.sub.3                                                                            N                                         6-CH.sub.3                                                                          CH═CH                                                                              C.sub.6 H.sub.5                                                                       CH.sub.3                                                                            CH.sub.3                                                                             N                                         6-Cl  CH═CH                                                                              H       CH.sub.3                                                                            CH.sub.3                                                                             CH                                        6-Cl  CH═CH                                                                              H       CH.sub.3                                                                            OCH.sub.3                                                                            CH                                        6-Cl  CH═CH                                                                              H       OCH.sub.3                                                                           OCH.sub.3                                                                            CH                                        6-Cl  CH═CH                                                                              H       Cl    OCH.sub.3                                                                            CH                                        6-Cl  CH═CH                                                                              H       CH.sub.3                                                                            OCH.sub.3                                                                            N                                         6-Cl  CH═CH                                                                              H       OCH.sub.3                                                                           OCH.sub.3                                                                            N                                         6-Cl  CH═CH                                                                              H       CH.sub.3                                                                            CH.sub.3                                                                             N                                         6-Cl  CH═CH                                                                              CH.sub.3                                                                              CH.sub.3                                                                            CH.sub.3                                                                             CH                                        6-Cl  CH═CH                                                                              CH.sub.3                                                                              OCH.sub.3                                                                           CH.sub.3                                                                             CH                                        6-Cl  CH═CH                                                                              CH.sub.3                                                                              OCH.sub.3                                                                           OCH.sub.3                                                                            CH                                        6-Cl  CH═CH                                                                              CH.sub.3                                                                              Cl    OCH.sub.3                                                                            CH                                        6-Cl  CH═CH                                                                              CH.sub.3                                                                              CH.sub.3                                                                            OCH.sub.3                                                                            N                                         6-Cl  CH═CH                                                                              CH.sub.3                                                                              OCH.sub.3                                                                           OCH.sub.3                                                                            N                                         6-Cl  CH═CH                                                                              CH.sub.3                                                                              CH.sub.3                                                                            CH.sub.3                                                                             N                                         6-Cl  CH═CH                                                                              C.sub.6 H.sub.5                                                                       CH.sub.3                                                                            CH.sub.3                                                                             CH                                        6-Cl  CH═CH                                                                              C.sub.6 H.sub.5                                                                       CH.sub.3                                                                            OCH.sub.3                                                                            CH                                        6-Cl  CH═CH                                                                              C.sub.6 H.sub.5                                                                       OCH.sub.3                                                                           OCH.sub.3                                                                            CH                                        6-Cl  CH═CH                                                                              C.sub.6 H.sub.5                                                                       Cl    OCH.sub.3                                                                            CH                                        6-Cl  CH═CH                                                                              C.sub.6 H.sub.5                                                                       CH.sub.3                                                                            OCH.sub.3                                                                            N                                         6-Cl  CH═CH                                                                              C.sub.6 H.sub.5                                                                       OCH.sub.3                                                                           OCH.sub.3                                                                            N                                         6-Cl  CH═CH                                                                              C.sub.6 H.sub.5                                                                       CH.sub.3                                                                            CH.sub.3                                                                             N                                         ______________________________________                                    

                  TABLE 4a                                                        ______________________________________                                        General Formula 4a                                                            R.sub.1                                                                              J       R.sub.5                                                                              X      Y     Z     m.p.(°C.)                     ______________________________________                                        H      C═O H      CH.sub.3                                                                             CH.sub.3                                                                            CH                                         H      C═O H      CH.sub.3                                                                             OCH.sub.3                                                                           CH                                         H      C═O H      OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                         H      C═O H      Cl     OCH.sub.3                                                                           CH                                         H      C═O H      CH.sub.3                                                                             OCH.sub.3                                                                           N                                          H      C═O H      OCH.sub.3                                                                            OCH.sub.3                                                                           N                                          H      C═O H      CH.sub.3                                                                             CH.sub.3                                                                            N                                          H      C═O CH.sub.3                                                                             CH.sub.3                                                                             CH.sub.3                                                                            CH                                         H      C═O CH.sub.3                                                                             CH.sub.3                                                                             OCH.sub.3                                                                           CH                                         H      C═O CH.sub.3                                                                             OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                         H      C═O CH.sub.3                                                                             Cl     OCH.sub.3                                                                           CH                                         H      C═O CH.sub.3                                                                             CH.sub.3                                                                             OCH.sub.3                                                                           N                                          H      C═O CH.sub.3                                                                             OCH.sub.3                                                                            OCH.sub.3                                                                           N                                          H      C═O CH.sub.3                                                                             CH.sub.3                                                                             CH.sub.3                                                                            N                                          H      CH.sub.2                                                                              CH.sub.3                                                                             CH.sub.3                                                                             CH.sub.3                                                                            CH                                         H      CH.sub.2                                                                              CH.sub.3                                                                             CH.sub.3                                                                             OCH.sub.3                                                                           CH                                         H      CH.sub.2                                                                              CH.sub.3                                                                             OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                         H      CH.sub.2                                                                              CH.sub.3                                                                             Cl     OCH.sub.3                                                                           CH                                         H      CH.sub.2                                                                              CH.sub.3                                                                             CH.sub.3                                                                             OCH.sub.3                                                                           N                                          H      CH.sub.2                                                                              CH.sub.3                                                                             OCH.sub.3                                                                            OCH.sub.3                                                                           N                                          H      CH.sub.2                                                                              CH.sub.3                                                                             CH.sub.3                                                                             CH.sub.3                                                                            N                                          H      S       CH.sub.3                                                                             CH.sub.3                                                                             CH.sub.3                                                                            CH                                         H      S       CH.sub.3                                                                             CH.sub.3                                                                             OCH.sub.3                                                                           CH                                         H      S       CH.sub.3                                                                             OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                         H      S       CH.sub.3                                                                             Cl     OCH.sub.3                                                                           CH                                         H      S       CH.sub.3                                                                             CH.sub.3                                                                             OCH.sub.3                                                                           N                                          H      S       CH.sub.3                                                                             OCH.sub.3                                                                            OCH.sub.3                                                                           N                                          H      S       CH.sub.3                                                                             CH.sub.3                                                                             CH.sub.3                                                                            N                                          H      SO.sub.2                                                                              H      CH.sub.3                                                                             CH.sub.3                                                                            CH                                         H      SO.sub.2                                                                              H      CH.sub.3                                                                             OCH.sub.3                                                                           CH                                         H      SO.sub.2                                                                              H      OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                         H      SO.sub.2                                                                              H      Cl     OCH.sub.3                                                                           CH                                         H      SO.sub.2                                                                              H      CH.sub.3                                                                             OCH.sub.3                                                                           N                                          H      SO.sub.2                                                                              H      OCH.sub.3                                                                            OCH.sub.3                                                                           N                                          H      SO.sub.2                                                                              H      CH.sub.3                                                                             CH.sub.3                                                                            N                                          H      SO.sub.2                                                                              CH.sub.3                                                                             CH.sub.3                                                                             CH.sub.3                                                                            CH                                         H      SO.sub.2                                                                              CH.sub.3                                                                             CH.sub.3                                                                             OCH.sub.3                                                                           CH                                         H      SO.sub.2                                                                              CH.sub.3                                                                             OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                         H      SO.sub.2                                                                              CH.sub.3                                                                             Cl     OCH.sub.3                                                                           CH                                         H      SO.sub.2                                                                              CH.sub. 3                                                                            CH.sub.3                                                                             OCH.sub.3                                                                           N                                          H      SO.sub.2                                                                              CH.sub.3                                                                             OCH.sub.3                                                                            OCH.sub.3                                                                           N                                          H      SO.sub.2                                                                              CH.sub.3                                                                             CH.sub.3                                                                             CH.sub.3                                                                            N                                          H      O       CH.sub.3                                                                             CH.sub.3                                                                             CH.sub.3                                                                            CH                                         H      O       CH.sub.3                                                                             CH.sub.3                                                                             OCH.sub.3                                                                           CH                                         H      O       CH.sub.3                                                                             OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                         H      O       CH.sub.3                                                                             Cl     OCH.sub.3                                                                           CH                                         H      O       CH.sub.3                                                                             CH.sub.3                                                                             OCH.sub.3                                                                           N                                          H      O       CH.sub.3                                                                             OCH.sub.3                                                                            OCH.sub.3                                                                           N                                          H      O       CH.sub.3                                                                             CH.sub.3                                                                             CH.sub.3                                                                            N                                          6-CH.sub.3                                                                           C═O H      CH.sub.3                                                                             CH.sub.3                                                                            CH                                         6-CH.sub.3                                                                           C═O H      CH.sub.3                                                                             OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                           C═O H      OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                           C═O H      Cl     OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                           C═O H      CH.sub.3                                                                             OCH.sub.3                                                                           N                                          6-CH.sub.3                                                                           C═O H      OCH.sub.3                                                                            OCH.sub.3                                                                           N                                          6-CH.sub.3                                                                           C═O H      CH.sub.3                                                                             CH.sub.3                                                                            N                                          6-CH.sub.3                                                                           C═O CH.sub.3                                                                             CH.sub.3                                                                             CH.sub.3                                                                            CH                                         6-CH.sub.3                                                                           C═O CH.sub.3                                                                             CH.sub.3                                                                             OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                           C═O CH.sub.3                                                                             OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                           C═O CH.sub.3                                                                             Cl     OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                           C═O CH.sub.3                                                                             CH.sub.3                                                                             OCH.sub.3                                                                           N                                          6-CH.sub.3                                                                           C═O CH.sub.3                                                                             OCH.sub.3                                                                            OCH.sub.3                                                                           N                                          6-CH.sub.3                                                                           C═O CH.sub.3                                                                             CH.sub.3                                                                             CH.sub.3                                                                            N                                          6-CH.sub.3                                                                           CH.sub.2                                                                              CH.sub.3                                                                             CH.sub.3                                                                             CH.sub.3                                                                            CH                                         6-CH.sub.3                                                                           CH.sub.2                                                                              CH.sub.3                                                                             CH.sub.3                                                                             OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                           CH.sub.2                                                                              CH.sub.3                                                                             OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                           CH.sub.2                                                                              CH.sub.3                                                                             Cl     OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                           CH.sub.2                                                                              CH.sub.3                                                                             CH.sub.3                                                                             OCH.sub.3                                                                           N                                          6-CH.sub.3                                                                           CH.sub.2                                                                              CH.sub.3                                                                             OCH.sub.3                                                                            OCH.sub.3                                                                           N                                          6-CH.sub.3                                                                           CH.sub.2                                                                              CH.sub.3                                                                             CH.sub.3                                                                             CH.sub.3                                                                            N                                          6-CH.sub.3                                                                           S       CH.sub.3                                                                             CH.sub.3                                                                             CH.sub.3                                                                            CH                                         6-CH.sub.3                                                                           S       CH.sub.3                                                                             CH.sub.3                                                                             OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                           S       CH.sub.3                                                                             OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                           S       CH.sub.3                                                                             Cl     OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                           S       CH.sub.3                                                                             CH.sub.3                                                                             OCH.sub.3                                                                           N                                          6-CH.sub.3                                                                           S       CH.sub.3                                                                             OCH.sub.3                                                                            OCH.sub.3                                                                           N                                          6-CH.sub.3                                                                           S       CH.sub.3                                                                             CH.sub.3                                                                             CH.sub.3                                                                            N                                          5-NO.sub.2                                                                           C═O H      CH.sub.3                                                                             CH.sub.3                                                                            CH                                         5-NO.sub.2                                                                           C═O H      CH.sub.3                                                                             OCH.sub.3                                                                           CH                                         5-NO.sub.2                                                                           C═O H      OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                         5-NO.sub.2                                                                           C═O H      Cl     OCH.sub.3                                                                           CH                                         5-NO.sub.2                                                                           C═O H      CH.sub.3                                                                             OCH.sub.3                                                                           N                                          5-NO.sub.2                                                                           C═O H      OCH.sub.3                                                                            OCH.sub.3                                                                           N                                          5-NO.sub.2                                                                           C═O H      CH.sub.3                                                                             CH.sub.3                                                                            N                                          5-NO.sub.2                                                                           C═O CH.sub.3                                                                             CH.sub.3                                                                             CH.sub.3                                                                            CH                                         5-NO.sub.2                                                                           C═O CH.sub.3                                                                             CH.sub.3                                                                             OCH.sub.3                                                                           CH                                         5-NO.sub.2                                                                           C═O CH.sub.3                                                                             OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                         5-NO.sub.2                                                                           C═O CH.sub.3                                                                             Cl     OCH.sub.3                                                                           CH                                         5-NO.sub.2                                                                           C═O CH.sub.3                                                                             CH.sub.3                                                                             OCH.sub.3                                                                           N                                          5-NO.sub.2                                                                           C═O CH.sub.3                                                                             OCH.sub.3                                                                            OCH.sub.3                                                                           N                                          5-NO.sub.2                                                                           C═O CH.sub.3                                                                             CH.sub.3                                                                             CH.sub.3                                                                            N                                          5-NO.sub.2                                                                           CH.sub.2                                                                              CH.sub.3                                                                             CH.sub.3                                                                             CH.sub.3                                                                            CH                                         5-NO.sub.2                                                                           CH.sub.2                                                                              CH.sub.3                                                                             CH.sub.3                                                                             OCH.sub.3                                                                           CH                                         5-NO.sub.2                                                                           CH.sub.2                                                                              CH.sub.3                                                                             OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                         5-NO.sub.2                                                                           CH.sub.2                                                                              CH.sub.3                                                                             Cl     OCH.sub.3                                                                           CH                                         5-NO.sub.2                                                                           CH.sub.2                                                                              CH.sub.3                                                                             CH.sub.3                                                                             OCH.sub.3                                                                           N                                          5-NO.sub.2                                                                           CH.sub.2                                                                              CH.sub.3                                                                             OCH.sub.3                                                                            OCH.sub.3                                                                           N                                          5-NO.sub.2                                                                           CH.sub.2                                                                              CH.sub.3                                                                             CH.sub.3                                                                             CH.sub.3                                                                            N                                          5-NO.sub. 2                                                                          S       CH.sub.3                                                                             CH.sub.3                                                                             CH.sub.3                                                                            CH                                         5-NO.sub.2                                                                           S       CH.sub.3                                                                             CH.sub.3                                                                             OCH.sub.3                                                                           CH                                         5-NO.sub.2                                                                           S       CH.sub.3                                                                             OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                         5-NO.sub.2                                                                           S       CH.sub.3                                                                             Cl     OCH.sub.3                                                                           CH                                         5-NO.sub.2                                                                           S       CH.sub.3                                                                             CH.sub.3                                                                             OCH.sub.3                                                                           N                                          5-NO.sub.2                                                                           S       CH.sub.3                                                                             OCH.sub.3                                                                            OCH.sub.3                                                                           N                                          5-NO.sub.2                                                                           S       CH.sub.3                                                                             CH.sub.3                                                                             CH.sub.3                                                                            N                                          6-CH.sub.3                                                                           SO.sub.2                                                                              H      CH.sub.3                                                                             CH.sub.3                                                                            CH                                         6-CH.sub.3                                                                           SO.sub.2                                                                              H      CH.sub.3                                                                             OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                           SO.sub.2                                                                              H      OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                           SO.sub.2                                                                              H      Cl     OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                           SO.sub.2                                                                              H      CH.sub.3                                                                             OCH.sub.3                                                                           N                                          6-CH.sub.3                                                                           SO.sub.2                                                                              H      OCH.sub.3                                                                            OCH.sub.3                                                                           N                                          6-CH.sub.3                                                                           SO.sub.2                                                                              H      CH.sub.3                                                                             CH.sub.3                                                                            N                                          6-CH.sub.3                                                                           SO.sub.2                                                                              CH.sub.3                                                                             CH.sub.3                                                                             CH.sub.3                                                                            CH                                         6-CH.sub.3                                                                           SO.sub.2                                                                              CH.sub.3                                                                             CH.sub.3                                                                             OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                           SO.sub.2                                                                              CH.sub.3                                                                             OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                           SO.sub.2                                                                              CH.sub.3                                                                             Cl     OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                           SO.sub.2                                                                              CH.sub.3                                                                             CH.sub.3                                                                             OCH.sub.3                                                                           N                                          6-CH.sub.3                                                                           SO.sub.2                                                                              CH.sub.3                                                                             OCH.sub.3                                                                            OCH.sub. 3                                                                          N                                          6-CH.sub.3                                                                           SO.sub.2                                                                              CH.sub.3                                                                             CH.sub.3                                                                             CH.sub.3                                                                            N                                          6-CH.sub.3                                                                           O       CH.sub.3                                                                             CH.sub.3                                                                             CH.sub.3                                                                            CH                                         6-CH.sub.3                                                                           O       CH.sub.3                                                                             CH.sub.3                                                                             OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                           O       CH.sub.3                                                                             OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                           O       CH.sub.3                                                                             Cl     OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                           O       CH.sub.3                                                                             CH.sub.3                                                                             OCH.sub.3                                                                           N                                          6-CH.sub.3                                                                           O       CH.sub.3                                                                             OCH.sub.3                                                                            OCH.sub.3                                                                           N                                          6-CH.sub.3                                                                           O       CH.sub.3                                                                             CH.sub.3                                                                             CH.sub.3                                                                            N                                          ______________________________________                                    

                  TABLE 4b                                                        ______________________________________                                        General Formula 4b                                                            R.sub.1                                                                             G        R.sub.5 X     Y     Z     m.p.(°C.)                     ______________________________________                                        H     CH.sub.2 H       CH.sub.3                                                                            CH.sub.3                                                                            CH                                         H     CH.sub.2 H       CH.sub.3                                                                            OCH.sub.3                                                                           CH                                         H     CH.sub.2 H       OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                         H     CH.sub.2 H       Cl    OCH.sub.3                                                                           CH                                         H     CH.sub.2 H       CH.sub.3                                                                            OCH.sub.3                                                                           N                                          H     CH.sub.2 H       OCH.sub.3                                                                           OCH.sub.3                                                                           N                                          H     CH.sub.2 H       CH.sub.3                                                                            CH.sub.3                                                                            N                                          H     CH.sub.2 CH.sub.3                                                                              CH.sub.3                                                                            CH.sub.3                                                                            CH                                         H     CH.sub.2 CH.sub.3                                                                              CH.sub.3                                                                            OCH.sub.3                                                                           CH                                         H     CH.sub.2 CH.sub.3                                                                              OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                         H     CH.sub.2 CH.sub.3                                                                              Cl    OCH.sub.3                                                                           CH                                         H     CH.sub.2 CH.sub.3                                                                              CH.sub.3                                                                            OCH.sub.3                                                                           N                                          H     CH.sub.2 CH.sub.3                                                                              OCH.sub.3                                                                           OCH.sub.3                                                                           N                                          H     CH.sub.2 CH.sub.3                                                                              CH.sub.3                                                                            CH.sub.3                                                                            N                                          6-CH.sub.3                                                                          CH.sub.2 H       CH.sub.3                                                                            CH.sub.3                                                                            CH                                         6-CH.sub.3                                                                          CH.sub.2 H       CH.sub.3                                                                            OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                          CH.sub.2 H       OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                          CH.sub.2 H       Cl    OCH.sub. 3                                                                          CH                                         6-CH.sub.3                                                                          CH.sub.2 H       CH.sub.3                                                                            OCH.sub.3                                                                           N                                          6-CH.sub.3                                                                          CH.sub.2 H       OCH.sub.3                                                                           OCH.sub.3                                                                           N                                          6-CH.sub.3                                                                          CH.sub.2 H       CH.sub.3                                                                            CH.sub.3                                                                            N                                          6-CH.sub.3                                                                          CH.sub.2 CH.sub.3                                                                              CH.sub.3                                                                            CH.sub.3                                                                            CH                                         6-CH.sub.3                                                                          CH.sub.2 CH.sub.3                                                                              CH.sub.3                                                                            OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                          CH.sub.2 CH.sub.3                                                                              OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                          CH.sub.2 CH.sub.3                                                                              Cl    OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                          CH.sub.2 CH.sub.3                                                                              CH.sub.3                                                                            OCH.sub.3                                                                           N                                          6-CH.sub.3                                                                          CH.sub.2 CH.sub.3                                                                              OCH.sub.3                                                                           OCH.sub.3                                                                           N                                          6-CH.sub.3                                                                          CH.sub.2 CH.sub.3                                                                              CH.sub.3                                                                            CH.sub.3                                                                            N                                          H     CH.sub.2 CH.sub.2                                                                      H       CH.sub.3                                                                            CH.sub.3                                                                            CH                                         H     CH.sub.2 CH.sub.2                                                                      H       CH.sub.3                                                                            OCH.sub.3                                                                           CH                                         H     CH.sub.2 CH.sub.2                                                                      H       OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                         H     CH.sub.2 CH.sub.2                                                                      H       Cl    OCH.sub.3                                                                           CH                                         H     CH.sub.2 CH.sub.2                                                                      H       CH.sub.3                                                                            OCH.sub.3                                                                           N                                          H     CH.sub.2 CH.sub.2                                                                      H       OCH.sub.3                                                                           OCH.sub.3                                                                           N                                          H     CH.sub.2 CH.sub.2                                                                      H       CH.sub.3                                                                            CH.sub.3                                                                            N                                          H     CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              CH.sub.3                                                                            CH.sub.3                                                                            CH                                         H     CH.sub.2 CH.sub. 2                                                                     CH.sub.3                                                                              CH.sub.3                                                                            OCH.sub.3                                                                           CH                                         H     CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                         H     CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              Cl    OCH.sub.3                                                                           CH                                         H     CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              CH.sub.3                                                                            OCH.sub.3                                                                           N                                          H     CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              OCH.sub.3                                                                           OCH.sub.3                                                                           N                                          H     CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              CH.sub.3                                                                            CH.sub.3                                                                            N                                          6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                      H       CH.sub.3                                                                            CH.sub.3                                                                            CH                                         6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                      H       CH.sub.3                                                                            OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                      H       OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                      H       Cl    OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                      H       CH.sub.3                                                                            OCH.sub.3                                                                           N                                          6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                      H       OCH.sub.3                                                                           OCH.sub.3                                                                           N                                          6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                      H       CH.sub.3                                                                            CH.sub.3                                                                            N                                          6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              CH.sub.3                                                                            CH.sub.3                                                                            CH                                         6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              CH.sub.3                                                                            OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              Cl    OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              CH.sub.3                                                                            OCH.sub.3                                                                           N                                          6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              OCH.sub.3                                                                           OCH.sub.3                                                                           N                                          6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              CH.sub.3                                                                            CH.sub.3                                                                            N                                          H     CH═CH                                                                              H       CH.sub.3                                                                            CH.sub.3                                                                            CH                                         H     CH═CH                                                                              H       CH.sub.3                                                                            OCH.sub.3                                                                           CH                                         H     CH═CH                                                                              H       OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                         H     CH═CH                                                                              H       Cl    OCH.sub.3                                                                           CH                                         H     CH═CH                                                                              H       CH.sub.3                                                                            OCH.sub.3                                                                           N                                          H     CH═CH                                                                              H       OCH.sub.3                                                                           OCH.sub.3                                                                           N                                          H     CH═CH                                                                              H       CH.sub.3                                                                            CH.sub.3                                                                            N                                          H     CH═CH                                                                              CH.sub.3                                                                              CH.sub.3                                                                            CH.sub.3                                                                            CH                                         H     CH═CH                                                                              CH.sub.3                                                                              CH.sub.3                                                                            OCH.sub.3                                                                           CH                                         H     CH═CH                                                                              CH.sub.3                                                                              OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                         H     CH═CH                                                                              CH.sub.3                                                                              Cl    OCH.sub.3                                                                           CH                                         H     CH═CH                                                                              CH.sub.3                                                                              CH.sub.3                                                                            OCH.sub.3                                                                           N                                          H     CH═CH                                                                              CH.sub.3                                                                              OCH.sub.3                                                                           OCH.sub.3                                                                           N                                          H     CH═CH                                                                              CH.sub.3                                                                              CH.sub.3                                                                            CH.sub.3                                                                            N                                          6-CH.sub.3                                                                          CH═CH                                                                              H       CH.sub.3                                                                            CH.sub. 3                                                                           CH                                         6-CH.sub.3                                                                          CH═CH                                                                              H       CH.sub.3                                                                            OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                          CH═CH                                                                              H       OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                          CH═CH                                                                              H       Cl    OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                          CH═CH                                                                              H       CH.sub.3                                                                            OCH.sub.3                                                                           N                                          6-CH.sub.3                                                                          CH═CH                                                                              H       OCH.sub.3                                                                           OCH.sub.3                                                                           N                                          6-CH.sub.3                                                                          CH═CH                                                                              H       CH.sub.3                                                                            CH.sub.3                                                                            N                                          6-CH.sub.3                                                                          CH═CH                                                                              CH.sub.3                                                                              CH.sub.3                                                                            CH.sub.3                                                                            CH                                         6-CH.sub.3                                                                          CH═CH                                                                              CH.sub.3                                                                              CH.sub.3                                                                            OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                          CH═CH                                                                              CH.sub.3                                                                              OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                          CH═CH                                                                              CH.sub.3                                                                              Cl    OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                          CH═CH                                                                              CH.sub.3                                                                              CH.sub.3                                                                            OCH.sub.3                                                                           N                                          6-CH.sub.3                                                                          CH═CH                                                                              CH.sub.3                                                                              OCH.sub.3                                                                           OCH.sub.3                                                                           N                                          6-CH.sub.3                                                                          CH═CH                                                                              CH.sub.3                                                                              CH.sub.3                                                                            CH.sub.3                                                                            N                                          ______________________________________                                    

                  TABLE 5a                                                        ______________________________________                                        General Formula 5a                                                            R.sub.1                                                                             J       R.sub.12                                                                              X     Y      Z    m.p.(°C.)                      ______________________________________                                        H     C═O H       CH.sub.3                                                                            CH.sub.3                                                                             CH                                         H     C═O H       CH.sub.3                                                                            OCH.sub.3                                                                            CH                                         H     C═O H       OCH.sub.3                                                                           OCH.sub.3                                                                            CH                                         H     C═O H       Cl    OCH.sub.3                                                                            CH                                         H     C═O H       CH.sub.3                                                                            OCH.sub.3                                                                            N                                          H     C═O H       OCH.sub.3                                                                           OCH.sub.3                                                                            N                                          H     C═O H       CH.sub.3                                                                            CH.sub.3                                                                             N                                          H     C═O CH.sub.3                                                                              CH.sub.3                                                                            CH.sub.3                                                                             CH                                         H     C═O CH.sub.3                                                                              CH.sub.3                                                                            OCH.sub.3                                                                            CH                                         H     C═O CH.sub.3                                                                              OCH.sub.3                                                                           OCH.sub.3                                                                            CH                                         H     C═O CH.sub.3                                                                              Cl    OCH.sub.3                                                                            CH                                         H     C═O CH.sub.3                                                                              CH.sub.3                                                                            OCH.sub.3                                                                            N                                          H     C═O CH.sub.3                                                                              OCH.sub.3                                                                           OCH.sub.3                                                                            N                                          H     C═O CH.sub.3                                                                              CH.sub.3                                                                            CH.sub.3                                                                             N                                          H     CH.sub.2                                                                              CH.sub.3                                                                              CH    CH.sub.3                                                                             CH                                         H     CH.sub.2                                                                              CH.sub.3                                                                              CH.sub.3                                                                            OCH.sub.3                                                                            CH                                         H     CH.sub.2                                                                              CH.sub.3                                                                              OCH.sub.3                                                                           OCH.sub.3                                                                            CH                                         H     CH.sub.2                                                                              CH.sub.3                                                                              Cl    OCH.sub.3                                                                            CH                                         H     CH.sub.2                                                                              CH.sub.3                                                                              CH.sub.3                                                                            OCH.sub.3                                                                            N                                          H     CH.sub.2                                                                              CH.sub.3                                                                              OCH.sub.3                                                                           OCH.sub.3                                                                            N                                          H     CH.sub.2                                                                              CH.sub.3                                                                              CH.sub.3                                                                            CH.sub.3                                                                             N                                          H     S       CH.sub.3                                                                              CH.sub.3                                                                            CH.sub.3                                                                             CH                                         H     S       CH.sub.3                                                                              CH.sub.3                                                                            OCH.sub.3                                                                            CH                                         H     S       CH.sub.3                                                                              OCH.sub.3                                                                           OCH.sub.3                                                                            CH                                         H     S       CH.sub.3                                                                              Cl    OCH.sub.3                                                                            CH                                         H     S       CH.sub.3                                                                              CH.sub.3                                                                            OCH.sub.3                                                                            N                                          H     S       CH.sub.3                                                                              OCH.sub.3                                                                           OCH.sub.3                                                                            N                                          H     S       CH.sub.3                                                                              CH.sub.3                                                                            CH.sub.3                                                                             N                                          H     SO.sub.2                                                                              CH.sub.3                                                                              CH.sub.3                                                                            CH.sub.3                                                                             CH                                         H     SO.sub.2                                                                              CH.sub.3                                                                              CH.sub.3                                                                            OCH.sub.3                                                                            CH                                         H     SO.sub.2                                                                              CH.sub.3                                                                              OCH.sub.3                                                                           OCH.sub.3                                                                            CH                                         H     SO.sub.2                                                                              CH.sub.3                                                                              Cl    OCH.sub.3                                                                            CH                                         H     SO.sub.2                                                                              CH.sub.3                                                                              CH.sub.3                                                                            OCH.sub.3                                                                            N                                          H     SO.sub.2                                                                              CH      OCH.sub.3                                                                           OCH.sub.3                                                                            N                                          H     SO.sub.2                                                                              CH.sub.3                                                                              CH.sub.3                                                                            CH.sub.3                                                                             N                                          H     NH      CH.sub.3                                                                              CH    CH.sub.3                                                                             CH                                         H     NH      CH.sub.3                                                                              CH.sub.3                                                                            OCH.sub.3                                                                            CH                                         H     NH      CH.sub.3                                                                              OCH.sub.3                                                                           OCH.sub.3                                                                            CH                                         H     NH      CH.sub.3                                                                              Cl    OCH.sub.3                                                                            CH                                         H     NH      CH.sub.3                                                                              CH.sub. 3                                                                           OCH.sub.3                                                                            N                                          H     NH      CH.sub.3                                                                              OCH.sub.3                                                                           OCH.sub.3                                                                            N                                          H     NH      CH.sub.3                                                                              CH.sub.3                                                                            CH.sub.3                                                                             N                                          H     O       CH.sub.3                                                                              CH.sub.3                                                                            CH.sub.3                                                                             CH                                         H     O       CH.sub.3                                                                              CH.sub.3                                                                            OCH.sub.3                                                                            CH                                         H     O       CH.sub.3                                                                              OCH.sub.3                                                                           OCH.sub.3                                                                            CH                                         H     O       CH.sub.3                                                                              Cl    OCH.sub.3                                                                            CH                                         H     O       CH.sub.3                                                                              CH.sub.3                                                                            OCH.sub.3                                                                            N                                          H     O       CH.sub.3                                                                              OCH.sub.3                                                                           OCH.sub.3                                                                            N                                          H     O       CH.sub.3                                                                              CH.sub.3                                                                            CH.sub.3                                                                             N                                          6-Cl  C═O H       CH.sub.3                                                                            CH.sub.3                                                                             CH                                         6-Cl  C═O H       CH.sub.3                                                                            OCH.sub.3                                                                            CH                                         6-Cl  C═O H       OCH.sub.3                                                                           OCH.sub.3                                                                            CH                                         6-Cl  C═O H       Cl    OCH.sub.3                                                                            CH                                         6-Cl  C═O H       CH.sub.3                                                                            OCH.sub.3                                                                            N                                          6-Cl  C═O H       OCH.sub.3                                                                           OCH.sub.3                                                                            N                                          6-Cl  C═O H       CH.sub.3                                                                            CH.sub.3                                                                             N                                          6-Cl  C═O CH.sub.3                                                                              CH.sub.3                                                                            CH.sub.3                                                                             CH                                         6-Cl  C═O CH.sub.3                                                                              CH.sub.3                                                                            OCH.sub.3                                                                            CH                                         6-Cl  C═O CH.sub.3                                                                              OCH.sub.3                                                                           OCH.sub.3                                                                            CH                                         6-Cl  C═O CH.sub.3                                                                              Cl    OCH.sub.3                                                                            CH                                         6-Cl  C═O CH.sub.3                                                                              CH.sub.3                                                                            OCH.sub.3                                                                            N                                          6-Cl  C═O CH.sub.3                                                                              OCH.sub.3                                                                           OCH.sub.3                                                                            N                                          6-Cl  C═O CH.sub.3                                                                              CH.sub.3                                                                            CH.sub.3                                                                             N                                          6-Cl  CH.sub.2                                                                              CH.sub.3                                                                              CH.sub.3                                                                            CH.sub.3                                                                             CH                                         6-Cl  CH.sub.2                                                                              CH.sub.3                                                                              CH.sub.3                                                                            OCH.sub.3                                                                            CH                                         6-Cl  CH.sub.2                                                                              CH.sub.3                                                                              OCH.sub.3                                                                           OCH.sub.3                                                                            CH                                         6-Cl  CH.sub.2                                                                              CH.sub.3                                                                              Cl    OCH.sub.3                                                                            CH                                         6-Cl  CH.sub.2                                                                              CH.sub.3                                                                              CH.sub.3                                                                            OCH.sub.3                                                                            N                                          6-Cl  CH.sub.2                                                                              CH.sub.3                                                                              OCH.sub.3                                                                           OCH.sub.3                                                                            N                                          6-Cl  CH.sub.2                                                                              CH.sub.3                                                                              CH.sub.3                                                                            CH.sub.3                                                                             N                                          6-Cl  S       CH.sub.3                                                                              CH.sub.3                                                                            CH.sub.3                                                                             CH                                         6-Cl  S       CH.sub.3                                                                              CH.sub.3                                                                            OCH.sub.3                                                                            CH                                         6-Cl  S       CH.sub.3                                                                              OCH.sub.3                                                                           OCH.sub.3                                                                            CH                                         6-Cl  S       CH.sub.3                                                                              Cl    OCH.sub.3                                                                            CH                                         6-Cl  S       CH.sub.3                                                                              CH.sub.3                                                                            OCH.sub.3                                                                            N                                          6-Cl  S       CH.sub.3                                                                              OCH.sub.3                                                                           OCH.sub.3                                                                            N                                          6-Cl  S       CH.sub.3                                                                              CH.sub.3                                                                            CH.sub.3                                                                             N                                          6-Cl  SO.sub.2                                                                              CH.sub.3                                                                              CH.sub.3                                                                            CH.sub.3                                                                             CH                                         6-Cl  SO.sub.2                                                                              CH.sub.3                                                                              CH.sub.3                                                                            OCH.sub.3                                                                            CH                                         6-Cl  SO.sub.2                                                                              CH.sub.3                                                                              OCH.sub.3                                                                           OCH.sub.3                                                                            CH                                         6-Cl  SO.sub.2                                                                              CH.sub.3                                                                              Cl    OCH.sub.3                                                                            CH                                         6-Cl  SO.sub.2                                                                              CH.sub.3                                                                              CH.sub.3                                                                            OCH.sub.3                                                                            N                                          6-Cl  SO.sub.2                                                                              CH      OCH.sub.3                                                                           OCH.sub.3                                                                            N                                          6-Cl  SO.sub.2                                                                              CH.sub.3                                                                              CH.sub.3                                                                            CH.sub.3                                                                             N                                          6-Cl  NH      CH.sub.3                                                                              CH    CH.sub.3                                                                             CH                                         6-Cl  NH      CH.sub.3                                                                              CH.sub.3                                                                            OCH.sub.3                                                                            CH                                         6-Cl  NH      CH.sub.3                                                                              OCH.sub.3                                                                           OCH.sub.3                                                                            CH                                         6-Cl  NH      CH.sub.3                                                                              Cl    OCH.sub.3                                                                            CH                                         6-Cl  NH      CH.sub.3                                                                              CH.sub.3                                                                            OCH.sub.3                                                                            N                                          6-Cl  NH      CH.sub.3                                                                              OCH.sub.3                                                                           OCH.sub.3                                                                            N                                          6-Cl  NH      CH.sub.3                                                                              CH.sub.3                                                                            CH.sub.3                                                                             N                                          6-Cl  O       CH.sub.3                                                                              CH.sub.3                                                                            CH.sub.3                                                                             CH                                         6-Cl  O       CH.sub.3                                                                              CH.sub.3                                                                            OCH.sub.3                                                                            CH                                         6-Cl  O       CH.sub.3                                                                              OCH.sub.3                                                                           OCH.sub.3                                                                            CH                                         6-Cl  O       CH.sub.3                                                                              Cl    OCH.sub.3                                                                            CH                                         6-Cl  O       CH.sub.3                                                                              CH.sub.3                                                                            OCH.sub.3                                                                            N                                          6-Cl  O       CH.sub.3                                                                              OCH.sub.3                                                                           OCH.sub.3                                                                            N                                          6-Cl  O       CH.sub.3                                                                              CH.sub.3                                                                            CH.sub.3                                                                             N                                          ______________________________________                                    

                  TABLE 5b                                                        ______________________________________                                        General Formula 5b                                                            R.sub.1                                                                             G        R.sub.12                                                                              X     Y      Z    m.p. (°C.)                    ______________________________________                                        H     CH.sub.2 H       CH.sub.3                                                                            CH.sub.3                                                                             CH                                        H     CH.sub.2 H       CH.sub.3                                                                            OCH.sub.3                                                                            CH                                        H     CH.sub.2 H       OCH.sub.3                                                                           OCH.sub.3                                                                            CH                                        H     CH.sub.2 H       Cl    OCH.sub.3                                                                            CH                                        H     CH.sub.2 H       CH.sub.3                                                                            OCH.sub.3                                                                            N                                         H     CH.sub.2 H       OCH.sub.3                                                                           OCH.sub.3                                                                            N                                         H     CH.sub.2 H       CH.sub.3                                                                            CH.sub.3                                                                             N                                         H     CH.sub.2 CH.sub.3                                                                              CH.sub.3                                                                            CH.sub.3                                                                             CH                                        H     CH.sub.2 CH.sub.3                                                                              CH.sub.3                                                                            OCH.sub.3                                                                            CH                                        H     CH.sub.2 CH.sub.3                                                                              OCH.sub.3                                                                           OCH.sub.3                                                                            CH                                        H     CH.sub.2 CH.sub.3                                                                              Cl    OCH.sub.3                                                                            CH                                        H     CH.sub.2 CH.sub.3                                                                              CH.sub.3                                                                            OCH.sub.3                                                                            N                                         H     CH.sub.2 CH.sub.3                                                                              OCH.sub.3                                                                           OCH.sub.3                                                                            N                                         H     CH.sub.2 CH.sub.3                                                                              CH.sub.3                                                                            CH.sub.3                                                                             N                                         6-Cl  CH.sub.2 H       CH.sub.3                                                                            CH.sub.3                                                                             CH                                        6-Cl  CH.sub.2 H       CH.sub.3                                                                            OCH.sub.3                                                                            CH                                        6-Cl  CH.sub.2 H       OCH.sub.3                                                                           OCH.sub.3                                                                            CH                                        6-Cl  CH.sub.2 H       Cl    OCH.sub.3                                                                            CH                                        6-Cl  CH.sub.2 H       CH.sub.3                                                                            OCH.sub.3                                                                            N                                         6-Cl  CH.sub.2 H       OCH.sub.3                                                                           OCH.sub.3                                                                            N                                         6-Cl  CH.sub.2 H       CH.sub.3                                                                            CH.sub.3                                                                             N                                         6-Cl  CH.sub.2 CH.sub.3                                                                              CH.sub.3                                                                            CH.sub.3                                                                             CH                                        6-Cl  CH.sub.2 CH.sub.3                                                                              CH.sub.3                                                                            OCH.sub.3                                                                            CH                                        6-Cl  CH.sub.2 CH.sub.3                                                                              OCH.sub.3                                                                           OCH.sub.3                                                                            CH                                        6-Cl  CH.sub.2 CH.sub.3                                                                              Cl    OCH.sub.3                                                                            CH                                        6-Cl  CH.sub.2 CH.sub.3                                                                              CH.sub.3                                                                            OCH.sub.3                                                                            N                                         6-Cl  CH.sub.2 CH.sub.3                                                                              OCH.sub.3                                                                           OCH.sub.3                                                                            N                                         6-Cl  CH.sub.2 CH.sub.3                                                                              CH.sub.3                                                                            CH.sub.3                                                                             N                                         H     CH.sub.2 CH.sub.2                                                                      H       CH.sub.3                                                                            CH.sub.3                                                                             CH                                        H     CH.sub.2 CH.sub.2                                                                      H       CH.sub.3                                                                            OCH.sub.3                                                                            CH                                        H     CH.sub.2 CH.sub.2                                                                      H       OCH.sub.3                                                                           OCH.sub.3                                                                            CH                                        H     CH.sub.2 CH.sub.2                                                                      H       Cl    OCH.sub.3                                                                            CH                                        H     CH.sub.2 CH.sub.2                                                                      H       CH.sub.3                                                                            OCH.sub.3                                                                            N                                         H     CH.sub.2 CH.sub.2                                                                      H       OCH.sub.3                                                                           OCH.sub.3                                                                            N                                         H     CH.sub.2 CH.sub.2                                                                      H       CH.sub.3                                                                            CH.sub.3                                                                             N                                         H     CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              CH.sub.3                                                                            CH.sub.3                                                                             CH                                        H     CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              CH.sub.3                                                                            OCH.sub.3                                                                            CH                                        H     CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              OCH.sub.3                                                                           OCH.sub.3                                                                            CH                                        H     CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              Cl    OCH.sub.3                                                                            CH                                        H     CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              CH.sub.3                                                                            OCH.sub.3                                                                            N                                         H     CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              OCH.sub.3                                                                           OCH.sub.3                                                                            N                                         H     CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              CH.sub.3                                                                            CH.sub.3                                                                             N                                         6-Cl  CH.sub.2 CH.sub.2                                                                      H       CH.sub.3                                                                            CH.sub.3                                                                             CH                                        6-Cl  CH.sub.2 CH.sub.2                                                                      H       CH.sub.3                                                                            OCH.sub.3                                                                            CH                                        6-Cl  CH.sub.2 CH.sub.2                                                                      H       OCH.sub.3                                                                           OCH.sub.3                                                                            CH                                        6-Cl  CH.sub.2 CH.sub.2                                                                      H       Cl    OCH.sub.3                                                                            CH                                        6-Cl  CH.sub.2 CH.sub.2                                                                      H       CH.sub.3                                                                            OCH.sub.3                                                                            N                                         6-Cl  CH.sub.2 CH.sub.2                                                                      H       OCH.sub.3                                                                           OCH.sub.3                                                                            N                                         6-Cl  CH.sub.2 CH.sub.2                                                                      H       CH.sub.3                                                                            CH.sub.3                                                                             N                                         6-Cl  CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              CH.sub.3                                                                            CH.sub.3                                                                             CH                                        6-Cl  CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              CH.sub.3                                                                            OCH.sub.3                                                                            CH                                        6-Cl  CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              OCH.sub.3                                                                           OCH.sub.3                                                                            CH                                        6-Cl  CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              Cl    OCH.sub.3                                                                            CH                                        6-Cl  CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              CH.sub.3                                                                            OCH.sub.3                                                                            N                                         6-Cl  CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              OCH.sub.3                                                                           OCH.sub.3                                                                            N                                         6-Cl  CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              CH.sub.3                                                                            CH.sub.3                                                                             N                                         H     CH═CH                                                                              H       CH.sub.3                                                                            CH.sub.3                                                                             CH                                        H     CH═CH                                                                              H       CH.sub.3                                                                            OCH.sub.3                                                                            CH                                        H     CH═CH                                                                              H       OCH.sub.3                                                                           OCH.sub.3                                                                            CH                                        H     CH═CH                                                                              H       Cl    OCH.sub.3                                                                            CH                                        H     CH═CH                                                                              H       CH.sub.3                                                                            OCH.sub.3                                                                            N                                         H     CH═CH                                                                              H       OCH.sub.3                                                                           OCH.sub.3                                                                            N                                         H     CH═CH                                                                              H       CH.sub.3                                                                            CH.sub.3                                                                             N                                         H     CH═CH                                                                              CH.sub.3                                                                              CH.sub.3                                                                            CH.sub.3                                                                             CH                                        H     CH═CH                                                                              CH.sub.3                                                                              CH.sub.3                                                                            OCH.sub.3                                                                            CH                                        H     CH═CH                                                                              CH.sub.3                                                                              OCH.sub.3                                                                           OCH.sub.3                                                                            CH                                        H     CH═CH                                                                              CH.sub.3                                                                              Cl    OCH.sub.3                                                                            CH                                        H     CH═CH                                                                              CH.sub.3                                                                              CH.sub.3                                                                            OCH.sub.3                                                                            N                                         H     CH═CH                                                                              CH.sub.3                                                                              OCH.sub.3                                                                           OCH.sub.3                                                                            N                                         H     CH═CH                                                                              CH.sub.3                                                                              CH.sub.3                                                                            CH.sub.3                                                                             N                                         6-Cl  CH═CH                                                                              H       CH.sub.3                                                                            CH.sub.3                                                                             CH                                        6-Cl  CH═CH                                                                              H       CH.sub.3                                                                            OCH.sub.3                                                                            CH                                        6-Cl  CH═CH                                                                              H       OCH.sub.3                                                                           OCH.sub.3                                                                            CH                                        6-Cl  CH═CH                                                                              H       Cl    OCH.sub.3                                                                            CH                                        6-Cl  CH═CH                                                                              H       CH.sub.3                                                                            OCH.sub.3                                                                            N                                         6-Cl  CH═CH                                                                              H       OCH.sub.3                                                                           OCH.sub.3                                                                            N                                         6-Cl  CH═CH                                                                              H       CH.sub.3                                                                            CH.sub.3                                                                             N                                         6-Cl  CH═CH                                                                              CH.sub.3                                                                              CH.sub.3                                                                            CH.sub.3                                                                             CH                                        6-Cl  CH═CH                                                                              CH.sub.3                                                                              CH.sub.3                                                                            OCH.sub.3                                                                            CH                                        6-Cl  CH═CH                                                                              CH.sub.3                                                                              OCH.sub.3                                                                           OCH.sub.3                                                                            CH                                        6-Cl  CH═CH                                                                              CH.sub.3                                                                              Cl    OCH.sub.3                                                                            CH                                        6-Cl  CH═CH                                                                              CH.sub.3                                                                              CH.sub.3                                                                            OCH.sub.3                                                                            N                                         6-Cl  CH═CH                                                                              CH.sub.3                                                                              OCH.sub.3                                                                           OCH.sub.3                                                                            N                                         6-Cl  CH═CH                                                                              CH.sub.3                                                                              CH.sub.3                                                                            CH.sub.3                                                                             N                                         ______________________________________                                    

                  TABLE 6                                                         ______________________________________                                        General Formula 6                                                             R.sub.1  J        X        Y      Z    m.p. (°C.)                      ______________________________________                                        H        C═O  CH.sub.3 CH.sub.3                                                                             CH                                          H        C═O  CH.sub.3 OCH.sub.3                                                                            CH                                          H        C═O  OCH.sub.3                                                                              OCH.sub.3                                                                            CH                                          H        C═O  Cl       OCH.sub.3                                                                            CH                                          H        C═O  CH.sub.3 OCH.sub.3                                                                            N                                           H        C═O  OCH.sub.3                                                                              OCH.sub.3                                                                            N                                           H        C═O  CH.sub.3 CH.sub.3                                                                             N                                           H        SO.sub.2 CH.sub.3 CH.sub.3                                                                             CH                                          H        SO.sub.2 CH.sub.3 OCH.sub.3                                                                            CH                                          H        SO.sub.2 OCH.sub.3                                                                              OCH.sub.3                                                                            CH                                          H        SO.sub.2 Cl       OCH.sub.3                                                                            CH                                          H        SO.sub.2 CH.sub.3 OCH.sub.3                                                                            N                                           H        SO.sub.2 OCH.sub.3                                                                              OCH.sub.3                                                                            N                                           H        SO.sub.2 CH.sub.3 CH.sub.3                                                                             N                                           H        NH       CH       CH.sub.3                                                                             CH                                          H        NH       CH.sub.3 OCH.sub.3                                                                            CH                                          H        NH       OCH.sub.3                                                                              OCH.sub.3                                                                            CH                                          H        NH       Cl       OCH.sub.3                                                                            CH                                          H        NH       CH.sub.3 OCH.sub.3                                                                            N                                           H        NH       OCH.sub.3                                                                              OCH.sub.3                                                                            N                                           H        NH       CH.sub.3 CH.sub.3                                                                             N                                           H        O        CH.sub.3 CH.sub.3                                                                             CH                                          H        O        CH.sub.3 OCH.sub.3                                                                            CH                                          H        O        OCH.sub.3                                                                              OCH.sub.3                                                                            CH                                          H        O        Cl       OCH.sub.3                                                                            CH                                          H        O        CH.sub.3 OCH.sub.3                                                                            N                                           H        O        OCH.sub.3                                                                              OCH.sub.3                                                                            N                                           H        O        CH.sub.3 CH.sub.3                                                                             N                                           6-Cl     C═O  CH.sub.3 CH.sub.3                                                                             CH                                          6-Cl     C═O  CH.sub.3 OCH.sub.3                                                                            CH                                          6-Cl     C═O  OCH.sub.3                                                                              OCH.sub.3                                                                            CH                                          6-Cl     C═O  Cl       OCH.sub.3                                                                            CH                                          6-Cl     C═O  CH.sub.3 OCH.sub.3                                                                            N                                           6-Cl     C═O  OCH.sub.3                                                                              OCH.sub.3                                                                            N                                           6-Cl     C═O  CH.sub.3 CH.sub.3                                                                             N                                           6-Cl     SO.sub.2 CH.sub.3 CH.sub.3                                                                             CH                                          6-Cl     SO.sub.2 CH.sub.3 OCH.sub.3                                                                            CH                                          6-Cl     SO.sub.2 OCH.sub.3                                                                              OCH.sub.3                                                                            CH                                          6-Cl     SO.sub.2 Cl       OCH.sub.3                                                                            CH                                          6-Cl     SO.sub.2 CH.sub.3 OCH.sub.3                                                                            N                                           6-Cl     SO.sub.2 OCH.sub.3                                                                              OCH.sub.3                                                                            N                                           6-Cl     SO.sub.2 CH.sub.3 CH.sub.3                                                                             N                                           6-Cl     NH       CH       CH.sub.3                                                                             CH                                          6-Cl     NH       CH.sub.3 OCH.sub.3                                                                            CH                                          6-Cl     NH       OCH.sub.3                                                                              OCH.sub.3                                                                            CH                                          6-Cl     NH       Cl       OCH.sub.3                                                                            CH                                          6-Cl     NH       CH.sub.3 OCH.sub.3                                                                            N                                           6-Cl     NH       OCH.sub.3                                                                              OCH.sub.3                                                                            N                                           6-Cl     NH       CH.sub.3 CH.sub.3                                                                             N                                           6-Cl     O        CH.sub.3 CH.sub.3                                                                             CH                                          6-Cl     O        CH.sub.3 OCH.sub.3                                                                            CH                                          6-Cl     O        OCH.sub.3                                                                              OCH.sub.3                                                                            CH                                          6-Cl     O        Cl       OCH.sub.3                                                                            CH                                          6-Cl     O        CH.sub.3 OCH.sub.3                                                                            N                                           6-Cl     O        OCH.sub.3                                                                              OCH.sub.3                                                                            N                                           6-Cl     O        CH.sub.3 CH.sub.3                                                                             N                                           5-SCH.sub.3                                                                            C═O  CH.sub.3 CH.sub.3                                                                             CH                                          5-SCH.sub.3                                                                            C═O  CH.sub.3 OCH.sub.3                                                                            CH                                          5-SCH.sub.3                                                                            C═O  OCH.sub.3                                                                              OCH.sub.3                                                                            CH                                          5-SCH.sub.3                                                                            C═O  Cl       OCH.sub.3                                                                            CH                                          5-SCH.sub.3                                                                            C═O  CH.sub.3 OCH.sub.3                                                                            N                                           5-SCH.sub.3                                                                            C═O  OCH.sub.3                                                                              OCH.sub.3                                                                            N                                           5-SCH.sub.3                                                                            C═O  CH.sub.3 CH.sub.3                                                                             N                                           5-SCH.sub.3                                                                            SO.sub.2 CH.sub.3 CH.sub.3                                                                             CH                                          5-SCH.sub.3                                                                            SO.sub.2 CH.sub.3 OCH.sub.3                                                                            CH                                          5-SCH.sub.3                                                                            SO.sub.2 OCH.sub.3                                                                              OCH.sub.3                                                                            CH                                          5-SCH.sub.3                                                                            SO.sub.2 Cl       OCH.sub.3                                                                            CH                                          5-SCH.sub.3                                                                            SO.sub.2 CH.sub.3 OCH.sub.3                                                                            N                                           5-SCH.sub.3                                                                            SO.sub.2 OCH.sub.3                                                                              OCH.sub.3                                                                            N                                           5-SCH.sub.3                                                                            SO.sub.2 CH.sub.3 CH.sub. 3                                                                            N                                           5-SCH.sub.3                                                                            NH       CH       CH.sub.3                                                                             CH                                          5-SCH.sub.3                                                                            NH       CH.sub.3 OCH.sub.3                                                                            CH                                          5-SCH.sub.3                                                                            NH       OCH.sub.3                                                                              OCH.sub.3                                                                            CH                                          5-SCH.sub.3                                                                            NH       Cl       OCH.sub.3                                                                            CH                                          5-SCH.sub.3                                                                            NH       CH.sub.3 OCH.sub.3                                                                            N                                           5-SCH.sub.3                                                                            NH       OCH.sub.3                                                                              OCH.sub.3                                                                            N                                           5-SCH.sub.3                                                                            NH       CH.sub.3 CH.sub.3                                                                             N                                           5-SCH.sub.3                                                                            O        CH.sub.3 CH.sub.3                                                                             CH                                          5-SCH.sub.3                                                                            O        CH.sub.3 OCH.sub.3                                                                            CH                                          5-SCH.sub.3                                                                            O        OCH.sub.3                                                                              OCH.sub.3                                                                            CH                                          5-SCH.sub.3                                                                            O        Cl       OCH.sub.3                                                                            CH                                          5-SCH.sub.3                                                                            O        CH.sub.3 OCH.sub.3                                                                            N                                           5-SCH.sub.3                                                                            O        OCH.sub.3                                                                              OCH.sub.3                                                                            N                                           5-SCH.sub.3                                                                            O        CH.sub.3 CH.sub.3                                                                             N                                           ______________________________________                                    

                  TABLE 7                                                         ______________________________________                                        General Formula 7                                                                                                           m.p.                            R.sub.1                                                                              J       R.sub.9                                                                              R.sub.13                                                                             X     Y     Z    (°C.)                    ______________________________________                                        H      C═O H      OCH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                                                                            CH                                   H      C═O H      OCH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   H      C═O H      OCH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   H      C═O H      OCH.sub.3                                                                            Cl    OCH.sub.3                                                                           CH                                   H      C═O H      OCH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           N                                    H      C═O H      OCH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    H      C═O H      OCH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                                                                            N                                    H      C═O CH.sub.3                                                                             SCH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                                                                            CH                                   H      C═O CH.sub.3                                                                             SCH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   H      C═O CH.sub.3                                                                             SCH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   H      C═O CH.sub.3                                                                             SCH.sub.3                                                                            Cl    OCH.sub.3                                                                           CH                                   H      C═O CH.sub.3                                                                             SCH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           N                                    H      C═O CH.sub.3                                                                             SCH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    H      C═O CH.sub.3                                                                             SCH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                                                                            N                                    H      SO.sub.2                                                                              CH.sub.3                                                                             OCH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                                                                            CH                                   H      SO.sub.2                                                                              CH.sub.3                                                                             OCH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   H      SO.sub.2                                                                              CH.sub.3                                                                             OCH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   H      SO.sub.2                                                                              CH.sub.3                                                                             OCH.sub.3                                                                            Cl    OCH.sub.3                                                                           CH                                   H      SO.sub.2                                                                              CH.sub.3                                                                             OCH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           N                                    H      SO.sub.2                                                                              CH.sub.3                                                                             OCH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    H      SO.sub.2                                                                              CH.sub.3                                                                             OCH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                                                                            N                                    H      C═O H      CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            CH                                   H      C═O H      CH.sub.3                                                                             CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   H      C═O H      CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   H      C═O H      CH.sub.3                                                                             Cl    OCH.sub.3                                                                           CH                                   H      C═O H      CH.sub.3                                                                             CH.sub.3                                                                            OCH.sub.3                                                                           N                                    H      C═O H      CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    H      C═O H      CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            N                                    H      SO.sub.2                                                                              H      CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            CH                                   H      SO.sub.2                                                                              H      CH.sub.3                                                                             CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   H      SO.sub.2                                                                              H      CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   H      SO.sub.2                                                                              H      CH.sub.3                                                                             Cl    OCH.sub.3                                                                           CH                                   H      SO.sub.2                                                                              H      CH.sub.3                                                                             CH.sub.3                                                                            OCH.sub.3                                                                           N                                    H      SO.sub.2                                                                              H      CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    H      SO.sub.2                                                                              H      CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            N                                    H      CH.sub.2                                                                              H      OCH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                                                                            CH                                   H      CH.sub.2                                                                              H      OCH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   H      CH.sub.2                                                                              H      OCH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   H      CH.sub.2                                                                              H      OCH.sub.3                                                                            Cl    OCH.sub.3                                                                           CH                                   H      CH.sub.2                                                                              H      OCH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           N                                    H      CH.sub.2                                                                              H      OCH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    H      CH.sub.2                                                                              H      OCH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                                                                            N                                    H      CH.sub.2                                                                              CH.sub.3                                                                             SCH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                                                                            CH                                   H      CH.sub.2                                                                              CH.sub.3                                                                             SCH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   H      CH.sub.2                                                                              CH.sub.3                                                                             SCH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   H      CH.sub.2                                                                              CH.sub.3                                                                             SCH.sub.3                                                                            Cl    OCH.sub.3                                                                           CH                                   H      CH.sub.2                                                                              CH.sub.3                                                                             SCH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           N                                    H      CH.sub.2                                                                              CH.sub.3                                                                             SCH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    H      CH.sub.2                                                                              CH.sub.3                                                                             SCH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                                                                            N                                    H      CH.sub.2                                                                              CH.sub.3                                                                             CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            CH                                   H      CH.sub.2                                                                              CH.sub.3                                                                             CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            CH                                   H      CH.sub.2                                                                              CH.sub.3                                                                             CH.sub.3                                                                             CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   H      CH.sub.2                                                                              CH.sub.3                                                                             CH.sub.3                                                                             OCH.sub.3                                                                           Cl    CH                                   H      CH.sub.2                                                                              CH.sub.3                                                                             CH.sub.3                                                                             CH.sub.3                                                                            OCH.sub.3                                                                           N                                    H      CH.sub.2                                                                              CH.sub.3                                                                             CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    H      CH.sub.2                                                                              CH.sub.3                                                                             CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            N                                    H      O       H      CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            CH                                   H      O       H      CH.sub.3                                                                             CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   H      O       H      CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   H      O       H      CH.sub.3                                                                             Cl    OCH.sub.3                                                                           CH                                   H      O       H      CH.sub.3                                                                             CH.sub.3                                                                            OCH.sub.3                                                                           N                                    H      O       H      CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    H      O       H      CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            N                                    H      O       H      OCH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                                                                            CH                                   H      O       H      OCH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   H      O       H      OCH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   H      O       H      OCH.sub.3                                                                            Cl    OCH.sub.3                                                                           CH                                   H      O       H      OCH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           N                                    H      O       H      OCH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    H      O       H      OCH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                                                                            N                                    6-CH.sub.3                                                                           C═O H      OCH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                                                                            CH                                   6-CH.sub.3                                                                           C═O H      OCH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   6-CH.sub.3                                                                           C═O H      OCH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   6-CH.sub.3                                                                           C═O H      OCH.sub.3                                                                            Cl    OCH.sub.3                                                                           CH                                   6-CH.sub.3                                                                           C═O H      OCH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           N                                    6-CH.sub.3                                                                           C═O H      OCH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    6-CH.sub.3                                                                           C═O H      OCH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                                                                            N                                    6-CH.sub.3                                                                           C═O CH.sub.3                                                                             SCH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                                                                            CH                                   6-CH.sub.3                                                                           C═O CH.sub.3                                                                             SCH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   6-CH.sub.3                                                                           C═O CH.sub.3                                                                             SCH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   6-CH.sub.3                                                                           C═O CH.sub.3                                                                             SCH.sub.3                                                                            Cl    OCH.sub.3                                                                           CH                                   6-CH.sub.3                                                                           C═O CH.sub.3                                                                             SCH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           N                                    6-CH.sub.3                                                                           C═O CH.sub.3                                                                             SCH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    6-CH.sub.3                                                                           C═O CH.sub.3                                                                             SCH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                                                                            N                                    6-CH.sub.3                                                                           SO.sub.2                                                                              CH.sub.3                                                                             OCH.sub.3                                                                            CH    CH.sub.3                                                                            CH                                   6-CH.sub.3                                                                           SO.sub.2                                                                              CH.sub.3                                                                             OCH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   6-CH.sub.3                                                                           SO.sub.2                                                                              CH.sub.3                                                                             OCH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   6-CH.sub.3                                                                           SO.sub.2                                                                              CH.sub.3                                                                             OCH.sub.3                                                                            Cl    OCH.sub.3                                                                           CH                                   6-CH.sub.3                                                                           SO.sub.2                                                                              CH.sub.3                                                                             OCH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           N                                    6-CH.sub.3                                                                           SO.sub.2                                                                              CH.sub.3                                                                             OCH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    6-CH.sub.3                                                                           SO.sub.2                                                                              CH.sub.3                                                                             OCH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                                                                            N                                    6-CH.sub.3                                                                           C═O H      CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            CH                                   6-CH.sub.3                                                                           C═O H      CH.sub.3                                                                             CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   6-CH.sub.3                                                                           C═ O                                                                              H      CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   6-CH.sub.3                                                                           C═O H      CH.sub.3                                                                             Cl    OCH.sub.3                                                                           CH                                   6-CH.sub.3                                                                           C═O H      CH.sub.3                                                                             CH.sub.3                                                                            OCH.sub.3                                                                           N                                    6-CH.sub.3                                                                           C═O H      CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3 N                                6-CH.sub.3                                                                           C═O H      CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            N                                    6-CH.sub.3                                                                           SO.sub.2                                                                              H      CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            CH                                   6-CH.sub.3                                                                           SO.sub.2                                                                              H      CH.sub.3                                                                             CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   6-CH.sub.3                                                                           SO.sub.2                                                                              H      CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   6-CH.sub.3                                                                           SO.sub.2                                                                              H      CH.sub.3                                                                             Cl    OCH.sub.3                                                                           CH                                   6-CH.sub.3                                                                           SO.sub.2                                                                              H      CH.sub.3                                                                             CH.sub.3                                                                            OCH.sub.3                                                                           N                                    6-CH.sub.3                                                                           SO.sub.2                                                                              H      CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    6-CH.sub.3                                                                           SO.sub.2                                                                              H      CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            N                                    6-CH.sub.3                                                                           CH.sub.2                                                                              H      OCH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                                                                            CH                                   6-CH.sub.3                                                                           CH.sub.2                                                                              H      OCH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   6-CH.sub.3                                                                           CH.sub.2                                                                              H      OCH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   6-CH.sub.3                                                                           CH.sub.2                                                                              H      OCH.sub.3                                                                            Cl    OCH.sub.3                                                                           CH                                   6-CH.sub.3                                                                           CH.sub.2                                                                              H      OCH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           N                                    6-CH.sub.3                                                                           CH.sub.2                                                                              H      OCH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    6-CH.sub.3                                                                           CH.sub.2                                                                              H      OCH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                                                                            N                                    6-CH.sub.3                                                                           CH.sub.2                                                                              CH.sub.3                                                                             SCH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                                                                            CH                                   6-CH.sub.3                                                                           CH.sub.2                                                                              CH.sub.3                                                                             SCH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   6-CH.sub.3                                                                           CH.sub.2                                                                              CH.sub.3                                                                             SCH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   6-CH.sub.3                                                                           CH.sub.2                                                                              CH.sub.3                                                                             SCH.sub.3                                                                            Cl    OCH.sub.3                                                                           CH                                   6-CH.sub.3                                                                           CH.sub.2                                                                              CH.sub.3                                                                             SCH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           N                                    6-CH.sub.3                                                                           CH.sub.2                                                                              CH.sub.3                                                                             SCH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    6-CH.sub.3                                                                           CH.sub.2                                                                              CH.sub.3                                                                             SCH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                                                                            N                                    6-CH.sub.3                                                                           CH.sub.2                                                                              CH.sub.3                                                                             CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            CH                                   6-CH.sub.3                                                                           CH.sub.2                                                                              CH.sub.3                                                                             CH.sub.3                                                                             CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   6-CH.sub.3                                                                           CH.sub.2                                                                              CH.sub.3                                                                             CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   6-CH.sub.3                                                                           CH.sub.2                                                                              CH.sub.3                                                                             CH.sub.3                                                                             OCH.sub.3                                                                           Cl    CH                                   6-CH.sub.3                                                                           CH.sub.2                                                                              CH.sub.3                                                                             CH.sub.3                                                                             CH.sub.3                                                                            OCH.sub.3                                                                           N                                    6-CH.sub.3                                                                           CH.sub.2                                                                              CH.sub.3                                                                             CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    6-CH.sub.3                                                                           CH.sub.2                                                                              CH.sub.3                                                                             CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            N                                    6-CH.sub.3                                                                           O       H      CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            CH                                   6-CH.sub.3                                                                           O       H      CH.sub.3                                                                             CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   6-CH.sub.3                                                                           O       H      CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   6-CH.sub.3                                                                           O       H      CH.sub.3                                                                             Cl    OCH.sub.3                                                                           CH                                   6-CH.sub.3                                                                           O       H      CH.sub.3                                                                             CH.sub.3                                                                            OCH.sub.3                                                                           N                                    6-CH.sub.3                                                                           O       H      CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    6-CH.sub.3                                                                           O       H      CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            N                                    6-CH.sub.3                                                                           O       H      OCH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                                                                            CH                                   6-CH.sub.3                                                                           O       H      OCH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   6-CH.sub.3                                                                           O       H      OCH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   6-CH.sub.3                                                                           O       H      OCH.sub.3                                                                            Cl    OCH.sub.3                                                                           CH                                   6-CH.sub.3                                                                           O       H      OCH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           N                                    6-CH.sub.3                                                                           O       H      OCH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    6-CH.sub.3                                                                           O       H      OCH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                                                                            N                                    5-OCH.sub.3                                                                          C═O H      OCH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                                                                            CH                                   5-OCH.sub.3                                                                          C═O H      OCH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   5-OCH.sub.3                                                                          C═O H      OCH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   5-OCH.sub.3                                                                          C═O H      OCH.sub.3                                                                            Cl    OCH.sub.3                                                                           CH                                   5-OCH.sub.3                                                                          C═O H      OCH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           N                                    5-OCH.sub.3                                                                          C═O H      OCH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    5-OCH.sub.3                                                                          C═O H      OCH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                                                                            N                                    5-OCH.sub.3                                                                          C═O CH.sub.3                                                                             SCH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                                                                            CH                                   5-OCH.sub.3                                                                          C═O CH.sub.3                                                                             SCH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   5-OCH.sub.3                                                                          C═O CH.sub.3                                                                             SCH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   5-OCH.sub.3                                                                          C═O CH.sub.3                                                                             SCH.sub.3                                                                            Cl    OCH.sub.3                                                                           CH                                   5-OCH.sub.3                                                                          C═O CH.sub.3                                                                             SCH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           N                                    5-OCH.sub.3                                                                          C═O CH.sub.3                                                                             SCH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    5-OCH.sub.3                                                                          C═O CH.sub.3                                                                             SCH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                                                                            N                                    5-OCH.sub.3                                                                          SO.sub.2                                                                              CH.sub.3                                                                             OCH.sub.3                                                                            CH    CH.sub.3                                                                            CH                                   5-OCH.sub.3                                                                          SO.sub.2                                                                              CH.sub.3                                                                             OCH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   5-OCH.sub.3                                                                          SO.sub.2                                                                              CH.sub.3                                                                             OCH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   5-OCH.sub.3                                                                          SO.sub.2                                                                              CH.sub.3                                                                             OCH.sub.3                                                                            Cl    OCH.sub.3                                                                           CH                                   5-OCH.sub.3                                                                          SO.sub.2                                                                              CH.sub.3                                                                             OCH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           N                                    5-OCH.sub.3                                                                          SO.sub.2                                                                              CH.sub.3                                                                             OCH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    5-OCH.sub.3                                                                          SO.sub.2                                                                              CH.sub.3                                                                             OCH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                                                                            N                                    5-OCH.sub.3                                                                          C═O H      CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            CH                                   5-OCH.sub.3                                                                          C═O H      CH.sub.3                                                                             CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   5-OCH.sub.3                                                                          C═O H      CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   5-OCH.sub.3                                                                          C═O H      CH.sub.3                                                                             Cl    OCH.sub.3                                                                           CH                                   5-OCH.sub.3                                                                          C═O H      CH.sub.3                                                                             CH.sub.3                                                                            OCH.sub.3                                                                           N                                    5-OCH.sub.3                                                                          C═O H      CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    5-OCH.sub.3                                                                          C═O H      CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            N                                    5-OCH.sub.3                                                                          SO.sub.2                                                                              H      CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            CH                                   5-OCH.sub.3                                                                          SO.sub.2                                                                              H      CH.sub.3                                                                             CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   5-OCH.sub.3                                                                          SO.sub.2                                                                              H      CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   5-OCH.sub.3                                                                          SO.sub.2                                                                              H      CH.sub.3                                                                             Cl    OCH.sub.3                                                                           CH                                   5-OCH.sub.3                                                                          SO.sub.2                                                                              H      CH.sub.3                                                                             CH.sub.3                                                                            OCH.sub.3                                                                           N                                    5-OCH.sub.3                                                                          SO.sub.2                                                                              H      CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    5-OCH.sub.3                                                                          SO.sub.2                                                                              H      CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            N                                    5-OCH.sub.3                                                                          CH.sub.2                                                                              H      OCH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                                                                            CH                                   5-OCH.sub.3                                                                          CH.sub.2                                                                              H      OCH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   5-OCH.sub.3                                                                          CH.sub.2                                                                              H      OCH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   5-OCH.sub.3                                                                          CH.sub.2                                                                              H      OCH.sub.3                                                                            Cl    OCH.sub.3                                                                           CH                                   5-OCH.sub.3                                                                          CH.sub.2                                                                              H      OCH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           N                                    5-OCH.sub.3                                                                          CH.sub.2                                                                              H      OCH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    5-OCH.sub.3                                                                          CH.sub.2                                                                              H      OCH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                                                                            N                                    5-OCH.sub.3                                                                          CH.sub.2                                                                              CH.sub.3                                                                             SCH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                                                                            N                                    5-OCH.sub.3                                                                          CH.sub.2                                                                              CH.sub.3                                                                             SCH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   5-OCH.sub.3                                                                          CH.sub.2                                                                              CH.sub.3                                                                             SCH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   5-OCH.sub.3                                                                          CH.sub.2                                                                              CH.sub.3                                                                             SCH    Cl    OCH.sub.3                                                                           CH                                   5-OCH.sub.3                                                                          CH.sub.2                                                                              CH.sub.3                                                                             SCH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           N                                    5-OCH.sub.3                                                                          CH.sub.2                                                                              CH.sub.3                                                                             SCH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    5-OCH.sub.3                                                                          CH.sub.2                                                                              CH.sub.3                                                                             SCH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                                                                            N                                    5-OCH.sub.3                                                                          CH.sub.2                                                                              CH.sub.3                                                                             CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            CH                                   5-OCH.sub.3                                                                          CH.sub.2                                                                              CH.sub.3                                                                             CH.sub.3                                                                             CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   5-OCH.sub.3                                                                          CH.sub.2                                                                              CH.sub.3                                                                             CH.sub. 3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   5-OCH.sub.3                                                                          CH.sub.2                                                                              CH.sub.3                                                                             CH.sub.3                                                                             OCH.sub.3                                                                           Cl    CH                                   5-OCH.sub.3                                                                          CH.sub.2                                                                              CH.sub.3                                                                             CH.sub.3                                                                             CH.sub.3                                                                            OCH.sub.3                                                                           N                                    5-OCH.sub.3                                                                          CH.sub.2                                                                              CH.sub.3                                                                             CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    5-OCH.sub.3                                                                          CH.sub.2                                                                              CH.sub.3                                                                             CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            N                                    5-OCH.sub.3                                                                          O       H      CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            CH                                   5-OCH.sub.3                                                                          O       H      CH.sub.3                                                                             CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   5-OCH.sub.3                                                                          O       H      CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   5-OCH.sub.3                                                                          O       H      CH.sub.3                                                                             Cl    OCH.sub.3                                                                           CH                                   5-OCH.sub.3                                                                          O       H      CH.sub.3                                                                             CH.sub.3                                                                            OCH.sub.3                                                                           N                                    5-OCH.sub.3                                                                          O       H      CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    5-OCH.sub.3                                                                          O       H      CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            N                                    5-OCH.sub.3                                                                          O       H      OCH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                                                                            CH                                   5-OCH.sub.3                                                                          O       OCH.sub.3                                                                            CH.sub.3                                                                             OCH.sub.3                                                                           CH                                         5-OCH.sub.3                                                                          O       H      OCH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   5-OCH.sub.3                                                                          O       H      OCH.sub.3                                                                            Cl    OCH.sub.3                                                                           CH                                   5-OCH.sub.3                                                                          O       H      OCH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           N                                    5-OCH.sub.3                                                                          O       H      OCH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    5-OCH.sub.3                                                                          O       H      OCH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                                                                            N                                    ______________________________________                                    

                  TABLE 8                                                         ______________________________________                                        General Formula 8                                                                                                           m.p.                            R.sub.1                                                                             J       R.sub.8 R.sub.11                                                                             X     Y     Z    (°C.)                    ______________________________________                                        H     C═O H       CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            CH                                   H     C═O H       CH.sub.3                                                                             CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   H     C═O H       CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   H     C═O H       CH.sub.3                                                                             Cl    OCH.sub.3                                                                           CH                                   H     C═O H       CH.sub.3                                                                             CH.sub.3                                                                            OCH.sub.3                                                                           N                                    H     C═O H       CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    H     C═O H       CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            N                                    H     C═O CH.sub.3                                                                              CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            CH                                   H     C═O CH.sub.3                                                                              CH.sub.3                                                                             CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   H     C═O CH.sub.3                                                                              CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   H     C═O CH.sub.3                                                                              CH.sub.3                                                                             Cl    OCH.sub.3                                                                           CH                                   H     C═O CH.sub.3                                                                              CH.sub.3                                                                             CH.sub.3                                                                            OCH.sub.3                                                                           N                                    H     C═O CH.sub.3                                                                              CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    H     C═O CH.sub.3                                                                              CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            N                                    H     SO.sub.2                                                                              CH.sub.3                                                                              CH.sub.3                                                                             CH    CH.sub.3                                                                            CH                                   H     SO.sub.2                                                                              CH.sub.3                                                                              CH.sub.3                                                                             CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   H     SO.sub.2                                                                              CH.sub.3                                                                              CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   H     SO.sub.2                                                                              CH.sub.3                                                                              CH.sub.3                                                                             Cl    OCH.sub.3                                                                           CH                                   H     SO      CH.sub.3                                                                              CH.sub.3                                                                             CH.sub.3                                                                            OCH.sub.3                                                                           N                                    H     SO      CH.sub.3                                                                              CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    H     SO.sub.2                                                                              CH.sub.3                                                                              CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            N                                    H     C═O CH.sub.3                                                                              N(CH.sub.3).sub.2                                                                    CH.sub.3                                                                            CH.sub.3                                                                            CH                                   H     C═O CH      N(CH.sub.3).sub.2                                                                    CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   H     C═O CH.sub.3                                                                              N(CH.sub.3).sub.2                                                                    OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   H     C═O CH.sub.3                                                                              N(CH.sub.3).sub.2                                                                    Cl    OCH.sub.3                                                                           CH                                   H     C═O CH.sub.3                                                                              N(CH.sub.3).sub.2                                                                    CH.sub.3                                                                            OCH.sub.3                                                                           N                                    H     C═O CH.sub.3                                                                              N(CH.sub.3).sub.2                                                                    OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    H     C═O CH.sub.3                                                                              N(CH.sub.3).sub.2                                                                    CH.sub.3                                                                            CH.sub.3                                                                            N                                    H     SO.sub.2                                                                              H       CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            CH                                   H     SO.sub.2                                                                              H       CH.sub.3                                                                             CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   H     SO.sub.2                                                                              H       CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   H     SO.sub.2                                                                              H       CH.sub.3                                                                             Cl    OCH.sub.3                                                                           CH                                   H     SO.sub.2                                                                              H       CH.sub.3                                                                             CH.sub.3                                                                            OCH.sub.3                                                                           N                                    H     SO.sub.2                                                                              H       CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    H     SO.sub.2                                                                              H       CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            N                                    H     C═O CH.sub.3                                                                              OCH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                                                                            CH                                   H     C═O CH.sub.3                                                                              OCH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   H     C═O CH.sub.3                                                                              OCH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   H     C═O CH.sub.3                                                                              OCH.sub.3                                                                            Cl    OCH.sub.3                                                                           CH                                   H     C═O CH.sub.3                                                                              OCH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           N                                    H     C═O CH.sub.3                                                                              OCH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    H     C═O CH.sub.3                                                                              OCH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                                                                            N                                    H     SO.sub.2                                                                              CH.sub.3                                                                              OCH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   H     SO.sub.2                                                                              CH.sub.3                                                                              OCH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   H     SO.sub.2                                                                              CH.sub.3                                                                              OCH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   H     SO.sub.2                                                                              CH.sub.3                                                                              OCH.sub.3                                                                            Cl    OCH.sub.3                                                                           CH                                   H     SO.sub.2                                                                              CH.sub.3                                                                              OCH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           N                                    H     SO.sub.2                                                                              CH.sub.3                                                                              OCH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    H     SO.sub.2                                                                              CH.sub.3                                                                              OCH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                                                                            N                                    H     CH.sub.2                                                                              H       CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            CH                                   H     CH.sub.2                                                                              H       CH.sub.3                                                                             CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   H     CH.sub.2                                                                              H       CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   H     CH.sub.2                                                                              H       CH.sub.3                                                                             Cl    OCH.sub.3                                                                           CH                                   H     CH.sub.2                                                                              H       CH.sub.3                                                                             CH.sub.3                                                                            OCH.sub.3                                                                           N                                    H     CH.sub.2                                                                              H       CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    H     CH.sub.2                                                                              H       CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            N                                    H     CH.sub.2                                                                              CH.sub.3                                                                              CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            CH                                   H     CH.sub.2                                                                              CH.sub.3                                                                              CH.sub.3                                                                             CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   H     CH.sub.2                                                                              CH.sub.3                                                                              CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   H     CH.sub.2                                                                              CH.sub.3                                                                              CH.sub.3                                                                             Cl    OCH.sub.3                                                                           CH                                   H     CH.sub.2                                                                              CH.sub.3                                                                              CH.sub.3                                                                             CH.sub.3                                                                            OCH.sub.3                                                                           N                                    H     CH.sub.2                                                                              CH.sub.3                                                                              CH.sub.3                                                                             CH.sub.3                                                                            OCH.sub.3                                                                           N                                    H     CH.sub.2                                                                              CH.sub.3                                                                              CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            N                                    H     CH.sub.2                                                                              CH.sub.3                                                                              SCH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                                                                            CH                                   H     CH.sub.2                                                                              CH.sub.3                                                                              SCH.sub.3                                                                            CH.sub. 3                                                                           OCH.sub.3                                                                           CH                                   H     CH.sub.2                                                                              CH.sub.3                                                                              SCH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   H     CH.sub.2                                                                              CH.sub.3                                                                              SCH.sub.3                                                                            Cl    OCH.sub.3                                                                           CH                                   H     CH.sub.2                                                                              CH.sub.3                                                                              SCH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           N                                    H     CH.sub.2                                                                              CH.sub.3                                                                              SCH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    H     CH.sub.2                                                                              CH.sub.3                                                                              SCH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                                                                            N                                    H     O       H       CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            CH                                   H     O       H       CH.sub.3                                                                             CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   H     O       H       CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   H     O       H       CH.sub.3                                                                             Cl    OCH.sub.3                                                                           CH                                   H     O       H       CH.sub.3                                                                             CH.sub.3                                                                            OCH.sub.3                                                                           N                                    H     O       H       CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    H     O       H       CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            N                                    H     O       H       OCH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                                                                            CH                                   H     O       H       OCH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   H     O       H       OCH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   H     O       H       OCH.sub.3                                                                            Cl    OCH.sub.3                                                                           CH                                   H     O       H       OCH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           N                                    H     O       H       OCH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    H     O       H       OCH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                                                                            N                                    H     O       CH.sub.3                                                                              CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            CH                                   H     O       CH.sub.3                                                                              CH.sub.3                                                                             CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   H     O       CH.sub.3                                                                              CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   H     O       CH.sub.3                                                                              CH.sub.3                                                                             Cl    OCH.sub.3                                                                           CH                                   H     O       CH.sub.3                                                                              CH.sub.3                                                                             CH.sub.3                                                                            OCH.sub.3                                                                           N                                    H     O       CH.sub.3                                                                              CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    H     O       CH.sub.3                                                                              CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            N                                    6-CH.sub.3                                                                          C═O H       CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            CH                                   6-CH.sub.3                                                                          C═O H       CH.sub.3                                                                             CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   6-CH.sub.3                                                                          C═O H       CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   6-CH.sub.3                                                                          C═O H       CH.sub.3                                                                             Cl    OCH.sub.3                                                                           CH                                   6-CH.sub.3                                                                          C═O H       CH.sub.3                                                                             CH.sub.3                                                                            OCH.sub.3                                                                           N                                    6-CH.sub.3                                                                          C═O H       CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    6-CH.sub.3                                                                          C═O H       CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            N                                    6-CH.sub.3                                                                          C═O CH.sub.3                                                                              CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            CH                                   6-CH.sub.3                                                                          C═O CH.sub.3                                                                              CH.sub.3                                                                             CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   6-CH.sub.3                                                                          C═O CH.sub.3                                                                              CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   6-CH.sub. 3                                                                         C═O CH.sub.3                                                                              CH.sub.3                                                                             Cl    OCH.sub.3                                                                           CH                                   6-CH.sub.3                                                                          C═O CH.sub.3                                                                              CH.sub.3                                                                             CH.sub.3                                                                            OCH.sub.3                                                                           N                                    6-CH.sub.3                                                                          C═O CH.sub.3                                                                              CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    6-CH.sub.3                                                                          C═O CH.sub.3                                                                              CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            N                                    6-CH.sub.3                                                                          SO.sub.2                                                                              CH.sub.3                                                                              CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            CH                                   6-CH.sub.3                                                                          SO.sub.2                                                                              CH.sub.3                                                                              CH.sub.3                                                                             CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   6-CH.sub.3                                                                          SO.sub.2                                                                              CH.sub.3                                                                              CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   6-CH.sub.3                                                                          SO.sub.2                                                                              CH.sub.3                                                                              CH.sub.3                                                                             Cl    OCH.sub.3                                                                           CH                                   6-CH.sub.3                                                                          SO.sub.2                                                                              CH.sub.3                                                                              CH.sub.3                                                                             CH.sub.3                                                                            OCH.sub.3                                                                           N                                    6-CH.sub.3                                                                          SO.sub.2                                                                              CH.sub.3                                                                              CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    6-CH.sub.3                                                                          SO.sub.2                                                                              CH.sub.3                                                                              CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            N                                    6-CH.sub.3                                                                          C═O CH.sub.3                                                                              N(CH.sub.3).sub.2                                                                    CH.sub.3                                                                            CH.sub.3                                                                            CH                                   6 CH.sub.3                                                                          C═O CH.sub.3                                                                              N(CH.sub.3).sub.2                                                                    CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   6-CH.sub.3                                                                          C═O CH.sub.3                                                                              N(CH.sub.3).sub.2                                                                    OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   6-CH.sub.3                                                                          C═O CH.sub.3                                                                              N(CH.sub.3).sub.2                                                                    Cl    OCH.sub.3                                                                           CH                                   6-CH.sub.3                                                                          C═O CH.sub.3                                                                              N(CH.sub.3).sub.2                                                                    CH.sub.3                                                                            OCH.sub.3                                                                           N                                    6-CH.sub.3                                                                          C═O CH.sub.3                                                                              N(CH.sub.3).sub.2                                                                    OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    6-CH.sub.3                                                                          C═O CH.sub.3                                                                              N(CH.sub.3).sub.2                                                                    CH.sub.3                                                                            CH.sub.3                                                                            N                                    6-CH.sub.3                                                                          SO.sub.2                                                                              H       CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            CH                                   6-CH.sub.3                                                                          SO.sub.2                                                                              H       CH.sub.3                                                                             CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   6-CH.sub.3                                                                          SO.sub.2                                                                              H       CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   6-CH.sub.3                                                                          SO.sub.2                                                                              H       CH.sub.3                                                                             Cl    OCH.sub.3                                                                           CH                                   6-CH.sub.3                                                                          SO.sub.2                                                                              H       CH.sub.3                                                                             CH.sub.3                                                                            OCH.sub.3                                                                           N                                    6-CH.sub.3                                                                          SO.sub.2                                                                              H       CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    6-CH.sub.3                                                                          SO.sub.2                                                                              H       CH.sub.3                                                                             CH.sub.3                                                                            OCH.sub.3                                                                           N                                    6-CH.sub.3                                                                          C═O CH.sub.3                                                                              OCH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                                                                            CH                                   6-CH.sub.3                                                                          C═O CH.sub.3                                                                              OCH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   6-CH.sub.3                                                                          C═O CH.sub.3                                                                              OCH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   6-CH.sub.3                                                                          C═O CH.sub.3                                                                              OCH.sub.3                                                                            Cl    OCH.sub.3                                                                           CH                                   6-CH.sub.3                                                                          C═O CH.sub.3                                                                              OCH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           N                                    6-CH.sub.3                                                                          C═O CH.sub.3                                                                              OCH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    6-CH.sub.3                                                                          C═O CH.sub.3                                                                              OCH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                                                                            N                                    6-CH.sub.3                                                                          SO.sub.2                                                                              CH.sub.3                                                                              OCH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                                                                            CH                                   6-CH.sub.3                                                                          SO.sub.2                                                                              CH.sub.3                                                                              OCH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   6-CH.sub.3                                                                          SO.sub.2                                                                              CH.sub.3                                                                              OCH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   6-CH.sub.3                                                                          SO.sub.2                                                                              CH.sub.3                                                                              OCH.sub.3                                                                            Cl    OCH.sub.3                                                                           CH                                   6-CH.sub.3                                                                          SO.sub.2                                                                              CH.sub.3                                                                              OCH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           N                                    6-CH.sub.3                                                                          SO.sub.2                                                                              CH.sub.3                                                                              OCH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    6-CH.sub.3                                                                          SO.sub.2                                                                              CH.sub.3                                                                              OCH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                                                                            N                                    6-CH.sub.3                                                                          CH.sub.2                                                                              H       CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            CH                                   6-CH.sub.3                                                                          CH.sub.2                                                                              H       CH.sub.3                                                                             CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   6-CH.sub.3                                                                          CH.sub.2                                                                              H       CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   6-CH.sub.3                                                                          CH.sub.2                                                                              H       CH.sub.3                                                                             Cl    OCH.sub.3                                                                           CH                                   6-CH.sub.3                                                                          CH.sub.2                                                                              H       CH.sub.3                                                                             CH.sub.3                                                                            OCH.sub.3                                                                           N                                    6-CH.sub.3                                                                          CH.sub.2                                                                              H       CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    6-CH.sub.3                                                                          CH.sub.2                                                                              H       CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            N                                    6-CH.sub.3                                                                          CH.sub.2                                                                              CH.sub.3                                                                              CH.sub.3                                                                             CH.sub. 3                                                                           CH.sub.3                                                                            CH                                   6-CH.sub.3                                                                          CH.sub.2                                                                              CH.sub.3                                                                              CH.sub.3                                                                             CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   6-CH.sub.3                                                                          CH.sub.2                                                                              CH.sub.3                                                                              CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   6-CH.sub.3                                                                          CH.sub.2                                                                              CH.sub.3                                                                              CH.sub.3                                                                             Cl    OCH.sub.3                                                                           CH                                   6-CH.sub.3                                                                          CH.sub.2                                                                              CH.sub.3                                                                              CH.sub.3                                                                             CH.sub.3                                                                            OCH.sub.3                                                                           N                                    6-CH.sub.3                                                                          CH.sub.2                                                                              CH.sub.3                                                                              CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    6-CH.sub.3                                                                          CH.sub.2                                                                              CH.sub.3                                                                              CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            N                                    6-CH.sub.3                                                                          CH.sub.2                                                                              CH.sub.3                                                                              SCH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                                                                            CH                                   6-CH.sub.3                                                                          CH.sub.2                                                                              CH.sub.3                                                                              SCH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   6-CH.sub.3                                                                          CH.sub.2                                                                              CH.sub.3                                                                              SCH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   6-CH.sub.3                                                                          CH.sub.2                                                                              CH.sub.3                                                                              SCH.sub.3                                                                            Cl    OCH.sub.3                                                                           CH                                   6-CH.sub.3                                                                          CH.sub.2                                                                              CH.sub.3                                                                              SCH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           N                                    6-CH.sub.3                                                                          CH.sub.2                                                                              CH.sub.3                                                                              SCH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    6-CH.sub.3                                                                          CH.sub.2                                                                              CH.sub.3                                                                              SCH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                                                                            N                                    6-CH.sub.3                                                                          O       H       CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            CH                                   6-CH.sub.3                                                                          O       H       CH.sub.3                                                                             CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   6-CH.sub.3                                                                          O       H       CH.sub.3                                                                             OCH.sub. 3                                                                          OCH.sub.3                                                                           CH                                   6-CH.sub.3                                                                          O       H       CH.sub.3                                                                             Cl    OCH.sub.3                                                                           CH                                   6-CH.sub.3                                                                          O       H       CH.sub.3                                                                             CH.sub.3                                                                            OCH.sub.3                                                                           N                                    6-CH.sub.3                                                                          O       H       CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    6-CH.sub.3                                                                          O       H       CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            N                                    6-CH.sub.3                                                                          O       H       OCH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                                                                            CH                                   6-CH.sub.3                                                                          O       H       OCH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   6-CH.sub.3                                                                          O       H       OCH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   6-CH.sub.3                                                                          O       H       OCH.sub.3                                                                            Cl    OCH.sub.3                                                                           CH                                   6-CH.sub.3                                                                          O       H       OCH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           N                                    6-CH.sub.3                                                                          O       H       OCH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    6-CH.sub.3                                                                          O       H       OCH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                                                                            N                                    6-CH.sub.3                                                                          O       CH.sub.3                                                                              CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            CH                                   6-CH.sub.3                                                                          O       CH.sub.3                                                                              CH.sub.3                                                                             CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   6-CH.sub.3                                                                          O       CH.sub.3                                                                              CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   6-CH.sub.3                                                                          O       CH.sub.3                                                                              CH.sub.3                                                                             Cl    OCH.sub.3                                                                           CH                                   6-CH.sub.3                                                                          O       CH.sub.3                                                                              CH.sub.3                                                                             CH.sub.3                                                                            OCH.sub.3                                                                           N                                    6-CH.sub.3                                                                          O       CH.sub.3                                                                              CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    6-CH.sub.3                                                                          O       CH.sub.3                                                                              CH.sub. 3                                                                            CH.sub.3                                                                            CH.sub.3                                                                            N                                    ______________________________________                                    

                  TABLE 9                                                         ______________________________________                                        General Formula 9                                                             R.sub.1  J        X        Y      Z    m.p. (°C.)                      ______________________________________                                        H        C═O  CH.sub.3 CH.sub.3                                                                             CH                                          H        C═O  CH.sub.3 OCH.sub.3                                                                            CH                                          H        C═O  OCH.sub.3                                                                              OCH.sub.3                                                                            CH                                          H        C═O  Cl       OCH.sub.3                                                                            CH                                          H        C═O  CH.sub.3 OCH.sub.3                                                                            N                                           H        C═O  OCH.sub.3                                                                              OCH.sub.3                                                                            N                                           H        C═O  CH.sub.3 CH.sub.3                                                                             N                                           H        S        CH.sub.3 CH.sub.3                                                                             CH                                          H        S        CH.sub.3 OCH.sub.3                                                                            CH                                          H        S        OCH.sub.3                                                                              OCH.sub.3                                                                            CH                                          H        S        Cl       OCH.sub.3                                                                            CH                                          H        S        CH.sub.3 OCH.sub.3                                                                            N                                           H        S        OCH.sub.3                                                                              OCH.sub.3                                                                            N                                           H        S        CH.sub.3 CH.sub.3                                                                             N                                           H        SO.sub.2 CH.sub.3 CH.sub.3                                                                             CH                                          H        SO.sub.2 CH.sub.3 OCH.sub.3                                                                            CH                                          H        SO.sub.2 OCH.sub.3                                                                              OCH.sub.3                                                                            CH                                          H        SO.sub.2 Cl       OCH.sub.3                                                                            CH                                          H        SO.sub.2 CH.sub.3 OCH.sub.3                                                                            N                                           H        SO.sub.2 OCH.sub.3                                                                              OCH.sub.3                                                                            N                                           H        SO.sub.2 CH.sub.3 CH.sub.3                                                                             N                                           H        CH.sub.2 CH.sub.3 CH.sub.3                                                                             CH                                          H        CH.sub.2 CH.sub.3 OCH.sub.3                                                                            CH                                          H        CH.sub.2 OCH.sub.3                                                                              OCH.sub.3                                                                            CH                                          H        CH.sub.2 Cl       OCH.sub.3                                                                            CH                                          H        CH.sub.2 CH.sub.3 OCH.sub.3                                                                            N                                           H        CH.sub.2 OCH.sub.3                                                                              OCH.sub.3                                                                            N                                           H        CH.sub.2 CH.sub.3 CH.sub.3                                                                             N                                           6-CH.sub.3                                                                             C═O  CH.sub.3 CH.sub.3                                                                             CH                                          6-CH.sub.3                                                                             C═O  CH.sub.3 OCH.sub.3                                                                            CH                                          6-CH.sub.3                                                                             C═O  OCH.sub.3                                                                              OCH.sub.3                                                                            CH                                          6-CH.sub.3                                                                             C═O  Cl       OCH.sub.3                                                                            CH                                          6-CH.sub.3                                                                             C═O  CH.sub.3 OCH.sub.3                                                                            N                                           6-CH.sub.3                                                                             C═O  OCH.sub.3                                                                              OCH.sub.3                                                                            N                                           6-CH.sub.3                                                                             C═O  CH.sub.3 CH.sub.3                                                                             N                                           6-CH.sub.3                                                                             S        CH.sub.3 CH.sub.3                                                                             CH                                          6-CH.sub.3                                                                             S        CH.sub.3 OCH.sub.3                                                                            CH                                          6-CH.sub.3                                                                             S        OCH.sub.3                                                                              OCH.sub.3                                                                            CH                                          6-CH.sub.3                                                                             S        Cl       OCH.sub.3                                                                            CH                                          6-CH.sub.3                                                                             S        CH.sub.3 OCH.sub.3                                                                            N                                           6-CH.sub.3                                                                             S        OCH.sub.3                                                                              OCH.sub.3                                                                            N                                           6-CH.sub.3                                                                             S        CH.sub.3 CH.sub.3                                                                             N                                           6-CH.sub.3                                                                             SO.sub.2 CH.sub.3 CH.sub.3                                                                             CH                                          6-CH.sub.3                                                                             SO.sub.2 CH.sub.3 OCH.sub.3                                                                            CH                                          6-CH.sub.3                                                                             SO.sub.2 OCH.sub.3                                                                              OCH.sub.3                                                                            CH                                          6-CH.sub.3                                                                             SO.sub.2 Cl       OCH.sub.3                                                                            CH                                          6-CH.sub.3                                                                             SO.sub.2 CH.sub.3 OCH.sub.3                                                                            N                                           6-CH.sub.3                                                                             SO.sub.2 OCH.sub.3                                                                              OCH.sub.3                                                                            N                                           6-CH.sub.3                                                                             SO.sub.2 CH.sub.3 CH.sub.3                                                                             N                                           6-CH.sub.3                                                                             CH.sub.2 CH.sub.3 CH.sub.3                                                                             CH                                          6-CH.sub.3                                                                             CH.sub.2 CH.sub.3 OCH.sub.3                                                                            CH                                          6-CH.sub.3                                                                             CH.sub.2 OCH.sub.3                                                                              OCH.sub.3                                                                            CH                                          6-CH.sub.3                                                                             CH.sub.2 Cl       OCH.sub.3                                                                            CH                                          6-CH.sub.3                                                                             CH.sub.2 Cl       OCH.sub.3                                                                            N                                           6-CH.sub.3                                                                             CH.sub.2 OCH.sub.3                                                                              OCH.sub.3                                                                            N                                           6-CH.sub.3                                                                             CH.sub.2 CH.sub.3 CH.sub.3                                                                             N                                           ______________________________________                                    

                  TABLE 10                                                        ______________________________________                                        General Formula 10                                                            R.sub.1  J        X        Y      Z    m.p. (°C.)                      ______________________________________                                        H        C═O  CH.sub.3 CH.sub.3                                                                             CH                                          H        C═O  CH.sub.3 OCH.sub.3                                                                            CH                                          H        C═O  OCH.sub.3                                                                              OCH.sub.3                                                                            CH                                          H        C═O  Cl       OCH.sub.3                                                                            CH                                          H        C═O  CH.sub.3 OCH.sub.3                                                                            N                                           H        C═O  OCH.sub.3                                                                              OCH.sub.3                                                                            N                                           H        C═O  CH.sub.3 CH.sub.3                                                                             N                                           H        SO.sub.2 CH.sub.3 CH.sub.3                                                                             CH                                          H        SO.sub.2 CH.sub.3 OCH.sub.3                                                                            CH                                          H        SO.sub.2 OCH.sub.3                                                                              OCH.sub.3                                                                            CH                                          H        SO.sub.2 Cl       OCH.sub.3                                                                            CH                                          H        SO.sub.2 CH.sub.3 OCH.sub.3                                                                            N                                           H        SO.sub.2 OCH.sub.3                                                                              OCH.sub.3                                                                            N                                           H        SO.sub.2 CH.sub.3 CH.sub.3                                                                             N                                           H        CH.sub.2 CH.sub.3 CH.sub.3                                                                             CH                                          H        CH.sub.2 CH.sub.3 OCH.sub.3                                                                            CH                                          H        CH.sub.2 OCH.sub.3                                                                              OCH.sub.3                                                                            CH                                          H        CH.sub.2 Cl       OCH.sub.3                                                                            CH                                          H        CH.sub.2 CH.sub.3 OCH.sub.3                                                                            N                                           H        CH.sub.2 OCH.sub.3                                                                              OCH.sub.3                                                                            N                                           H        CH.sub.2 CH.sub.3 CH.sub.3                                                                             N                                           6-CH.sub.3                                                                             C═O  CH.sub.3 CH.sub.3                                                                             CH                                          6-CH.sub.3                                                                             C═O  CH.sub.3 OCH.sub.3                                                                            CH                                          6-CH.sub.3                                                                             C═O  OCH.sub.3                                                                              OCH.sub.3                                                                            CH                                          6-CH.sub.3                                                                             C═O  Cl       OCH.sub.3                                                                            CH                                          6-CH.sub.3                                                                             C═O  CH.sub.3 OCH.sub.3                                                                            N                                           6-CH.sub.3                                                                             C═O  OCH.sub.3                                                                              OCH.sub.3                                                                            N                                           6-CH.sub.3                                                                             C═O  CH.sub.3 CH.sub.3                                                                             N                                           6-CH.sub.3                                                                             SO.sub.2 CH.sub.3 CH.sub.3                                                                             CH                                          6-CH.sub.3                                                                             SO.sub.2 CH.sub.3 OCH.sub.3                                                                            CH                                          6-CH.sub.3                                                                             SO.sub.2 OCH.sub.3                                                                              OCH.sub.3                                                                            CH                                          6-CH.sub.3                                                                             SO.sub.2 Cl       OCH.sub.3                                                                            CH                                          6-CH.sub.3                                                                             SO.sub.2 CH.sub.3 OCH.sub.3                                                                            N                                           6-CH.sub.3                                                                             SO.sub.2 OCH.sub.3                                                                              OCH.sub.3                                                                            N                                           6-CH.sub.3                                                                             SO.sub.2 CH.sub.3 CH.sub.3                                                                             N                                           6-CH.sub.3                                                                             CH.sub.2 CH.sub.3 CH.sub.3                                                                             CH                                          6-CH.sub.3                                                                             CH.sub.2 CH.sub.3 OCH.sub.3                                                                            CH                                          6-CH.sub.3                                                                             CH.sub.2 OCH.sub.3                                                                              OCH.sub.3                                                                            CH                                          6-CH.sub.3                                                                             CH.sub.2 Cl       OCH.sub.3                                                                            CH                                          6-CH.sub.3                                                                             CH.sub.2 CH.sub.3 OCH.sub.3                                                                            N                                           6-CH.sub.3                                                                             CH.sub.2 OCH.sub.3                                                                              OCH.sub.3                                                                            N                                           6-CH.sub.3                                                                             CH.sub.2 CH.sub.3 CH.sub.3                                                                             N                                           ______________________________________                                    

                  TABLE 11                                                        ______________________________________                                        General Formula 11                                                                                                          m.p.                            R.sub.1                                                                             J       R.sub.8 R.sub.11                                                                             X     Y     Z    (°C.)                    ______________________________________                                        H     C═O CH.sub.3                                                                              SCH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                                                                            CH                                   H     C═O CH.sub.3                                                                              SCH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   H     C═O CH.sub.3                                                                              SCH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   H     C═O CH.sub.3                                                                              SCH.sub.3                                                                            Cl    OCH.sub.3                                                                           CH                                   H     C═O CH.sub.3                                                                              SCH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           N                                    H     C═O CH.sub.3                                                                              SCH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    H     C═O CH.sub.3                                                                              SCH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                                                                            N                                    H     C═O SCH.sub.3                                                                             SCH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                                                                            CH                                   H     C═O SCH.sub.3                                                                             SCH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   H     C═O SCH.sub.3                                                                             SCH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   H     C═O SCH.sub.3                                                                             SCH.sub.3                                                                            Cl    OCH.sub.3                                                                           CH                                   H     C═O SCH.sub.3                                                                             SCH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           N                                    H     C═O SCH.sub.3                                                                             SCH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    H     C═ O                                                                              SCH.sub.3                                                                             SCH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                                                                            N                                    H     SO.sub.2                                                                              CH.sub.3                                                                              SCH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                                                                            CH                                   H     SO.sub.2                                                                              CH.sub.3                                                                              SCH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   H     SO.sub.2                                                                              CH.sub.3                                                                              SCH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   H     SO.sub.2                                                                              CH.sub.3                                                                              SCH.sub.3                                                                            Cl    OCH.sub.3                                                                           CH                                   H     SO.sub.2                                                                              CH.sub.3                                                                              SCH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           N                                    H     SO.sub.2                                                                              CH.sub.3                                                                              SCH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    H     SO.sub.2                                                                              CH.sub.3                                                                              SCH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                                                                            N                                    H     CH.sub.2                                                                              CH.sub.3                                                                              SCH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                                                                            CH                                   H     CH.sub.2                                                                              CH.sub.3                                                                              SCH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   H     CH.sub.2                                                                              CH.sub.3                                                                              SCH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   H     CH.sub.2                                                                              CH.sub.3                                                                              SCH.sub.3                                                                            Cl    OCH.sub.3                                                                           CH                                   H     CH.sub.2                                                                              CH.sub.3                                                                              SCH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           N                                    H     CH.sub.2                                                                              CH.sub.3                                                                              SCH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    H     CH.sub.2                                                                              CH.sub.3                                                                              SCH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                                                                            N                                    H     CH.sub.2                                                                              CH.sub.3                                                                              OCH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                                                                            CH                                   H     CH.sub.2                                                                              CH.sub.3                                                                              OCH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   H     CH.sub.2                                                                              CH.sub.3                                                                              OCH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   H     CH.sub.2                                                                              CH.sub.3                                                                              OCH.sub.3                                                                            Cl    OCH.sub.3                                                                           CH                                   H     CH.sub.2                                                                              CH.sub.3                                                                              OCH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           N                                    H     CH.sub.2                                                                              CH.sub.3                                                                              OCH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    H     CH.sub.2                                                                              CH.sub.3                                                                              OCH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                                                                            N                                    H     CH.sub.2                                                                              CH.sub.3                                                                              CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            CH                                   H     CH.sub.2                                                                              CH.sub.3                                                                              CH.sub.3                                                                             CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   H     CH.sub.2                                                                              CH.sub.3                                                                              CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   H     CH.sub.2                                                                              CH.sub.3                                                                              CH.sub.3                                                                             Cl    OCH.sub.3                                                                           CH                                   H     CH.sub.2                                                                              CH.sub.3                                                                              CH.sub.3                                                                             CH.sub.3                                                                            OCH.sub.3                                                                           N                                    H     CH.sub.2                                                                              CH.sub.3                                                                              CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    H     CH.sub.2                                                                              CH.sub.3                                                                              CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            N                                    H     C═O CH.sub.3                                                                              N(CH.sub.3).sub.2                                                                    CH.sub.3                                                                            CH.sub.3                                                                            CH                                   H     C═O CH.sub.3                                                                              N(CH.sub.3).sub.2                                                                    CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   H     C═O CH.sub.3                                                                              N(CH.sub.3).sub.2                                                                    OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   H     C═O CH.sub.3                                                                              N(CH.sub.3).sub.2                                                                    Cl    OCH.sub.3                                                                           CH                                   H     C═O CH.sub. 3                                                                             N(CH.sub.3).sub.2                                                                    CH.sub.3                                                                            OCH.sub.3                                                                           N                                    H     C═O CH.sub.3                                                                              N(CH.sub.3).sub.2                                                                    OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    H     C═O CH.sub.3                                                                              N(CH.sub.3).sub.2                                                                    CH.sub.3                                                                            CH.sub.3                                                                            N                                    H     C═O CH.sub.3                                                                              OCH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                                                                            CH                                   H     C═O CH.sub.3                                                                              OCH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   H     C═O CH.sub.3                                                                              OCH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   H     C═O CH.sub.3                                                                              OCH.sub.3                                                                            Cl    OCH.sub.3                                                                           CH                                   H     C═O CH.sub.3                                                                              OCH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           N                                    H     C═O CH.sub.3                                                                              OCH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    H     C═O CH.sub.3                                                                              OCH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                                                                            N                                    H     SO.sub.2                                                                              CH.sub.3                                                                              OCH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                                                                            CH                                   H     SO.sub.2                                                                              CH.sub.3                                                                              OCH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   H     SO.sub.2                                                                              CH.sub.3                                                                              OCH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   H     SO.sub.2                                                                              CH.sub.3                                                                              OCH.sub.3                                                                            Cl    OCH.sub.3                                                                           CH                                   H     SO.sub.2                                                                              CH.sub.3                                                                              OCH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           N                                    H     SO.sub.2                                                                              CH.sub.3                                                                              OCH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    H     SO.sub.2                                                                              CH.sub.3                                                                              OCH.sub.3                                                                            CH.sub. 3                                                                           CH.sub.3                                                                            N                                    6-Cl  C═O CH.sub.3                                                                              SCH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                                                                            CH                                   6-Cl  C═O CH.sub.3                                                                              SCH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   6-Cl  C═O CH.sub.3                                                                              SCH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   6-Cl  C═O CH.sub.3                                                                              SCH.sub.3                                                                            Cl    OCH.sub.3                                                                           CH                                   6-Cl  C═O CH.sub.3                                                                              SCH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           N                                    6-Cl  C═O CH.sub.3                                                                              SCH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    6-Cl  C═O CH.sub.3                                                                              SCH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                                                                            N                                    6-Cl  C═O SCH.sub.3                                                                             SCH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                                                                            CH                                   6-Cl  C═O SCH.sub.3                                                                             SCH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   6-Cl  C═O SCH.sub.3                                                                             SCH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   6-Cl  C═O SCH.sub.3                                                                             SCH.sub.3                                                                            Cl    OCH.sub.3                                                                           CH                                   6-Cl  C═O SCH.sub.3                                                                             SCH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           N                                    6-Cl  C═O SCH.sub.3                                                                             SCH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    6-Cl  C═O SCH.sub.3                                                                             SCH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                                                                            N                                    6-Cl  SO.sub.2                                                                              CH.sub.3                                                                              SCH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                                                                            CH                                   6-Cl  SO.sub.2                                                                              CH.sub.3                                                                              SCH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   6-Cl  SO.sub.2                                                                              CH.sub.3                                                                              SCH.sub. 3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   6-Cl  SO.sub.2                                                                              CH.sub.3                                                                              SCH.sub.3                                                                            Cl    OCH.sub.3                                                                           CH                                   6-Cl  SO.sub.2                                                                              CH.sub.3                                                                              SCH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           N                                    6-Cl  SO.sub.2                                                                              CH.sub.3                                                                              SCH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    6-Cl  SO.sub.2                                                                              CH.sub.3                                                                              SCH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                                                                            N                                    6-Cl  CH.sub.2                                                                              CH.sub.3                                                                              SCH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                                                                            CH                                   6-Cl  CH.sub.2                                                                              CH.sub.3                                                                              SCH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   6-Cl  CH.sub.2                                                                              CH.sub.3                                                                              SCH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   6-Cl  CH.sub.2                                                                              CH.sub.3                                                                              SCH.sub.3                                                                            Cl    OCH.sub.3                                                                           CH                                   6-Cl  CH.sub.2                                                                              CH.sub.3                                                                              SCH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           N                                    6-Cl  CH.sub.2                                                                              CH.sub.3                                                                              SCH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    6-Cl  CH.sub.2                                                                              CH.sub.3                                                                              SCH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                                                                            N                                    5-OCH.sub.3                                                                         CH.sub.2                                                                              CH.sub.3                                                                              OCH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                                                                            CH                                   5-OCH.sub.3                                                                         CH.sub.2                                                                              CH.sub.3                                                                              OCH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   5-OCH.sub.3                                                                         CH.sub.2                                                                              CH.sub.3                                                                              OCH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   5-OCH.sub.3                                                                         CH.sub.2                                                                              CH.sub.3                                                                              OCH.sub.3                                                                            Cl    OCH.sub.3                                                                           CH                                   5-OCH.sub.3                                                                         CH.sub.2                                                                              CH.sub.3                                                                              OCH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           N                                    5-OCH.sub.3                                                                         CH.sub.2                                                                              CH.sub.3                                                                              OCH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    5-OCH.sub.3                                                                         CH.sub.2                                                                              CH.sub.3                                                                              OCH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                                                                            N                                    5-OCH.sub.3                                                                         CH.sub.2                                                                              CH.sub.3                                                                              CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            CH                                   5-OCH.sub.3                                                                         CH.sub.2                                                                              CH.sub.3                                                                              CH.sub.3                                                                             CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   5-OCH.sub.3                                                                         CH.sub.2                                                                              CH.sub.3                                                                              CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   5-OCH.sub.3                                                                         CH.sub.2                                                                              CH.sub.3                                                                              CH.sub.3                                                                             Cl    OCH.sub.3                                                                           CH                                   5-OCH.sub.3                                                                         CH.sub.2                                                                              CH.sub.3                                                                              CH.sub.3                                                                             CH.sub.3                                                                            OCH.sub.3                                                                           N                                    5-OCH.sub.3                                                                         CH.sub.2                                                                              CH.sub.3                                                                              CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    5-OCH.sub.3                                                                         CH.sub.2                                                                              CH.sub.3                                                                              CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            N                                    5-OCH.sub.3                                                                         C═O CH.sub.3                                                                              N(CH.sub.3).sub.2                                                                    CH.sub.3                                                                            CH.sub.3                                                                            CH                                   5-OCH.sub.3                                                                         C═O CH.sub.3                                                                              N(CH.sub.3).sub.2                                                                    CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   5-OCH.sub.3                                                                         C═O CH.sub.3                                                                              N(CH.sub.3).sub.2                                                                    OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   5-OCH.sub.3                                                                         C═O CH.sub.3                                                                              N(CH.sub.3).sub.2                                                                    Cl    OCH.sub.3                                                                           CH                                   5-OCH.sub.3                                                                         C═O CH.sub.3                                                                              N(CH.sub.3).sub.2                                                                    CH.sub.3                                                                            OCH.sub.3                                                                           N                                    5-OCH.sub.3                                                                         C═O CH.sub.3                                                                              N(CH.sub.3).sub.2                                                                    OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    5-OCH.sub.3                                                                         C═O CH.sub.3                                                                              N(CH.sub.3).sub.2                                                                    CH.sub.3                                                                            CH.sub.3                                                                            N                                    5-OCH.sub.3                                                                         C═O CH.sub.3                                                                              OCH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                                                                            CH                                   5-OCH.sub.3                                                                         C═O CH.sub.3                                                                              OCH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   5-OCH.sub.3                                                                         C═O CH.sub.3                                                                              OCH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   5-OCH.sub.3                                                                         C═O CH.sub.3                                                                              OCH.sub.3                                                                            Cl    OCH.sub.3                                                                           CH                                   5-OCH.sub.3                                                                         C═O CH.sub.3                                                                              OCH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           N                                    5-OCH.sub.3                                                                         C═O CH.sub.3                                                                              OCH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    5-OCH.sub.3                                                                         C═O CH.sub.3                                                                              OCH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                                                                            N                                    5-OCH.sub.3                                                                         SO.sub.2                                                                              CH.sub.3                                                                              OCH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                                                                            CH                                   5-OCH.sub.3                                                                         SO.sub.2                                                                              CH.sub.3                                                                              OCH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   5-OCH.sub.3                                                                         SO.sub.2                                                                              CH.sub.3                                                                              OCH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   5-OCH.sub.3                                                                         SO.sub.2                                                                              CH.sub.3                                                                              OCH.sub.3                                                                            Cl    OCH.sub.3                                                                           CH                                   5-OCH.sub.3                                                                         SO.sub.2                                                                              CH.sub.3                                                                              OCH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           N                                    5-OCH.sub.3                                                                         SO.sub.2                                                                              CH.sub.3                                                                              OCH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    5-OCH.sub.3                                                                         SO.sub.2                                                                              CH.sub.3                                                                              OCH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                                                                            N                                    ______________________________________                                    

                  TABLE 12                                                        ______________________________________                                        General Formula 12                                                            R.sub.1                                                                             J       R.sub.8 X      Y     Z     m.p. (°C.)                    ______________________________________                                        H     C═O H       CH.sub.3                                                                             CH.sub.3                                                                            CH                                         H     C═O H       CH.sub.3                                                                             OCH.sub.3                                                                           CH                                         H     C═O H       OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                         H     C═O H       Cl     OCH.sub.3                                                                           CH                                         H     C═O H       CH.sub.3                                                                             OCH.sub.3                                                                           N                                          H     C═O H       OCH.sub.3                                                                            OCH.sub.3                                                                           N                                          H     C═O H       CH.sub.3                                                                             CH.sub.3                                                                            N                                          H     C═O CH.sub.3                                                                              CH.sub.3                                                                             CH.sub.3                                                                            CH                                         H     C═O CH.sub.3                                                                              CH.sub.3                                                                             OCH.sub.3                                                                           CH                                         H     C═O CH.sub.3                                                                              OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                         H     C═O CH.sub.3                                                                              Cl     OCH.sub.3                                                                           CH                                         H     C═O CH.sub.3                                                                              CH.sub.3                                                                             OCH.sub.3                                                                           N                                          H     C═O CH.sub.3                                                                              OCH.sub.3                                                                            OCH.sub.3                                                                           N                                          H     C═O CH.sub.3                                                                              CH.sub.3                                                                             CH.sub.3                                                                            N                                          H     SO.sub.2                                                                              CH.sub.3                                                                              CH.sub.3                                                                             CH.sub.3                                                                            CH                                         H     SO.sub.2                                                                              CH.sub.3                                                                              CH.sub.3                                                                             OCH.sub.3                                                                           CH                                         H     SO.sub.2                                                                              CH.sub.3                                                                              OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                         H     SO.sub.2                                                                              CH.sub.3                                                                              Cl     OCH.sub.3                                                                           CH                                         H     SO.sub.2                                                                              CH.sub.3                                                                              CH.sub.3                                                                             OCH.sub.3                                                                           N                                          H     SO.sub.2                                                                              CH.sub.3                                                                              OCH.sub.3                                                                            OCH.sub.3                                                                           N                                          H     SO.sub.2                                                                              CH.sub.3                                                                              CH.sub.3                                                                             CH.sub.3                                                                            N                                          H     SO.sub.2                                                                              H       CH.sub.3                                                                             CH.sub.3                                                                            CH                                         H     SO.sub.2                                                                              H       CH.sub.3                                                                             OCH.sub.3                                                                           CH                                         H     SO.sub.2                                                                              H       OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                         H     SO.sub.2                                                                              H       Cl     OCH.sub.3                                                                           CH                                         H     SO.sub.2                                                                              H       CH.sub.3                                                                             OCH.sub.3                                                                           N                                          H     SO.sub.2                                                                              H       OCH.sub.3                                                                            OCH.sub.3                                                                           N                                          H     SO.sub.2                                                                              H       CH.sub.3                                                                             CH.sub.3                                                                            N                                          H     CH.sub.2                                                                              H       CH.sub.3                                                                             CH.sub.3                                                                            CH                                         H     CH.sub.2                                                                              H       CH.sub.3                                                                             OCH.sub.3                                                                           CH                                         H     CH.sub.2                                                                              H       OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                         H     CH.sub.2                                                                              H       Cl     OCH.sub.3                                                                           CH                                         H     CH.sub.2                                                                              H       CH.sub.3                                                                             OCH.sub.3                                                                           N                                          H     CH.sub.2                                                                              H       OCH.sub.3                                                                            OCH.sub.3                                                                           N                                          H     CH.sub.2                                                                              H       CH.sub.3                                                                             CH.sub.3                                                                            N                                          H     CH.sub.2                                                                              CH.sub.3                                                                              CH.sub.3                                                                             CH.sub.3                                                                            CH                                         H     CH.sub.2                                                                              CH.sub.3                                                                              CH.sub.3                                                                             OCH.sub.3                                                                           CH                                         H     CH.sub.2                                                                              CH.sub.3                                                                              OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                         H     CH.sub.2                                                                              CH.sub.3                                                                              Cl     OCH.sub.3                                                                           CH                                         H     CH.sub.2                                                                              CH.sub. 3                                                                             CH.sub.3                                                                             OCH.sub.3                                                                           N                                          H     CH.sub.2                                                                              CH.sub.3                                                                              OCH.sub.3                                                                            OCH.sub.3                                                                           N                                          H     CH.sub.2                                                                              CH.sub.3                                                                              CH.sub.3                                                                             CH.sub.3                                                                            N                                          5-OCH.sub.3                                                                         C═O H       CH.sub.3                                                                             CH.sub.3                                                                            CH                                         5-OCH.sub.3                                                                         C═O H       CH.sub.3                                                                             OCH.sub.3                                                                           CH                                         5-OCH.sub.3                                                                         C═O H       OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                         5-OCH.sub.3                                                                         C═O H       Cl     OCH.sub.3                                                                           CH                                         5-OCH.sub.3                                                                         C═O H       CH.sub.3                                                                             OCH.sub.3                                                                           N                                          5-OCH.sub.3                                                                         C═O H       OCH.sub.3                                                                            OCH.sub.3                                                                           N                                          5-OCH.sub.3                                                                         C═O H       CH.sub.3                                                                             CH.sub.3                                                                            N                                          5-OCH.sub.3                                                                         C═O CH.sub.3                                                                              CH.sub.3                                                                             CH.sub.3                                                                            CH                                         5-OCH.sub.3                                                                         C═O CH.sub.3                                                                              CH.sub.3                                                                             OCH.sub.3                                                                           CH                                         5-OCH.sub.3                                                                         C═O CH.sub.3                                                                              OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                         5-OCH.sub.3                                                                         C═O CH.sub.3                                                                              Cl     OCH.sub.3                                                                           CH                                         5-OCH.sub.3                                                                         C═O CH.sub.3                                                                              CH.sub.3                                                                             OCH.sub.3                                                                           N                                          5-OCH.sub.3                                                                         C═O CH.sub.3                                                                              OCH.sub.3                                                                            OCH.sub.3                                                                           N                                          5-OCH.sub.3                                                                         C═O CH.sub.3                                                                              CH.sub.3                                                                             CH.sub.3                                                                            N                                          5-OCH.sub.3                                                                         SO.sub.2                                                                              CH.sub.3                                                                              CH.sub.3                                                                             CH.sub.3                                                                            CH                                         5-OCH.sub.3                                                                         SO.sub.2                                                                              CH.sub.3                                                                              CH.sub.3                                                                             OCH.sub.3                                                                           CH                                         5-OCH.sub.3                                                                         SO.sub.2                                                                              CH.sub.3                                                                              OCH.sub. 3                                                                           OCH.sub.3                                                                           CH                                         5-OCH.sub.3                                                                         SO.sub.2                                                                              CH.sub.3                                                                              Cl     OCH.sub.3                                                                           CH                                         5-OCH.sub.3                                                                         SO.sub.2                                                                              CH.sub.3                                                                              CH.sub.3                                                                             OCH.sub.3                                                                           N                                          5-OCH.sub.3                                                                         SO.sub.2                                                                              CH.sub.3                                                                              OCH.sub.3                                                                            OCH.sub.3                                                                           N                                          5-OCH.sub.3                                                                         SO.sub.2                                                                              CH.sub.3                                                                              CH.sub.3                                                                             CH.sub.3                                                                            N                                          5-OCH.sub.3                                                                         SO.sub.2                                                                              H       CH.sub.3                                                                             CH.sub.3                                                                            CH                                         5-OCH.sub.3                                                                         SO.sub.2                                                                              H       CH.sub.3                                                                             OCH.sub.3                                                                           CH                                         5-OCH.sub.3                                                                         SO.sub.2                                                                              H       OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                         5-OCH.sub.3                                                                         SO.sub.2                                                                              H       Cl     OCH.sub.3                                                                           CH                                         5-OCH.sub.3                                                                         SO.sub.2                                                                              H       CH.sub.3                                                                             OCH.sub.3                                                                           N                                          5-OCH.sub.3                                                                         SO.sub.2                                                                              H       OCH.sub.3                                                                            OCH.sub.3                                                                           N                                          5-OCH.sub.3                                                                         SO.sub.2                                                                              H       CH.sub.3                                                                             CH.sub.3                                                                            N                                          5-OCH.sub.3                                                                         CH.sub.2                                                                              H       CH.sub.3                                                                             CH.sub.3                                                                            CH                                         5-OCH.sub.3                                                                         CH.sub.2                                                                              H       CH.sub.3                                                                             OCH.sub.3                                                                           CH                                         5-OCH.sub.3                                                                         CH.sub.2                                                                              H       OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                         5-OCH.sub.3                                                                         CH.sub.2                                                                              H       Cl     OCH.sub.3                                                                           CH                                         5-OCH.sub.3                                                                         CH.sub.2                                                                              H       CH.sub.3                                                                             OCH.sub.3                                                                           N                                          5-OCH.sub.3                                                                         CH.sub.2                                                                              H       OCH.sub.3                                                                            OCH.sub.3                                                                           N                                          5-OCH.sub.3                                                                         CH.sub.2                                                                              H       CH.sub.3                                                                             CH.sub.3                                                                            N                                          5-OCH.sub.3                                                                         CH.sub.2                                                                              CH.sub.3                                                                              CH.sub.3                                                                             CH.sub.3                                                                            CH                                         5-OCH.sub.3                                                                         CH.sub.2                                                                              CH.sub.3                                                                              CH.sub.3                                                                             OCH.sub.3                                                                           CH                                         5-OCH.sub.3                                                                         CH.sub.2                                                                              CH.sub.3                                                                              OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                         5-OCH.sub.3                                                                         CH.sub.2                                                                              CH.sub.3                                                                              Cl     OCH.sub.3                                                                           CH                                         5-OCH.sub.3                                                                         CH.sub.2                                                                              CH.sub.3                                                                              CH.sub.3                                                                             OCH.sub.3                                                                           N                                          5-OCH.sub.3                                                                         CH.sub.2                                                                              CH.sub.3                                                                              OCH.sub.3                                                                            OCH.sub.3                                                                           N                                          5-OCH.sub.3                                                                         CH.sub.2                                                                              CH.sub.3                                                                              CH.sub.3                                                                             CH.sub.3                                                                            N                                          ______________________________________                                    

                  TABLE 13                                                        ______________________________________                                        General Formula 13                                                            R.sub.1                                                                             G        R.sub.14                                                                              X      Y     Z    m.p. (°C.)                    ______________________________________                                        H     CH.sub.2 H       CH.sub.3                                                                             CH.sub.3                                                                            CH                                        H     CH.sub.2 H       CH.sub.3                                                                             OCH.sub.3                                                                           CH                                        H     CH.sub.2 H       OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     CH.sub.2 H       Cl     OCH.sub.3                                                                           CH                                        H     CH.sub.2 H       CH.sub.3                                                                             OCH.sub.3                                                                           N                                         H     CH.sub.2 H       OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         H     CH.sub.2 H       CH.sub.3                                                                             CH.sub.3                                                                            N                                         H     CH.sub.2 7-NO.sub.2                                                                            CH.sub.3                                                                             CH.sub.3                                                                            CH                                        H     CH.sub.2 7-NO.sub.2                                                                            CH.sub.3                                                                             OCH.sub.3                                                                           CH                                        H     CH.sub.2 7-NO.sub.2                                                                            OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     CH.sub.2 7-NO.sub.2                                                                            Cl     OCH.sub.3                                                                           CH                                        H     CH.sub.2 7-NO.sub.2                                                                            CH.sub.3                                                                             OCH.sub.3                                                                           N                                         H     CH.sub.2 7-NO.sub.2                                                                            OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         H     CH.sub.2 7-NO.sub.2                                                                            CH.sub.3                                                                             CH.sub.3                                                                            N                                         H     CH.sub.2 8-Cl    CH.sub.3                                                                             CH.sub.3                                                                            CH                                        H     CH.sub.2 8-Cl    CH.sub.3                                                                             OCH.sub.3                                                                           CH                                        H     CH.sub.2 8-Cl    OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     CH.sub.2 8-Cl    Cl     OCH.sub.3                                                                           CH                                        H     CH.sub.2 8-Cl    CH.sub.3                                                                             OCH.sub.3                                                                           N                                         H     CH.sub.2 8-Cl    OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         H     CH.sub.2 8-Cl    CH.sub.3                                                                             CH.sub.3                                                                            N                                         H     CH.sub.2 9-OCH.sub.3                                                                           CH.sub.3                                                                             CH.sub.3                                                                            CH                                        H     CH.sub.2 9-OCH.sub.3                                                                           CH.sub.3                                                                             OCH.sub.3                                                                           CH                                        H     CH.sub.2 9-OCH.sub.3                                                                           OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     CH.sub.2 9-OCH.sub.3                                                                           Cl     OCH.sub.3                                                                           CH                                        H     CH.sub.2 9-OCH.sub.3                                                                           H      OCH.sub.3                                                                           N                                         H     CH.sub.2 9-OCH.sub.3                                                                           OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         H     CH.sub.2 9-OCH.sub.3                                                                           CH.sub.3                                                                             CH.sub.3                                                                            N                                         H     CH.sub.2 10-CH.sub.3                                                                           CH.sub.3                                                                             CH.sub.3                                                                            CH                                        H     CH.sub.2 10-CH.sub.3                                                                           CH.sub.3                                                                             OCH.sub.3                                                                           CH                                        H     CH.sub.2 10-CH.sub.3                                                                           OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     CH.sub.2 10-CH.sub.3                                                                           Cl     OCH.sub.3                                                                           CH                                        H     CH.sub.2 10-CH.sub.3                                                                           CH.sub.3                                                                             OCH.sub.3                                                                           N                                         H     CH.sub.2 10-CH.sub.3                                                                           OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         H     CH.sub.2 10-CH.sub.3                                                                           CH.sub.3                                                                             CH.sub.3                                                                            N                                         H     CH.sub.2 7-F     CH.sub.3                                                                             CH.sub.3                                                                            CH                                        H     CH.sub.2 7-F     CH.sub.3                                                                             OCH.sub.3                                                                           CH                                        H     CH.sub.2 7-F     OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     CH.sub.2 7-F     Cl     OCH.sub.3                                                                           CH                                        H     CH.sub. 2                                                                              7-F     CH.sub.3                                                                             OCH.sub.3                                                                           N                                         H     CH.sub.2 7-F     OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         H     CH.sub.2 7-F     CH.sub.3                                                                             CH.sub.3                                                                            N                                         6-Cl  CH.sub.2 H       CH.sub.3                                                                             CH.sub.3                                                                            CH                                        6-Cl  CH.sub.2 H       CH.sub.3                                                                             OCH.sub.3                                                                           CH                                        6-Cl  CH.sub.2 H       OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-Cl  CH.sub.2 H       Cl     OCH.sub.3                                                                           CH                                        6-Cl  CH.sub.2 H       CH.sub.3                                                                             OCH.sub.3                                                                           N                                         6-Cl  CH.sub.2 H       OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         6-Cl  CH.sub.2 H       CH.sub.3                                                                             CH.sub.3                                                                            N                                         6-Cl  CH.sub.2 8-NO.sub.2                                                                            CH.sub.3                                                                             CH.sub.3                                                                            CH                                        6-Cl  CH.sub.2 8-NO.sub.2                                                                            CH.sub.3                                                                             OCH.sub.3                                                                           CH                                        6-Cl  CH.sub.2 8-NO.sub.2                                                                            OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-Cl  CH.sub.2 8-NO.sub.2                                                                            Cl     OCH.sub.3                                                                           CH                                        6-Cl  CH.sub.2 8-NO.sub.2                                                                            CH.sub.3                                                                             OCH.sub.3                                                                           N                                         6-Cl  CH.sub.2 8-NO.sub.2                                                                            OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         6-Cl  CH.sub.2 8-NO.sub.2                                                                            CH.sub.3                                                                             CH.sub.3                                                                            N                                         6-Cl  CH.sub.2 9-Cl    CH.sub.3                                                                             CH.sub.3                                                                            CH                                        6-Cl  CH.sub.2 9-Cl    CH.sub.3                                                                             OCH.sub.3                                                                           CH                                        6-Cl  CH.sub.2 9-Cl    OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-Cl  CH.sub.2 9-Cl    Cl     OCH.sub.3                                                                           CH                                        6-Cl  CH.sub.2 9-Cl    CH.sub.3                                                                             OCH.sub.3                                                                           N                                         6-Cl  CH.sub.2 9-Cl    OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         6-Cl  CH.sub.2 9-Cl    CH.sub.3                                                                             CH.sub.3                                                                            N                                         6-CH.sub.3                                                                          CH.sub.2 7-OCH.sub.3                                                                           CH.sub.3                                                                             CH.sub.3                                                                            CH                                        6-CH.sub.3                                                                          CH.sub.2 7-OCH.sub.3                                                                           CH.sub.3                                                                             OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          CH.sub.2 7-OCH.sub.3                                                                           OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          CH.sub.2 7-OCH.sub.3                                                                           Cl     OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          CH.sub.2 7-OCH.sub.3                                                                           H      OCH.sub.3                                                                           N                                         6-CH.sub.3                                                                          CH.sub.2 7-OCH.sub.3                                                                           OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         6-CH.sub.3                                                                          CH.sub.2 7-OCH.sub.3                                                                           CH.sub.3                                                                             CH.sub.3                                                                            N                                         6-CH.sub.3                                                                          CH.sub.2 10-CH.sub.3                                                                           CH.sub.3                                                                             CH.sub.3                                                                            CH                                        6-CH.sub.3                                                                          CH.sub.2 10-CH.sub.3                                                                           CH.sub.3                                                                             OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          CH.sub.2 10-CH.sub.3                                                                           OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          CH.sub.2 10-CH.sub.3                                                                           Cl     OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          CH.sub.2 10-CH.sub.3                                                                           CH.sub.3                                                                             OCH.sub.3                                                                           N                                         6-CH.sub.3                                                                          CH.sub.2 10-CH.sub.3                                                                           OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         6-CH.sub.3                                                                          CH.sub.2 10-CH.sub.3                                                                           CH.sub.3                                                                             CH.sub.3                                                                            N                                         6-CH.sub.3                                                                          CH.sub.2 9-F     CH.sub.3                                                                             CH.sub.3                                                                            CH                                        6-CH.sub.3                                                                          CH.sub.2 9-F     CH.sub.3                                                                             OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          CH.sub.2 9-F     OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-CH.sub. 3                                                                         CH.sub.2 9-F     Cl     OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          CH.sub.2 9-F     CH.sub.3                                                                             OCH.sub.3                                                                           N                                         6-CH.sub.3                                                                          CH.sub.2 9-F     OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         6-CH.sub.3                                                                          CH.sub.2 9-F     CH.sub.3                                                                             CH.sub.3                                                                            N                                         H     CH.sub.2 CH.sub.2                                                                      H       CH.sub.3                                                                             CH.sub.3                                                                            CH                                        H     CH.sub.2 CH.sub.2                                                                      H       CH.sub.3                                                                             OCH.sub.3                                                                           CH                                        H     CH.sub.2 CH.sub.2                                                                      H       OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     CH.sub.2 CH.sub.2                                                                      H       Cl     OCH.sub.3                                                                           CH                                        H     CH.sub.2 CH.sub.2                                                                      H       CH.sub.3                                                                             OCH.sub.3                                                                           N                                         H     CH.sub.2 CH.sub.2                                                                      H       OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         H     CH.sub.2 CH.sub.2                                                                      H       CH.sub.3                                                                             CH.sub.3                                                                            N                                         H     CH.sub.2 CH.sub.2                                                                      7-NO.sub.2                                                                            CH.sub.3                                                                             CH.sub.3                                                                            CH                                        H     CH.sub.2 CH.sub.2                                                                      7-NO.sub.2                                                                            CH.sub.3                                                                             OCH.sub.3                                                                           CH                                        H     CH.sub.2 CH.sub.2                                                                      7-NO.sub.2                                                                            OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     CH.sub.2 CH.sub.2                                                                      7-NO.sub.2                                                                            Cl     OCH.sub.3                                                                           CH                                        H     CH.sub.2 CH.sub.2                                                                      7-NO.sub.2                                                                            CH.sub.3                                                                             OCH.sub.3                                                                           N                                         H     CH.sub.2 CH.sub.2                                                                      7-NO.sub.2                                                                            OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         H     CH.sub.2 CH.sub.2                                                                      7-NO.sub.2                                                                            CH.sub.3                                                                             CH.sub.3                                                                            N                                         H     CH.sub.2 CH.sub.2                                                                      8-Cl    CH.sub.3                                                                             CH.sub.3                                                                            CH                                        H     CH.sub.2 CH.sub.2                                                                      8-Cl    CH.sub.3                                                                             OCH.sub.3                                                                           CH                                        H     CH.sub.2 CH.sub.2                                                                      8-Cl    OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     CH.sub.2 CH.sub.2                                                                      8-Cl    Cl     OCH.sub.3                                                                           CH                                        H     CH.sub.2 CH.sub.2                                                                      8-Cl    CH.sub.3                                                                             OCH.sub.3                                                                           N                                         H     CH.sub.2 CH.sub.2                                                                      8-Cl    OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         H     CH.sub.2 CH.sub.2                                                                      8-Cl    CH.sub.3                                                                             CH.sub.3                                                                            N                                         H     CH.sub.2 CH.sub.2                                                                      9-OCH.sub.3                                                                           CH.sub.3                                                                             CH.sub.3                                                                            CH                                        H     CH.sub.2 CH.sub.2                                                                      9-OCH.sub.3                                                                           CH.sub.3                                                                             OCH.sub.3                                                                           CH                                        H     CH.sub.2 CH.sub.2                                                                      9-OCH.sub.3                                                                           OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     CH.sub.2 CH.sub.2                                                                      9-OCH.sub.3                                                                           Cl     OCH.sub.3                                                                           CH                                        H     CH.sub.2 CH.sub.2                                                                      9-OCH.sub.3                                                                           H      OCH.sub.3                                                                           N                                         H     CH.sub.2 CH.sub.2                                                                      9-OCH.sub.3                                                                           OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         H     CH.sub.2 CH.sub.2                                                                      9-OCH.sub.3                                                                           CH.sub.3                                                                             CH.sub.3                                                                            N                                         H     CH.sub.2 CH.sub.2                                                                      10-CH.sub.3                                                                           CH.sub.3                                                                             CH.sub.3                                                                            CH                                        H     CH.sub.2 CH.sub.2                                                                      10-CH.sub.3                                                                           CH.sub.3                                                                             OCH.sub.3                                                                           CH                                        H     CH.sub.2 CH.sub.2                                                                      10-CH.sub.3                                                                           OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     CH.sub.2 CH.sub.2                                                                      10-CH.sub.3                                                                           Cl     OCH.sub. 3                                                                          CH                                        H     CH.sub.2 CH.sub.2                                                                      10-CH.sub.3                                                                           CH.sub.3                                                                             OCH.sub.3                                                                           N                                         H     CH.sub.2 CH.sub.2                                                                      10-CH.sub.3                                                                           OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         H     CH.sub.2 CH.sub.2                                                                      10-CH.sub.3                                                                           CH.sub.3                                                                             CH.sub.3                                                                            N                                         H     CH.sub.2 CH.sub.2                                                                      7-F     CH.sub.3                                                                             CH.sub.3                                                                            CH                                        H     CH.sub.2 CH.sub.2                                                                      7-F     CH.sub.3                                                                             OCH.sub.3                                                                           CH                                        H     CH.sub.2 CH.sub.2                                                                      7-F     OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     CH.sub.2 CH.sub.2                                                                      7-F     Cl     OCH.sub.3                                                                           CH                                        H     CH.sub.2 CH.sub.2                                                                      7-F     CH.sub.3                                                                             OCH.sub.3                                                                           N                                         H     CH.sub.2 CH.sub.2                                                                      7-F     OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         H     CH.sub.2 CH.sub.2                                                                      7-F     CH.sub.3                                                                             CH.sub.3                                                                            N                                         6-Cl  CH.sub.2 CH.sub.2                                                                      H       CH.sub.3                                                                             CH.sub.3                                                                            CH                                        6-Cl  CH.sub.2 CH.sub.2                                                                      H       CH.sub.3                                                                             OCH.sub.3                                                                           CH                                        6-Cl  CH.sub.2 CH.sub.2                                                                      H       OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-Cl  CH.sub.2 CH.sub.2                                                                      H       Cl     OCH.sub.3                                                                           CH                                        6-Cl  CH.sub.2 CH.sub.2                                                                      H       CH.sub.3                                                                             OCH.sub.3                                                                           N                                         6-Cl  CH.sub.2 CH.sub.2                                                                      H       OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         6-Cl  CH.sub.2 CH.sub.2                                                                      H       CH.sub.3                                                                             CH.sub.3                                                                            N                                         6-Cl  CH.sub.2 CH.sub.2                                                                      8-NO.sub.2                                                                            CH.sub.3                                                                             CH.sub. 3                                                                           CH                                        6-Cl  CH.sub.2 CH.sub.2                                                                      8-NO.sub.2                                                                            CH.sub.3                                                                             OCH.sub.3                                                                           CH                                        6-Cl  CH.sub.2 CH.sub.2                                                                      8-NO.sub.2                                                                            OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-Cl  CH.sub.2 CH.sub.2                                                                      8-NO.sub.2                                                                            Cl     OCH.sub.3                                                                           CH                                        6-Cl  CH.sub.2 CH.sub.2                                                                      8-NO.sub.2                                                                            CH.sub.3                                                                             OCH.sub.3                                                                           N                                         6-Cl  CH.sub.2 CH.sub.2                                                                      8-NO.sub.2                                                                            OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         6-Cl  CH.sub.2 CH.sub.2                                                                      8-NO.sub.2                                                                            CH.sub.3                                                                             CH.sub.3                                                                            N                                         6-Cl  CH.sub.2 CH.sub.2                                                                      9-Cl    CH.sub.3                                                                             CH.sub.3                                                                            CH                                        6-Cl  CH.sub.2 CH.sub.2                                                                      9-Cl    CH.sub.3                                                                             OCH.sub.3                                                                           CH                                        6-Cl  CH.sub.2 CH.sub.2                                                                      9-Cl    OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-Cl  CH.sub.2 CH.sub.2                                                                      9-Cl    Cl     OCH.sub.3                                                                           CH                                        6-Cl  CH.sub.2 CH.sub.2                                                                      9-Cl    CH.sub.3                                                                             OCH.sub.3                                                                           N                                         6-Cl  CH.sub.2 CH.sub.2                                                                      9-Cl    OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         6-Cl  CH.sub.2 CH.sub.2                                                                      9-Cl    CH.sub.3                                                                             CH.sub.3                                                                            N                                         6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                      7-OCH.sub.3                                                                           CH.sub.3                                                                             CH.sub.3                                                                            CH                                        6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                      7-OCH.sub.3                                                                           CH.sub.3                                                                             OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                      7-OCH.sub.3                                                                           OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                      7-OCH.sub.3                                                                           Cl     OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                      7-OCH.sub.3                                                                           H      OCH.sub.3                                                                           N                                         6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                      7-OCH.sub.3                                                                           OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                      7-OCH.sub.3                                                                           CH.sub.3                                                                             CH.sub.3                                                                            N                                         6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                      10-CH.sub.3                                                                           CH.sub.3                                                                             CH.sub.3                                                                            CH                                        6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                      10-CH.sub.3                                                                           CH.sub.3                                                                             OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                      10-CH.sub.3                                                                           OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                      10-CH.sub.3                                                                           Cl     OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                      10-CH.sub.3                                                                           CH.sub.3                                                                             OCH.sub.3                                                                           N                                         6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                      10-CH.sub.3                                                                           OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                      10-CH.sub.3                                                                           CH.sub.3                                                                             CH.sub.3                                                                            N                                         6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                      9-F     CH.sub.3                                                                             CH.sub.3                                                                            CH                                        6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                      9-F     CH.sub.3                                                                             OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                      9-F     OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                      9-F     Cl     OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                      9-F     CH.sub.3                                                                             OCH.sub.3                                                                           N                                         6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                      9-F     OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         6-CH.sub. 3                                                                         CH.sub.2 CH.sub.2                                                                      9-F     CH.sub.3                                                                             CH.sub.3                                                                            N                                         H     CH═CH                                                                              H       CH.sub.3                                                                             CH.sub.3                                                                            CH                                        H     CH═CH                                                                              H       CH.sub.3                                                                             OCH.sub.3                                                                           CH                                        H     CH═CH                                                                              H       OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     CH═CH                                                                              H       Cl     OCH.sub.3                                                                           CH                                        H     CH═CH                                                                              H       CH.sub.3                                                                             OCH.sub.3                                                                           N                                         H     CH═CH                                                                              H       OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         H     CH═CH                                                                              H       CH.sub.3                                                                             CH.sub.3                                                                            N                                         H     CH═CH                                                                              7-NO.sub.2                                                                            CH.sub.3                                                                             CH.sub.3                                                                            CH                                        H     CH═CH                                                                              7-NO.sub.2                                                                            CH.sub.3                                                                             OCH.sub.3                                                                           CH                                        H     CH═CH                                                                              7-NO.sub.2                                                                            OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     CH═CH                                                                              7-NO.sub.2                                                                            Cl     OCH.sub.3                                                                           CH                                        H     CH═CH                                                                              7-NO.sub.2                                                                            CH.sub.3                                                                             OCH.sub.3                                                                           N                                         H     CH═CH                                                                              7-NO.sub.2                                                                            OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         H     CH═CH                                                                              7-NO.sub.2                                                                            CH.sub.3                                                                             CH.sub.3                                                                            N                                         H     CH═CH                                                                              8-Cl    CH.sub.3                                                                             CH.sub.3                                                                            CH                                        H     CH═CH                                                                              8-Cl    CH.sub.3                                                                             OCH.sub.3                                                                           CH                                        H     CH═CH                                                                              8-Cl    OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     CH═CH                                                                              8-Cl    Cl     OCH.sub.3                                                                           CH                                        H     CH═CH                                                                              8-Cl    CH.sub.3                                                                             OCH.sub.3                                                                           N                                         H     CH═CH                                                                              8-Cl    OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         H     CH═CH                                                                              8-Cl    CH.sub. 3                                                                            CH.sub.3                                                                            N                                         H     CH═CH                                                                              9-OCH.sub.3                                                                           CH.sub.3                                                                             CH.sub.3                                                                            CH                                        H     CH═CH                                                                              9-OCH.sub.3                                                                           CH.sub.3                                                                             OCH.sub.3                                                                           CH                                        H     CH═CH                                                                              9-OCH.sub.3                                                                           OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     CH═CH                                                                              9-OCH.sub.3                                                                           Cl     OCH.sub.3                                                                           CH                                        H     CH═CH                                                                              9-OCH.sub.3                                                                           H      OCH.sub.3                                                                           N                                         H     CH═CH                                                                              9-OCH.sub.3                                                                           OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         H     CH═CH                                                                              9-OCH.sub.3                                                                           CH.sub.3                                                                             CH.sub.3                                                                            N                                         H     CH═CH                                                                              10-CH.sub.3                                                                           CH.sub.3                                                                             CH.sub.3                                                                            CH                                        H     CH═CH                                                                              10-CH.sub.3                                                                           CH.sub.3                                                                             OCH.sub.3                                                                           CH                                        H     CH═CH                                                                              10-CH.sub.3                                                                           OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     CH═CH                                                                              10-CH.sub.3                                                                           Cl     OCH.sub.3                                                                           CH                                        H     CH═CH                                                                              10-CH.sub.3                                                                           CH.sub.3                                                                             OCH.sub.3                                                                           N                                         H     CH═CH                                                                              10-CH.sub.3                                                                           OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         H     CH═CH                                                                              10-CH.sub.3                                                                           CH.sub.3                                                                             CH.sub.3                                                                            N                                         H     CH═CH                                                                              7-F     CH.sub.3                                                                             CH.sub.3                                                                            CH                                        H     CH═CH                                                                              7-F     CH.sub.3                                                                             OCH.sub.3                                                                           CH                                        H     CH═CH                                                                              7-F     OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     CH═CH                                                                              7-F     Cl     OCH.sub.3                                                                           CH                                        H     CH═CH                                                                              7-F     CH.sub.3                                                                             OCH.sub.3                                                                           N                                         H     CH═CH                                                                              7-F     OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         H     CH═CH                                                                              7-F     CH.sub.3                                                                             CH.sub.3                                                                            N                                         6-Cl  CH═CH                                                                              H       CH.sub.3                                                                             CH.sub.3                                                                            CH                                        6-Cl  CH═CH                                                                              H       CH.sub.3                                                                             OCH.sub.3                                                                           CH                                        6-Cl  CH═CH                                                                              H       OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-Cl  CH═CH                                                                              H       Cl     OCH.sub.3                                                                           CH                                        6-Cl  CH═CH                                                                              H       CH.sub.3                                                                             OCH.sub.3                                                                           N                                         6-Cl  CH═CH                                                                              H       OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         6-Cl  CH═CH                                                                              H       CH.sub.3                                                                             CH.sub.3                                                                            N                                         6-Cl  CH═CH                                                                              8-NO.sub.2                                                                            CH.sub.3                                                                             CH.sub.3                                                                            CH                                        6-Cl  CH═CH                                                                              8-NO.sub.2                                                                            CH.sub.3                                                                             OCH.sub.3                                                                           CH                                        6-Cl  CH═CH                                                                              8-NO.sub.2                                                                            OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-Cl  CH═CH                                                                              8-NO.sub.2                                                                            Cl     OCH.sub.3                                                                           CH                                        6-Cl  CH═CH                                                                              8-NO.sub.2                                                                            CH.sub.3                                                                             OCH.sub.3                                                                           N                                         6-Cl  CH═CH                                                                              8-NO.sub.2                                                                            OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         6-Cl  CH═CH                                                                              8-NO.sub.2                                                                            CH.sub.3                                                                             CH.sub.3                                                                            N                                         6-Cl  CH═CH                                                                              9-Cl    CH.sub.3                                                                             CH.sub.3                                                                            CH                                        6-Cl  CH═CH                                                                              9-Cl    CH.sub.3                                                                             OCH.sub.3                                                                           CH                                        6-Cl  CH═CH                                                                              9-Cl    OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-Cl  CH═CH                                                                              9-Cl    Cl     OCH.sub.3                                                                           CH                                        6-Cl  CH═CH                                                                              9-Cl    CH.sub.3                                                                             OCH.sub.3                                                                           N                                         6-Cl  CH═CH                                                                              9-Cl    OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         6-Cl  CH═CH                                                                              9-Cl    CH.sub.3                                                                             CH.sub.3                                                                            N                                         6-CH.sub.3                                                                          CH═CH                                                                              7-OCH.sub.3                                                                           CH.sub.3                                                                             CH.sub.3                                                                            CH                                        6-CH.sub.3                                                                          CH═CH                                                                              7-OCH.sub.3                                                                           CH.sub.3                                                                             OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          CH═CH                                                                              7-OCH.sub.3                                                                           OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          CH═CH                                                                              7-OCH.sub.3                                                                           Cl     OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          CH═CH                                                                              7-OCH.sub.3                                                                           H      OCH.sub.3                                                                           N                                         6-CH.sub.3                                                                          CH═CH                                                                              7-OCH.sub.3                                                                           OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         6-CH.sub.3                                                                          CH═CH                                                                              7-OCH.sub.3                                                                           CH.sub.3                                                                             CH.sub.3                                                                            N                                         6-CH.sub.3                                                                          CH═CH                                                                              10-CH.sub.3                                                                           CH.sub.3                                                                             CH.sub.3                                                                            CH                                        6-CH.sub.3                                                                          CH═CH                                                                              10-CH.sub.3                                                                           CH.sub.3                                                                             OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          CH═CH                                                                              10-CH.sub.3                                                                           OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          CH═CH                                                                              10-CH.sub.3                                                                           Cl     OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          CH═CH                                                                              10-CH.sub.3                                                                           CH.sub.3                                                                             OCH.sub.3                                                                           N                                         6-CH.sub.3                                                                          CH═CH                                                                              9-F     CH.sub.3                                                                             CH.sub.3                                                                            CH                                        6-CH.sub.3                                                                          CH═CH                                                                              9-F     CH.sub.3                                                                             OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          CH═CH                                                                              9-F     OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          CH═CH                                                                              9-F     Cl     OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          CH═CH                                                                              9-F     CH.sub.3                                                                             OCH.sub.3                                                                           N                                         6-CH.sub.3                                                                          CH═CH                                                                              9-F     OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         6-CH.sub.3                                                                          CH═CH                                                                              9-F     CH.sub. 3                                                                            CH.sub.3                                                                            N                                         ______________________________________                                    

                  TABLE 14                                                        ______________________________________                                        General Formula 14                                                                                                            m.p.                          R   R.sub.1 J        E    n   X      Y     Z    (°C.)                  ______________________________________                                        H   H       CH.sub.2 N    0   CH.sub.3                                                                             CH.sub.3                                                                            CH                                 H   H       CH.sub.2 N    0   CH.sub.3                                                                             OCH.sub.3                                                                           CH                                 H   H       CH.sub.2 N    0   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                 H   H       CH.sub.2 N    0   CH.sub.3                                                                             CH.sub.3                                                                            N                                  H   H       CH.sub.2 N    0   CH.sub.3                                                                             OCH.sub.3                                                                           N                                  H   H       CH.sub.2 N    0   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                  H   H       CH.sub.2 N    1   CH.sub.3                                                                             CH.sub.3                                                                            CH                                 H   H       CH.sub.2 N    1   CH.sub.3                                                                             OCH.sub.3                                                                           CH                                 H   H       CH.sub.2 N    1   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                 H   H       CH.sub.2 N    1   CH.sub.3                                                                             CH.sub.3                                                                            N                                  H   H       CH.sub.2 N    1   CH.sub.3                                                                             OCH.sub.3                                                                           N                                  H   H       CH.sub.2 N    1   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                  H   H       CH.sub.2 N    1   OCH.sub.3                                                                            Cl    CH                                 CH.sub.3                                                                          H       C═O  N    0   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                 H   H       C═O  CH   0   CH.sub.3                                                                             CH.sub.3                                                                            CH                                 H   H       C═O  CH   0   CH.sub.3                                                                             OCH.sub.3                                                                           CH                                 H   H       C═O  CH   0   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                 H   H       C═O  CH   0   CH.sub.3                                                                             CH.sub.3                                                                            N                                  H   H       C═O  CH   0   CH.sub.3                                                                             OCH.sub.3                                                                           N                                  H   H       C═O  CH   0   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                  H   H       C═O  CH   1   CH.sub.3                                                                             CH.sub.3                                                                            CH                                 H   H       C═O  CH   1   CH.sub.3                                                                             OCH.sub.3                                                                           CH                                 H   H       C═O  CH   1   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                 H   H       C═O  CH   1   CH.sub.3                                                                             CH.sub.3                                                                            N                                  H   H       C═O  CH   1   CH.sub.3                                                                             OCH.sub.3                                                                           N                                  H   H       C═O  CH   1   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                  H   H       C═O  CH   1   OCH.sub.3                                                                            Cl    CH                                 H   CH.sub.3                                                                              C═O  CH   1   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                 H   6-CH.sub.3                                                                            CH.sub.2 N    0   CH.sub.3                                                                             CH.sub.3                                                                            CH                                 H   6-CH.sub.3                                                                            CH.sub.2 N    0   CH.sub.3                                                                             OCH.sub.3                                                                           CH                                 H   6-CH.sub.3                                                                            CH.sub.2 N    0   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                 H   6-CH.sub.3                                                                            CH.sub.2 N    0   CH.sub.3                                                                             CH.sub. 3                                                                           N                                  H   6-CH.sub.3                                                                            CH.sub.2 N    0   CH.sub.3                                                                             OCH.sub.3                                                                           N                                  H   6-CH.sub.3                                                                            CH.sub.2 N    0   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                  H   6-CH.sub.3                                                                            CH.sub.2 N    1   CH.sub.3                                                                             CH.sub.3                                                                            CH                                 H   6-CH.sub.3                                                                            CH.sub.2 N    1   CH.sub.3                                                                             OCH.sub.3                                                                           CH                                 H   6-CH.sub.3                                                                            CH.sub.2 N    1   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                 H   6-CH.sub.3                                                                            CH.sub.2 N    1   CH.sub.3                                                                             CH.sub.3                                                                            N                                  H   6-CH.sub.3                                                                            CH.sub.2 N    1   CH.sub.3                                                                             OCH.sub.3                                                                           N                                  H   6-CH.sub.3                                                                            CH.sub.2 N    1   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                  H   6-CH.sub.3                                                                            CH.sub.2 N    1   OCH.sub.3                                                                            Cl    CH                                 CH.sub.3                                                                          6-CH.sub.3                                                                            CH.sub.2 N    0   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                 H   6-CH.sub.3                                                                            C═O  CH   0   CH.sub.3                                                                             CH.sub.3                                                                            CH                                 H   6-CH.sub.3                                                                            C═O  CH   0   CH.sub.3                                                                             OCH.sub.3                                                                           CH                                 H   6-CH.sub.3                                                                            C═O  CH   0   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                 H   6-CH.sub.3                                                                            C═O  CH   0   CH.sub.3                                                                             CH.sub.3                                                                            N                                  H   6-CH.sub.3                                                                            C═O  CH   0   CH.sub.3                                                                             OCH.sub.3                                                                           N                                  H   6-CH.sub.3                                                                            C═O  CH   0   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                  H   6-CH.sub.3                                                                            C═O  CH   1   CH.sub.3                                                                             CH.sub.3                                                                            CH                                 H   6-CH.sub.3                                                                            C═O  CH   1   CH.sub.3                                                                             OCH.sub.3                                                                           CH                                 H   6-CH.sub.3                                                                            C═O  CH   1   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                 H   6-CH.sub.3                                                                            C═O  CH   1   CH.sub.3                                                                             CH.sub.3                                                                            N                                  H   6-CH.sub.3                                                                            C═O  CH   1   CH.sub.3                                                                             OCH.sub.3                                                                           N                                  H   6-CH.sub.3                                                                            C═O  CH   1   OCH.sub.3                                                                            OCH.sub.3                                                                           N                                  H   6-CH.sub.3                                                                            C═O  CH   1   OCH.sub.3                                                                            Cl    CH                                 H   6-CH.sub.3                                                                            C═O  CH   1   OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                 ______________________________________                                    

                  TABLE 15                                                        ______________________________________                                        General Formula 15                                                                                                          m.p.                            R.sub.1                                                                             G        W'      R.sub.9                                                                             X     Y     Z    (°C.)                    ______________________________________                                        H     CH.sub.2 O       H     CH.sub.3                                                                            CH.sub.3                                                                            CH                                   H     CH.sub.2 O       H     CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   H     CH.sub.2 O       H     OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   H     CH.sub.2 O       H     Cl    OCH.sub.3                                                                           CH                                   H     CH.sub.2 O       H     CH.sub.3                                                                            OCH.sub.3                                                                           N                                    H     CH.sub.2 O       H     OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    H     CH.sub.2 O       H     CH.sub.3                                                                            CH.sub.3                                                                            N                                    H     CH.sub.2 S       CH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                                                                            CH                                   H     CH.sub.2 S       CH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   H     CH.sub.2 S       CH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   H     CH.sub.2 S       CH.sub.3                                                                            Cl    OCH.sub.3                                                                           CH                                   H     CH.sub.2 S       CH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           N                                    H     CH.sub.2 S       CH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    H     CH.sub.2 S       CH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                                                                            N                                    H     CH.sub.2 NH      H     CH.sub.3                                                                            CH.sub.3                                                                            CH                                   H     CH.sub.2 NH      H     CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   H     CH.sub.2 NH      H     OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   H     CH.sub.2 NH      H     Cl    OCH.sub.3                                                                           CH                                   H     CH.sub.2 NH      H     CH.sub.3                                                                            OCH.sub.3                                                                           N                                    H     CH.sub.2 NH      H     OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    H     CH.sub.2 NH      H     CH.sub.3                                                                            CH.sub.3                                                                            N                                    6-Cl  CH.sub.2 O       H     CH.sub.3                                                                            CH.sub.3                                                                            CH                                   6-Cl  CH.sub.2 O       H     CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   6-Cl  CH.sub.2 O       H     OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   6-Cl  CH.sub.2 O       H     Cl    OCH.sub.3                                                                           CH                                   6-Cl  CH.sub.2 O       H     CH.sub.3                                                                            OCH.sub.3                                                                           N                                    6-Cl  CH.sub.2 O       H     OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    6-Cl  CH.sub.2 O       H     CH.sub.3                                                                            CH.sub.3                                                                            N                                    6-Cl  CH.sub.2 S       CH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                                                                            CH                                   6-Cl  CH.sub.2 S       CH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   6-Cl  CH.sub.2 S       CH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   6-Cl  CH.sub.2 S       CH.sub.3                                                                            Cl    OCH.sub.3                                                                           CH                                   6-Cl  CH.sub.2 S       CH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           N                                    6-Cl  CH.sub.2 S       CH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    6-Cl  CH.sub.2 S       CH.sub.3                                                                            CH.sub.3                                                                            CH.sub. 3                                                                           N                                    6-Cl  CH.sub.2 NH      H     CH    CH.sub.3                                                                            CH                                   6-Cl  CH.sub.2 NH      H     CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   6-Cl  CH.sub.2 NH      H     OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   6-Cl  CH.sub.2 NH      H     Cl    OCH.sub.3                                                                           CH                                   6-Cl  CH.sub.2 NH      H     CH.sub.3                                                                            OCH.sub.3                                                                           N                                    6-Cl  CH.sub.2 NH      H     OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    6-Cl  CH.sub.2 NH      H     CH.sub.3                                                                            CH.sub.3                                                                            N                                    H     CH.sub.2 S       H     OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   H     CH.sub.2 S       H     CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   H     CH.sub.2 S       H     CH.sub.3                                                                            CH.sub.3                                                                            CH                                   H     CH.sub.2 S       H     CH.sub.3                                                                            OCH.sub.3                                                                           N                                    H     CH.sub.2 S       H     OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    H     CH.sub.2 S       H     Cl    OCH.sub.3                                                                           CH                                   H     CH.sub.2 NCH.sub.3                                                                             H     OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   H     CH.sub.2 NCH.sub.3                                                                             H     CH.sub.3                                                                            OCH.sub.3                                                                           N                                    H     CH.sub.2 CH.sub.2                                                                      O       H     CH.sub.3                                                                            CH.sub.3                                                                            CH                                   H     CH.sub.2 CH.sub.2                                                                      O       H     CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   H     CH.sub.2 CH.sub.2                                                                      O       H     OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   H     CH.sub.2 CH.sub.2                                                                      O       H     Cl    OCH.sub.3                                                                           CH                                   H     CH.sub. 2 CH.sub.2                                                                     O       H     CH.sub.3                                                                            OCH.sub.3                                                                           N                                    H     CH.sub.2 CH.sub.2                                                                      O       H     OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    H     CH.sub.2 CH.sub.2                                                                      O       H     CH.sub.3                                                                            CH.sub.3                                                                            N                                    H     CH.sub.2 CH.sub.2                                                                      S       CH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                                                                            CH                                   H     CH.sub.2 CH.sub.2                                                                      S       CH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   H     CH.sub.2 CH.sub.2                                                                      S       CH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   H     CH.sub.2 CH.sub.2                                                                      S       CH.sub.3                                                                            Cl    OCH.sub.3                                                                           CH                                   H     CH.sub.2 CH.sub.2                                                                      S       CH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           N                                    H     CH.sub.2 CH.sub.2                                                                      S       CH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    H     CH.sub.2 CH.sub.2                                                                      S       CH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                                                                            N                                    H     CH.sub.2 CH.sub.2                                                                      NH      H     CH.sub.3                                                                            CH.sub.3                                                                            CH                                   H     CH.sub.2 CH.sub.2                                                                      NH      H     CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   H     CH.sub.2 CH.sub.2                                                                      NH      H     OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   H     CH.sub.2 CH.sub.2                                                                      NH      H     Cl    OCH.sub.3                                                                           CH                                   H     CH.sub.2 CH.sub.2                                                                      NH      H     CH.sub.3                                                                            OCH.sub.3                                                                           N                                    H     CH.sub.2 CH.sub.2                                                                      NH      H     OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    H     CH.sub.2 CH.sub.2                                                                      NH      H     CH.sub.3                                                                            CH.sub.3                                                                            N                                    6-Cl  CH.sub.2 CH.sub.2                                                                      O       H     CH.sub.3                                                                            CH.sub.3                                                                            CH                                   6-Cl  CH.sub.2 CH.sub.2                                                                      O       H     CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   6-Cl  CH.sub.2 CH.sub.2                                                                      O       H     OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   6-Cl  CH.sub.2 CH.sub.2                                                                      O       H     Cl    OCH.sub.3                                                                           CH                                   6-Cl  CH.sub.2 CH.sub.2                                                                      O       H     CH.sub.3                                                                            OCH.sub.3                                                                           N                                    6-Cl  CH.sub.2 CH.sub.2                                                                      O       H     OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    6-Cl  CH.sub.2 CH.sub.2                                                                      O       H     CH.sub.3                                                                            CH.sub.3                                                                            N                                    6-Cl  CH.sub.2 CH.sub.2                                                                      S       CH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                                                                            CH                                   6-Cl  CH.sub.2 CH.sub.2                                                                      S       CH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   6-Cl  CH.sub.2 CH.sub.2                                                                      S       CH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   6-Cl  CH.sub.2 CH.sub.2                                                                      S       CH.sub.3                                                                            Cl    OCH.sub.3                                                                           CH                                   6-Cl  CH.sub.2 CH.sub.2                                                                      S       CH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           N                                    6-Cl  CH.sub.2 CH.sub.2                                                                      S       CH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    6-Cl  CH.sub.2 CH.sub.2                                                                      S       CH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                                                                            N                                    6-Cl  CH.sub.2 CH.sub.2                                                                      NH      H     CH    CH.sub.3                                                                            CH                                   6-Cl  CH.sub.2 CH.sub.2                                                                      NH      H     CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   6-Cl  CH.sub.2 CH.sub.2                                                                      NH      H     OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   6-Cl  CH.sub.2 CH.sub.2                                                                      NH      H     Cl    OCH.sub.3                                                                           CH                                   6-Cl  CH.sub.2 CH.sub.2                                                                      NH      H     CH.sub.3                                                                            OCH.sub.3                                                                           N                                    6-Cl  CH.sub.2 CH.sub.2                                                                      NH      H     OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    6-Cl  CH.sub.2 CH.sub.2                                                                      NH      H     CH.sub.3                                                                            CH.sub.3                                                                            N                                    H     CH.sub.2 CH.sub.2                                                                      S       H     OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   H     CH.sub.2 CH.sub.2                                                                      S       H     CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   H     CH.sub.2 CH.sub.2                                                                      S       H     CH.sub.3                                                                            CH.sub.3                                                                            CH                                   H     CH.sub.2 CH.sub.2                                                                      S       H     CH.sub.3                                                                            OCH.sub.3                                                                           N                                    H     CH.sub.2 CH.sub.2                                                                      S       H     OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    H     CH.sub.2 CH.sub.2                                                                      S       H     Cl    OCH.sub.3                                                                           CH                                   H     CH.sub.2 CH.sub.2                                                                      NCH.sub.3                                                                             H     OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   H     CH.sub.2 CH.sub.2                                                                      NCH.sub.3                                                                             H     CH.sub.3                                                                            OCH.sub.3                                                                           N                                    H     CH═CH                                                                              O       H     CH.sub.3                                                                            CH.sub.3                                                                            CH                                   H     CH═CH                                                                              O       H     CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   H     CH═CH                                                                              O       H     OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   H     CH═CH                                                                              O       H     Cl    OCH.sub.3                                                                           CH                                   H     CH═CH                                                                              O       H     CH.sub.3                                                                            OCH.sub.3                                                                           N                                    H     CH═CH                                                                              O       H     OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    H     CH═CH                                                                              O       H     CH.sub.3                                                                            CH.sub.3                                                                            N                                    H     CH═CH                                                                              S       CH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                                                                            CH                                   H     CH═CH                                                                              S       CH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   H     CH═CH                                                                              S       CH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   H     CH═CH                                                                              S       CH.sub.3                                                                            Cl    OCH.sub.3                                                                           CH                                   H     CH═CH                                                                              S       CH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           N                                    H     CH═CH                                                                              S       CH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    H     CH═CH                                                                              S       CH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                                                                            N                                    H     CH═CH                                                                              NH      H     CH.sub.3                                                                            CH.sub.3                                                                            CH                                   H     CH═CH                                                                              NH      H     CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   H     CH═CH                                                                              NH      H     OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   H     CH═CH                                                                              NH      H     Cl    OCH.sub.3                                                                           CH                                   H     CH═CH                                                                              NH      H     CH.sub.3                                                                            OCH.sub.3                                                                           N                                    H     CH═CH                                                                              NH      H     OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    H     CH═CH                                                                              NH      H     CH.sub.3                                                                            CH.sub.3                                                                            N                                    6-Cl  CH═CH                                                                              O       H     CH.sub.3                                                                            CH.sub.3                                                                            CH                                   6-Cl  CH═CH                                                                              O       H     CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   6-Cl  CH═CH                                                                              O       H     OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   6-Cl  CH═CH                                                                              O       H     Cl    OCH.sub.3                                                                           CH                                   6-Cl  CH═CH                                                                              O       H     CH.sub.3                                                                            OCH.sub.3                                                                           N                                    6-Cl  CH═CH                                                                              O       H     OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    6-Cl  CH═CH                                                                              O       H     CH.sub.3                                                                            CH.sub.3                                                                            N                                    6-Cl  CH═CH                                                                              S       CH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                                                                            CH                                   6-Cl  CH═CH                                                                              S       CH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   6-Cl  CH═CH                                                                              S       CH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   6-Cl  CH═CH                                                                              S       CH.sub.3                                                                            Cl    OCH.sub.3                                                                           CH                                   6-Cl  CH═CH                                                                              S       CH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           N                                    6-Cl  CH═CH                                                                              S       CH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    6-Cl  CH═CH                                                                              S       CH.sub.3                                                                            CH.sub.3                                                                            CH.sub.3                                                                            N                                    6-Cl  CH═CH                                                                              NH      H     CH    CH.sub.3                                                                            CH                                   6-Cl  CH═CH                                                                              NH      H     CH.sub.3                                                                            OCH.sub.3                                                                           CH                                   6-Cl  CH═CH                                                                              NH      H     OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   6-Cl  CH═CH                                                                              NH      H     Cl    OCH.sub.3                                                                           CH                                   6-Cl  CH═CH                                                                              NH      H     CH.sub.3                                                                            OCH.sub.3                                                                           N                                    6-Cl  CH═CH                                                                              NH      H     OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    6-Cl  CH═CH                                                                              NH      H     CH.sub.3                                                                            CH.sub.3                                                                            N                                    H     CH═CH                                                                              S       H     OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   H     CH═CH                                                                              S       H     CH.sub. 3                                                                           OCH.sub.3                                                                           CH                                   H     CH═CH                                                                              S       H     CH.sub.3                                                                            CH.sub.3                                                                            CH                                   H     CH═CH                                                                              S       H     CH.sub.3                                                                            OCH.sub.3                                                                           N                                    H     CH═CH                                                                              S       H     OCH.sub.3                                                                           OCH.sub.3                                                                           N                                    H     CH═CH                                                                              S       H     Cl    OCH.sub.3                                                                           CH                                   H     CH═CH                                                                              NCH.sub.3                                                                             H     OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                   H     CH═CH                                                                              NCH.sub.3                                                                             H     CH.sub.3                                                                            OCH.sub.3                                                                           N                                    ______________________________________                                    

                  TABLE 16                                                        ______________________________________                                        General Formula 16                                                            R.sub.1 G        X        Y      Z     m.p. (20 C.)                           ______________________________________                                        H       CH.sub.2 OCH.sub.3                                                                              OCH.sub.3                                                                            CH                                           H       CH.sub.2 CH.sub.3 OCH.sub.3                                                                            CH                                           H       CH.sub.2 Cl       OCH.sub.3                                                                            CH                                           H       CH.sub.2 CH.sub.3 CH.sub.3                                                                             CH                                           H       CH.sub.2 OCH.sub.3                                                                              OCH.sub.3                                                                            N                                            H       CH.sub.2 CH.sub.3 OCH.sub.3                                                                            N                                            H       CH.sub.2 CH.sub.2                                                                      OCH.sub.3                                                                              OCH.sub.3                                                                            CH                                           H       CH.sub.2 CH.sub.2                                                                      CH.sub.3 OCH.sub.3                                                                            CH                                           H       CH.sub.2 CH.sub.2                                                                      Cl       OCH.sub.3                                                                            CH                                           H       CH.sub.2 CH.sub.2                                                                      CH.sub.3 CH.sub.3                                                                             CH                                           H       CH.sub.2 CH.sub.2                                                                      OCH.sub.3                                                                              OCH.sub.3                                                                            N                                            H       CH.sub.2 CH.sub.2                                                                      CH.sub.3 OCH.sub.3                                                                            N                                            H       CH═CH                                                                              OCH.sub.3                                                                              OCH.sub.3                                                                            CH                                           H       CH═CH                                                                              OCH.sub.3                                                                              OCH.sub.3                                                                            N                                            H       CH═CH                                                                              CH.sub.3 OCH.sub.3                                                                            CH                                           H       CH═CH                                                                              CH.sub.3 CH.sub.3                                                                             CH                                           H       CH═CH                                                                              CH.sub.3 OCH.sub.3                                                                            N                                            H       CH═CH                                                                              Cl       OCH.sub.3                                                                            N                                            6-CH.sub.3                                                                            CH.sub.2 OCH.sub.3                                                                              OCH.sub.3                                                                            CH                                           6-CH.sub.3                                                                            CH.sub.2 CH.sub.3 OCH.sub.3                                                                            CH                                           6-CH.sub.3                                                                            CH.sub.2 CH.sub.3 OCH.sub.3                                                                            N                                            6-Cl    CH.sub.2 OCH.sub.3                                                                              OCH.sub.3                                                                            CH                                           6-Cl    CH.sub.2 OCH.sub.3                                                                              OCH.sub.3                                                                            N                                            6-Cl    CH.sub.2 CH.sub.3 OCH.sub.3                                                                            CH                                           5-OCH.sub.3                                                                           CH.sub.2 OCH.sub.3                                                                              OCH.sub.3                                                                            CH                                           5-OCH.sub.3                                                                           CH.sub.2 CH.sub.3 OCH.sub.3                                                                            CH                                           6-CH.sub.3                                                                            CH.sub.2 CH.sub.2                                                                      OCH.sub.3                                                                              OCH.sub.3                                                                            CH                                           6-CH.sub.3                                                                            CH.sub.2 CH.sub.2                                                                      CH.sub.3 OCH.sub.3                                                                            CH                                           6-Cl    CH.sub.2 CH.sub.2                                                                      OCH.sub.3                                                                              OCH.sub.3                                                                            CH                                           6-Cl    CH.sub.2 CH.sub.2                                                                      CH.sub.3 OCH.sub.3                                                                            CH                                           5-OCH.sub.3                                                                           CH.sub.2 CH.sub.2                                                                      OCH.sub.3                                                                              OCH.sub.3                                                                            CH                                           5-OCH.sub.3                                                                           CH.sub.2 CH.sub.2                                                                      CH.sub.3 OCH.sub.3                                                                            CH                                           6-CH.sub.3                                                                            CH═CH                                                                              OCH.sub.3                                                                              OCH.sub.3                                                                            CH                                           6-CH.sub.3                                                                            CH═CH                                                                              CH.sub.3 OCH.sub.3                                                                            CH                                           6-Cl    CH═CH                                                                              OCH.sub.3                                                                              OCH.sub.3                                                                            CH                                           6-Cl    CH═CH                                                                              CH.sub.3 OCH.sub.3                                                                            CH                                           ______________________________________                                    

                  TABLE 17                                                        ______________________________________                                        General Formula 17                                                            R.sub.1                                                                             G        R.sub.12                                                                              X      Y     Z    m.p. (°C.)                    ______________________________________                                        H     CH.sub.2 H       CH.sub.3                                                                             CH.sub.3                                                                            CH                                        H     CH.sub.2 H       CH.sub.3                                                                             OCH.sub.3                                                                           CH                                        H     CH.sub.2 H       OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     CH.sub.2 H       Cl     OCH.sub.3                                                                           CH                                        H     CH.sub.2 H       CH.sub.3                                                                             OCH.sub.3                                                                           N                                         H     CH.sub.2 H       OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         H     CH.sub.2 H       CH.sub.3                                                                             CH.sub.3                                                                            N                                         H     CH.sub.2 CH.sub.3                                                                              CH.sub.3                                                                             CH.sub.3                                                                            CH                                        H     CH.sub.2 CH.sub.3                                                                              CH.sub.3                                                                             OCH.sub.3                                                                           CH                                        H     CH.sub.2 CH.sub.3                                                                              OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     CH.sub.2 CH.sub.3                                                                              Cl     OCH.sub.3                                                                           CH                                        H     CH.sub.2 CH.sub.3                                                                              CH.sub.3                                                                             OCH.sub.3                                                                           N                                         H     CH.sub.2 CH.sub.3                                                                              OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         H     CH.sub.2 CH.sub.3                                                                              CH.sub.3                                                                             CH.sub.3                                                                            N                                         H     CH.sub.2 C.sub.6 H.sub.5                                                                       CH.sub.3                                                                             CH.sub.3                                                                            CH                                        H     CH.sub.2 C.sub.6 H.sub.5                                                                       CH.sub.3                                                                             OCH.sub.3                                                                           CH                                        H     CH.sub.2 C.sub.6 H.sub.5                                                                       OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     CH.sub.2 C.sub.6 H.sub.5                                                                       Cl     OCH.sub.3                                                                           CH                                        H     CH.sub.2 C.sub.6 H.sub.5                                                                       CH.sub.3                                                                             OCH.sub.3                                                                           N                                         H     CH.sub.2 C.sub.6 H.sub.5                                                                       OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         H     CH.sub.2 C.sub.6 H.sub.5                                                                       CH.sub.3                                                                             CH.sub.3                                                                            N                                         6-CH.sub.3                                                                          CH.sub.2 H       CH.sub.3                                                                             CH.sub.3                                                                            CH                                        6-CH.sub.3                                                                          CH.sub.2 H       CH.sub.3                                                                             OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          CH.sub.2 H       OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          CH.sub.2 H       Cl     OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          CH.sub.2 H       CH.sub.3                                                                             OCH.sub.3                                                                           N                                         6-CH.sub.3                                                                          CH.sub.2 H       OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         6-CH.sub.3                                                                          CH.sub.2 H       CH.sub.3                                                                             CH.sub.3                                                                            N                                         6-CH.sub.3                                                                          CH.sub.2 CH.sub.3                                                                              CH.sub.3                                                                             CH.sub.3                                                                            CH                                        6-CH.sub.3                                                                          CH.sub.2 CH.sub.3                                                                              OCH.sub.3                                                                            CH.sub.3                                                                            CH                                        6-CH.sub.3                                                                          CH.sub.2 CH.sub.3                                                                              OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          CH.sub.2 CH.sub.3                                                                              Cl     OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          CH.sub.2 CH.sub.3                                                                              CH.sub.3                                                                             OCH.sub.3                                                                           N                                         6-CH.sub.3                                                                          CH.sub.2 CH.sub.3                                                                              OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         6-CH.sub.3                                                                          CH.sub.2 CH.sub.3                                                                              CH.sub.3                                                                             CH.sub.3                                                                            N                                         6-CH.sub.3                                                                          CH.sub.2 C.sub.6 H.sub.5                                                                       CH.sub.3                                                                             CH.sub.3                                                                            CH                                        6-CH.sub.3                                                                          CH.sub.2 C.sub.6 H.sub.5                                                                       CH.sub.3                                                                             OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          CH.sub.2 C.sub.6 H.sub.5                                                                       OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          CH.sub.2 C.sub.6 H.sub.5                                                                       Cl     OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          CH.sub.2 C.sub.6 H.sub.5                                                                       CH.sub.3                                                                             OCH.sub.3                                                                           N                                         6-CH.sub.3                                                                          CH.sub.2 C.sub.6 H.sub.5                                                                       OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         6-CH.sub.3                                                                          CH.sub.2 C.sub.6 H.sub.5                                                                       CH.sub.3                                                                             CH.sub.3                                                                            N                                         6-Cl  CH.sub.2 H       CH.sub.3                                                                             CH.sub.3                                                                            CH                                        6-Cl  CH.sub.2 H       CH.sub.3                                                                             OCH.sub.3                                                                           CH                                        6-Cl  CH.sub.2 H       OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-Cl  CH.sub.2 H       Cl     OCH.sub.3                                                                           CH                                        6-Cl  CH.sub.2 H       CH.sub.3                                                                             OCH.sub.3                                                                           N                                         6-Cl  CH.sub.2 H       OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         6-Cl  CH.sub.2 H       CH.sub.3                                                                             CH.sub.3                                                                            N                                         6-Cl  CH.sub.2 CH.sub.3                                                                              CH.sub.3                                                                             CH.sub.3                                                                            CH                                        6-Cl  CH.sub.2 CH.sub.3                                                                              OCH.sub.3                                                                            CH.sub.3                                                                            CH                                        6-Cl  CH.sub.2 CH.sub.3                                                                              OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-Cl  CH.sub.2 CH.sub.3                                                                              Cl     OCH.sub.3                                                                           CH                                        6-Cl  CH.sub.2 CH.sub.3                                                                              CH.sub.3                                                                             OCH.sub.3                                                                           N                                         6-Cl  CH.sub.2 CH.sub.3                                                                              OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         6-Cl  CH.sub.2 CH.sub.3                                                                              CH.sub.3                                                                             CH.sub.3                                                                            N                                         6-Cl  CH.sub.2 C.sub.6 H.sub.5                                                                       CH.sub.3                                                                             CH.sub.3                                                                            CH                                        6-Cl  CH.sub.2 C.sub.6 H.sub.5                                                                       CH.sub.3                                                                             OCH.sub.3                                                                           CH                                        6-Cl  CH.sub.2 C.sub.6 H.sub.5                                                                       OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-Cl  CH.sub.2 C.sub.6 H.sub.5                                                                       Cl     OCH.sub.3                                                                           CH                                        6-Cl  CH.sub.2 C.sub.6 H.sub.5                                                                       CH.sub.3                                                                             OCH.sub.3                                                                           N                                         6-Cl  CH.sub.2 C.sub.6 H.sub.5                                                                       OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         6-Cl  CH.sub.2 C.sub.6 H.sub.5                                                                       CH.sub.3                                                                             CH.sub.3                                                                            N                                         H     CH.sub.2 CH.sub.2                                                                      H       CH.sub.3                                                                             CH.sub.3                                                                            CH                                        H     CH.sub.2 CH.sub.2                                                                      H       CH.sub.3                                                                             OCH.sub.3                                                                           CH                                        H     CH.sub.2 CH.sub.2                                                                      H       OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     CH.sub.2 CH.sub.2                                                                      H       Cl     OCH.sub.3                                                                           CH                                        H     CH.sub.2 CH.sub.2                                                                      H       CH.sub.3                                                                             OCH.sub.3                                                                           N                                         H     CH.sub.2 CH.sub.2                                                                      H       OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         H     CH.sub.2 CH.sub.2                                                                      H       CH.sub.3                                                                             CH.sub.3                                                                            N                                         H     CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              CH.sub.3                                                                             CH.sub.3                                                                            CH                                        H     CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              CH.sub.3                                                                             OCH.sub.3                                                                           CH                                        H     CH.sub.2 CH.sub. 2                                                                     CH.sub.3                                                                              OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              Cl     OCH.sub.3                                                                           CH                                        H     CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              CH.sub.3                                                                             OCH.sub.3                                                                           N                                         H     CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         H     CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              CH.sub.3                                                                             CH.sub.3                                                                            N                                         H     CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                       CH.sub.3                                                                             CH.sub.3                                                                            CH                                        H     CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                       CH.sub.3                                                                             OCH.sub.3                                                                           CH                                        H     CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                       OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                       Cl     OCH.sub.3                                                                           CH                                        H     CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                       CH.sub.3                                                                             OCH.sub.3                                                                           N                                         H     CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                       OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         H     CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                       CH.sub.3                                                                             CH.sub.3                                                                            N                                         6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                      H       CH.sub.3                                                                             CH.sub.3                                                                            CH                                        6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                      H       CH.sub.3                                                                             OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                      H       OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                      H       Cl     OCH.sub.3                                                                           CH                                        6-CH.sub. 3                                                                         CH.sub.2 CH.sub.2                                                                      H       CH.sub.3                                                                             OCH.sub.3                                                                           N                                         6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                      H       OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                      H       CH.sub.3                                                                             CH.sub.3                                                                            N                                         6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              CH.sub.3                                                                             CH.sub.3                                                                            CH                                        6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              OCH.sub.3                                                                            CH.sub.3                                                                            CH                                        6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              Cl     OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              CH.sub.3                                                                             OCH.sub.3                                                                           N                                         6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              CH.sub.3                                                                             CH.sub.3                                                                            N                                         6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                       CH.sub.3                                                                             CH.sub.3                                                                            CH                                        6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                       CH.sub.3                                                                             OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                       OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                       Cl     OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                       CH.sub.3                                                                             OCH.sub.3                                                                           N                                         6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                       OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                       CH.sub.3                                                                             CH.sub.3                                                                            N                                         6-Cl  CH.sub.2 CH.sub.2                                                                      H       CH.sub.3                                                                             CH.sub.3                                                                            CH                                        6-Cl  CH.sub.2 CH.sub.2                                                                      H       CH.sub.3                                                                             OCH.sub.3                                                                           CH                                        6-Cl  CH.sub.2 CH.sub.2                                                                      H       OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-Cl  CH.sub.2 CH.sub.2                                                                      H       Cl     OCH.sub.3                                                                           CH                                        6-Cl  CH.sub.2 CH.sub.2                                                                      H       CH.sub.3                                                                             OCH.sub.3                                                                           N                                         6-Cl  CH.sub.2 CH.sub.2                                                                      H       OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         6-Cl  CH.sub.2 CH.sub.2                                                                      H       CH.sub.3                                                                             CH.sub.3                                                                            N                                         6-Cl  CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              CH.sub.3                                                                             CH.sub.3                                                                            CH                                        6-Cl  CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              OCH.sub.3                                                                            CH.sub.3                                                                            CH                                        6-Cl  CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-Cl  CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              Cl     OCH.sub.3                                                                           CH                                        6-Cl  CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              CH.sub.3                                                                             OCH.sub.3                                                                           N                                         6-Cl  CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         6-Cl  CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              CH.sub.3                                                                             CH.sub.3                                                                            N                                         6-Cl  CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                       CH.sub.3                                                                             CH.sub.3                                                                            CH                                        6-Cl  CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                       CH.sub.3                                                                             OCH.sub.3                                                                           CH                                        6-Cl  CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                       OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-Cl  CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                       Cl     OCH.sub.3                                                                           CH                                        6-Cl  CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                       CH.sub.3                                                                             OCH.sub.3                                                                           N                                         6-Cl  CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                       OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         6-Cl  CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                       CH.sub.3                                                                             CH.sub.3                                                                            N                                         H     CH═CH                                                                              H       CH.sub.3                                                                             CH.sub.3                                                                            CH                                        H     CH═CH                                                                              H       CH.sub.3                                                                             OCH.sub.3                                                                           CH                                        H     CH═CH                                                                              H       OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     CH═CH                                                                              H       Cl     OCH.sub.3                                                                           CH                                        H     CH═CH                                                                              H       CH.sub.3                                                                             OCH.sub.3                                                                           N                                         H     CH═CH                                                                              H       OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         H     CH═CH                                                                              H       CH.sub.3                                                                             CH.sub.3                                                                            N                                         H     CH═CH                                                                              CH.sub.3                                                                              CH.sub.3                                                                             CH.sub.3                                                                            CH                                        H     CH═CH                                                                              CH.sub.3                                                                              CH.sub.3                                                                             OCH.sub.3                                                                           CH                                        H     CH═CH                                                                              CH.sub.3                                                                              OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     CH═CH                                                                              CH.sub.3                                                                              Cl     OCH.sub.3                                                                           CH                                        H     CH═CH                                                                              CH.sub.3                                                                              CH.sub.3                                                                             OCH.sub.3                                                                           N                                         H     CH═CH                                                                              CH.sub.3                                                                              OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         H     CH═CH                                                                              CH.sub.3                                                                              CH.sub.3                                                                             CH.sub.3                                                                            N                                         H     CH═CH                                                                              C.sub.6 H.sub.5                                                                       CH.sub.3                                                                             CH.sub.3                                                                            CH                                        H     CH═CH                                                                              C.sub.6 H.sub.5                                                                       CH.sub.3                                                                             OCH.sub.3                                                                           CH                                        H     CH═CH                                                                              C.sub.6 H.sub.5                                                                       OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     CH═CH                                                                              C.sub.6 H.sub.5                                                                       Cl     OCH.sub.3                                                                           CH                                        H     CH═CH                                                                              C.sub.6 H.sub.5                                                                       CH.sub.3                                                                             OCH.sub.3                                                                           N                                         H     CH═CH                                                                              C.sub.6 H.sub.5                                                                       OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         H     CH═CH                                                                              C.sub.6 H.sub.5                                                                       CH.sub.3                                                                             CH.sub.3                                                                            N                                         6-CH.sub.3                                                                          CH═CH                                                                              H       CH.sub.3                                                                             CH.sub.3                                                                            CH                                        6-CH.sub.3                                                                          CH═CH                                                                              H       CH.sub.3                                                                             OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          CH═CH                                                                              H       OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          CH═CH                                                                              H       Cl     OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          CH═CH                                                                              H       CH.sub.3                                                                             OCH.sub.3                                                                           N                                         6-CH.sub.3                                                                          CH═CH                                                                              H       OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         6-CH.sub.3                                                                          CH═CH                                                                              H       CH.sub.3                                                                             CH.sub.3                                                                            N                                         6-CH.sub.3                                                                          CH═CH                                                                              CH.sub.3                                                                              CH.sub.3                                                                             CH.sub.3                                                                            CH                                        6-CH.sub.3                                                                          CH═CH                                                                              CH.sub.3                                                                              OCH.sub.3                                                                            CH.sub.3                                                                            CH                                        6-CH.sub.3                                                                          CH═CH                                                                              CH.sub.3                                                                              OCH.sub.3                                                                            OCH.sub. 3                                                                          CH                                        6-CH.sub.3                                                                          CH═CH                                                                              CH.sub.3                                                                              Cl     OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          CH═CH                                                                              CH.sub.3                                                                              CH.sub.3                                                                             OCH.sub.3                                                                           N                                         6-CH.sub.3                                                                          CH═CH                                                                              CH.sub.3                                                                              OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         6-CH.sub.3                                                                          CH═CH                                                                              CH.sub.3                                                                              CH.sub.3                                                                             CH.sub.3                                                                            N                                         6-CH.sub.3                                                                          CH═CH                                                                              C.sub.6 H.sub.5                                                                       CH.sub.3                                                                             CH.sub.3                                                                            CH                                        6-CH.sub.3                                                                          CH═CH                                                                              C.sub.6 H.sub.5                                                                       CH.sub.3                                                                             OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          CH═CH                                                                              C.sub.6 H.sub.5                                                                       OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          CH═CH                                                                              C.sub.6 H.sub.5                                                                       Cl     OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          CH═CH                                                                              C.sub.6 H.sub.5                                                                       CH.sub.3                                                                             OCH.sub.3                                                                           N                                         6-CH.sub.3                                                                          CH═CH                                                                              C.sub.6 H.sub.5                                                                       OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         6-CH.sub.3                                                                          CH═CH                                                                              C.sub.6 H.sub.5                                                                       CH.sub.3                                                                             CH.sub.3                                                                            N                                         6-Cl  CH═CH                                                                              H       CH.sub.3                                                                             CH.sub.3                                                                            CH                                        6-Cl  CH═CH                                                                              H       CH.sub.3                                                                             OCH.sub.3                                                                           CH                                        6-Cl  CH═CH                                                                              H       OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-Cl  CH═CH                                                                              H       Cl     OCH.sub.3                                                                           CH                                        6-Cl  CH═CH                                                                              H       CH.sub.3                                                                             OCH.sub.3                                                                           N                                         6-Cl  CH═CH                                                                              H       OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         6-Cl  CH═CH                                                                              H       CH.sub.3                                                                             CH.sub.3                                                                            N                                         6-Cl  CH═CH                                                                              CH.sub.3                                                                              CH.sub.3                                                                             CH.sub.3                                                                            CH                                        6-Cl  CH═CH                                                                              CH.sub.3                                                                              OCH.sub.3                                                                            CH.sub.3                                                                            CH                                        6-Cl  CH═CH                                                                              CH.sub.3                                                                              OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-Cl  CH═CH                                                                              CH.sub.3                                                                              Cl     OCH.sub.3                                                                           CH                                        6-Cl  CH═CH                                                                              CH.sub.3                                                                              CH.sub.3                                                                             OCH.sub.3                                                                           N                                         6-Cl  CH═CH                                                                              CH.sub.3                                                                              OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         6-Cl  CH═CH                                                                              CH.sub.3                                                                              CH.sub.3                                                                             CH.sub.3                                                                            N                                         6-Cl  CH═CH                                                                              C.sub.6 H.sub.5                                                                       CH.sub.3                                                                             CH.sub.3                                                                            CH                                        6-Cl  CH═CH                                                                              C.sub.6 H.sub.5                                                                       CH.sub.3                                                                             OCH.sub.3                                                                           CH                                        6-Cl  CH═CH                                                                              C.sub.6 H.sub.5                                                                       OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-Cl  CH═CH                                                                              C.sub.6 H.sub.5                                                                       Cl     OCH.sub.3                                                                           CH                                        6-Cl  CH═CH                                                                              C.sub.6 H.sub.5                                                                       CH.sub.3                                                                             OCH.sub.3                                                                           N                                         6-Cl  CH═CH                                                                              C.sub.6 H.sub.5                                                                       OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         6-Cl  CH═CH                                                                              C.sub.6 H.sub.5                                                                       CH.sub.3                                                                             CH.sub.3                                                                            N                                         ______________________________________                                    

                  TABLE 18                                                        ______________________________________                                        General Formula 18                                                            R.sub.1                                                                             G         R.sub.12                                                                             X      Y     Z     m.p. (°C.)                   ______________________________________                                        H     CH.sub.2  H      CH.sub.3                                                                             CH.sub.3                                                                            CH                                        H     CH.sub.2  H      CH.sub.3                                                                             OCH.sub.3                                                                           CH                                        H     CH.sub.2  H      OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     CH.sub.2  H      Cl     OCH.sub.3                                                                           CH                                        H     CH.sub.2  H      CH.sub.3                                                                             OCH.sub.3                                                                           N                                         H     CH.sub.2  H      OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         H     CH.sub.2  H      CH.sub.3                                                                             CH.sub.3                                                                            N                                         H     CH.sub.2  CH.sub.3                                                                             CH.sub.3                                                                             CH.sub.3                                                                            CH                                        H     CH.sub.2  CH.sub.3                                                                             CH.sub.3                                                                             OCH.sub.3                                                                           CH                                        H     CH.sub.2  CH.sub.3                                                                             OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     CH.sub.2  CH.sub.3                                                                             Cl     OCH.sub.3                                                                           CH                                        H     CH.sub.2  CH.sub.3                                                                             CH.sub.3                                                                             OCH.sub.3                                                                           N                                         H     CH.sub.2  CH.sub.3                                                                             OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         H     CH.sub.2  CH.sub.3                                                                             CH.sub.3                                                                             CH.sub.3                                                                            N                                         H     CH.sub.2  C.sub.6 H.sub.5                                                                      CH.sub.3                                                                             CH.sub.3                                                                            CH                                        H     CH.sub.2  C.sub.6 H.sub.5                                                                      CH.sub.3                                                                             OCH.sub.3                                                                           CH                                        H     CH.sub.2  C.sub.6 H.sub.5                                                                      OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     CH.sub.2  C.sub.6 H.sub.5                                                                      Cl     OCH.sub.3                                                                           CH                                        H     CH.sub.2  C.sub.6 H.sub.5                                                                      CH.sub.3                                                                             OCH.sub.3                                                                           N                                         H     CH.sub.2  C.sub.6 H.sub.5                                                                      OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         H     CH.sub.2  C.sub.6 H.sub.5                                                                      CH.sub.3                                                                             CH.sub.3                                                                            N                                         6-CH.sub.3                                                                          CH.sub.2  H      CH.sub.3                                                                             CH.sub.3                                                                            CH                                        6-CH.sub.3                                                                          CH.sub.2  H      CH.sub.3                                                                             OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          CH.sub.2  H      OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          CH.sub.2  H      Cl     OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          CH.sub.2  H      CH.sub.3                                                                             OCH.sub.3                                                                           N                                         6-CH.sub.3                                                                          CH.sub.2  H      OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         6-CH.sub.3                                                                          CH.sub.2  H      CH.sub.3                                                                             CH.sub.3                                                                            N                                         6-CH.sub.3                                                                          CH.sub.2  CH.sub.3                                                                             CH.sub.3                                                                             CH.sub.3                                                                            CH                                        6-CH.sub.3                                                                          CH.sub.2  CH.sub.3                                                                             OCH.sub.3                                                                            CH.sub.3                                                                            CH                                        6-CH.sub.3                                                                          CH.sub.2  CH.sub.3                                                                             OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          CH.sub.2  CH.sub.3                                                                             Cl     OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          CH.sub.2  CH.sub.3                                                                             CH.sub.3                                                                             OCH.sub.3                                                                           N                                         6-CH.sub.3                                                                          CH.sub.2  CH.sub.3                                                                             OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         6-CH.sub.3                                                                          CH.sub.2  CH.sub.3                                                                             CH.sub.3                                                                             CH.sub.3                                                                            N                                         6-CH.sub.3                                                                          CH.sub.2  C.sub.6 H.sub.5                                                                      CH.sub.3                                                                             CH.sub.3                                                                            CH                                        6-CH.sub.3                                                                          CH.sub.2  C.sub.6 H.sub.5                                                                      CH.sub.3                                                                             OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          CH.sub.2  C.sub.6 H.sub.5                                                                      OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          CH.sub.2  C.sub.6 H.sub.5                                                                      Cl     OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          CH.sub.2  C.sub.6 H.sub.5                                                                      CH.sub.3                                                                             OCH.sub.3                                                                           N                                         6-CH.sub.3                                                                          CH.sub.2  C.sub.6 H.sub.5                                                                      OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         6-CH.sub.3                                                                          CH.sub.2  C.sub.6 H.sub.5                                                                      CH.sub.3                                                                             CH.sub.3                                                                            N                                         6-Cl  CH.sub.2  H      CH.sub.3                                                                             CH.sub.3                                                                            CH                                        6-Cl  CH.sub.2  H      CH.sub.3                                                                             OCH.sub.3                                                                           CH                                        6-Cl  CH.sub.2  H      OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-Cl  CH.sub.2  H      Cl     OCH.sub.3                                                                           CH                                        6-Cl  CH.sub.2  H      CH.sub.3                                                                             OCH.sub.3                                                                           N                                         6-Cl  CH.sub.2  H      OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         6-Cl  CH.sub.2  H      CH.sub.3                                                                             CH.sub.3                                                                            N                                         6-Cl  CH.sub.2  CH.sub.3                                                                             CH.sub.3                                                                             CH.sub.3                                                                            CH                                        6-Cl  CH.sub.2  CH.sub.3                                                                             OCH.sub.3                                                                            CH.sub.3                                                                            CH                                        6-Cl  CH.sub.2  CH.sub.3                                                                             OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-Cl  CH.sub.2  CH.sub.3                                                                             Cl     OCH.sub.3                                                                           CH                                        6-Cl  CH.sub.2  CH.sub.3                                                                             CH     OCH.sub.3                                                                           N                                         6-Cl  CH.sub.2  CH.sub.3                                                                             OCH.sub.3                                                                            OCH.sub. 3                                                                          N                                         6-Cl  CH.sub.2  CH.sub.3                                                                             CH.sub.3                                                                             CH.sub.3                                                                            N                                         6-Cl  CH.sub.2  C.sub.6 H.sub.5                                                                      CH.sub.3                                                                             CH.sub.3                                                                            CH                                        6-Cl  CH.sub.2  C.sub.6 H.sub.5                                                                      CH.sub.3                                                                             OCH.sub.3                                                                           CH                                        6-Cl  CH.sub.2  C.sub.6 H.sub.5                                                                      OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-Cl  CH.sub.2  C.sub.6 H.sub.5                                                                      Cl     OCH.sub.3                                                                           CH                                        6-Cl  CH.sub.2  C.sub.6 H.sub.5                                                                      CH.sub.3                                                                             OCH.sub.3                                                                           N                                         6-Cl  CH.sub.2  C.sub.6 H.sub.5                                                                      OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         6-Cl  CH.sub.2  C.sub.6 H.sub.5                                                                      CH.sub.3                                                                             CH.sub.3                                                                            N                                         H     CH.sub.2 CH.sub.2                                                                       H      CH.sub.3                                                                             CH.sub.3                                                                            CH                                        H     CH.sub.2 CH.sub.2                                                                       H      CH.sub.3                                                                             OCH.sub.3                                                                           CH                                        H     CH.sub.2 CH.sub.2                                                                       H      OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     CH.sub.2 CH.sub.2                                                                       H      Cl     OCH.sub.3                                                                           CH                                        H     CH.sub.2 CH.sub.2                                                                       H      CH.sub.3                                                                             OCH.sub.3                                                                           N                                         H     CH.sub.2 CH.sub.2                                                                       H      OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         H     CH.sub.2 CH.sub.2                                                                       H      CH.sub.3                                                                             CH.sub.3                                                                            N                                         H     CH.sub.2 CH.sub.2                                                                       CH.sub.3                                                                             CH.sub.3                                                                             CH.sub.3                                                                            CH                                        H     CH.sub.2 CH.sub.2                                                                       CH.sub.3                                                                             CH.sub.3                                                                             OCH.sub.3                                                                           CH                                        H     CH.sub.2 CH.sub.2                                                                       CH.sub. 3                                                                            OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     CH.sub.2 CH.sub.2                                                                       CH.sub.3                                                                             Cl     OCH.sub.3                                                                           CH                                        H     CH.sub.2 CH.sub.2                                                                       CH.sub.3                                                                             CH.sub.3                                                                             OCH.sub.3                                                                           N                                         H     CH.sub.2 CH.sub.2                                                                       CH.sub.3                                                                             OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         H     CH.sub.2 CH.sub.2                                                                       CH.sub.3                                                                             CH.sub.3                                                                             CH.sub.3                                                                            N                                         H     CH.sub.2 CH.sub.2                                                                       C.sub.6 H.sub.5                                                                      CH.sub.3                                                                             CH.sub.3                                                                            CH                                        H     CH.sub.2 CH.sub.2                                                                       C.sub.6 H.sub.5                                                                      CH.sub.3                                                                             OCH.sub.3                                                                           CH                                        H     CH.sub.2 CH.sub.2                                                                       C.sub.6 H.sub.5                                                                      OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     CH.sub.2 CH.sub.2                                                                       C.sub.6 H.sub.5                                                                      Cl     OCH.sub.3                                                                           CH                                        H     CH.sub.2 CH.sub.2                                                                       C.sub.6 H.sub.5                                                                      CH.sub.3                                                                             OCH.sub.3                                                                           N                                         H     CH.sub.2 CH.sub.2                                                                       C.sub.6 H.sub.5                                                                      OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         H     CH.sub.2 CH.sub.2                                                                       C.sub.6 H.sub.5                                                                      CH.sub.3                                                                             CH.sub.3                                                                            N                                         6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                       H      CH.sub.3                                                                             CH.sub.3                                                                            CH                                        6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                       H      CH.sub.3                                                                             OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                       H      OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                       H      Cl     OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          CH.sub. 2 CH.sub.2                                                                      H      CH.sub.3                                                                             OCH.sub.3                                                                           N                                         6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                       H      OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                       H      CH.sub.3                                                                             CH.sub.3                                                                            N                                         6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                       CH.sub.3                                                                             CH.sub.3                                                                             CH.sub.3                                                                            CH                                        6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                       CH.sub.3                                                                             OCH.sub.3                                                                            CH.sub.3                                                                            CH                                        6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                       CH.sub.3                                                                             OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                       CH.sub.3                                                                             Cl     OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                       CH.sub.3                                                                             CH.sub.3                                                                             OCH.sub.3                                                                           N                                         6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                       CH.sub.3                                                                             OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                       CH.sub.3                                                                             CH.sub.3                                                                             CH.sub.3                                                                            N                                         6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                       C.sub.6 H.sub.5                                                                      CH.sub.3                                                                             CH.sub.3                                                                            CH                                        6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                       C.sub.6 H.sub.5                                                                      CH.sub.3                                                                             OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                       C.sub.6 H.sub.5                                                                      OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                       C.sub.6 H.sub.5                                                                      Cl     OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                       C.sub.6 H.sub.5                                                                      CH.sub.3                                                                             OCH.sub.3                                                                           N                                         6-CH.sub.3                                                                          CH.sub. 2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                       C.sub.6 H.sub.5                                                                      CH.sub.3                                                                             CH.sub.3                                                                            N                                         6-Cl  CH.sub.2 CH.sub.2                                                                       H      CH.sub.3                                                                             CH.sub.3                                                                            CH                                        6-Cl  CH.sub.2 CH.sub.2                                                                       H      CH.sub.3                                                                             OCH.sub.3                                                                           CH                                        6-Cl  CH.sub.2 CH.sub.2                                                                       H      OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-Cl  CH.sub.2 CH.sub.2                                                                       H      Cl     OCH.sub.3                                                                           CH                                        6-Cl  CH.sub.2 CH.sub.2                                                                       H      CH.sub.3                                                                             OCH.sub.3                                                                           N                                         6-Cl  CH.sub.2 CH.sub.2                                                                       H      OCH.sub.3                                                                            OCH.sub.3                                                                           N -6-Cl CH.sub.2 CH.sub.2 H CH.sub.3 C                                        H.sub.3 N                                 6-Cl  CH.sub.2 CH.sub.2                                                                       CH.sub.3                                                                             CH.sub.3                                                                             CH.sub.3                                                                            CH                                        6-Cl  CH.sub.2 CH.sub.2                                                                       CH.sub.3                                                                             OCH.sub.3                                                                            CH.sub.3                                                                            CH                                        6-Cl  CH.sub.2 CH.sub.2                                                                       CH.sub.3                                                                             OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-Cl  CH.sub.2 CH.sub.2                                                                       CH.sub.3                                                                             Cl     OCH.sub.3                                                                           CH                                        6-Cl  CH.sub.2 CH.sub.2                                                                       CH.sub.3                                                                             CH.sub.3                                                                             OCH.sub.3                                                                           N                                         6-Cl  CH.sub.2 CH.sub.2                                                                       CH.sub.3                                                                             OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         6-Cl  CH.sub.2 CH.sub.2                                                                       CH.sub.3                                                                             CH.sub.3                                                                             CH.sub.3                                                                            N                                         6-Cl  CH.sub.2 CH.sub.2                                                                       C.sub.6 H.sub.5                                                                      CH.sub.3                                                                             CH.sub.3                                                                            CH                                        6-Cl  CH.sub.2 CH.sub.2                                                                       C.sub.6 H.sub.5                                                                      CH.sub.3                                                                             OCH.sub.3                                                                           CH                                        6-Cl  CH.sub.2 CH.sub.2                                                                       C.sub.6 H.sub.5                                                                      OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-Cl  CH.sub.2 CH.sub.2                                                                       C.sub.6 H.sub.5                                                                      Cl     OCH.sub.3                                                                           CH                                        6-Cl  CH.sub.2 CH.sub.2                                                                       C.sub.6 H.sub.5                                                                      CH.sub.3                                                                             OCH.sub.3                                                                           N                                         6-Cl  CH.sub.2 CH.sub.2                                                                       C.sub.6 H.sub.5                                                                      OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         6-Cl  CH.sub.2 CH.sub.2                                                                       C.sub.6 H.sub.5                                                                      CH.sub.3                                                                             CH.sub.3                                                                            N                                         H     CH═CH H      CH.sub.3                                                                             CH.sub.3                                                                            CH                                        H     CH═CH H      CH.sub.3                                                                             OCH.sub.3                                                                           CH                                        H     CH═CH H      OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     CH═CH H      Cl     OCH.sub.3                                                                           CH                                        H     CH═CH H      CH.sub.3                                                                             OCH.sub.3                                                                           N                                         H     CH═CH H      OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         H     CH═CH H      CH.sub.3                                                                             CH.sub.3                                                                            N                                         H     CH═CH CH.sub.3                                                                             CH.sub.3                                                                             CH.sub.3                                                                            CH                                        H     CH═CH CH.sub.3                                                                             CH.sub.3                                                                             OCH.sub.3                                                                           CH                                        H     CH═CH CH.sub.3                                                                             OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     CH═CH CH.sub.3                                                                             Cl     OCH.sub.3                                                                           CH                                        H     CH═CH CH.sub.3                                                                             CH.sub.3                                                                             OCH.sub.3                                                                           N                                         H     CH═CH CH.sub.3                                                                             OCH.sub. 3                                                                           OCH.sub.3                                                                           N                                         H     CH═CH CH.sub.3                                                                             CH.sub.3                                                                             CH.sub.3                                                                            N                                         H     CH═CH C.sub.6 H.sub.5                                                                      CH.sub.3                                                                             CH.sub.3                                                                            CH                                        H     CH═CH C.sub.6 H.sub.5                                                                      CH.sub.3                                                                             OCH.sub.3                                                                           CH                                        H     CH═CH C.sub.6 H.sub.5                                                                      OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        H     CH═CH C.sub.6 H.sub.5                                                                      Cl     OCH.sub.3                                                                           CH                                        H     CH═CH C.sub.6 H.sub.5                                                                      CH.sub.3                                                                             OCH.sub.3                                                                           N                                         H     CH═CH C.sub.6 H.sub.5                                                                      OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         H     CH═CH C.sub.6 H.sub.5                                                                      CH.sub.3                                                                             CH.sub.3                                                                            N                                         6-CH.sub.3                                                                          CH═CH H      CH.sub.3                                                                             CH.sub.3                                                                            CH                                        6-CH.sub.3                                                                          CH═CH H      CH.sub.3                                                                             OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          CH═CH H      OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          CH═CH H      Cl     OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          CH═CH H      CH.sub.3                                                                             OCH.sub.3                                                                           N                                         6-CH.sub.3                                                                          CH═CH H      OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         6-CH.sub.3                                                                          CH═CH H      CH.sub.3                                                                             CH.sub.3                                                                            N                                         6-CH.sub.3                                                                          CH═CH CH.sub.3                                                                             CH.sub.3                                                                             CH.sub.3                                                                            CH                                        6-CH.sub.3                                                                          CH═CH CH.sub.3                                                                             OCH.sub.3                                                                            CH.sub.3                                                                            CH                                        6-CH.sub.3                                                                          CH═CH CH.sub.3                                                                             OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-CH.sub. 3                                                                         CH═CH CH.sub.3                                                                             Cl     OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          CH═CH CH.sub.3                                                                             CH.sub.3                                                                             OCH.sub.3                                                                           N                                         6-CH.sub.3                                                                          CH═CH CH.sub.3                                                                             OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         6-CH.sub.3                                                                          CH═CH CH.sub.3                                                                             CH.sub.3                                                                             CH.sub.3                                                                            N                                         6-CH.sub.3                                                                          CH═CH C.sub.6 H.sub.5                                                                      CH.sub.3                                                                             CH.sub.3                                                                            CH                                        6-CH.sub.3                                                                          CH═CH C.sub.6 H.sub.5                                                                      CH.sub.3                                                                             OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          CH═CH C.sub.6 H.sub.5                                                                      OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          CH═CH C.sub.6 H.sub.5                                                                      Cl     OCH.sub.3                                                                           CH                                        6-CH.sub.3                                                                          CH═CH C.sub.6 H.sub.5                                                                      CH.sub.3                                                                             OCH.sub.3                                                                           N                                         6-CH.sub.3                                                                          CH═CH C.sub.6 H.sub.5                                                                      OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         6-CH.sub.3                                                                          CH═CH C.sub.6 H.sub.5                                                                      CH.sub.3                                                                             CH.sub.3                                                                            N                                         6-Cl  CH═CH H      CH.sub.3                                                                             CH.sub.3                                                                            CH                                        6-Cl  CH═CH H      CH.sub.3                                                                             OCH.sub.3                                                                           CH                                        6-Cl  CH═CH H      OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-Cl  CH═CH H      Cl     OCH.sub.3                                                                           CH                                        6-Cl  CH═CH H      CH.sub.3                                                                             OCH.sub.3                                                                           N                                         6-Cl  CH═CH H      OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         6-Cl  CH═CH H      CH.sub.3                                                                             CH.sub.3                                                                            N                                         6-Cl  CH═CH CH.sub.3                                                                             CH.sub. 3                                                                            CH.sub.3                                                                            CH                                        6-Cl  CH═CH CH.sub.3                                                                             OCH.sub.3                                                                            CH.sub.3                                                                            CH                                        6-Cl  CH═CH CH.sub.3                                                                             OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-Cl  CH═CH CH.sub.3                                                                             Cl     OCH.sub.3                                                                           CH                                        6-Cl  CH═CH CH.sub.3                                                                             CH.sub.3                                                                             OCH.sub.3                                                                           N                                         6-Cl  CH═CH CH.sub.3                                                                             OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         6-Cl  CH═CH CH.sub.3                                                                             CH.sub.3                                                                             CH.sub.3                                                                            N                                         6-Cl  CH═CH C.sub.6 H.sub.5                                                                      CH.sub.3                                                                             CH.sub.3                                                                            CH                                        6-Cl  CH═CH C.sub.6 H.sub.5                                                                      CH.sub.3                                                                             OCH.sub.3                                                                           CH                                        6-Cl  CH═CH C.sub.6 H.sub.5                                                                      OCH.sub.3                                                                            OCH.sub.3                                                                           CH                                        6-Cl  CH═CH C.sub.6 H.sub.5                                                                      Cl     OCH.sub.3                                                                           CH                                        6-Cl  CH═CH C.sub.6 H.sub.5                                                                      CH.sub.3                                                                             OCH.sub.3                                                                           N                                         6-Cl  CH═CH C.sub.6 H.sub.5                                                                      OCH.sub.3                                                                            OCH.sub.3                                                                           N                                         6-Cl  CH═CH C.sub.6 H.sub.5                                                                      CH.sub.3                                                                             CH.sub.3                                                                            N                                         ______________________________________                                    

                  TABLE 19                                                        ______________________________________                                        General Formula 19                                                            R.sub.1                                                                           G        R.sub.9                                                                              R.sub.13                                                                            X     Y     Z    m.p. (°C.)                  ______________________________________                                        H   CH.sub.2 H      OCH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      H   CH.sub.2 H      OCH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       H   CH.sub.2 H      OCH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H   CH.sub.2 H      OCH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           N                                       H   CH.sub.2 CH.sub.2                                                                      H      OCH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      H   CH.sub.2 CH.sub.2                                                                      H      OCH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       H   CH.sub.2 CH.sub.2                                                                      H      OCH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H   CH.sub.2 CH.sub.2                                                                      H      OCH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           N                                       H   CH═CH                                                                              H      OCH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      H   CH═CH                                                                              H      OCH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       H   CH═CH                                                                              H      OCH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H   CH═CH                                                                              H      OCH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           N                                       H   CH.sub.2 CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      H   CH.sub.2 CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       H   CH.sub.2 CH.sub.3                                                                             OCH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H   CH.sub.2 CH.sub.3                                                                             OCH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           N                                       H   CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      H   CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       H   CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             OCH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H   CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             OCH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           N                                       H   CH═CH                                                                              CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      H   CH═CH                                                                              CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       H   CH═CH                                                                              CH.sub.3                                                                             OCH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H   CH═CH                                                                              CH.sub.3                                                                             OCH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           N                                       H   CH.sub.2 H      CH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      H   CH.sub.2 H      CH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H   CH.sub.2 CH.sub.2                                                                      H      CH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      H   CH.sub.2 CH.sub.2                                                                      H      CH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H   CH═CH                                                                              H      CH.sub.3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      H   CH═CH                                                                              H      CH.sub.3                                                                            CH.sub.3                                                                            OCH.sub.3                                                                           N                                       H   CH.sub.2 H      SCH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      H   CH.sub.2 H      SCH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H   CH.sub.2 CH.sub.2                                                                      H      SCH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      H   CH.sub.2 CH.sub.2                                                                      H      SCH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H   CH═CH                                                                              H      SCH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      H   CH═CH                                                                              H      SCH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      ______________________________________                                    

                  TABLE 20                                                        ______________________________________                                        General Formula 20                                                            R.sub.1                                                                            G        R.sub.6                                                                              R.sub.7                                                                            X     Y     Z    m.p. (°C.)                  ______________________________________                                        H    CH.sub.2 H      CH.sub.3                                                                           CH.sub.3                                                                            CH.sub.3                                                                            CH                                      H    CH.sub.2 H      CH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H    CH.sub.2 H      CH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      H    CH.sub.2 H      CH.sub.3                                                                           Cl    OCH.sub.3                                                                           CH                                      H    CH.sub.2 H      CH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           N                                       H    CH.sub.2 H      CH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       H    CH.sub.2 H      CH.sub.3                                                                           CH.sub.3                                                                            CH.sub.3                                                                            N                                       H    CH.sub.2 CH.sub.3                                                                             CH.sub.3                                                                           CH.sub.3                                                                            CH.sub.3                                                                            CH                                      H    CH.sub.2 CH.sub.3                                                                             CH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H    CH.sub.2 CH.sub.3                                                                             CH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      H    CH.sub.2 CH.sub.3                                                                             CH.sub.3                                                                           Cl    OCH.sub.3                                                                           CH                                      H    CH.sub.2 CH.sub.3                                                                             CH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           N                                       H    CH.sub.2 CH.sub.3                                                                             CH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       H    CH.sub.2 CH.sub.3                                                                             CH.sub.3                                                                           CH.sub.3                                                                            CH.sub.3                                                                            N                                       H    CH.sub.2 C.sub. 6 H.sub.5                                                                     CH.sub.3                                                                           CH.sub.3                                                                            CH.sub.3                                                                            CH                                      H    CH.sub.2 C.sub.6 H.sub.5                                                                      CH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H    CH.sub.2 C.sub.6 H.sub.5                                                                      CH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      H    CH.sub.2 C.sub.6 H.sub.5                                                                      CH.sub.3                                                                           Cl    OCH.sub.3                                                                           CH                                      H    CH.sub.2 C.sub.6 H.sub.5                                                                      CH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           N                                       H    CH.sub.2 C.sub.6 H.sub.5                                                                      CH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       H    CH.sub.2 C.sub.6 H.sub.5                                                                      CH.sub.3                                                                           CH.sub.3                                                                            CH.sub.3                                                                            N                                       H    CH.sub.2 H      H    CH.sub.3                                                                            CH.sub.3                                                                            CH                                      H    CH.sub.2 H      H    CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H    CH.sub.2 H      H    OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      H    CH.sub.2 H      H    Cl    OCH.sub.3                                                                           CH                                      H    CH.sub.2 H      H    CH.sub.3                                                                            OCH.sub.3                                                                           N                                       H    CH.sub.2 H      H    OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       H    CH.sub.2 H      H    CH.sub.3                                                                            CH.sub.3                                                                            N                                       H    CH.sub.2 C.sub.6 H.sub.5                                                                      H    CH.sub.3                                                                            CH.sub.3                                                                            CH                                      H    CH.sub.2 C.sub.6 H.sub.5                                                                      H    CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H    CH.sub.2 C.sub.6 H.sub.5                                                                      H    OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      H    CH.sub.2 C.sub.6 H.sub.5                                                                      H    Cl    OCH.sub.3                                                                           CH                                      H    CH.sub.2 C.sub.6 H.sub.5                                                                      H    CH.sub.3                                                                            OCH.sub.3                                                                           N                                       H    CH.sub.2 C.sub.6 H.sub.5                                                                      H    OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       H    CH.sub.2 C.sub.6 H.sub.5                                                                      H    CH.sub.3                                                                            CH.sub.3                                                                            N                                       6-Cl CH.sub.2 CH.sub.3                                                                             H    CH.sub.3                                                                            CH.sub.3                                                                            CH                                      6-Cl CH.sub.2 CH.sub.3                                                                             H    CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-Cl CH.sub.2 CH.sub.3                                                                             H    OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      6-Cl CH.sub.2 CH.sub.3                                                                             H    Cl    OCH.sub.3                                                                           CH                                      6-Cl CH.sub.2 CH.sub.3                                                                             H    CH.sub.3                                                                            OCH.sub.3                                                                           N                                       6-Cl CH.sub.2 CH.sub.3                                                                             H    OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       6-Cl CH.sub.2 C.sub.6 H.sub.5                                                                      H    CH.sub.3                                                                            CH.sub.3                                                                            CH                                      6-Cl CH.sub.2 C.sub.6 H.sub.5                                                                      H    CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-Cl CH.sub.2 C.sub.6 H.sub.5                                                                      H    OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      6-Cl CH.sub.2 C.sub.6 H.sub.5                                                                      H    Cl    OCH.sub.3                                                                           CH                                      6-Cl CH.sub.2 C.sub.6 H.sub.5                                                                      H    CH.sub.3                                                                            OCH.sub.3                                                                           N                                       6-Cl CH.sub.2 C.sub.6 H.sub.5                                                                      H    OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       H    CH.sub.2 CH.sub.2                                                                      H      CH.sub.3                                                                           CH.sub.3                                                                            CH.sub.3                                                                            CH                                      H    CH.sub.2 CH.sub.2                                                                      H      CH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H    CH.sub.2 CH.sub.2                                                                      H      CH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      H    CH.sub.2 CH.sub.2                                                                      H      CH.sub.3                                                                           Cl    OCH.sub.3                                                                           CH                                      H    CH.sub.2 CH.sub.2                                                                      H      CH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           N                                       H    CH.sub.2 CH.sub.2                                                                      H      CH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       H    CH.sub.2 CH.sub.2                                                                      H      CH.sub.3                                                                           CH.sub.3                                                                            CH.sub.3                                                                            N                                       H    CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             CH.sub.3                                                                           CH.sub.3                                                                            CH.sub.3                                                                            CH                                      H    CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             CH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H    CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             CH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      H    CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             CH.sub.3                                                                           Cl    OCH.sub.3                                                                           CH                                      H    CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             CH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           N                                       H    CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             CH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       H    CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             CH.sub.3                                                                           CH.sub.3                                                                            CH.sub.3                                                                            N                                       H    CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      CH.sub.3                                                                           CH.sub.3                                                                            CH.sub.3                                                                            CH                                      H    CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      CH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H    CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      CH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      H    CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      CH.sub.3                                                                           Cl    OCH.sub.3                                                                           CH                                      H    CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      CH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           N                                       H    CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      CH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       H    CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      CH.sub.3                                                                           CH.sub.3                                                                            CH.sub.3                                                                            N                                       H    CH.sub.2 CH.sub.2                                                                      H      H    CH.sub.3                                                                            CH.sub.3                                                                            CH                                      H    CH.sub.2 CH.sub.2                                                                      H      H    CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H    CH.sub.2 CH.sub.2                                                                      H      H    OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      H    CH.sub.2 CH.sub.2                                                                      H      H    Cl    OCH.sub.3                                                                           CH                                      H    CH.sub.2 CH.sub.2                                                                      H      H    CH.sub.3                                                                            OCH.sub.3                                                                           N                                       H    CH.sub.2 CH.sub.2                                                                      H      H    OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       H    CH.sub.2 CH.sub.2                                                                      H      H    CH.sub.3                                                                            CH.sub.3                                                                            N                                       H    CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      H    CH.sub.3                                                                            CH.sub.3                                                                            CH                                      H    CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      H    CH.sub. 3                                                                           OCH.sub.3                                                                           CH                                      H    CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      H    OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      H    CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      H    Cl    OCH.sub.3                                                                           CH                                      H    CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      H    CH.sub.3                                                                            OCH.sub.3                                                                           N                                       H    CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      H    OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       H    CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      H    CH.sub.3                                                                            CH.sub.3                                                                            N                                       6-Cl CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             H    CH.sub.3                                                                            CH.sub.3                                                                            CH                                      6-Cl CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             H    CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-Cl CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             H    OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      6-Cl CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             H    Cl    OCH.sub.3                                                                           CH                                      6-Cl CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             H    CH.sub.3                                                                            OCH.sub.3                                                                           N                                       6-Cl CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             H    OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       6-Cl CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      H    CH.sub.3                                                                            CH.sub.3                                                                            CH                                      6-Cl CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      H    CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-Cl CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      H    OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      6-Cl CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      H    Cl    OCH.sub.3                                                                           CH                                      6-Cl CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      H    CH.sub.3                                                                            OCH.sub.3                                                                           N                                       6-Cl CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      H    OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       H    CH═CH                                                                              H      CH.sub.3                                                                           CH.sub.3                                                                            CH.sub.3                                                                            CH                                      H    CH═CH                                                                              H      CH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H    CH═CH                                                                              H      CH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      H    CH═CH                                                                              H      CH.sub.3                                                                           Cl    OCH.sub.3                                                                           CH                                      H    CH═CH                                                                              H      CH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           N                                       H    CH═CH                                                                              H      CH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       H    CH═CH                                                                              H      CH.sub.3                                                                           CH.sub.3                                                                            CH.sub.3                                                                            N                                       H    CH═CH                                                                              CH.sub.3                                                                             CH.sub.3                                                                           CH.sub.3                                                                            CH.sub.3                                                                            CH                                      H    CH═CH                                                                              CH.sub.3                                                                             CH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H    CH═CH                                                                              CH.sub.3                                                                             CH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      H    CH═CH                                                                              CH.sub.3                                                                             CH.sub.3                                                                           Cl    OCH.sub.3                                                                           CH                                      H    CH═CH                                                                              CH.sub.3                                                                             CH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           N                                       H    CH═CH                                                                              CH.sub.3                                                                             CH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       H    CH═CH                                                                              CH.sub.3                                                                             CH.sub.3                                                                           CH.sub.3                                                                            CH.sub.3                                                                            N                                       H    CH═CH                                                                              C.sub.6 H.sub.5                                                                      CH.sub.3                                                                           CH.sub.3                                                                            CH.sub.3                                                                            CH                                      H    CH═CH                                                                              C.sub.6 H.sub.5                                                                      CH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H    CH═CH                                                                              C.sub.6 H.sub.5                                                                      CH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      H    CH═CH                                                                              C.sub.6 H.sub.5                                                                      CH.sub.3                                                                           Cl    OCH.sub.3                                                                           CH                                      H    CH═CH                                                                              C.sub.6 H.sub.5                                                                      CH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           N                                       H    CH═CH                                                                              C.sub.6 H.sub.5                                                                      CH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       H    CH═CH                                                                              C.sub.6 H.sub.5                                                                      CH.sub.3                                                                           CH.sub.3                                                                            CH.sub.3                                                                            N                                       H    CH═CH                                                                              H      H    CH.sub.3                                                                            CH.sub.3                                                                            CH                                      H    CH═CH                                                                              H      H    CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H    CH═CH                                                                              H      H    OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      H    CH═CH                                                                              H      H    Cl    OCH.sub.3                                                                           CH                                      H    CH═CH                                                                              H      H    CH.sub.3                                                                            OCH.sub.3                                                                           N                                       H    CH═CH                                                                              H      H    OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       H    CH═CH                                                                              H      H    CH.sub.3                                                                            CH.sub.3                                                                            N                                       H    CH═CH                                                                              C.sub.6 H.sub.5                                                                      H    CH.sub.3                                                                            CH.sub.3                                                                            CH                                      H    CH═CH                                                                              C.sub.6 H.sub.5                                                                      H    CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H    CH═CH                                                                              C.sub.6 H.sub.5                                                                      H    OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      H    CH═CH                                                                              C.sub.6 H.sub.5                                                                      H    Cl    OCH.sub.3                                                                           CH                                      H    CH═CH                                                                              C.sub.6 H.sub.5                                                                      H    CH.sub.3                                                                            OCH.sub.3                                                                           N                                       H    CH═CH                                                                              C.sub.6 H.sub.5                                                                      H    OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       H    CH═CH                                                                              C.sub.6 H.sub.5                                                                      H    CH.sub.3                                                                            CH.sub.3                                                                            N                                       6-Cl CH═CH                                                                              CH.sub.3                                                                             H    CH.sub.3                                                                            CH.sub.3                                                                            CH                                      6-Cl CH═CH                                                                              CH.sub.3                                                                             H    CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-Cl CH═CH                                                                              CH.sub.3                                                                             H    OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      6-Cl CH═CH                                                                              CH.sub.3                                                                             H    Cl    OCH.sub.3                                                                           CH                                      6-Cl CH═CH                                                                              CH.sub.3                                                                             H    CH.sub.3                                                                            OCH.sub.3                                                                           N                                       6-Cl CH═CH                                                                              CH.sub.3                                                                             H    OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       6-Cl CH═CH                                                                              C.sub.6 H.sub.5                                                                      H    CH.sub.3                                                                            CH.sub.3                                                                            CH                                      6-Cl CH═CH                                                                              C.sub.6 H.sub.5                                                                      H    CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-Cl CH═CH                                                                              C.sub.6 H.sub.5                                                                      H    OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      6-Cl CH═CH                                                                              C.sub.6 H.sub.5                                                                      H    Cl    OCH.sub.3                                                                           CH                                      6-Cl CH═CH                                                                              C.sub.6 H.sub.5                                                                      H    CH.sub.3                                                                            OCH.sub.3                                                                           N                                       6-Cl CH═CH                                                                              C.sub.6 H.sub.5                                                                      H    OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       H    CH.sub.2 CH.sub.3                                                                             H    OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      H    CH.sub.2 CH.sub.3                                                                             H    OCH.sub.3                                                                           CH.sub.3                                                                            CH                                      H    CH.sub.2 CH.sub.3                                                                             H    CH.sub.3                                                                            CH.sub.3                                                                            CH                                      H    CH.sub.2 CH.sub.3                                                                             H    OCH.sub.3                                                                           Cl.sub.3                                                                            CH                                      H    CH.sub.2 CH.sub.3                                                                             H    OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       H    CH.sub.2 CH.sub.3                                                                             H    OCH.sub.3                                                                           CH.sub.3                                                                            N                                       H    CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             H    OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      H    CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             H    OCH.sub.3                                                                           CH.sub.3                                                                            CH                                      H    CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             H    CH.sub.3                                                                            CH.sub.3                                                                            CH                                      H    CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             H    OCH.sub.3                                                                           Cl.sub.3                                                                            CH                                      H    CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             H    OCH.sub.3                                                                           CH.sub.3                                                                            N                                       H    CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             H    OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       H    CH═CH                                                                              CH.sub.3                                                                             H    OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      H    CH═CH                                                                              CH.sub.3                                                                             H    OCH.sub.3                                                                           CH.sub.3                                                                            CH                                      H    CH═CH                                                                              CH.sub.3                                                                             H    CH.sub.3                                                                            CH.sub.3                                                                            CH                                      H    CH═CH                                                                              CH.sub.3                                                                             H    OCH.sub.3                                                                           Cl.sub.3                                                                            CH                                      H    CH═CH                                                                              CH.sub.3                                                                             H    OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       H    CH═CH                                                                              CH.sub.3                                                                             H    OCH.sub.3                                                                           CH.sub.3                                                                            N                                       ______________________________________                                    

                  TABLE 21                                                        ______________________________________                                        General Formula 21                                                            R.sub.1                                                                            G        R.sub.6                                                                              R.sub.7                                                                            X     Y     Z    m.p. (°C.)                  ______________________________________                                        H    CH.sub.2 H      CH.sub.3                                                                           CH.sub.3                                                                            CH.sub.3                                                                            CH                                      H    CH.sub.2 H      CH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H    CH.sub.2 H      CH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      H    CH.sub.2 H      CH.sub.3                                                                           Cl    OCH.sub.3                                                                           CH                                      H    CH.sub.2 H      CH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           N                                       H    CH.sub.2 H      CH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       H    CH.sub.2 H      CH.sub.3                                                                           CH.sub.3                                                                            CH.sub.3                                                                            N                                       H    CH.sub.2 CH.sub.3                                                                             CH.sub.3                                                                           CH.sub.3                                                                            CH.sub.3                                                                            CH                                      H    CH.sub.2 CH.sub.3                                                                             CH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H    CH.sub.2 CH.sub.3                                                                             CH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      H    CH.sub.2 CH.sub.3                                                                             CH.sub.3                                                                           Cl    OCH.sub.3                                                                           CH                                      H    CH.sub.2 CH.sub.3                                                                             CH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           N                                       H    CH.sub.2 CH.sub.3                                                                             CH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       H    CH.sub.2 CH.sub.3                                                                             CH.sub.3                                                                           CH.sub.3                                                                            CH.sub.3                                                                            N                                       H    CH.sub. 2                                                                              C.sub.6 H.sub.5                                                                      CH.sub.3                                                                           CH.sub.3                                                                            CH.sub.3                                                                            CH                                      H    CH.sub.2 C.sub.6 H.sub.5                                                                      CH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H    CH.sub.2 C.sub.6 H.sub.5                                                                      CH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      H    CH.sub.2 C.sub.6 H.sub.5                                                                      CH.sub.3                                                                           Cl    OCH.sub.3                                                                           CH                                      H    CH.sub.2 C.sub.6 H.sub.5                                                                      CH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           N                                       H    CH.sub.2 C.sub.6 H.sub.5                                                                      CH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       H    CH.sub.2 C.sub.6 H.sub.5                                                                      CH.sub.3                                                                           CH.sub.3                                                                            CH.sub.3                                                                            N                                       H    CH.sub.2 H      H    CH.sub.3                                                                            CH.sub.3                                                                            CH                                      H    CH.sub.2 H      H    CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H    CH.sub.2 H      H    OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      H    CH.sub.2 H      H    Cl    OCH.sub.3                                                                           CH                                      H    CH.sub.2 H      H    CH.sub.3                                                                            OCH.sub.3                                                                           N                                       H    CH.sub.2 H      H    OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       H    CH.sub.2 H      H    CH.sub.3                                                                            CH.sub.3                                                                            N                                       H    CH.sub.2 C.sub.6 H.sub.5                                                                      H    CH.sub.3                                                                            CH.sub.3                                                                            CH                                      H    CH.sub.2 C.sub.6 H.sub.5                                                                      H    CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H    CH.sub.2 C.sub.6 H.sub.5                                                                      H    OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      H    CH.sub.2 C.sub.6 H.sub.5                                                                      H    Cl    OCH.sub.3                                                                           CH                                      H    CH.sub.2 C.sub.6 H.sub.5                                                                      H    CH.sub.3                                                                            OCH.sub.3                                                                           N                                       H    CH.sub.2 C.sub.6 H.sub.5                                                                      H    OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       H    CH.sub.2 C.sub.6 H.sub.5                                                                      H    CH.sub.3                                                                            CH.sub.3                                                                            N                                       6-Cl CH.sub.2 CH.sub.3                                                                             H    CH.sub.3                                                                            CH.sub.3                                                                            CH                                      6-Cl CH.sub.2 CH.sub.3                                                                             H    CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-Cl CH.sub.2 CH.sub.3                                                                             H    OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      6-Cl CH.sub.2 CH.sub.3                                                                             H    Cl    OCH.sub.3                                                                           CH                                      6-Cl CH.sub.2 CH.sub.3                                                                             H    CH.sub.3                                                                            OCH.sub.3                                                                           N                                       6-Cl CH.sub.2 CH.sub.3                                                                             H    OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       6-Cl CH.sub.2 C.sub.6 H.sub.5                                                                      H    CH.sub.3                                                                            CH.sub.3                                                                            CH                                      6-Cl CH.sub.2 C.sub.6 H.sub.5                                                                      H    CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-Cl CH.sub.2 C.sub.6 H.sub.5                                                                      H    OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      6-Cl CH.sub.2 C.sub.6 H.sub.5                                                                      H    Cl    OCH.sub.3                                                                           CH                                      6-Cl CH.sub.2 C.sub.6 H.sub.5                                                                      H    CH.sub.3                                                                            OCH.sub.3                                                                           N                                       6-Cl CH.sub.2 C.sub.6 H.sub.5                                                                      H    OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       H    CH.sub.2 CH.sub. 2                                                                     H      CH.sub.3                                                                           CH.sub.3                                                                            CH.sub.3                                                                            CH                                      H    CH.sub.2 CH.sub.2                                                                      H      CH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H    CH.sub.2 CH.sub.2                                                                      H      CH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      H    CH.sub.2 CH.sub.2                                                                      H      CH.sub.3                                                                           Cl    OCH.sub.3                                                                           CH                                      H    CH.sub.2 CH.sub.2                                                                      H      CH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           N                                       H    CH.sub.2 CH.sub.2                                                                      H      CH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       H    CH.sub.2 CH.sub.2                                                                      H      CH.sub.3                                                                           CH.sub.3                                                                            CH.sub.3                                                                            N                                       H    CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             CH.sub.3                                                                           CH.sub.3                                                                            CH.sub.3                                                                            CH                                      H    CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             CH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H    CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             CH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      H    CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             CH.sub.3                                                                           Cl    OCH.sub.3                                                                           CH                                      H    CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             CH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           N                                       H    CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             CH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       H    CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             CH.sub.3                                                                           CH.sub.3                                                                            CH.sub.3                                                                            N                                       H    CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      CH.sub.3                                                                           CH.sub.3                                                                            CH.sub.3                                                                            CH                                      H    CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      CH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H    CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      CH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      H    CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      CH.sub.3                                                                           Cl    OCH.sub.3                                                                           CH                                      H    CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      CH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           N                                       H    CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      CH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       H    CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      CH.sub.3                                                                           CH.sub.3                                                                            CH.sub.3                                                                            N                                       H    CH.sub.2 CH.sub.2                                                                      H      H    CH.sub.3                                                                            CH.sub.3                                                                            CH                                      H    CH.sub.2 CH.sub.2                                                                      H      H    CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H    CH.sub.2 CH.sub.2                                                                      H      H    OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      H    CH.sub.2 CH.sub.2                                                                      H      H    Cl    OCH.sub.3                                                                           CH                                      H    CH.sub.2 CH.sub.2                                                                      H      H    CH.sub.3                                                                            OCH.sub.3                                                                           N                                       H    CH.sub.2 CH.sub.2                                                                      H      H    OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       H    CH.sub.2 CH.sub.2                                                                      H      H    CH.sub.3                                                                            CH.sub.3                                                                            N                                       H    CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      H    CH.sub.3                                                                            CH.sub.3                                                                            CH                                      H    CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub. 5                                                                     H    CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H    CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      H    OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      H    CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      H    Cl    OCH.sub.3                                                                           CH                                      H    CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      H    CH.sub.3                                                                            OCH.sub.3                                                                           N                                       H    CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      H    OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       H    CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      H    CH.sub.3                                                                            CH.sub.3                                                                            N                                       6-Cl CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             H    CH.sub.3                                                                            CH.sub.3                                                                            CH                                      6-Cl CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             H    CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-Cl CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             H    OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      6-Cl CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             H    Cl    OCH.sub.3                                                                           CH                                      6-Cl CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             H    CH.sub.3                                                                            OCH.sub.3                                                                           N                                       6-Cl CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             H    OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       6-Cl CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      H    CH.sub.3                                                                            CH.sub.3                                                                            CH                                      6-Cl CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      H    CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-Cl CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      H    OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      6-Cl CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      H    Cl    OCH.sub.3                                                                           CH                                      6-Cl CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      H    CH.sub.3                                                                            OCH.sub.3                                                                           N                                       6-Cl CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      H    OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       H    CH═CH                                                                              H      CH.sub.3                                                                           CH.sub.3                                                                            CH.sub.3                                                                            CH                                      H    CH═CH                                                                              H      CH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H    CH═CH                                                                              H      CH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      H    CH═CH                                                                              H      CH.sub.3                                                                           Cl    OCH.sub.3                                                                           CH                                      H    CH═CH                                                                              H      CH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           N                                       H    CH═CH                                                                              H      CH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       H    CH═CH                                                                              H      CH.sub.3                                                                           CH.sub.3                                                                            CH.sub.3                                                                            N                                       H    CH═CH                                                                              CH.sub.3                                                                             CH.sub.3                                                                           CH.sub.3                                                                            CH.sub.3                                                                            CH                                      H    CH═CH                                                                              CH.sub.3                                                                             CH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H    CH═CH                                                                              CH.sub.3                                                                             CH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      H    CH═CH                                                                              CH.sub.3                                                                             CH.sub.3                                                                           Cl    OCH.sub.3                                                                           CH                                      H    CH═CH                                                                              CH.sub.3                                                                             CH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           N                                       H    CH═CH                                                                              CH.sub.3                                                                             CH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       H    CH═CH                                                                              CH.sub.3                                                                             CH.sub. 3                                                                          CH.sub.3                                                                            CH.sub.3                                                                            N                                       H    CH═CH                                                                              C.sub.6 H.sub.5                                                                      CH.sub.3                                                                           CH.sub.3                                                                            CH.sub.3                                                                            CH                                      H    CH═CH                                                                              C.sub.6 H.sub.5                                                                      CH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H    CH═CH                                                                              C.sub.6 H.sub.5                                                                      CH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      H    CH═CH                                                                              C.sub.6 H.sub.5                                                                      CH.sub.3                                                                           Cl    OCH.sub.3                                                                           CH                                      H    CH═CH                                                                              C.sub.6 H.sub.5                                                                      CH.sub.3                                                                           CH.sub.3                                                                            OCH.sub.3                                                                           N                                       H    CH═CH                                                                              C.sub.6 H.sub.5                                                                      CH.sub.3                                                                           OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       H    CH═CH                                                                              C.sub.6 H.sub.5                                                                      CH.sub.3                                                                           CH.sub.3                                                                            CH.sub.3                                                                            N                                       H    CH═CH                                                                              H      H    CH.sub.3                                                                            CH.sub.3                                                                            CH                                      H    CH═CH                                                                              H      H    CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H    CH═CH                                                                              H      H    OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      H    CH═CH                                                                              H      H    Cl    OCH.sub.3                                                                           CH                                      H    CH═CH                                                                              H      H    CH.sub.3                                                                            OCH.sub.3                                                                           N                                       H    CH═CH                                                                              H      H    OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       H    CH═CH                                                                              H      H    CH.sub.3                                                                            CH.sub.3                                                                            N                                       H    CH═CH                                                                              C.sub.6 H.sub.5                                                                      H    CH.sub.3                                                                            CH.sub.3                                                                            CH                                      H    CH═CH                                                                              C.sub.6 H.sub.5                                                                      H    CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      H    CH═ CH                                                                             C.sub.6 H.sub.5                                                                      H    OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      H    CH═CH                                                                              C.sub.6 H.sub.5                                                                      H    Cl    OCH.sub.3                                                                           CH                                      H    CH═CH                                                                              C.sub.6 H.sub.5                                                                      H    CH.sub.3                                                                            OCH.sub.3                                                                           N                                       H    CH═CH                                                                              C.sub.6 H.sub.5                                                                      H    OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       H    CH═CH                                                                              C.sub.6 H.sub.5                                                                      H    CH.sub.3                                                                            CH.sub.3                                                                            N                                       6-Cl CH═CH                                                                              CH.sub.3                                                                             H    CH.sub.3                                                                            CH.sub.3                                                                            CH                                      6-Cl CH═CH                                                                              CH.sub.3                                                                             H    CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-Cl CH═CH                                                                              CH.sub.3                                                                             H    OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      6-Cl CH═CH                                                                              CH.sub.3                                                                             H    Cl    OCH.sub.3                                                                           CH                                      6-Cl CH═CH                                                                              CH.sub.3                                                                             H    CH.sub.3                                                                            OCH.sub.3                                                                           N                                       6-Cl CH═CH                                                                              CH.sub.3                                                                             H    OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       6-Cl CH═CH                                                                              C.sub.6 H.sub.5                                                                      H    CH.sub.3                                                                            CH.sub.3                                                                            CH                                      6-Cl CH═CH                                                                              C.sub.6 H.sub.5                                                                      H    CH.sub.3                                                                            OCH.sub.3                                                                           CH                                      6-Cl CH═CH                                                                              C.sub.6 H.sub.5                                                                      H    OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      6-Cl CH═CH                                                                              C.sub.6 H.sub.5                                                                      H    Cl    OCH.sub.3                                                                           CH                                      6-Cl CH═CH                                                                              C.sub.6 H.sub.5                                                                      H    CH.sub.3                                                                            OCH.sub.3                                                                           N                                       6-Cl CH═CH                                                                              C.sub.6 H.sub.5                                                                      H    OCH.sub. 3                                                                          OCH.sub.3                                                                           N                                       H    CH.sub.2 CH.sub.3                                                                             H    OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      H    CH.sub.2 CH.sub.3                                                                             H    OCH.sub.3                                                                           CH.sub.3                                                                            CH                                      H    CH.sub.2 CH.sub.3                                                                             H    CH.sub.3                                                                            CH.sub.3                                                                            CH                                      H    CH.sub.2 CH.sub.3                                                                             H    OCH.sub.3                                                                           C1.sub.3                                                                            CH                                      H    CH.sub.2 CH.sub.3                                                                             H    OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       H    CH.sub.2 CH.sub.3                                                                             H    OCH.sub.3                                                                           CH.sub.3                                                                            N                                       H    CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             H    OCH.sub.3                                                                           OCH.sub.3                                                                           CH   173-180 (d)                        H    CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             H    OCH.sub.3                                                                           CH.sub.3                                                                            CH                                      H    CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             H    CH.sub.3                                                                            CH.sub.3                                                                            CH                                      H    CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             H    OCH.sub.3                                                                           Cl.sub.3                                                                            CH                                      H    CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             H    OCH.sub.3                                                                           CH.sub.3                                                                            N                                       H    CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             H    OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       H    CH═CH                                                                              CH.sub.3                                                                             H    OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                      H    CH═CH                                                                              CH.sub.3                                                                             H    OCH.sub.3                                                                           CH.sub.3                                                                            CH                                      H    CH═CH                                                                              CH.sub.3                                                                             H    CH.sub.3                                                                            CH.sub.3                                                                            CH                                      H    CH═CH                                                                              CH.sub.3                                                                             H    OCH.sub.3                                                                           Cl.sub.3                                                                            CH                                      H    CH═CH                                                                              CH.sub.3                                                                             H    OCH.sub.3                                                                           OCH.sub.3                                                                           N                                       H    CH═CH                                                                              CH.sub.3                                                                             H    OCH.sub.3                                                                           CH.sub.3                                                                            N                                       ______________________________________                                    

                  TABLE 22                                                        ______________________________________                                        General Formula 22                                                            R.sub.1   X        Y         Z     m.p. (°C.)                          ______________________________________                                        H         OCH.sub.3                                                                              OCH.sub.3 N                                                H         OCH.sub.3                                                                              OCH.sub.3 CH                                               H         CH.sub.3 OCH.sub.3 N                                                H         CH.sub.3 OCH.sub.3 CH                                               H         Cl       OCH.sub.3 CH                                               H         CH.sub.3 CH.sub.3  CH                                               6-CH.sub.3                                                                              OCH.sub.3                                                                              OCH.sub.3 N                                                6-CH.sub.3                                                                              OCH.sub.3                                                                              OCH.sub.3 CH                                               6-CH.sub.3                                                                              CH.sub.3 OCH.sub.3 N                                                6-CH.sub.3                                                                              CH.sub.3 OCH.sub.3 CH                                               6-CH.sub.3                                                                              Cl       OCH.sub.3 CH                                               6-CH.sub.3                                                                              CH.sub.3 CH.sub.3  CH                                               6-Cl      OCH.sub.3                                                                              OCH.sub.3 N                                                6-Cl      OCH.sub.3                                                                              OCH.sub.3 CH                                               6-Cl      CH.sub.3 OCH.sub.3 N                                                6-Cl      CH.sub.3 OCH.sub.3 CH                                               6-Cl      Cl       OCH.sub.3 CH                                               6-Cl      CH.sub.3 CH.sub.3  CH                                               6-OCH.sub.3                                                                             OCH.sub.3                                                                              OCH.sub.3 N                                                6-OCH.sub.3                                                                             OCH.sub.3                                                                              OCH.sub.3 CH                                               6-OCH.sub.3                                                                             CH.sub.3 OCH.sub.3 N                                                6-OCH.sub.3                                                                             CH.sub.3 OCH.sub.3 CH                                               6-OCH.sub.3                                                                             Cl       OCH.sub.3 CH                                               6-OCH.sub.3                                                                             CH.sub.3 CH.sub.3  CH                                               5-Cl      OCH.sub.3                                                                              OCH.sub.3 N                                                5-Cl      OCH.sub.3                                                                              OCH.sub.3 CH                                               5-Cl      CH.sub.3 OCH.sub.3 N                                                5-Cl      CH.sub.3 OCH.sub. 3                                                                              CH                                               5-Cl      Cl       OCH.sub.3 CH                                               5-Cl      CH.sub.3 CH.sub.3  CH                                               5-OCH.sub.3                                                                             OCH.sub.3                                                                              OCH.sub.3 N                                                5-OCH.sub.3                                                                             OCH.sub.3                                                                              OCH.sub.3 CH                                               5-OCH.sub.3                                                                             CH.sub.3 OCH.sub.3 N                                                5-OCH.sub.3                                                                             CH.sub.3 OCH.sub.3 CH                                               5-OCH.sub.3                                                                             Cl       OCH.sub.3 CH                                               5-OCH.sub.3                                                                             CH.sub.3 CH.sub.3  CH                                               5-SCH.sub.3                                                                             OCH.sub.3                                                                              OCH.sub.3 N                                                5-SCH.sub.3                                                                             OCH.sub.3                                                                              OCH.sub.3 CH                                               5-SCH.sub.3                                                                             CH.sub.3 OCH.sub.3 N                                                5-SCH.sub.3                                                                             CH.sub.3 OCH.sub.3 CH                                               5-SCH.sub.3                                                                             Cl       OCH.sub.3 CH                                               5-SCH.sub.3                                                                             CH.sub.3 CH.sub.3  CH                                               ______________________________________                                    

                  TABLE 23                                                        ______________________________________                                        General Formula 23                                                            R.sub.1   X        Y         Z     m.p. (°C.)                          ______________________________________                                        H         OCH.sub.3                                                                              OCH.sub.3 N                                                H         OCH.sub.3                                                                              OCH.sub.3 CH                                               H         CH.sub.3 OCH.sub.3 N                                                H         CH.sub.3 OCH.sub.3 CH                                               H         Cl       OCH.sub.3 CH                                               H         CH.sub.3 CH.sub.3  CH                                               6-CH.sub.3                                                                              OCH.sub.3                                                                              OCH.sub.3 N                                                6-CH.sub.3                                                                              OCH.sub.3                                                                              OCH.sub.3 CH                                               6-CH.sub.3                                                                              CH.sub.3 OCH.sub.3 N                                                6-CH.sub.3                                                                              CH.sub.3 OCH.sub.3 CH                                               6-CH.sub.3                                                                              Cl       OCH.sub.3 CH                                               6-CH.sub.3                                                                              CH.sub.3 CH.sub.3  CH                                               6-Cl      OCH.sub.3                                                                              OCH.sub.3 CH                                               6-Cl      OCH.sub.3                                                                              OCH.sub.3 CH                                               6-Cl      CH.sub.3 OCH.sub.3 N                                                6-Cl      CH.sub.3 OCH.sub.3 CH                                               6-Cl      Cl       OCH.sub.3 CH                                               6-Cl      CH.sub.3 CH.sub.3  CH                                               6-OCH.sub.3                                                                             OCH.sub.3                                                                              OCH.sub.3 N                                                6-OCH.sub.3                                                                             OCH.sub.3                                                                              OCH.sub.3 CH                                               6-OCH.sub.3                                                                             CH.sub.3 OCH.sub.3 N                                                6-OCH.sub.3                                                                             CH.sub.3 OCH.sub.3 CH                                               6-OCH.sub.3                                                                             Cl       OCH.sub.3 CH                                               6-OCH.sub.3                                                                             CH.sub.3 CH.sub.3  CH                                               5-Cl      OCH.sub.3                                                                              OCH.sub.3 N                                                5-Cl      OCH.sub.3                                                                              OCH.sub.3 CH                                               5-Cl      CH.sub.3 OCH.sub.3 N                                                5-Cl      CH.sub.3 OCH.sub. 3                                                                              CH                                               5-Cl      Cl       OCH.sub.3 CH                                               5-Cl      CH.sub.3 CH.sub.3  CH                                               5-OCH.sub.3                                                                             OCH.sub.3                                                                              OCH.sub.3 N                                                5-OCH.sub.3                                                                             OCH.sub.3                                                                              OCH.sub.3 CH                                               5-OCH.sub.3                                                                             CH.sub.3 OCH.sub.3 N                                                5-OCH.sub.3                                                                             CH.sub.3 OCH.sub.3 CH                                               5-OCH.sub.3                                                                             Cl       OCH.sub.3 CH                                               5-OCH.sub.3                                                                             CH.sub.3 CH.sub.3  CH                                               5-SCH.sub.3                                                                             OCH.sub.3                                                                              OCH.sub.3 N                                                5-SCH.sub.3                                                                             OCH.sub.3                                                                              OCH.sub.3 CH                                               5-SCH.sub.3                                                                             CH.sub.3 OCH.sub.3 N                                                5-SCH.sub.3                                                                             CH.sub.3 OCH.sub.3 CH                                               5-SCH.sub.3                                                                             Cl       OCH.sub.3 CH                                               5-SCH.sub.3                                                                             CH.sub.3 CH.sub.3  CH                                               ______________________________________                                    

                  TABLE 24                                                        ______________________________________                                        General Formula 24                                                            R.sub.1                                                                              G        R.sub.10                                                                             X     Y     Z    m.p. (°C.)                     ______________________________________                                        H      CH.sub.2 H      CH.sub.3                                                                            CH.sub.3                                                                            CH                                         H      CH.sub.2 H      CH.sub.3                                                                            OCH.sub.3                                                                           CH                                         H      CH.sub.2 H      OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                         H      CH.sub.2 H      Cl    OCH.sub.3                                                                           CH                                         H      CH.sub.2 H      CH.sub.3                                                                            OCH.sub.3                                                                           N                                          H      CH.sub.2 H      OCH.sub.3                                                                           OCH.sub.3                                                                           N                                          H      CH.sub.2 H      CH.sub.3                                                                            CH.sub.3                                                                            N                                          H      CH.sub.2 CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            CH                                         H      CH.sub.2 CH.sub.3                                                                             CH.sub.3                                                                            OCH.sub.3                                                                           CH                                         H      CH.sub.2 CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                         H      CH.sub.2 CH.sub.3                                                                             Cl    OCH.sub.3                                                                           CH                                         H      CH.sub.2 CH.sub.3                                                                             CH.sub.3                                                                            OCH.sub.3                                                                           N                                          H      CH.sub.2 CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           N                                          H      CH.sub.2 CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            N                                          H      CH.sub.2 C.sub.6 H.sub.5                                                                      CH.sub.3                                                                            CH.sub.3                                                                            CH                                         H      CH.sub.2 C.sub.6 H.sub.5                                                                      CH.sub.3                                                                            OCH.sub.3                                                                           CH                                         H      CH.sub.2 C.sub.6 H.sub.5                                                                      OCH.sub.3                                                                           OCH.sub. 3                                                                          CH                                         H      CH.sub.2 C.sub.6 H.sub.5                                                                      Cl    OCH.sub.3                                                                           CH                                         H      CH.sub.2 C.sub.6 H.sub.5                                                                      CH.sub.3                                                                            OCH.sub.3                                                                           N                                          H      CH.sub.2 C.sub.6 H.sub.5                                                                      OCH.sub.3                                                                           OCH.sub.3                                                                           N                                          H      CH.sub.2 C.sub.6 H.sub.5                                                                      CH.sub.3                                                                            CH.sub.3                                                                            N                                          6-CH.sub.3                                                                           CH.sub.2 H      CH.sub.3                                                                            CH.sub.3                                                                            CH                                         6-CH.sub.3                                                                           CH.sub.2 H      CH.sub.3                                                                            OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                           CH.sub.2 H      OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                           CH.sub.2 H      Cl    OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                           CH.sub.2 H      CH.sub.3                                                                            OCH.sub.3                                                                           N                                          6-CH.sub.3                                                                           CH.sub.2 H      OCH.sub.3                                                                           OCH.sub.3                                                                           N                                          6-CH.sub.3                                                                           CH.sub.2 H      CH.sub.3                                                                            CH.sub.3                                                                            N                                          6-CH.sub.3                                                                           CH.sub.2 CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            CH                                         6-CH.sub.3                                                                           CH.sub.2 CH.sub.3                                                                             OCH.sub.3                                                                           CH.sub.3                                                                            CH                                         6-CH.sub.3                                                                           CH.sub.2 CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                           CH.sub.2 CH.sub.3                                                                             Cl    OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                           CH.sub.2 CH.sub.3                                                                             CH.sub.3                                                                            OCH.sub.3                                                                           N                                          6-CH.sub.3                                                                           CH.sub.2 CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           N                                          6-CH.sub.3                                                                           CH.sub.2 CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            N                                          6-CH.sub.3                                                                           CH.sub.2 C.sub.6 H.sub.5                                                                      CH.sub.3                                                                            CH.sub.3                                                                            CH                                         6-CH.sub.3                                                                           CH.sub.2 C.sub.6 H.sub.5                                                                      CH.sub.3                                                                            OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                           CH.sub.2 C.sub.6 H.sub.5                                                                      OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                           CH.sub.2 C.sub.6 H.sub.5                                                                      Cl    OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                           CH.sub.2 C.sub.6 H.sub.5                                                                      CH.sub.3                                                                            OCH.sub.3                                                                           N                                          6-CH.sub.3                                                                           CH.sub.2 C.sub.6 H.sub.5                                                                      OCH.sub.3                                                                           OCH.sub.3                                                                           N                                          6-CH.sub.3                                                                           CH.sub.2 C.sub.6 H.sub.5                                                                      CH.sub.3                                                                            CH.sub.3                                                                            N                                          6-Cl   CH.sub.2 H      CH.sub.3                                                                            CH.sub.3                                                                            CH                                         6-Cl   CH.sub.2 H      CH.sub.3                                                                            OCH.sub.3                                                                           CH                                         6-Cl   CH.sub.2 H      OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                         6-Cl   CH.sub.2 H      Cl    OCH.sub.3                                                                           CH                                         6-Cl   CH.sub.2 H      CH.sub.3                                                                            OCH.sub.3                                                                           N                                          6-Cl   CH.sub.2 H      OCH.sub.3                                                                           OCH.sub.3                                                                           N                                          6-Cl   CH.sub.2 H      CH.sub.3                                                                            CH.sub.3                                                                            N                                          6-Cl   CH.sub.2 CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            CH                                         6-Cl   CH.sub.2 CH.sub.3                                                                             OCH.sub.3                                                                           CH.sub.3                                                                            CH                                         6-Cl   CH.sub.2 CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                         6-Cl   CH.sub.2 CH.sub.3                                                                             Cl    OCH.sub.3                                                                           CH                                         6-Cl   CH.sub.2 CH.sub.3                                                                             CH.sub.3                                                                            OCH.sub.3                                                                           N                                          6-Cl   CH.sub.2 CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           N                                          6-Cl   CH.sub.2 CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            N                                          6-Cl   CH.sub.2 C.sub.6 H.sub.5                                                                      CH.sub.3                                                                            CH.sub.3                                                                            CH                                         6-Cl   CH.sub.2 C.sub.6 H.sub.5                                                                      CH.sub.3                                                                            OCH.sub.3                                                                           CH                                         6-Cl   CH.sub.2 C.sub.6 H.sub.5                                                                      OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                         6-Cl   CH.sub.2 C.sub.6 H.sub.5                                                                      Cl    OCH.sub.3                                                                           CH                                         6-Cl   CH.sub.2 C.sub.6 H.sub.5                                                                      CH.sub.3                                                                            OCH.sub.3                                                                           N                                          6-Cl   CH.sub.2 C.sub.6 H.sub.5                                                                      OCH.sub.3                                                                           OCH.sub.3                                                                           N                                          6-Cl   CH.sub.2 C.sub.6 H.sub.5                                                                      CH.sub.3                                                                            CH.sub.3                                                                            N                                          H      CH.sub.2 CH.sub.2                                                                      H      CH.sub.3                                                                            CH.sub.3                                                                            CH                                         H      CH.sub.2 CH.sub.2                                                                      H      CH.sub.3                                                                            OCH.sub.3                                                                           CH                                         H      CH.sub.2 CH.sub.2                                                                      H      OCH.sub.3                                                                           OCH.sub.3                                                                           CH   189-192 (d)                           H      CH.sub.2 CH.sub.2                                                                      H      Cl    OCH.sub.3                                                                           CH                                         H      CH.sub.2 CH.sub.2                                                                      H      CH.sub.3                                                                            OCH.sub.3                                                                           N                                          H      CH.sub.2 CH.sub.2                                                                      H      OCH.sub.3                                                                           OCH.sub.3                                                                           N    147-150                               H      CH.sub.2 CH.sub.2                                                                      H      CH.sub.3                                                                            CH.sub.3                                                                            N                                          H      CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            CH                                         H      CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             CH.sub.3                                                                            OCH.sub.3                                                                           CH                                         H      CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                         H      CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             Cl    OCH.sub.3                                                                           CH                                         H      CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             CH.sub.3                                                                            OCH.sub.3                                                                           N                                          H      CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           N                                          H      CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            N                                          H      CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      CH.sub.3                                                                            CH.sub.3                                                                            CH                                         H      CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      CH.sub.3                                                                            OCH.sub.3                                                                           CH                                         H      CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                         H      CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      Cl    OCH.sub.3                                                                           CH                                         H      CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      CH.sub.3                                                                            OCH.sub.3                                                                           N                                          H      CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      OCH.sub.3                                                                           OCH.sub.3                                                                           N                                          H      CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      CH.sub.3                                                                            CH.sub.3                                                                            N                                          6-CH.sub.3                                                                           CH.sub.2 CH.sub.2                                                                      H      CH.sub.3                                                                            CH.sub.3                                                                            CH                                         6-CH.sub.3                                                                           CH.sub.2 CH.sub.2                                                                      H      CH.sub.3                                                                            OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                           CH.sub.2 CH.sub.2                                                                      H      OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                           CH.sub.2 CH.sub. 2                                                                     H      Cl    OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                           CH.sub.2 CH.sub.2                                                                      H      CH.sub.3                                                                            OCH.sub.3                                                                           N                                          6-CH.sub.3                                                                           CH.sub.2 CH.sub.2                                                                      H      OCH.sub.3                                                                           OCH.sub.3                                                                           N                                          6-CH.sub.3                                                                           CH.sub.2 CH.sub.2                                                                      H      CH.sub.3                                                                            CH.sub.3                                                                            N                                          6-CH.sub.3                                                                           CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            CH                                         6-CH.sub.3                                                                           CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             OCH.sub.3                                                                           CH.sub.3                                                                            CH                                         6-CH.sub.3                                                                           CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                           CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             Cl    OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                           CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             CH.sub.3                                                                            OCH.sub.3                                                                           N                                          6-CH.sub.3                                                                           CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           N                                          6-CH.sub.3                                                                           CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            N                                          6-CH.sub.3                                                                           CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      CH.sub.3                                                                            CH.sub.3                                                                            CH                                         6-CH.sub.3                                                                           CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      CH.sub.3                                                                            OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                           CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                           CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      Cl    OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                           CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub. 5                                                                     CH.sub.3                                                                            OCH.sub.3                                                                           N                                          6-CH.sub.3                                                                           CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      OCH.sub.3                                                                           OCH.sub.3                                                                           N                                          6-CH.sub.3                                                                           CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      CH.sub.3                                                                            CH.sub.3                                                                            N                                          6-Cl   CH.sub.2 CH.sub.2                                                                      H      CH.sub.3                                                                            CH.sub.3                                                                            CH                                         6-Cl   CH.sub.2 CH.sub.2                                                                      H      CH.sub.3                                                                            OCH.sub.3                                                                           CH                                         6-Cl   CH.sub.2 CH.sub.2                                                                      H      OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                         6-Cl   CH.sub.2 CH.sub.2                                                                      H      Cl    OCH.sub.3                                                                           CH                                         6-Cl   CH.sub.2 CH.sub.2                                                                      H      CH.sub.3                                                                            OCH.sub.3                                                                           N                                          6-Cl   CH.sub.2 CH.sub.2                                                                      H      OCH.sub.3                                                                           OCH.sub.3                                                                           N                                          6-Cl   CH.sub.2 CH.sub.2                                                                      H      CH.sub.3                                                                            CH.sub.3                                                                            N                                          6-Cl   CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            CH                                         6-Cl   CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             OCH.sub.3                                                                           CH.sub.3                                                                            CH                                         6-Cl   CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                         6-Cl   CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             Cl    OCH.sub.3                                                                           CH                                         6-Cl   CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             CH.sub.3                                                                            OCH.sub.3                                                                           N                                          6-Cl   CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           N                                          6-Cl   CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            N                                          6-Cl   CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      CH.sub.3                                                                            CH.sub.3                                                                            CH                                         6-Cl   CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      CH.sub.3                                                                            OCH.sub.3                                                                           CH                                         6-Cl   CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                         6-Cl   CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      Cl    OCH.sub.3                                                                           CH                                         6-Cl   CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      CH.sub.3                                                                            OCH.sub.3                                                                           N                                          6-Cl   CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      OCH.sub.3                                                                           OCH.sub.3                                                                           N                                          6-Cl   CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      CH.sub.3                                                                            CH.sub.3                                                                            N                                          H      CH═CH                                                                              H      CH.sub.3                                                                            CH.sub.3                                                                            CH                                         H      CH═CH                                                                              H      CH.sub.3                                                                            OCH.sub.3                                                                           CH                                         H      CH═CH                                                                              H      OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                         H      CH═CH                                                                              H      Cl    OCH.sub.3                                                                           CH                                         H      CH═CH                                                                              H      CH.sub.3                                                                            OCH.sub.3                                                                           N                                          H      CH═CH                                                                              H      OCH.sub.3                                                                           OCH.sub.3                                                                           N                                          H      CH═CH                                                                              H      CH.sub.3                                                                            CH.sub.3                                                                            N                                          H      CH═CH                                                                              CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            CH                                         H      CH═CH                                                                              CH.sub.3                                                                             CH.sub.3                                                                            OCH.sub.3                                                                           CH                                         H      CH═CH                                                                              CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                         H      CH═CH                                                                              CH.sub.3                                                                             Cl    OCH.sub.3                                                                           CH                                         H      CH═CH                                                                              CH.sub.3                                                                             CH.sub.3                                                                            OCH.sub.3                                                                           N                                          H      CH═CH                                                                              CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           N                                          H      CH═CH                                                                              CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            N                                          H      CH═CH                                                                              C.sub.6 H.sub.5                                                                      CH.sub.3                                                                            CH.sub.3                                                                            CH                                         H      CH═CH                                                                              C.sub.6 H.sub.5                                                                      CH.sub.3                                                                            OCH.sub.3                                                                           CH                                         H      CH═CH                                                                              C.sub.6 H.sub.5                                                                      OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                         H      CH═CH                                                                              C.sub.6 H.sub.5                                                                      Cl    OCH.sub.3                                                                           CH                                         H      CH═CH                                                                              C.sub.6 H.sub.5                                                                      CH.sub.3                                                                            OCH.sub.3                                                                           N                                          H      CH═CH                                                                              C.sub.6 H.sub.5                                                                      OCH.sub.3                                                                           OCH.sub.3                                                                           N                                          H      CH═CH                                                                              C.sub.6 H.sub.5                                                                      CH.sub.3                                                                            CH.sub.3                                                                            N                                          6-CH.sub.3                                                                           CH═CH                                                                              H      CH.sub.3                                                                            CH.sub.3                                                                            CH                                         6-CH.sub.3                                                                           CH═CH                                                                              H      CH.sub.3                                                                            OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                           CH═CH                                                                              H      OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                           CH═CH                                                                              H      Cl    OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                           CH═CH                                                                              H      CH.sub.3                                                                            OCH.sub.3                                                                           N                                          6-CH.sub.3                                                                           CH═CH                                                                              H      OCH.sub.3                                                                           OCH.sub.3                                                                           N                                          6-CH.sub.3                                                                           CH═CH                                                                              H      CH.sub.3                                                                            CH.sub.3                                                                            N                                          6-CH.sub.3                                                                           CH═CH                                                                              CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            CH                                         6-CH.sub.3                                                                           CH═CH                                                                              CH.sub.3                                                                             OCH.sub.3                                                                           CH.sub.3                                                                            CH                                         6-CH.sub.3                                                                           CH═ CH                                                                             CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                           CH═CH                                                                              CH.sub.3                                                                             Cl    OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                           CH═CH                                                                              CH.sub.3                                                                             CH.sub.3                                                                            OCH.sub.3                                                                           N                                          6-CH.sub.3                                                                           CH═CH                                                                              CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           N                                          6-CH.sub.3                                                                           CH═CH                                                                              CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            N                                          6-CH.sub.3                                                                           CH═CH                                                                              C.sub.6 H.sub.5                                                                      CH.sub.3                                                                            CH.sub.3                                                                            CH                                         6-CH.sub.3                                                                           CH═CH                                                                              C.sub.6 H.sub.5                                                                      CH.sub.3                                                                            OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                           CH═CH                                                                              C.sub.6 H.sub.5                                                                      OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                           CH═CH                                                                              C.sub.6 H.sub.5                                                                      Cl    OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                           CH═CH                                                                              C.sub.6 H.sub.5                                                                      CH.sub.3                                                                            OCH.sub.3                                                                           N                                          6-CH.sub.3                                                                           CH═CH                                                                              C.sub.6 H.sub.5                                                                      OCH.sub.3                                                                           OCH.sub.3                                                                           N                                          6-CH.sub.3                                                                           CH═CH                                                                              C.sub.6 H.sub.5                                                                      CH.sub.3                                                                            CH.sub.3                                                                            N                                          6-Cl   CH═CH                                                                              H      CH.sub.3                                                                            CH.sub.3                                                                            CH                                         6-Cl   CH═CH                                                                              H      CH.sub.3                                                                            OCH.sub.3                                                                           CH                                         6-Cl   CH═CH                                                                              H      OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                         6-Cl   CH═CH                                                                              H      Cl    OCH.sub.3                                                                           CH                                         6-Cl   CH═CH                                                                              H      CH.sub.3                                                                            OCH.sub.3                                                                           N                                          6-Cl   CH═CH                                                                              H      OCH.sub.3                                                                           OCH.sub.3                                                                           N                                          6-Cl   CH═CH                                                                              H      CH.sub.3                                                                            CH.sub.3                                                                            N                                          6-Cl   CH═CH                                                                              CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            CH                                         6-Cl   CH═CH                                                                              CH.sub.3                                                                             OCH.sub.3                                                                           CH.sub.3                                                                            CH                                         6-Cl   CH═CH                                                                              CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                         6-Cl   CH═CH                                                                              CH.sub.3                                                                             Cl    OCH.sub.3                                                                           CH                                         6-Cl   CH═CH                                                                              CH.sub.3                                                                             CH.sub.3                                                                            OCH.sub.3                                                                           N                                          6-Cl   CH═CH                                                                              CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           N                                          6-Cl   CH═CH                                                                              CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            N                                          6-Cl   CH═CH                                                                              C.sub.6 H.sub.5                                                                      CH.sub.3                                                                            CH.sub.3                                                                            CH                                         6-Cl   CH═CH                                                                              C.sub.6 H.sub.5                                                                      CH.sub.3                                                                            OCH.sub.3                                                                           CH                                         6-Cl   CH═CH                                                                              C.sub.6 H.sub.5                                                                      OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                         6-Cl   CH═CH                                                                              C.sub.6 H.sub.5                                                                      Cl    OCH.sub.3                                                                           CH                                         6-Cl   CH═CH                                                                              C.sub.6 H.sub.5                                                                      CH.sub.3                                                                            OCH.sub.3                                                                           N                                          6-Cl   CH═CH                                                                              C.sub.6 H.sub.5                                                                      OCH.sub.3                                                                           OCH.sub.3                                                                           N                                          6-Cl   CH═CH                                                                              C.sub.6 H.sub.5                                                                      CH.sub.3                                                                            CH.sub.3                                                                            N                                          ______________________________________                                    

                  TABLE 25                                                        ______________________________________                                        General Formula 25                                                            R.sub.1                                                                              G        R.sub.10                                                                             X     Y     Z    m.p. (°C.)                     ______________________________________                                        H      CH.sub.2 H      CH.sub.3                                                                            CH.sub.3                                                                            CH                                         H      CH.sub.2 H      CH.sub.3                                                                            OCH.sub.3                                                                           CH                                         H      CH.sub.2 H      OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                         H      CH.sub.2 H      Cl    OCH.sub.3                                                                           CH                                         H      CH.sub.2 H      CH.sub.3                                                                            OCH.sub.3                                                                           N                                          H      CH.sub.2 H      OCH.sub.3                                                                           OCH.sub.3                                                                           N                                          H      CH.sub.2 H      CH.sub.3                                                                            CH.sub.3                                                                            N                                          H      CH.sub.2 CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            CH                                         H      CH.sub.2 CH.sub.3                                                                             CH.sub.3                                                                            OCH.sub.3                                                                           CH                                         H      CH.sub.2 CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                         H      CH.sub.2 CH.sub.3                                                                             Cl    OCH.sub.3                                                                           CH                                         H      CH.sub.2 CH.sub.3                                                                             CH.sub.3                                                                            OCH.sub.3                                                                           N                                          H      CH.sub.2 CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           N                                          H      CH.sub.2 CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            N                                          H      CH.sub.2 C.sub.6 H.sub.5                                                                      CH.sub.3                                                                            CH.sub.3                                                                            CH                                         H      CH.sub.2 C.sub.6 H.sub.5                                                                      CH.sub.3                                                                            OCH.sub.3                                                                           CH                                         H      CH.sub.2 C.sub.6 H.sub.5                                                                      OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                         H      CH.sub.2 C.sub.6 H.sub.5                                                                      Cl    OCH.sub.3                                                                           CH                                         H      CH.sub.2 C.sub.6 H.sub.5                                                                      CH.sub.3                                                                            OCH.sub.3                                                                           N                                          H      CH.sub.2 C.sub.6 H.sub.5                                                                      OCH.sub.3                                                                           OCH.sub.3                                                                           N                                          H      CH.sub.2 C.sub.6 H.sub.5                                                                      CH.sub.3                                                                            CH.sub.3                                                                            N                                          6-CH.sub.3                                                                           CH.sub.2 H      CH.sub.3                                                                            CH.sub.3                                                                            CH                                         6-CH.sub.3                                                                           CH.sub.2 H      CH.sub.3                                                                            OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                           CH.sub.2 H      OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                           CH.sub.2 H      Cl    OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                           CH.sub.2 H      CH.sub.3                                                                            OCH.sub.3                                                                           N                                          6-CH.sub.3                                                                           CH.sub.2 H      OCH.sub.3                                                                           OCH.sub.3                                                                           N                                          6-CH.sub.3                                                                           CH.sub.2 H      CH.sub.3                                                                            CH.sub.3                                                                            N                                          6-CH.sub.3                                                                           CH.sub.2 CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            CH                                         6-CH.sub.3                                                                           CH.sub.2 CH.sub.3                                                                             OCH.sub.3                                                                           CH.sub.3                                                                            CH                                         6-CH.sub.3                                                                           CH.sub.2 CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                           CH.sub.2 CH.sub.3                                                                             Cl    OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                           CH.sub.2 CH.sub.3                                                                             CH.sub.3                                                                            OCH.sub.3                                                                           N                                          6-CH.sub.3                                                                           CH.sub.2 CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           N                                          6-CH.sub.3                                                                           CH.sub.2 CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            N                                          6-CH.sub.3                                                                           CH.sub.2 C.sub.6 H.sub.5                                                                      CH.sub.3                                                                            CH.sub.3                                                                            CH                                         6-CH.sub.3                                                                           CH.sub.2 C.sub.6 H.sub.5                                                                      CH.sub.3                                                                            OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                           CH.sub.2 C.sub.6 H.sub.5                                                                      OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                           CH.sub.2 C.sub.6 H.sub.5                                                                      Cl    OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                           CH.sub.2 C.sub.6 H.sub.5                                                                      CH.sub.3                                                                            OCH.sub.3                                                                           N                                          6-CH.sub.3                                                                           CH.sub.2 C.sub.6 H.sub.5                                                                      OCH.sub.3                                                                           OCH.sub.3                                                                           N                                          6-CH.sub.3                                                                           CH.sub.2 C.sub.6 H.sub.5                                                                      CH.sub.3                                                                            CH.sub.3                                                                            N                                          6-Cl   CH.sub.2 H      CH.sub.3                                                                            CH.sub.3                                                                            CH                                         6-Cl   CH.sub.2 H      CH.sub.3                                                                            OCH.sub.3                                                                           CH                                         6-Cl   CH.sub.2 H      OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                         6-Cl   CH.sub.2 H      Cl    OCH.sub.3                                                                           CH                                         6-Cl   CH.sub.2 H      CH.sub.3                                                                            OCH.sub.3                                                                           N                                          6-Cl   CH.sub.2 H      OCH.sub.3                                                                           OCH.sub.3                                                                           N                                          6-Cl   CH.sub.2 H      CH.sub.3                                                                            CH.sub.3                                                                            N                                          6-Cl   CH.sub.2 CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            CH                                         6-Cl   CH.sub.2 CH.sub.3                                                                             OCH.sub.3                                                                           CH.sub.3                                                                            CH                                         6-Cl   CH.sub.2 CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                         6-Cl   CH.sub.2 CH.sub.3                                                                             Cl    OCH.sub.3                                                                           CH                                         6-Cl   CH.sub.2 CH.sub.3                                                                             CH.sub.3                                                                            OCH.sub.3                                                                           N                                          6-Cl   CH.sub.2 CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           N                                          6-Cl   CH.sub.2 CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            N                                          6-Cl   CH.sub.2 C.sub.6 H.sub.5                                                                      CH.sub.3                                                                            CH.sub.3                                                                            CH                                         6-Cl   CH.sub.2 C.sub.6 H.sub.5                                                                      CH.sub.3                                                                            OCH.sub.3                                                                           CH                                         6-Cl   CH.sub.2 C.sub.6 H.sub.5                                                                      OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                         6-Cl   CH.sub.2 C.sub.6 H.sub.5                                                                      Cl    OCH.sub.3                                                                           CH                                         6-Cl   CH.sub.2 C.sub.6 H.sub.5                                                                      CH.sub.3                                                                            OCH.sub.3                                                                           N                                          6-Cl   CH.sub.2 C.sub.6 H.sub.5                                                                      OCH.sub.3                                                                           OCH.sub.3                                                                           N                                          6-Cl   CH.sub.2 C.sub.6 H.sub.5                                                                      CH.sub.3                                                                            CH.sub.3                                                                            N                                          H      CH.sub.2 CH.sub.2                                                                      H      CH.sub.3                                                                            CH.sub.3                                                                            CH                                         H      CH.sub.2 CH.sub.2                                                                      H      CH.sub.3                                                                            OCH.sub.3                                                                           CH                                         H      CH.sub.2 CH.sub.2                                                                      H      OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                         H      CH.sub.2 CH.sub.2                                                                      H      Cl    OCH.sub.3                                                                           CH                                         H      CH.sub.2 CH.sub.2                                                                      H      CH.sub.3                                                                            OCH.sub.3                                                                           N                                          H      CH.sub.2 CH.sub.2                                                                      H      OCH.sub.3                                                                           OCH.sub.3                                                                           N                                          H      CH.sub.2 CH.sub.2                                                                      H      CH.sub.3                                                                            CH.sub.3                                                                            N                                          H      CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            CH                                         H      CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             CH.sub.3                                                                            OCH.sub.3                                                                           CH                                         H      CH.sub.2 CH.sub. 2                                                                     CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                         H      CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             Cl    OCH.sub.3                                                                           CH                                         H      CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             CH.sub.3                                                                            OCH.sub.3                                                                           N                                          H      CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           N                                          H      CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            N                                          H      CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      CH.sub.3                                                                            CH.sub.3                                                                            CH                                         H      CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      CH.sub.3                                                                            OCH.sub.3                                                                           CH                                         H      CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                         H      CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      Cl    OCH.sub.3                                                                           CH                                         H      CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      CH.sub.3                                                                            OCH.sub.3                                                                           N                                          H      CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      OCH.sub.3                                                                           OCH.sub.3                                                                           N                                          H      CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      CH.sub.3                                                                            CH.sub.3                                                                            N                                          6-CH.sub.3                                                                           CH.sub.2 CH.sub.2                                                                      H      CH.sub.3                                                                            CH.sub.3                                                                            CH                                         6-CH.sub.3                                                                           CH.sub.2 CH.sub.2                                                                      H      CH.sub.3                                                                            OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                           CH.sub.2 CH.sub.2                                                                      H      OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                           CH.sub.2 CH.sub.2                                                                      H      Cl    OCH.sub.3                                                                           CH                                         6-CH.sub. 3                                                                          CH.sub.2 CH.sub.2                                                                      H      CH.sub.3                                                                            OCH.sub.3                                                                           N                                          6-CH.sub.3                                                                           CH.sub.2 CH.sub.2                                                                      H      OCH.sub.3                                                                           OCH.sub.3                                                                           N                                          6-CH.sub.3                                                                           CH.sub.2 CH.sub.2                                                                      H      CH.sub.3                                                                            CH.sub.3                                                                            N                                          6-CH.sub.3                                                                           CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            CH                                         6-CH.sub.3                                                                           CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             OCH.sub.3                                                                           CH.sub.3                                                                            CH                                         6-CH.sub.3                                                                           CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                           CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             Cl    OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                           CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             CH.sub.3                                                                            OCH.sub.3                                                                           N                                          6-CH.sub.3                                                                           CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           N                                          6-CH.sub.3                                                                           CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            N                                          6-CH.sub.3                                                                           CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      CH.sub.3                                                                            CH.sub.3                                                                            CH                                         6-CH.sub.3                                                                           CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      CH.sub.3                                                                            OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                           CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                           CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      Cl    OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                           CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      CH.sub.3                                                                            OCH.sub.3                                                                           N                                          6-CH.sub. 3                                                                          CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      OCH.sub.3                                                                           OCH.sub.3                                                                           N                                          6-CH.sub.3                                                                           CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      CH.sub.3                                                                            CH.sub.3                                                                            N                                          6-Cl   CH.sub.2 CH.sub.2                                                                      H      CH.sub.3                                                                            CH.sub.3                                                                            CH                                         6-Cl   CH.sub.2 CH.sub.2                                                                      H      CH.sub.3                                                                            OCH.sub.3                                                                           CH                                         6-Cl   CH.sub.2 CH.sub.2                                                                      H      OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                         6-Cl   CH.sub.2 CH.sub.2                                                                      H      Cl    OCH.sub.3                                                                           CH                                         6-Cl   CH.sub.2 CH.sub.2                                                                      H      CH.sub.3                                                                            OCH.sub.3                                                                           N                                          6-Cl   CH.sub.2 CH.sub.2                                                                      H      OCH.sub.3                                                                           OCH.sub.3                                                                           N                                          6-Cl   CH.sub.2 CH.sub.2                                                                      H      CH.sub.3                                                                            CH.sub.3                                                                            N                                          6-Cl   CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            CH                                         6-Cl   CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             OCH.sub.3                                                                           CH.sub.3                                                                            CH                                         6-Cl   CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                         6-Cl   CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             Cl    OCH.sub.3                                                                           CH                                         6-Cl   CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             CH.sub.3                                                                            OCH.sub.3                                                                           N                                          6-Cl   CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           N                                          6-Cl   CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            N                                          6-Cl   CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      CH.sub.3                                                                            CH.sub. 3                                                                           CH                                         6-Cl   CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      CH.sub.3                                                                            OCH.sub.3                                                                           CH                                         6-Cl   CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                         6-Cl   CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      Cl    OCH.sub.3                                                                           CH                                         6-Cl   CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      CH.sub.3                                                                            OCH.sub.3                                                                           N                                          6-Cl   CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      OCH.sub.3                                                                           OCH.sub.3                                                                           N                                          6-Cl   CH.sub.2 CH.sub.2                                                                      C.sub.6 H.sub.5                                                                      CH.sub.3                                                                            CH.sub.3                                                                            N                                          H      CH═CH                                                                              H      CH.sub.3                                                                            CH.sub.3                                                                            CH                                         H      CH═CH                                                                              H      CH.sub.3                                                                            OCH.sub.3                                                                           CH                                         H      CH═CH                                                                              H      OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                         H      CH═CH                                                                              H      Cl    OCH.sub.3                                                                           CH                                         H      CH═CH                                                                              H      CH.sub.3                                                                            OCH.sub.3                                                                           N                                          H      CH═CH                                                                              H      OCH.sub.3                                                                           OCH.sub.3                                                                           N                                          H      CH═CH                                                                              H      CH.sub.3                                                                            CH.sub.3                                                                            N                                          H      CH═CH                                                                              CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            CH                                         H      CH═CH                                                                              CH.sub.3                                                                             CH.sub.3                                                                            OCH.sub.3                                                                           CH                                         H      CH═CH                                                                              CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                         H      CH═CH                                                                              CH.sub.3                                                                             Cl    OCH.sub.3                                                                           CH                                         H      CH═CH                                                                              CH.sub.3                                                                             CH.sub.3                                                                            OCH.sub.3                                                                           N                                          H      CH═CH                                                                              CH.sub. 3                                                                            OCH.sub.3                                                                           OCH.sub.3                                                                           N                                          H      CH═CH                                                                              CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            N                                          H      CH═CH                                                                              C.sub.6 H.sub.5                                                                      CH.sub.3                                                                            CH.sub.3                                                                            CH                                         H      CH═CH                                                                              C.sub.6 H.sub.5                                                                      CH.sub.3                                                                            OCH.sub.3                                                                           CH                                         H      CH═CH                                                                              C.sub.6 H.sub.5                                                                      OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                         H      CH═CH                                                                              C.sub.6 H.sub.5                                                                      Cl    OCH.sub.3                                                                           CH                                         H      CH═CH                                                                              C.sub.6 H.sub.5                                                                      CH.sub.3                                                                            OCH.sub.3                                                                           N                                          H      CH═CH                                                                              C.sub.6 H.sub.5                                                                      OCH.sub.3                                                                           OCH.sub.3                                                                           N                                          H      CH═CH                                                                              C.sub.6 H.sub.5                                                                      CH.sub.3                                                                            CH.sub.3                                                                            N                                          6-CH.sub.3                                                                           CH═CH                                                                              H      CH.sub.3                                                                            CH.sub.3                                                                            CH                                         6-CH.sub.3                                                                           CH═CH                                                                              H      CH.sub.3                                                                            OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                           CH═CH                                                                              H      OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                           CH═CH                                                                              H      Cl    OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                           CH═CH                                                                              H      CH.sub.3                                                                            OCH.sub.3                                                                           N                                          6-CH.sub.3                                                                           CH═CH                                                                              H      OCH.sub.3                                                                           OCH.sub.3                                                                           N                                          6-CH.sub.3                                                                           CH═CH                                                                              H      CH.sub.3                                                                            CH.sub.3                                                                            N                                          6-CH.sub.3                                                                           CH═CH                                                                              CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            CH                                         6-CH.sub.3                                                                           CH═CH                                                                              CH.sub.3                                                                             OCH.sub.3                                                                           CH.sub.3                                                                            CH                                         6-CH.sub.3                                                                           CH═CH                                                                              CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                           CH═CH                                                                              CH.sub.3                                                                             Cl    OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                           CH═CH                                                                              CH.sub.3                                                                             CH.sub.3                                                                            OCH.sub.3                                                                           N                                          6-CH.sub.3                                                                           CH═CH                                                                              CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           N                                          6-CH.sub.3                                                                           CH═CH                                                                              CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            N                                          6-CH.sub.3                                                                           CH═CH                                                                              C.sub.6 H.sub.5                                                                      CH.sub.3                                                                            CH.sub.3                                                                            CH                                         6-CH.sub.3                                                                           CH═CH                                                                              C.sub.6 H.sub.5                                                                      CH.sub.3                                                                            OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                           CH═CH                                                                              C.sub.6 H.sub.5                                                                      OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                           CH═CH                                                                              C.sub.6 H.sub.5                                                                      Cl    OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                           CH═CH                                                                              C.sub.6 H.sub.5                                                                      CH.sub.3                                                                            OCH.sub.3                                                                           N                                          6-CH.sub.3                                                                           CH═CH                                                                              C.sub.6 H.sub.5                                                                      OCH.sub.3                                                                           OCH.sub.3                                                                           N                                          6-CH.sub.3                                                                           CH═CH                                                                              C.sub.6 H.sub.5                                                                      CH.sub.3                                                                            CH.sub.3                                                                            N                                          6-Cl   CH═CH                                                                              H      CH.sub.3                                                                            CH.sub.3                                                                            CH                                         6-Cl   CH═CH                                                                              H      CH.sub.3                                                                            OCH.sub.3                                                                           CH                                         6-Cl   CH═CH                                                                              H      OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                         6-Cl   CH═CH                                                                              H      Cl    OCH.sub.3                                                                           CH                                         6-Cl   CH═CH                                                                              H      CH.sub.3                                                                            OCH.sub.3                                                                           N                                          6-Cl   CH═CH                                                                              H      OCH.sub.3                                                                           OCH.sub.3                                                                           N                                          6-Cl   CH═CH                                                                              H      CH.sub.3                                                                            CH.sub.3                                                                            N                                          6-Cl   CH═CH                                                                              CH.sub. 3                                                                            CH.sub.3                                                                            CH.sub.3                                                                            CH                                         6-Cl   CH═CH                                                                              CH.sub.3                                                                             OCH.sub.3                                                                           CH.sub.3                                                                            CH                                         6-Cl   CH═CH                                                                              CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                         6-Cl   CH═CH                                                                              CH.sub.3                                                                             Cl    OCH.sub.3                                                                           CH                                         6-Cl   CH═CH                                                                              CH.sub.3                                                                             CH.sub.3                                                                            OCH.sub.3                                                                           N                                          6-Cl   CH═CH                                                                              CH.sub.3                                                                             OCH.sub.3                                                                           OCH.sub.3                                                                           N                                          6-Cl   CH═CH                                                                              CH.sub.3                                                                             CH.sub.3                                                                            CH.sub.3                                                                            N                                          6-Cl   CH═CH                                                                              C.sub.6 H.sub.5                                                                      CH.sub.3                                                                            CH.sub.3                                                                            CH                                         6-Cl   CH═CH                                                                              C.sub.6 H.sub.5                                                                      CH.sub.3                                                                            OCH.sub.3                                                                           CH                                         6-Cl   CH═CH                                                                              C.sub.6 H.sub.5                                                                      OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                         6-Cl   CH═CH                                                                              C.sub.6 H.sub.5                                                                      Cl    OCH.sub.3                                                                           CH                                         6-Cl   CH═CH                                                                              C.sub.6 H.sub.5                                                                      CH.sub.3                                                                            OCH.sub.3                                                                           N                                          6-Cl   CH═CH                                                                              C.sub.6 H.sub.5                                                                      OCH.sub.3                                                                           OCH.sub.3                                                                           N                                          6-Cl   CH═CH                                                                              C.sub.6 H.sub.5                                                                      CH.sub.3                                                                            CH.sub.3                                                                            N                                          ______________________________________                                    

                  TABLE 26                                                        ______________________________________                                        General Formula 26                                                            R.sub.1                                                                             G        R.sub.5 X     Y     Z     m.p. (°C.)                    ______________________________________                                        H     CH.sub.2 H       CH.sub.3                                                                            CH.sub.3                                                                            CH                                         H     CH.sub.2 H       CH.sub.3                                                                            OCH.sub.3                                                                           CH                                         H     CH.sub.2 H       OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                         H     CH.sub.2 H       Cl    OCH.sub.3                                                                           CH                                         H     CH.sub.2 H       CH.sub.3                                                                            OCH.sub.3                                                                           N                                          H     CH.sub.2 H       OCH.sub.3                                                                           OCH.sub.3                                                                           N                                          H     CH.sub.2 H       CH.sub.3                                                                            CH.sub.3                                                                            N                                          H     CH.sub.2 CH.sub.3                                                                              CH.sub.3                                                                            CH.sub.3                                                                            CH                                         H     CH.sub.2 CH.sub.3                                                                              CH.sub.3                                                                            OCH.sub.3                                                                           CH                                         H     CH.sub.2 CH.sub.3                                                                              OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                         H     CH.sub.2 CH.sub.3                                                                              Cl    OCH.sub.3                                                                           CH                                         H     CH.sub.2 CH.sub.3                                                                              CH.sub.3                                                                            OCH.sub.3                                                                           N                                          H     CH.sub.2 CH.sub.3                                                                              OCH.sub.3                                                                           OCH.sub.3                                                                           N                                          H     CH.sub.2 CH.sub.3                                                                              CH.sub.3                                                                            CH.sub.3                                                                            N                                          6-CH.sub.3                                                                          CH.sub.2 H       CH.sub.3                                                                            CH.sub.3                                                                            CH                                         6-CH.sub.3                                                                          CH.sub.2 H       CH.sub.3                                                                            OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                          CH.sub.2 H       OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                          CH.sub.2 H       Cl    OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                          CH.sub.2 H       CH.sub.3                                                                            OCH.sub.3                                                                           N                                          6-CH.sub.3                                                                          CH.sub.2 H       OCH.sub.3                                                                           OCH.sub.3                                                                           N                                          6-CH.sub.3                                                                          CH.sub.2 H       CH.sub.3                                                                            CH.sub.3                                                                            N                                          6-CH.sub.3                                                                          CH.sub.2 CH.sub.3                                                                              CH.sub.3                                                                            CH.sub.3                                                                            CH                                         6-CH.sub.3                                                                          CH.sub.2 CH.sub.3                                                                              CH.sub.3                                                                            OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                          CH.sub.2 CH.sub.3                                                                              OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                          CH.sub.2 CH.sub.3                                                                              Cl    OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                          CH.sub.2 CH.sub.3                                                                              CH.sub.3                                                                            OCH.sub.3                                                                           N                                          6-CH.sub.3                                                                          CH.sub.2 CH.sub.3                                                                              OCH.sub.3                                                                           OCH.sub.3                                                                           N                                          6-CH.sub.3                                                                          CH.sub.2 CH.sub.3                                                                              CH.sub.3                                                                            CH.sub.3                                                                            N                                          H     CH.sub.2 CH.sub.2                                                                      H       CH.sub.3                                                                            CH.sub.3                                                                            CH                                         H     CH.sub.2 CH.sub.2                                                                      H       CH.sub.3                                                                            OCH.sub.3                                                                           CH                                         H     CH.sub.2 CH.sub.2                                                                      H       OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                         H     CH.sub.2 CH.sub.2                                                                      H       Cl    OCH.sub.3                                                                           CH                                         H     CH.sub.2 CH.sub.2                                                                      H       CH.sub.3                                                                            OCH.sub.3                                                                           N                                          H     CH.sub.2 CH.sub.2                                                                      H       OCH.sub.3                                                                           OCH.sub.3                                                                           N                                          H     CH.sub.2 CH.sub.2                                                                      H       CH.sub.3                                                                            CH.sub.3                                                                            N                                          H     CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              CH.sub.3                                                                            CH.sub.3                                                                            CH                                         H     CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              CH.sub.3                                                                            OCH.sub.3                                                                           CH                                         H     CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                         H     CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              Cl    OCH.sub.3                                                                           CH                                         H     CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              CH.sub.3                                                                            OCH.sub.3                                                                           N                                          H     CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              OCH.sub.3                                                                           OCH.sub.3                                                                           N                                          H     CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              CH.sub.3                                                                            CH.sub.3                                                                            N                                          6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                      H       CH.sub.3                                                                            CH.sub.3                                                                            CH                                         6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                      H       CH.sub.3                                                                            OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                      H       OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                      H       Cl    OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                      H       CH.sub.3                                                                            OCH.sub.3                                                                           N                                          6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                      H       OCH.sub.3                                                                           OCH.sub.3                                                                           N                                          6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                      H       CH.sub.3                                                                            CH.sub.3                                                                            N                                          6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              CH.sub.3                                                                            CH.sub.3                                                                            CH                                         6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              CH.sub.3                                                                            OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              Cl    OCH.sub. 3                                                                          CH                                         6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              CH.sub.3                                                                            OCH.sub.3                                                                           N                                          6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              OCH.sub.3                                                                           OCH.sub.3                                                                           N                                          6-CH.sub.3                                                                          CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              CH.sub.3                                                                            CH.sub.3                                                                            N                                          H     CH═CH                                                                              H       CH.sub.3                                                                            CH.sub.3                                                                            CH                                         H     CH═CH                                                                              H       CH.sub.3                                                                            OCH.sub.3                                                                           CH                                         H     CH═CH                                                                              H       OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                         H     CH═CH                                                                              H       Cl    OCH.sub.3                                                                           CH                                         H     CH═CH                                                                              H       CH.sub.3                                                                            OCH.sub.3                                                                           N                                          H     CH═CH                                                                              H       OCH.sub.3                                                                           OCH.sub.3                                                                           N                                          H     CH═CH                                                                              H       CH.sub.3                                                                            CH.sub.3                                                                            N                                          H     CH═CH                                                                              CH.sub.3                                                                              CH.sub.3                                                                            CH.sub.3                                                                            CH                                         H     CH═CH                                                                              CH.sub.3                                                                              CH.sub.3                                                                            OCH.sub.3                                                                           CH                                         H     CH═CH                                                                              CH.sub.3                                                                              OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                         H     CH═CH                                                                              CH.sub.3                                                                              Cl    OCH.sub.3                                                                           CH                                         H     CH═CH                                                                              CH.sub.3                                                                              CH.sub.3                                                                            OCH.sub.3                                                                           N                                          H     CH═CH                                                                              CH.sub.3                                                                              OCH.sub.3                                                                           OCH.sub.3                                                                           N                                          H     CH═CH                                                                              CH.sub.3                                                                              CH.sub.3                                                                            CH.sub.3                                                                            N                                          6-CH.sub.3                                                                          CH═CH                                                                              H       CH.sub.3                                                                            CH.sub.3                                                                            CH                                         6-CH.sub.3                                                                          CH═CH                                                                              H       CH.sub.3                                                                            OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                          CH═CH                                                                              H       OCH.sub.3                                                                           OCH.sub. 3                                                                          CH                                         6-CH.sub.3                                                                          CH═CH                                                                              H       Cl    OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                          CH═CH                                                                              H       CH.sub.3                                                                            OCH.sub.3                                                                           N                                          6-CH.sub.3                                                                          CH═CH                                                                              H       OCH.sub.3                                                                           OCH.sub.3                                                                           N                                          6-CH.sub.3                                                                          CH═CH                                                                              H       CH.sub.3                                                                            CH.sub.3                                                                            N                                          6-CH.sub.3                                                                          CH═CH                                                                              CH.sub.3                                                                              CH.sub.3                                                                            CH.sub.3                                                                            CH                                         6-CH.sub.3                                                                          CH═CH                                                                              CH.sub.3                                                                              CH.sub.3                                                                            OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                          CH═CH                                                                              CH.sub.3                                                                              OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                          CH═CH                                                                              CH.sub.3                                                                              Cl    OCH.sub.3                                                                           CH                                         6-CH.sub.3                                                                          CH═CH                                                                              CH.sub.3                                                                              CH.sub.3                                                                            OCH.sub.3                                                                           N                                          6-CH.sub.3                                                                          CH═CH                                                                              CH.sub.3                                                                              OCH.sub.3                                                                           OCH.sub.3                                                                           N                                          6-CH.sub.3                                                                          CH═CH                                                                              CH.sub.3                                                                              CH.sub.3                                                                            CH.sub.3                                                                            N                                          ______________________________________                                    

                  TABLE 27                                                        ______________________________________                                        General Formula 27                                                            R.sub.1                                                                             G        R.sub.12                                                                              X     Y     Z     m.p. (°C.)                    ______________________________________                                        H     CH.sub.2 H       CH.sub.3                                                                            CH.sub.3                                                                            CH                                         H     CH.sub.2 H       CH.sub.3                                                                            OCH.sub.3                                                                           CH                                         H     CH.sub.2 H       OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                         H     CH.sub.2 H       Cl    OCH.sub.3                                                                           CH                                         H     CH.sub.2 H       CH.sub.3                                                                            OCH.sub.3                                                                           N                                          H     CH.sub.2 H       OCH.sub.3                                                                           OCH.sub.3                                                                           N                                          H     CH.sub.2 H       CH.sub.3                                                                            CH.sub.3                                                                            N                                          H     CH.sub.2 CH.sub.3                                                                              CH.sub.3                                                                            CH.sub.3                                                                            CH                                         H     CH.sub.2 CH.sub.3                                                                              CH.sub.3                                                                            OCH.sub.3                                                                           CH                                         H     CH.sub.2 CH.sub.3                                                                              OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                         H     CH.sub.2 CH.sub.3                                                                              Cl    OCH.sub.3                                                                           CH                                         H     CH.sub.2 CH.sub.3                                                                              CH.sub.3                                                                            OCH.sub.3                                                                           N                                          H     CH.sub.2 CH.sub.3                                                                              OCH.sub.3                                                                           OCH.sub.3                                                                           N                                          H     CH.sub.2 CH.sub.3                                                                              CH.sub.3                                                                            CH.sub.3                                                                            N                                          6-Cl  CH.sub.2 H       CH.sub.3                                                                            CH.sub.3                                                                            CH                                         6-Cl  CH.sub.2 H       CH.sub.3                                                                            OCH.sub.3                                                                           CH                                         6-Cl  CH.sub.2 H       OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                         6-Cl  CH.sub.2 H       Cl    OCH.sub.3                                                                           CH                                         6-Cl  CH.sub.2 H       CH.sub.3                                                                            OCH.sub.3                                                                           N                                          6-Cl  CH.sub.2 H       OCH.sub.3                                                                           OCH.sub.3                                                                           N                                          6-Cl  CH.sub.2 H       CH.sub.3                                                                            CH.sub.3                                                                            N                                          6-Cl  CH.sub.2 CH.sub.3                                                                              CH.sub.3                                                                            CH.sub.3                                                                            CH                                         6-Cl  CH.sub.2 CH.sub.3                                                                              CH.sub.3                                                                            OCH.sub.3                                                                           CH                                         6-Cl  CH.sub.2 CH.sub.3                                                                              OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                         6-Cl  CH.sub.2 CH.sub.3                                                                              Cl    OCH.sub.3                                                                           CH                                         6-Cl  CH.sub.2 CH.sub.3                                                                              CH.sub.3                                                                            OCH.sub.3                                                                           N                                          6-Cl  CH.sub.2 CH.sub.3                                                                              OCH.sub.3                                                                           OCH.sub.3                                                                           N                                          6-Cl  CH.sub.2 CH.sub.3                                                                              CH.sub.3                                                                            CH.sub.3                                                                            N                                          H     CH.sub.2 CH.sub.2                                                                      H       CH.sub.3                                                                            CH.sub.3                                                                            CH                                         H     CH.sub.2 CH.sub.2                                                                      H       CH.sub.3                                                                            OCH.sub.3                                                                           CH                                         H     CH.sub.2 CH.sub.2                                                                      H       OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                         H     CH.sub.2 CH.sub.2                                                                      H       Cl    OCH.sub.3                                                                           CH                                         H     CH.sub.2 CH.sub.2                                                                      H       CH.sub.3                                                                            OCH.sub.3                                                                           N                                          H     CH.sub.2 CH.sub.2                                                                      H       OCH.sub.3                                                                           OCH.sub.3                                                                           N                                          H     CH.sub.2 CH.sub.2                                                                      H       CH.sub.3                                                                            CH.sub.3                                                                            N                                          H     CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              CH.sub.3                                                                            CH.sub.3                                                                            CH                                         H     CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              CH.sub.3                                                                            OCH.sub.3                                                                           CH                                         H     CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                         H     CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              Cl    OCH.sub.3                                                                           CH                                         H     CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              CH.sub.3                                                                            OCH.sub.3                                                                           N                                          H     CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              OCH.sub.3                                                                           OCH.sub.3                                                                           N                                          H     CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              CH.sub.3                                                                            CH.sub.3                                                                            N                                          6-Cl  CH.sub.2 CH.sub.2                                                                      H       CH.sub.3                                                                            CH.sub.3                                                                            CH                                         6-Cl  CH.sub.2 CH.sub.2                                                                      H       CH.sub.3                                                                            OCH.sub.3                                                                           CH                                         6-Cl  CH.sub.2 CH.sub.2                                                                      H       OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                         6-Cl  CH.sub.2 CH.sub.2                                                                      H       Cl    OCH.sub.3                                                                           CH                                         6-Cl  CH.sub.2 CH.sub.2                                                                      H       CH.sub.3                                                                            OCH.sub.3                                                                           N                                          6-Cl  CH.sub.2 CH.sub.2                                                                      H       OCH.sub.3                                                                           OCH.sub.3                                                                           N                                          6-Cl  CH.sub.2 CH.sub.2                                                                      H       CH.sub.3                                                                            CH.sub.3                                                                            N                                          6-Cl  CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              CH.sub.3                                                                            CH.sub.3                                                                            CH                                         6-Cl  CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              CH.sub.3                                                                            OCH.sub.3                                                                           CH                                         6-Cl  CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                         6-Cl  CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              Cl    OCH.sub.3                                                                           CH                                         6-Cl  CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              CH.sub.3                                                                            OCH.sub.3                                                                           N                                          6-Cl  CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              OCH.sub.3                                                                           OCH.sub.3                                                                           N                                          6-Cl  CH.sub.2 CH.sub.2                                                                      CH.sub.3                                                                              CH.sub.3                                                                            CH.sub.3                                                                            N                                          H     CH═CH                                                                              H       CH.sub.3                                                                            CH.sub.3                                                                            CH                                         H     CH═CH                                                                              H       CH.sub.3                                                                            OCH.sub.3                                                                           CH                                         H     CH═CH                                                                              H       OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                         H     CH═CH                                                                              H       Cl    OCH.sub.3                                                                           CH                                         H     CH═CH                                                                              H       CH.sub.3                                                                            OCH.sub.3                                                                           N                                          H     CH═CH                                                                              H       OCH.sub.3                                                                           OCH.sub.3                                                                           N                                          H     CH═CH                                                                              H       CH.sub.3                                                                            CH.sub.3                                                                            N                                          H     CH═CH                                                                              CH.sub.3                                                                              CH.sub.3                                                                            CH.sub.3                                                                            CH                                         H     CH═CH                                                                              CH.sub.3                                                                              CH.sub.3                                                                            OCH.sub.3                                                                           CH                                         H     CH═CH                                                                              CH.sub.3                                                                              OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                         H     CH═CH                                                                              CH.sub.3                                                                              Cl    OCH.sub.3                                                                           CH                                         H     CH═CH                                                                              CH.sub.3                                                                              CH.sub.3                                                                            OCH.sub.3                                                                           N                                          H     CH═CH                                                                              CH.sub.3                                                                              OCH.sub.3                                                                           OCH.sub.3                                                                           N                                          H     CH═CH                                                                              CH.sub.3                                                                              CH.sub.3                                                                            CH.sub.3                                                                            N                                          6-Cl  CH═CH                                                                              H       CH.sub.3                                                                            CH.sub.3                                                                            CH                                         6-Cl  CH═CH                                                                              H       CH.sub.3                                                                            OCH.sub.3                                                                           CH                                         6-Cl  CH═CH                                                                              H       OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                         6-Cl  CH═CH                                                                              H       Cl    OCH.sub.3                                                                           CH                                         6-Cl  CH═CH                                                                              H       CH.sub.3                                                                            OCH.sub.3                                                                           N                                          6-Cl  CH═CH                                                                              H       OCH.sub.3                                                                           OCH.sub.3                                                                           N                                          6-Cl  CH═CH                                                                              H       CH.sub.3                                                                            CH.sub.3                                                                            N                                          6-Cl  CH═CH                                                                              CH.sub.3                                                                              CH.sub.3                                                                            CH.sub.3                                                                            CH                                         6-Cl  CH═CH                                                                              CH.sub.3                                                                              CH.sub.3                                                                            OCH.sub.3                                                                           CH                                         6-Cl  CH═CH                                                                              CH.sub.3                                                                              OCH.sub.3                                                                           OCH.sub.3                                                                           CH                                         6-Cl  CH═CH                                                                              CH.sub.3                                                                              Cl    OCH.sub.3                                                                           CH                                         6-Cl  CH═CH                                                                              CH.sub.3                                                                              CH.sub.3                                                                            OCH.sub.3                                                                           N                                          6-Cl  CH═CH                                                                              CH.sub.3                                                                              OCH.sub.3                                                                           OCH.sub.3                                                                           N                                          6-Cl  CH═CH                                                                              CH.sub.3                                                                              CH.sub.3                                                                            CH.sub.3                                                                            N                                          ______________________________________                                    

                  TABLE 28                                                        ______________________________________                                        General Formula 28                                                            R.sub.1   X         Y        Z      m.p. (°C.)                         ______________________________________                                        H         OCH.sub.3 OCH.sub.3                                                                              N                                                H         OCH.sub.3 OCH.sub.3                                                                              CH                                               H         CH.sub.3  OCH.sub.3                                                                              N                                                H         CH.sub.3  OCH.sub.3                                                                              CH                                               H         Cl        OCH.sub.3                                                                              CH                                               H         CH.sub.3  CH.sub.3 CH                                               6-CH.sub.3                                                                              OCH.sub.3 OCH.sub.3                                                                              N                                                6-CH.sub.3                                                                              OCH.sub.3 OCH.sub.3                                                                              CH                                               6-CH.sub.3                                                                              CH.sub.3  OCH.sub.3                                                                              N                                                6-CH.sub.3                                                                              CH.sub.3  OCH.sub.3                                                                              CH                                               6-CH.sub.3                                                                              Cl        OCH.sub.3                                                                              CH                                               6-CH.sub.3                                                                              CH.sub.3  CH.sub.3 CH                                               6-Cl      OCH.sub.3 OCH.sub.3                                                                              N                                                6-Cl      OCH.sub.3 OCH.sub.3                                                                              CH                                               6-Cl      CH.sub.3  OCH.sub.3                                                                              N                                                6-Cl      CH.sub.3  OCH.sub.3                                                                              CH                                               6-Cl      Cl        OCH.sub.3                                                                              CH                                               6-Cl      CH.sub.3  CH.sub.3 CH                                               6-OCH.sub.3                                                                             OCH.sub.3 OCH.sub.3                                                                              N                                                6-OCH.sub.3                                                                             OCH.sub.3 OCH.sub.3                                                                              CH                                               6-OCH.sub.3                                                                             CH.sub.3  OCH.sub.3                                                                              N                                                6-OCH.sub.3                                                                             CH.sub.3  OCH.sub.3                                                                              CH                                               6-OCH.sub.3                                                                             Cl        OCH.sub.3                                                                              CH                                               6-OCH.sub.3                                                                             CH.sub.3  CH.sub.3 CH                                               5-Cl      OCH.sub.3 OCH.sub.3                                                                              N                                                5-Cl      OCH.sub.3 OCH.sub.3                                                                              CH                                               5-Cl      CH.sub.3  OCH.sub.3                                                                              N                                                5-Cl      CH.sub.3  OCH.sub. 3                                                                             CH                                               5-Cl      Cl        OCH.sub.3                                                                              CH                                               5-Cl      CH.sub.3  CH.sub.3 CH                                               5-OCH.sub.3                                                                             OCH.sub.3 OCH.sub.3                                                                              N                                                5-OCH.sub.3                                                                             OCH.sub.3 OCH.sub.3                                                                              CH                                               5-OCH.sub.3                                                                             CH.sub.3  OCH.sub.3                                                                              N                                                5-OCH.sub.3                                                                             CH.sub.3  OCH.sub.3                                                                              CH                                               5-OCH.sub.3                                                                             Cl        OCH.sub.3                                                                              CH                                               5-OCH.sub.3                                                                             CH.sub.3  CH.sub.3 CH                                               5-SCH.sub.3                                                                             OCH.sub.3 OCH.sub.3                                                                              N                                                5-SCH.sub.3                                                                             OCH.sub.3 OCH.sub.3                                                                              CH                                               5-SCH.sub.3                                                                             CH.sub.3  OCH.sub.3                                                                              N                                                5-SCH.sub.3                                                                             CH.sub.3  OCH.sub.3                                                                              CH                                               5-SCH.sub.3                                                                             Cl        OCH.sub.3                                                                              CH                                               5-SCH.sub.3                                                                             CH.sub.3  CH.sub.3 CH                                               ______________________________________                                    

Formulations

Useful formulations of the compounds of Formula I can be prepared inconventional ways. They include dusts, granules, pellets, solutions,suspensions, emulsions, wettable powders, emulsifiable concentrates andthe like. Many of these may be applied directly. Sprayable formulationscan be extended in suitable media and used at spray volumes of from afew liters to several hundred liters per hectare. High strengthcompositions are primarily used as intermediates for furtherformulation. The formulations, broadly, contain about 0.1% to 99% byweight of active ingredient(s) and at least one of (a) about 0.1% to 20%surfactant(s) and (b) about 1% to 99.9% solid or liquid inertdiluent(s). More specifically, they will contain these ingredients inthe following approximate proportions:

                  TABLE 29                                                        ______________________________________                                                    Active  Weight Percent*                                                       Ingredient                                                                            Diluent(s)                                                                              Surfactant(s)                                   ______________________________________                                        Wettable Powders                                                                            20-90      0-74     1-10                                        Oil Suspensions,                                                                             3-50     40-95     0-15                                        Emulsions, Solutions,                                                         (including Emulsifiable                                                       Concentrates)                                                                 Aqueous Suspension                                                                          10-50     40-84     1-20                                        Dusts          1-25     70-99     0-5                                         Granules and Pellets                                                                        0.1-95      5-99.9  0-15                                        High Strength 90-99      0-10     0-2                                         Compositions                                                                  ______________________________________                                         *Active ingredient plus at least one of a Surfactant or a Diluent equals      100 weight percent.                                                      

Lower or higher levels of active ingredient can, of course, be presentdepending on the intended use and the physical properties of thecompound. Higher ratios of surfactant to active ingredient are sometimesdesirable, and are achieved by incorporation into the formulation or bytank mixing.

Typical solid diluents are described in Watkins, et al., "Handbook ofInsecticide Dust Diluents and Carriers", 2nd Ed., Dorland Books,Caldwell, N.J., but other solids, either mined or manufactured, may beused. The more absorptive diluents are preferred for wettable powdersand the denser ones for dusts. Typical liquid diluents and solvents aredescribed in Marsden, "Solvents Guide," 2nd Ed., Interscience, New York,1950. Solubility under 0.1% is preferred for suspension concentrates;solution concentrates are preferably stable against phase separation at0° C. "McCutcheon's Detergents and Emulsifiers Annual", MC PublishingCorp., Ridgewood, N.J., as well as Sisely and Wood, "Encyclopedia ofSurface Active Agents", Chemical Publishing Co., Inc., New York, 1964,list surfactants and recommended uses. All formulations can containminor amounts of additives to reduce foaming, caking, corrosion,microbiological growth, etc.

The methods of making such compositions are well known. Solutions areprepared by simply mixing the ingredients. Fine solid compositions aremade by blending and, usually, grinding as in a hammer or fluid energymill. Suspensions are prepared by wet milling (see, for example,Littler, U.S. Pat. No. 3,060,084). Granules and pellets may be made byspraying the active material upon preformed granular carriers or byagglomeration techniques.

In the following examples, all parts are by weight unless otherwiseindicated.

EXAMPLE 17 Wettable Powder

N-[(4,6-dimethoxy-1,3,5-triazin-2-yl)aminocarbonyl]-1,4-dihydro-3-methyl-4-oxo-1-phenyl-indeno[1,2-C]pyrazole-5-sulfonamide:80%

sodium alkylnaphthalenesulfonate: 2%

sodium ligninsulfonate: 2%

synthetic amorphous silica: 3%

kaolinite: 13%

The ingredients are blended, hammer-milled until all the solids areessentially under 50 microns, reblended, and packaged.

EXAMPLE 18 Wettable Powder

N-[(4-methoxy-6-methylpyrimidin-2-yl)aminocarbonyl]-1,4-dihydro-3-methyl-4-oxo-1-phyenyl-indeno[1,2-C]pyrazole-5-sulfonamide:50%

sodium alkylnaphthalenesulfonate: 2%

low viscosity methyl cellulose: 2%

diatomaceous earth: 46%

The ingredients are blended, coarsely hammer-milled and then air-milledto produce particles essentially all below 10 microns in diameter. Theproduct is reblended before packaging.

EXAMPLE 19 Granule

Wettable Powder of Example 18: 5%

attapulgite granules (U.S.S. 20-40 mesh; 0.84-0.42 mm): 95%

A slurry of wettable powder containing 25% solids is sprayed on thesurface of attapulgite granules in a double-cone blender. The granulesare dried and packaged.

EXAMPLE 20 Extruded Pellet

N-[(4,6-dimethoxy-1,3,5-triazin-2-yl)aminocarbonyl]-1,4-dihydro-3-methyl-4-oxo-1-phenyl-indeno[1,2-C]pyrazole-5-sulfonamide:25%

anhydrous sodium sulfate: 10%

crude calcium ligninsulfonate: 5%

sodium alkylnaphthalenesulfonate: 1%

calcium/magnesium bentonite: 59%

The ingredients are blended, hammer-milled and then moistened with about12% water. The mixture is extruded as cylinders about 3 mm diameterwhich are cut to produce pellets about 3 mm long. These may be useddirectly after drying, or the dried pellets may be crushed to pass aU.S.S. No. 20 sieve (0.84 mm openings). The granules held on a U.S.S.No. 40 sieve (0.42 mm openings) may be packaged for use and the finesrecycled.

EXAMPLE 21 Oil Suspension

N-[(4-methoxy-6-methylpyrimidin-2-yl)aminocarbonyl]-1,4-dihydro-3-methyl-4-oxo-1-phenyl-indeno[1,2-C]pyrazole-5-sulfonamide:25%

polyoxyethylene sorbitol hexaoleate: 5%

highly aliphatic hydrocarbon oil: 70%

The ingredients are ground together in a sand mill until the solidparticles have been reduced to under about 5 microns. The resultingthick suspension may be applied directly, but preferably after beingextended with oils or emulsified in water.

EXAMPLE 22 Wettable Powder

N-[(4-methoxy-6-methylpyrimidin-2-yl)aminocarbonyl]-1,4-dihydro-3-methyl-4-oxo-1-phenyl-indeno[1,2-C]pyrazole-5-sulfonamide:20%

sodium alkylnaphthalenesulfonate: 4%

sodium ligninsulfonate: 4%

low viscosity methyl cellulose: 3%

attapulgite: 69%

The ingredients are thoroughly blended. After grinding in a hammer-millto produce particles essentially all below 100 microns, the material isreblended and sifted through a U.S.S. No. 50 sieve (0.3 mm opening) andpackaged.

EXAMPLE 23 Low Strength Granule

N-[(4,6-dimethoxy-1,3,5-triazin-2-yl)aminocarbonyl]-1,4-dihydro-3-methyl-4-oxo-1-phenyl-indeno[1,2-C]pyrazole-5-sulfonamide:1%

N,N-dimethylformamide: 9%

attapulgite granules (U.S.S. 20-40 sieve): 90%

The active ingredient is dissolved in the solvent and the solution issprayed upon dedusted granules in a double cone blender. After sprayingof the solution has been completed, the blender is allowed to run for ashort period and then the granules are packaged.

EXAMPLE 24 Aqueous Suspension

N-[(4-methoxy-6-methylpyrimidin-2-yl)aminocarbonyl]-1,4-dihydro-3-methyl-4-oxo-1-phenyl-indeno[1,2-C]pyrazole-5-sulfonamide:

polyacrylic acid thickener: 40%

dodecylphenol polyethylene glycol ether: 0.5%

disodium phosphate: 1%

monosodium phosphate: 0.5%

polyvinyl alcohol: 1.0%

water: 56.7%

The ingredients are blended and ground together in a sand mill toproduce particles essentially all under 5 microns in size.

EXAMPLE 25 Solution

N-[(4,6-dimethoxy-1,3,5-triazin-2-yl)aminocarbonyl]-1,4-dihydro-3-methyl-4-oxo-1-phenyl-indeno[1,2-C]pyrazole-5-sulfonamide,ammonium salt: 5%

water: 95%

The salt is added directly to the water with stirring to produce thesolution, which may then be packaged for use.

EXAMPLE 26 Low Strength Granule

N-[(4,6-dimethoxy-1,3,5-triazin-2-yl)aminocarbonyl]-1,4-dihydro-3-methyl-4-oxo-1-phenyl-indeno[1,2-C]pyrazole-5-sulfonamide:0.1%

attapulgite granules (U.S.S. 20-40 mesh): 99.9%

The active ingredient is dissolved in a solvent and the solution issprayed upon dedusted granules in a double-cone blender. After sprayingof the solution has been completed, the material is warmed to evaporatethe solvent. The material is allowed to cool and then packaged.

EXAMPLE 27 Granule

N-[(4-methoxy-6-methylpyrimidin-2-yl)aminocarbonyl]-1,4-dihydro-3-methyl-4-oxo-1-phenyl-indeno[1,2-C]pyrazole-5-sulfonamide:80%

wetting agent: 1%

crude ligninsulfonate salt (containing 5-20% of the natural sugars): 10%

attapulgite clay 9%

The ingredients are blended and milled to pass through a 100 meshscreen. This material is then added to a fluid bed granulator, the airflow is adjusted to gently fluidize the material, and a fine spray ofwater is sprayed onto the fluidized material. The fluidization andspraying are continued until granules of the desired size range aremade. The spraying is stopped, but fluidization is continued, optionallywith heat, until the water content is reduced to the desired level,generally less than 1%. The material is then discharged, screened to thedesired size range, generally 14-100 mesh (1410-149 microns), andpackaged for use.

EXAMPLE 28 High Strength Concentrate

N-[(4-methoxy-6-methylpyrimidin-2-yl)aminocarbonyl]-1,4-dihydro-3-methyl-4-oxo-1-phenyl-indeno[1,2-C]pyrazole-5-sulfonamide:99%

silica aerogel: 0.5%

synthetic amorphous silica: 0.5%

The ingredients are blended and ground in a hammer-mill to produce amaterial essentially all passing a U.S.S. No. 50 screen (0.3 mmopening). The concentrate may be formulated further if necessary.

EXAMPLE 29 Wettable Powder

N-[(4-methoxy-6-methylpyrimidin-2-yl)aminocarbonyl]-1,4-dihydro-3-methyl-4-oxo-1-phenyl-indeno[1,2-C]pyrazole-5-sulfonamide:90%

dioctyl sodium sulfosuccinate: 0.1%

synthetic fine silica: 9.9%

The ingredients are blended and ground in a hammer-mill to produceparticles essentially all below 100 microns. The material is siftedthrough a U.S.S. No. 50 screen and then packaged.

EXAMPLE 30 Wettable Powder

N-[(4,6-dimethoxy-1,3,5-triazin-2-yl)aminocarbonyl]-1,4-dihydro-3-methyl-4-oxo-1-phenyl-indeno[1,2-C]pyrazole-5-sulfonamide:40%

sodium ligninsulfonate: 20%

montmorillonite clay: 40%

The ingredients are thoroughly blended, coarsely hammer-milled and thenair-milled to produce particles essentially all below 10 microns insize. The material is reblended and then packaged.

EXAMPLE 31 Oil Suspension

N-[(4,6-dimethoxy-1,3,5-triazin-2-yl)aminocarbonyl]-1,4-dihydro-3-methyl-4-oxo-1-phenyl-indeno[1,2-C]pyrazole-5-sulfonamide:35%

blend of polyalcohol carboxylic esters and oil soluble petroleumsulfonates: 6%

xylene: 59%

The ingredients are combined and ground together in a sand mill toproduce particles essentially all below 5 microns. The product can beused directly, extended with oils, or emulsified in water.

EXAMPLE 32 Dust

N-[(4,6-dimethoxy-1,3,5-triazin-2-yl)aminocarbonyl]-1,4-dihydro-3-methyl-4-oxo-1-phenyl-indeno[1,2-C]pyrazole-5-sulfonamide:10%

attapulgite: 10%

Pyrophyllite: 80%

The active ingredient is blended with attapulgite and then passedthrough a hammer-mill to produce particles substantially all below 200microns. The ground concentrate is then blended with powderedpyrophyllite until homogeneous.

EXAMPLE 33 Emulsifiable Concentrate

N-[(4,6-dimethoxy-1,3,5-triazin-2-yl)aminocarbonyl]-1,4-dihydro-3-methyl-4-oxo-1-phenyl-indeno[1,2-C]pyrazole-5-sulfonamide:20%

chlorobenzene: 74%

sorbitan monostearate and polyoxyethylene condensates thereof: 6%

The ingredients are combined and stirred to produce a solution which canbe emulsified in water for application.

Utility

Test results indicate that the compounds of the present invention arehighly active preemergent or postemergent herbicides or plant growthregulants. Many of them have utility for broad-spectrum pre- and orpost-emergence weed control in areas where complete control of allvegetation is desired, such as around fuel storage tanks, ammunitiondepots, industrial storage areas, parking lots, drive-in theaters,around billboards, highway and railroad structures. Some of thecompounds have utility for selective weed control in crops such as rice,soybeans and wheat. Alternatively, the subject compounds are useful tomodify plant growth.

The rates of application for the compounds of the invention aredetermined by a number of factors, including their use as plant growthmodifiers or as herbicides, the crop species involved, the types ofweeds to be controlled, weather and climate, formulations selected, modeof application, amount of foliage present, etc. In general terms, thesubject compounds should be applied at levels of around 0.05 to 20kg/ha, the lower rates being suggested for use on lighter soils and/orthose having a low organic matter content, for selective weed control orfor situations where only short-term persistence is required.

The compounds of the invention may be used in combination with any othercommercial herbicide; examples of which are those of the triazine,triazole, uracil, urea, amide, diphenylether, carbamate and bipyridyliumtypes.

The herbicidal properties of the subject compounds were discovered in anumber of greenhouse tests. The test procedures and results follow.

TEST A

Seeds of crabgrass (Digitaria spp.), barnyardgrass (Echinochloacrusgalli), wild oats (Avena fatua), cheatgrass (Bromus secalinus),velvetleaf (Abutilon theophrasti), morningglory (Ipomoea spp.),cocklebur (Xanthium pennsylvanicum), sorghum, corn, soybean, sugarbeet,cotton, rice, wheat, and purple nutsedge (Cyperus rotundus) tubers wereplanted and treated preemergence with the test chemicals dissolved in anon-phytotoxic solvent. In some tests, velvetleaf and cheatgrass werenot included. At the same time, these crop and weed species were treatedwith a soil/foliage application. At the time of treatment, the plantsranged in height from 2 to 18 cm. Treated plants and controls weremaintained in a greenhouse for sixteen days, after which all specieswere compared to controls and visually rated for response to treatment.The ratings, summarized in Table A, are based on a numerical scaleextending from 0=no injury, to 10=complete kill. The accompanyingdescriptive symbols have the following meanings:

C=chlorosis/necrosis

B=burn

D=defoliation

E=emergence inhibition

G=growth retardation

H=formative effect

U=unusual pigmentation

X=axilliary stimulation

S=albinism

6Y=abscised buds or flowers.

    ______________________________________                                        COMPOUNDS                                                                     ______________________________________                                         ##STR66##                                                                    Compound R.sub.6       X        Y      Z                                      ______________________________________                                         1       C.sub.6 H.sub.5                                                                             OCH.sub.3                                                                              OCH.sub.3                                                                            N                                       2       C.sub.6 H.sub.5                                                                             OCH.sub.3                                                                              CH.sub.3                                                                             CH                                      3       CH.sub.3      CH.sub.3 CH.sub.3                                                                             CH                                      4       CH.sub.3      CH.sub.3 OCH.sub.3                                                                            CH                                      5       4-OCH.sub.3C.sub.6 H.sub.4                                                                  CH.sub.3 OCH.sub.3                                                                            CH                                      6       4-ClC.sub.6 H.sub.4                                                                         CH.sub.3 CH.sub.3                                                                             CH                                      7       4-ClC.sub.6 H.sub.4                                                                         Cl       OCH.sub.3                                                                            CH                                      8       4-ClC.sub.6 H.sub.4                                                                         OCH.sub.3                                                                              OCH.sub.3                                                                            CH                                      9       4-ClC.sub.6 H.sub.4                                                                         OCH.sub.3                                                                              OCH.sub.3                                                                            N                                      10       4-ClC.sub.6 H.sub.4                                                                         OCH.sub.3                                                                              CH.sub.3                                                                             CH                                     11       CH.sub.3      OCH.sub.3                                                                              CH.sub.3                                                                             N                                      12       CH.sub.3      OCH.sub.3                                                                              OCH.sub.3                                                                            CH                                     13       CH.sub.3      OCH.sub.3                                                                              OCH.sub.3                                                                            N                                      14       CH.sub.3      Cl       OCH.sub.3                                                                            CH                                     15       C.sub.6 H.sub.5                                                                             CH.sub.3 CH.sub.3                                                                             N                                      16       C.sub.6 H.sub.5                                                                             OCH.sub.3                                                                              OCH.sub.3                                                                            CH                                     17       C.sub.6 H.sub.5                                                                             OCH.sub.3                                                                              Cl     CH                                     18       C.sub.6 H.sub.5                                                                             OCH.sub.3                                                                              CH.sub.3                                                                             N                                      19       4-SO.sub.2 CH.sub.3C.sub.6 H.sub.4                                                          OCH.sub.3                                                                              OCH.sub.3                                                                            CH                                     20       4-SO.sub.2 CH.sub.3C.sub.6 H.sub.4                                                          OCH.sub.3                                                                              OCH.sub.3                                                                            N                                      21       4-SO.sub.2 CH.sub.3C.sub.6 H.sub.4                                                          CH.sub.3 CH.sub.3                                                                             CH                                     22       4-SO.sub.2 CH.sub.3C.sub.6 H.sub.4                                                          OCH.sub.3                                                                              CH.sub.3                                                                             CH                                     ______________________________________                                         ##STR67##                                                                     Compound    X          Y          Z                                          ______________________________________                                        23           OCH.sub.3  CH.sub.3   CH                                         24           OCH.sub.3  Cl         CH                                         25           OCH.sub.3  OCH.sub.3  N                                          ______________________________________                                         ##STR68##                                                                    Compound     X          Y          Z                                          ______________________________________                                        26           OCH.sub.3  OCH.sub.3  CH                                         27           OCH.sub.3  OCH.sub.3  N                                          ______________________________________                                         ##STR69##                                                                    Compound R.sub.6       X        Y      Z                                      ______________________________________                                        28       CH.sub.2 CH.sub.2 CH.sub.3                                                                  OCH.sub. 3                                                                             OCH.sub.3                                                                            CH                                     29       CH.sub.2 CH.sub.2 CH.sub.3                                                                  CH.sub.3 OCH.sub.3                                                                            CH                                     30       CH.sub.2 CH.sub.2 CH.sub.3                                                                  Cl       OCH.sub.3                                                                            CH                                     31       CH.sub.2 CH.sub.2 CH.sub.3                                                                  OCH.sub.3                                                                              OCH.sub.3                                                                            N                                      32       CH.sub.2 CH.sub.2 CH.sub.3                                                                  CH.sub.3 OCH.sub.3                                                                            N                                      33       CH.sub.3      Cl       OCH.sub.3                                                                            CH                                     34       CH.sub.3      CH.sub.3 CH.sub.3                                                                             CH                                     35       CH.sub.3      OCH.sub.3                                                                              OCH.sub.3                                                                            CH                                     36       CH.sub.3      CH.sub.3 OCH.sub.3                                                                            CH                                     37       CH.sub.3      CH.sub.3 OCH.sub.3                                                                            N                                      38       CH.sub.3      OCH.sub.3                                                                              OCH.sub.3                                                                            N                                      39       CH.sub.2 C.sub.6 H.sub.5                                                                    OCH.sub.3                                                                              OCH.sub.3                                                                            CH                                     40       CH.sub.2 C.sub.6 H.sub.5                                                                    CH.sub.3 OCH.sub.3                                                                            CH                                     41       CH.sub.2 C.sub.6 H.sub.5                                                                    CH.sub.3 CH.sub.3                                                                             CH                                     42       CH.sub.2 C.sub.6 H.sub.5                                                                    Cl       OCH.sub.3                                                                            CH                                     43       CH.sub.2 C.sub.6 H.sub.5                                                                    OCH.sub.3                                                                              OCH.sub.3                                                                            N                                      44       CH.sub.2 C.sub.6 H.sub.5                                                                    CH.sub.3 OCH.sub.3                                                                            N                                      45       3-FC.sub.6 H.sub.4                                                                          OCH.sub.3                                                                              OCH.sub.3                                                                            CH                                     46       3-FC.sub.6 H.sub.4                                                                          CH.sub.3 OCH.sub.3                                                                            CH                                     ______________________________________                                    

    TABLE A       Compound 1 Compound 2 Compound 3 Compound 4 Compound 5 Compound 6     Compound 7 Compound 8 Compound 9 Compound 10 Compound 11 Compound 12     Rate (kg/ha) 0.4 0.4 0.4 0.4 0.4 0.4 2.0 0.4 2.0 0.4 2.0 0.4 0.4 0.4     0.4   POSTEMERGENCE Morningglory 5C,9H 1C,4G 0 1C,5G 4G 0 0 0 0 0 0 0 0     0 5G Cocklebur 10C 5C,9H 3C,8H 5C,9H 2C,5H 0 0 0 0 0 0 3C,9H 0 8G,5H     5C,9H Velvetleaf 4C,9H 4C,8G 0 5C,9G 0 0 0 0 0 0 0 0 0 4G 5C,9H Nutsedge     2C,9G 0 0 0 0 0 0 0 0 0 0 0 0 0 5G Crabgrass 2C,5G 3G 0 2C,5G 0 0 0 0 0     0 0 0 0 0 0 Barnyardgrass 3C,9H 3C,8H 0 3C,9H 2C,6H 0 0 0 0 0 0 0 0     8G,3H 8H Cheatgrass 8G 3C,7G 0 2C,5G 0 0 0 0 0 0 0 0 0 0 6G Wild Oats 0     0 0 0 0 0 0 0 0 0 0 0 0 0 0 Wheat 3C,9G 0 0 3C,8G 0 0 0 0 0 0 0 0 0 5G     3G Corn 9C 3C,9H 0 5C,9H 0 0 0 0 0 0 0 0 0 5G,3H 9H Soybean 2G 0 0 2C,4H     1H 0 0 0 0 0 0 5G 0 0 3C,7G Rice 9C 6G 0 5C,9G 0 0 0 0 0 0 0 0 0 5G,3C     4C,9G Sorghum 5C,9H 3C,9H 0 5C,9H 0 0 0 0 0 0 0 0 0 7G,3H 2C,6H Sugar     Beets 5H 4C,9H 0 9C 3C,6G 0 0 0 0 2C,3H 0 0 2C,6G 3C 5H Cotton 3C,8H     4C,9H 0 2C,9G 5G 0 0 0 0 0 0 0 0 6G,3H 8H Bushbean Cassia Giant Foxtail     Sugar beet PREEMERGENCE Morningglory 2C,7H 2H 0 2C,3H 3C,5G 0 0 0 0 0 0     0 0 0 6G Cocklebur 9H 7H 8H 9H -- 0 0 0 0 0 0 2C 0 5G 8G Velvetleaf 7H     5G 0 8H 3G 0 0 0 0 0 0 0 0 0 8G Nutsedge 0 0 0 0 0 0 0 0 0 0 0 0 0 0 4G     Crabgrass 0 0 0 0 0 0 0 0 0 0 0 0 0 0 5G Barnyardgrass 3C,9H 5C,9H 0     2C,5H 3C,9H 0 0 2C 0 0 0 0 2C,8G 5G 9H Cheatgrass 5C,9H 2C,8G 0 3C,8G 7G     0 0 0 0 0 0 0 5G 0 4C,9G Wild Oats 5G 2C,6G 0 0 0 0 0 0 0 0 0 2G 0 0     2C,6G Wheat 5C,9H 8G 0 3C,9H 5G 0 0 0 0 0 0 5G 4G 7G 8G Corn 3C,8G 8H 0     3C,9G 4G 0 2C,8G 2 0 0 0 3G 0 3C 5G Soybean 0 0 0 0 2G 0 0 0 0 0 0 0 0 0     0 Rice 5C,9H 2C,7G 0 5C,9H 2C,5G 0 0 0 0 0 0 4G 4G 7G 8G Sorghum 5C,9H     9G 0 7C,9H 4C,9G 0 0 0 0 0 0 0 2C,6G 5G 8G Sugar Beets 6G 3C,8H 5G 5C,9G     8H 0 0 0 0 0 0 2G 5G 9C 8G Cotton 0 0 0 3C,4H 0 0 0 0 0 0 0 0 0 7C 5G     Bushbean Cassia Giant Foxtail Sugar beet               Com- Com- Com- Com- Com- Compound 13 Compound 14 Compound 15     Compound 16 Compound 17 Compound 18 Compound 19 Compound 20 pound 21     pound 22 pound 23 pound 24 pound 25 Rate (kg/ha) 0.4 0.4 0.4 0.05 0.4     0.05 0.4 0.05 0.4 0.05 0.4  0.4 0.4 0.4 0.4 0.4 2.0 0.4       POSTEMERGENCE Morningglory 3G 0 3C,7G 2C,4H 2C,4G 1C,1H 1H 0 9C 4C,9H     0 0  4G 0 0 0 0 3H Cocklebur 5G 5C,9H 5C,9G 4C,9G 3C,9H 3C,8H 5C,9G     3C,9H 10C 9C 0 0 0 0 5G,3C 3H 1C,5G 5G,5H Velvetleaf 3C,5H 5G 2C,6G 3G     3C,8G 2C,5G 3G 2G 5C,9G 3C,9G 0 0 0 0 6G 0 0 4G Nutsedge 0 0 0 0 0 0 0 0     9C 2C,9G 0 0 0 0 0 0 0 0 Crabgrass 3G 3G 2G 0 2G 0 0 0 3C,6G 2G 0 0 0 0     0 0 0 0 Barnyardgrass 0 2H 3C,9H 3C,8H 2C,8H 2C,7H 3C,9H 2C,5H 9C 4C,9H     0 0 0 0 6G,3H 0 0 0 Cheatgrass 0 0 2C,8G 0 2C,8G 2C,7G 0 0 4C,9G 4C,9G 0     0 0 0 0 0 0 0 Wild Oats 0 0 0 0 0 0 0 0 3G 0 0 0 0 0 0 0 0 0 Wheat 0 0     7G 0 7G 2G 0 0 3C,9G 9G 0 0 0 0 0 0 0 0 Corn 2U,5H 3H 3C,8H 3G 3C,9G     2C,8H 2C,6H 2C,6G 9C 9C 0 0 0 0 5G,3C 0 0 0 Soybean 0 0 2G 0 2G 0 0 0     2C,7G 2G 0 0 0 0 0 0 0 0 Rice 8G 3G 5C,9G 2C,6G 5C,9G 7G 4C,8H 7G 5C,9G     5C,9G 0 0 0 0 0 0 0 0 Sorghum 1C,4G 5G 4C,9H 3C,7H 4C,9H 2C,9H 1C,4G 1C     9C 4C,9H 0 0 0 0 0 0 0 0 Sugar Beets 2H 2H 4C,9G 3C,8H 3C,8H 2C,7H 3C,6H     3H 10C 9C 0 0 0 0 4G,3C 0 0 0 Cotton 5H 3G 2C,5H 2G 3C,8G 4G 1C,3G 3G     4C,9H 4C,9H 0 0 0 0 0 0 0 0 Bushbean                  Cassia          Giant Foxtail Sugar beet PREEMERGENCE Morningglory 0 6G 0 0 0 0 0 0 9     G 8G 0 0 0 2G 0 0 0 0 Cocklebur 5H 8H 8H 0 4G -- 2C,3H -- 8H 7H 0 -- 0 0     0 -- 0 0 Velvetleaf 4G 4G 0 0 1H 0 0 0 2C,9G 4G 0 0 0 0 0 0 0 0 Nutsedge     0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 Crabgrass 3G 5G 0 0 0 0 0 0 2C,5G 2G     0 0 0 0 0 0 0 0 Barnyardgrass 0 5G 2H 0 3C,8H 3C,3H 3C,7H 2C,2H 4C,9H     3C,6G 0 0 0 0 0 0 0 0 Cheatgrass 6G 0 0 0 8G 2G 5G 0 5C,9G 6G 0 0 0 0 0     0 0 0 Wild Oats 0 0 0 0 3G 0 0 0 2C,5G 1C 0 0 0 0 0 0 0 0 Wheat 8G 0 8G     0 8G 0 0 0 4C,9H 4C,9H 0 0 0 0 0 0 0 0 Corn 3C,3H 2G 2C,5G 0 8H 0 6G 4G     3C,5G 3C,7G 0 0 0 0 0 0 0 0 Soybean 0 0 0 0 0 0 0 0 2H 0 0 0 0 0 0 0 0 0     Rice 9H 2C,5G 3G 0 2C,4G 1C 6G 2G 4C,9H 2C,7G 0 0 0 0 0 0 0 0 Sorghum     4C,9G 8C,9H 4G 0 3C,9G 2C,6G 2C,8H 0 5C,9H 3C,9H 0 0 0 0 0 0 0 0 Sugar     Beets 5H 8H 8G 0 3G 0 6G 2H 5C,9G 5G 0 0 0 0 0 0 0 0 Cotton 0 9G 0 0 2G     0 0 -- 7G 0 0 0 0 0 0 0 0 0 Bushbean                  -- Cassia             -- Giant Foxtail Sugar beet           Cmpd.  Cmpd.     Com-  Compound 26 Compound 27 Compound 28     Compound 29 30 Cmpd. 31 32 Compound 33 Compound 34 Compound 35 Compound     36 pound 37 Compound 38 Rate (kg/ha) 0.05 0.01 0.05 0.01 0.4 0.05 0.4     0.05 0.05 0.05 0.05 0.4 0.05 0.4 0.05 0.4 0.05 0.4 0.05 0.4 0.05 0.4     0.05  POSTEMERGENCE Morningglory 9C 2C,7G 4C,8G 3C,8H 0 0 2C 1C 0 0 0 0     0 0 0 2G 2C,2H 1C 1C 0 0 0 0 Cocklebur 7H 3H 9H 4G 3C,8H 4C,9G 4C,9G     4C,9H 3C,7H 0 0 0 0 0 0 3C,9G 4C,9G 2C,3G 2C,4G 0 0 0 0 Velvetleaf 10C     9G 10C 4C,9G 3C,7G 2C,4G 3C,8H 2C,5G 0 0 0 0 0 0 0 3C,7G 2C,5G 1C 2C 0 0     0 0 Nutsedge 2C,8G 9G 9G 3C,8C 0 0 0 3G 0 0 0 0 0 0 0 3G 0 0 0 0 0 0 0     Crabgrass 7G 0 4G 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 Barnyardgrass     5C,9H 7H 10C 4H 0 0 0 3H 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 Cheatgrass 7G 5G     8G 2G 0 0 4G 5G 0 0 0 0 0 0 0 0 2C,6G 0 0 0 0 0 0 Wild Oats 2G 0 3C,7G     1C 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 Wheat 6G 0 0 0 0 0 4G 3G 0 0 0     0 0 0 0 0 0 0 0 0 0 0 0 Corn 5C,9G 4C,9G 3C,9H 3C,9H 4G 0 0 0 0 0 0 0 0     0 0 2C,5G 3C,8H 0 0 0 0 0 0 Barley 2C,6G 3G 4G 0 0 0 4G 0 0 0 0 -- -- --     -- -- -- -- -- -- -- -- --  Soybean 4C,9G 3C,8H 4C,9G 4C,9H 1C 1C 2C,3G     2C,3G 0 0 0 0 0 0 0 1C 2C,2H 0 0 0 0 0 0 Rice 5C,9G 3C,9G 5C,9G 4C,9G 0     0 0 0 0 0 0 0 0 0 0 2C,5G 3C,8G 0 0 0 0 0 0 Sorghum 2C,9G 3C,8H 4C,9H     2C,9H 4G 4G 3G 3G 2G 0 0 0 0 0 0 2C,3G 4C,9H 0 0 0 0 0 0 Sugar Beets     Cotton 4C,9G 8G 9C 4C,9G 3C,8G 3C,4G 3C,8H 3C,5G 2H 0 0 0 0 0 0 3C,8H     4C,9H 2C,5G 0 0 0 0 0 Bushbean Cassia Giant Foxtail 9C 8G 3C,9G 2C,4G 2G     0 0 0 3G 0 0 -- -- -- -- -- -- -- -- --  -- -- -- Sugar beet 5C,9G 7G     2C,9G 7H 2C,2H 3C,4G 3C,3H 3C,5G 0 0 0 0 0 0 0 3C,7G 4C,9G 2H 3C,5H 0 0     0 0 PREEMERGENCE Morningglory 9G 5G 9H 8G 0 0 3C 0 0 0 0 0 0 0 0 5G 0 6G 0      2G 0 2C,5G 0 Cocklebur 9H 5H -- 8H -- 3H 7G 2C -- 0 0 5G 0 0 0 8G 7G --     0 1H 0 0 0 Velvetleaf 9G 7G 3C,8G 6G 4G 0 2C,5G 0 0 0 0 0 0 0 0 5G 3G     2C,2H 0 0 0 0 0 Nutsedge 10E 6G 10E 0 0 0 0 0 0 0 0 0 0 0 0 2C,7G 0 0 0     0 0 0 0 Crabgrass 4G 2G 3G 0 0 0 0 0 0 0 0 0 0 0 0 2G 0 2C,5G 0 0 0 3G 0     Barnyardgrass 4C,9H 9H 9H 0 0 0 2C 0 0 0 0 0 0 0 0 2H 0 0 0 0 0 0 0     Cheatgrass 9H 9H 8H 5G 0 0 0 0 0 0 0 0 0 0 0 8G 0 2C,7G 0 0 0 0 0 Wild     Oats 2C,6G 2C 6G 0 0 0 0 0 0 0 0 0 0 0 0 2C,5G 0 0 0 0 0 0 0 Wheat 7G 8G     2G 0 0 0 0 0 0 0 0 0 0 0 0 8G 0 0 0 0 0 0 0 Corn 4C,9G 3C,9G 8H 2C,7G 0     0 0 0 0 0 0 0 0 0 0 2C,7G 0 2C,3G 0 0 0 0 0 Barley 9G 5G 8G 7G 0 0 0 0 0     0 0 -- -- -- -- -- -- -- -- -- --  -- -- Soybean 6H 3H 2C,5H 5H 0 0 1C 0     0 0 0 0 0 0 0 3G 0 0 0 0 0 0 0 Rice 10E 3C,9H 9H 7H 0 0 2G 0 0 0 2G 7G 0     0 0 3C,9G 0 3C,7G 0 3G 0 0 0 Sorghum 4C,9H 4C,9H 3C,9H 3C,8H 4G 3G 5G 0     0 0 0 5G 0 0 0 3C,9G 0 2C,4G 0 0 0 2G 0 Sugar Beets Cotton 9G 7G 9G 9G 0     0 2C 2G 0 0 0 0 0 0 0 6G 0 2C,2G 0 0 0 0 0 Bushbean Cassia Giant Foxtail     2C,9H 3C,6G 3H 0 0 0 2G 0 0 0 0 -- -- -- -- -- -- -- -- -- -- -- --     Sugar beet 9G 8G 8G 8G 9G 5G 9G 8G 5G 7G 5G 4G 0 0 0 4C,8G 0 5C,8G 0 2G     0 5G 0        Cmpd. 39 Cmpd. 40 Cmpd. 41 Cmpd. 42 Cmpd. 43 Cmpd. 44 Cmpd. 45 Cmpd.     46 Rate (kg/ha) 0.05 0.05 0.05 0.05 0.05 0.05 0.05 0.05       POSTEMERGENCE Morningglory 0 0 0 0 0 0 4C,8H 4C,9H Cocklebur 0 2H 0 0     0 0 10C 9C Velvetleaf 0 0 0 4G 0 0 4C,8H 4C,8H Nutsedge 0 0 0 0 0 0     3C,7G 3C,7G Crabgrass 0 0 0 0 0 0 0 0 Barnyardgrass 0 0 0 0 0 0 0 3C,7H     Cheatgrass 0 0 0 0 0 0 7G 3C,9G Wild Oats 0 0 0 0 0 0 3G 2C,5G Wheat 0 0     0 0 0 0 5G 3G Corn 0 0 0 0 0 0 1C,4G 3C,9H Barley 0 0 0 0 0 0 3C,7G     3C,9G Soybean 0 0 0 0 0 0 0 2G Rice 0 0 0 0 0 0 9C 4C,9G Sorghum 0 0 0 0     0 0 4C,9H 4C,9H Sugar Beets Cotton 0 0 0 0 0 0 4C,9G 9C Bushbean Cassia     Giant Foxtail 0 0 0 0 0 0 2G 3C,7G Sugar beet 0 0 0 0 0 0 9C 5C,9H     PREEMERGENCE Morningglory 0 0 0 0 0 0 2C,4G 2C,3G Cocklebur 0 0 0 0 0 0     8H 3C,7H Velvetleaf 0 0 0 0 0 0 8G 3C,6G Nutsedge 0 0 0 0 0 0 0 0     Crabgrass 0 0 0 0 0 0 0 1C Barnyardgrass 0 0 0 2G 0 0 2G 0 Cheatgrass 0     0 0 2G 0 0 2C,8G 3C,8G Wild Oats 0 0 0 0 0 0 0 3C,5G Wheat 0 0 0 3G 0 0     3G 7G Corn 0 0 0 7G 0 0 4G 2C,4G Barley 0 0 0 5G 0 0 4G 3G Soybean 0 0 0     0 0 0 2C,2H 0 Rice 0 0 0 5G 0 0 6G 3C,8G Sorghum 0 0 0 6G 0 0 2C,7G     3C,8H Sugar Beets Cotton 0 0 0 0 0 0 2G 3G Bushbean Cassia Giant Foxtail     0 0 0 3G 0 0 2G 2G Sugar beet 0 0 0 5G 0 0 8G 3C,8G

What is claimed is:
 1. A compound of the formula: ##STR70## wherein W isO or S;Q is ##STR71## G is CH₂, CH₂ CH₂, O, S, NH, NCH₃ or CH═CH; G₁ isCH₂, CH₂ CH₂ or CH═CH; J is CH₂, C═O, S(O)_(m), O, NH, NCH₃, CHOH,CHOCH₃, CH(CH₃) or C(CH₃)OH; J₁ is CH₂, C═O or SO₂ ; n and n₁ areindependently 0 or 1; m is 0, 1 or 2; E is a bridge of 3 or 4 atomscontaining 0 to 2 heteroatoms selected from the group consisting ofoxygen, sulfur or nitrogen, wherein 1 atom of sulfur may take the formof SO or SO₂, said bridge also containing 1 to 4 atoms of carbon wherein1 atom of carbon may take the form of C═O, said bridge together with twoattachment sites forming a non-aromatic heterocyclic or carbocyclic ringoptionally substituted by 1 to 3 substituent groups selected from thegroup L, or E is a bridge of 3 or 4 atoms containing 1-1 heteroatoms ofoxygen or sulfur and 0-3 heteroatoms of nitrogen, said bridge alsocontaining 0-4 atoms of carbon, said bridge together with two attachmentsites forming an aromatic heterocyclic or carbocyclic ring optionallysubstituted by 1 to 3 substituents selected from the group L, with theproviso that when E contains two oxygen atoms or two sulfur atoms saidatom must be separated by at least one atom of carbon and that oxygenand sulfur are only linked to each other if the sulfur is in the form ofSO or SO₂ ; L is C₁ -C₄ alkyl, C₁ -C₄ haloalkyl, C₁ -C₄ alkoxy, C₁ -C₄haloalkoxy, C₂ -C₈ alkoxyalkoxy, halogen, N(CH₃)₂, cyano, nitro, phenylor phenyl substituted with C₁ -C₃ alkyl, C₁ -C₃ haloalkyl, halogen, NO₂,C₁ -C₃ alkoxy, C₁ -C₃ alkylthio, C₁ -C₃ alkylsulfinyl or C₁ -C₃alkylsulfonyl;R is H or CH₃ ; R₁ is H, C₁ -C₃ alkyl, C₁ -C₃ haloalkyl,halogen, nitro, C₁ -C₃ alkoxy, SO₂ NR^(I) R^(II). C₁ -C₃ alkylthio, C₁-C₃ alkylsulfinyl, C₁ -C₃ alkylsulfonyl, CO₂ R^(III) or NR_(a) R_(b) ;R^(I) is H, C₁ -C₄ alkyl, C₂ -C₃ cyanoalkyl, methoxy or ethoxy; R^(II)is H, C₁ -C₄ alkyl or C₃ -C₄ alkenyl; or R^(I) and R^(II) may be takentogether as --(CH₂)₃ --, --(CH₂)₄ --, --(CH₂)₅ -- or --CH₂ CH₂ OCH₂ CH₂--; R^(III) is C₁ -C₄ alkyl, C₃ -C₄ alkenyl, C₃ -C₄ alkynyl, C₂ -C₄haloalkyl, C₁ -C₃ cyanoalkyl, C₅ -C₆ cycloalkyl, C₄ -C₇ cycloalkylalkylor C₂ -C₄ alkoxyalkyl; R_(a) and R_(b) are independently H or C₁ -C₂alkyl; A is ##STR72## X is H, C₁ -C₄ alkyl, C₁ -C₄ alkoxy, C₁ -C₄haloalkoxy, C₁ -C₄ haloalkyl, C₁ -C₄ haloalkylthio, C₁ -C₄ alkylthio,halogen, C₂ -C₅ alkoxyalkyl, C₂ -C₅ alkoxyalkoxy, amino, C₁ -C₃alkylamino or di(C₁ -C₃ alkyl)amino; Y is H, C₁ -C₄ alkyl, C₁ -C₄alkoxy, C₁ -C₄ haloalkoxy, haloalkylthio, C₁ -C₄ alkylthio, C₂ -C₅alkoxyalkyl, C₂ -C₅ alkoxyalkoxy, amino, C₁ -C₃ alkylamino, di(C₁ -C₃alkyl)amino, C₃ -C₄ alkenyloxy, C₃ -C₄ alkynyloxy, C₂ -C₅alkylthioalkyl, C₁ -C₄ haloalkyl, C₃ -C₅ cycloalkyl, C₂ -C₄ alkynyl,N(OCH₃)CH₃, ##STR73## p is 2 or 3; L₁ and L₂ are independently O or S;R₂ and R₃ are independently C₁ -C₂ alkyl; R₄ is H or CH₃ ; Z is CH;andtheir agriculturally suitable salts; provided that (a) when X is Cl, F,Br or I, then Y is OCH₃, OC₂ H₅, N(OCH₃)CH₃, NHCH₃, N(CH₃)₂ or OCF₂ H;(b) n and n₁ cannot simultaneously be O; (c) when G or G₁ is CH₂ CH₂ orCH═CH, then n is 0; (d) when Q is Q₁ and n is 1, then E must contain atleast one heteroatom selected from oxygen, sulfur or nitrogen; and (e)when W is S, then R is H, and Y is CH₃, OCH₃, OC₂ H₅, CH₂ OCH₃, C₂ H₅,CF₃, SCH₃, OCH₂ CH═CH₂, OCH₂ C.tbd.CH, OCH₂ CH₂ OCH₃, CH(OCH₃)₂##STR74##
 2. Compounds of claim 1 where W is O; G and G₁ are CH₂, CH₂CH₂ or CH═CH; J is CO, SO₂ or CH₂ ; R is H; X is CH₃, OCH₃, OCH₂ CH₃,Cl, F, Br, I, OCF₂ H, CH₂ F, OCH₂ CH₂ F, OCH₂ CHF₂, OCH₂ CF₃, CF₃, CH₂Cl or CH₂ Br; Y is H, CH₃, OCH₃, OC₂ H₅, CH₂ OCH₃, NHCH₃, N(OCH₃)CH₃,N(CH₃)₂, CH₂ CH₃, CF₃, SCH₃, OCH₂ CH═CH₂, OCH₂ C.tbd.CH, CH₂ OCH₂ CH₃,OCH₂ CH₂ OCH₃, CH₂ SCH₃, ##STR75## OCF₂ H, SCF₂ H, cyclopropyl, C.tbd.CHor or C.tbd.CCH₃.
 3. Compounds of claim 2 where R₁ is H, CH₃, halogen,OCH₃, SCH₃ or SO₂ CH₃ ; and L is halogen, CH₃, OCH₃, SCH₃, NO₂, N(CH₃)₂or phenyl.
 4. Compounds of claim 3 where Q is ##STR76## R₅ is H or C₃ ;R₆ is H, CH₃ or phenyl;R₇ is H or CH₃ ; R₈ is H or CH₃ ; R₉ is H, CH₃ orphenyl; R₁₀ is H or CH₃ ; R₁₁ is SCH₃, OCH₃, N(CH₃)₂ or CH₃ ; R₁₂ is Hor CH₃ ; R₁₃ is H, CH₃, OCH₃ or SCH₃ ; and R₁₄ is H, Cl, Br, F, CH₃,OCH₃ or NO₂.
 5. Compounds of claim 4 where X is CH₃, OCH₃, OCH₂ CH₃, Cl,OCF₂ H or OCH₂ CF₃ ; and Y is CH₃, OCH₃, CH₂ CH₃, CH₂ OCH₃, NHCH₃ orCH(OCH₃)₂.
 6. Compounds of claim 5 where n is O.
 7. Compounds of claim 5where n₁ is O.
 8. Compounds of claim 6 where Q is Q₁ -4, Q₁ -6, Q₁ -17,Q₁ -18, Q₁ -19, Q₁ -21, Q₁ -22, Q₁ -23, Q₂ -1 or Q₃ -1.
 9. Compounds ofclaim 7 where Q is Q₁ -2, Q₁ -3 or Q₁ -14.
 10. The compound of claim 1which isN-[(4,6-dimethoxypyrimidin-2-yl)aminocarbonyl]-1-phenyl-1H-[1]benzothieno[3,2-C]pyrazole-5-sulfonamide,4,4-dioxide.
 11. The compound of claim 1 which is4,5-dihydro-N-[(4,6-dimethoxypyrimidin-2-yl)aminocarbonyl]naphth[2,1-D]isoxazole-9sulfonamide.12. The compound of claim 1 which is4,5-dihydro-N-[(4-methoxy-6-methylpyrimidin-2-yl)aminocarbonyl]naphth[2,1-D]isoxazole-9-sulfonamide.13. A composition suitable for controlling the growth of undesiredvegetation which comprises an effective amount of a compound of claim 1and at least one of the following: surfactant, solid or liquid diluent.14. A composition suitable for controlling the growth of undesiredvegetation which comprises an effective amount of a compound of claim 2and at least one of the following: surfactant, solid or liquid diluent.15. A composition suitable for controlling the growth of undesiredvegetation which comprises an effective amount of a compound of claim 3and at least one of the following: surfactant, solid or liquid diluent.16. A composition suitable for controlling the growth of undesiredvegetation which comprises an effective amount of a compound of claim 4and at least one of the following: surfactant, solid or liquid diluent.17. A composition suitable for controlling the growth of undesiredvegetation which comprises an effective amount of a compound of claim 5and at least one of the following: surfactant, solid or liquid diluent.18. A composition suitable for controlling the growth of undesiredvegetation which comprises an effective amount of a compound of claim 6and at least one of the following: surfactant, solid or liquid diluent.19. A composition suitable for controlling the growth of undesiredvegetation which comprises an effective amount of a compound of claim 7and at least one of the following: surfactant, solid or liquid diluent.20. A composition suitable for controlling the growth of undesiredvegetation which comprises an effective amount of a compound of claim 8and at least one of the following: surfactant, solid or liquid diluent.21. A method for controlling the growth of undesired vegetation whichcomprises applying to the locus to be protected an effective amount of acompound of claim
 1. 22. A method for controlling the growth ofundesired vegetation which comprises applying to the locus to beprotected an effective amount of a compound of claim
 2. 23. A method forcontrolling the growth of undesired vegetation which comprises applyingto the locus to be protected an effective amount of a compound of claim3.
 24. A method for controlling the growth of undesired vegetation whichcomprises applying to the locus to be protected an effective amount of acompound of claim
 4. 25. A method for controlling the growth ofundesired vegetation which comprises applying to the locus to beprotected an effective amount of a compound of claim
 5. 26. A method forcontrolling the growth of undesired vegetation which comprises applyingto the locus to be protected an effective amount of a compound of claim6.
 27. A method for controlling the growth of undesired vegetation whichcomprises applying to the locus to be protected an effective amount of acompound of claim
 7. 28. A method for controlling the growth ofundesired vegetation which comprises applying to the locus to beprotected an effective amount of a compound of claim 8.